Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.523 productos)
- Apoptosis(5.792 productos)
- Ciclo celular / Checkpoint(4.449 productos)
- Cromatina / Epigenética(2.238 productos)
- Señalización citoesquelética(1.383 productos)
- Daño al ADN / Reparación del ADN(2.825 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.526 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.202 productos)
- Transportador de membrana / canal de iones(2.790 productos)
- Metabolismo(9.448 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.926 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.016 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66641 productos de "Inhibidores"
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N-Benzylnaltrindole hydrochloride
CAS:<p>δ2 opioid receptor antagonist</p>Fórmula:C33H33ClN2O3Pureza:98%Forma y color:SolidPeso molecular:541.08SIRT-IN-1
CAS:<p>SIRT-IN-1 is a potent SIRT1/2/3 inhibitor(IC50s of 15, 10, 33 μM, respectively).</p>Fórmula:C19H27N5O2SPureza:99.29%Forma y color:SolidPeso molecular:389.52ZINC08792355
CAS:<p>ZINC08792355 is a novel inhibitor of SIRT1.</p>Fórmula:C31H24N4O3Forma y color:SolidPeso molecular:500.55MC2590
CAS:<p>MC2590 is a histone deacetylase (HDAC) inhibitor that inhibits HDAC1-3, -6, -8, and -10 activities, induces cell cycle arrest, and promotes apoptosis.</p>Fórmula:C20H17N3O3Pureza:99.64%Forma y color:SolidPeso molecular:347.37DC 432
CAS:<p>DC 432, a potent peptidomimetic inhibitor of N-terminal methyltransferase 1/2 (NTMT1/2) with an IC50 value of 54 nM, incorporates a BM30 peptide enhanced by</p>Fórmula:C55H100N28O10Forma y color:SolidPeso molecular:1313.59ICMT-IN-23
CAS:<p>ICMT-IN-23 (compound 36) serves as an inhibitor of ICMT, exhibiting a half-maximal inhibitory concentration (IC50) of 0.123 μM [1].</p>Fórmula:C22H26N2OForma y color:SolidPeso molecular:334.45AL-38022A
CAS:<p>AL-38022A: selective 5-HT2 ligand, Ki ≤2.2 nM; >100-fold less binding to other 5-HT; minimal interaction with non-5-HT targets; full agonist.</p>Fórmula:C13H17N3OForma y color:SolidPeso molecular:231.29ATM-IN-1
CAS:<p>ATM-IN-1 is a potent inhibitor of ATM. ATM-IN-1 has shown research potential in cancer and neurological diseases.</p>Fórmula:C30H36N6O3Forma y color:SolidPeso molecular:528.65CI-949
CAS:<p>CI-949 inhibits LTC4/D4, histamine, TXB2 release (IC50: 0.5, 11.4, 0.1 μM).</p>Fórmula:C20H20N6O3Pureza:98%Forma y color:SolidPeso molecular:392.41ROCK2-IN-7
CAS:<p>ROCK2 inhibitor is a chemical compound associated with the therapeutic management of psoriasis.</p>Fórmula:C26H28FN5OPureza:98%Forma y color:SolidPeso molecular:445.53AZD1092
CAS:<p>AZD1092 is the glucokinase enzyme activator.</p>Fórmula:C24H26N4O5Pureza:98%Forma y color:SolidPeso molecular:450.49Lagociclovir valactate
CAS:<p>Lagociclovir valactate is a prodrug of Lagociclovir . Lagociclovir valactate is an orally active anti- HBV agent [1] .</p>Fórmula:C18H25FN6O6Forma y color:SolidPeso molecular:440.43Etiroxate
CAS:<p>Etiroxate (CG-635) is a lipid-lowering agent utilized in hyperlipoproteinemia studies [1].</p>Fórmula:C18H17I4NO4Forma y color:SolidPeso molecular:818.95ICMT-IN-24
CAS:<p>ICMT-IN-24 (compound 63) is an inhibitor of isoprenylcysteine carboxyl methyltransferase (ICMT), exhibiting potent activity with an IC50 value of 0.19 μM [1].</p>Fórmula:C22H28ClNO2Forma y color:SolidPeso molecular:373.92Antiproliferative agent-38
CAS:<p>Antiproliferative Agent-38 (COM 18), a tetracyclic compound, features a reactive ring nitrogen (likely the quinoline moiety) that resists N-alkylation.</p>Fórmula:C15H10N2Forma y color:SolidPeso molecular:218.25ICMT-IN-29
CAS:<p>ICMT-IN-29, also known as compound 66, effectively inhibits ICMT with an IC50 value of 0.019 μM [1].</p>Fórmula:C20H27NO2SForma y color:SolidPeso molecular:345.5Larixol
CAS:<p>Larixol acts as both an fMLP inhibitor and a modulator of various signaling pathways by inhibiting Src kinase, ERK1/2, p38, and AKT phosphorylation critical for</p>Fórmula:C20H34O2Pureza:98%Forma y color:SolidPeso molecular:306.48Kv3 modulator 4
CAS:<p>Kv3 modulator 4 is a Kv3.1 (pEC50=5.45) and Kv3.2 modulator .Cyclobutyl structure.</p>Fórmula:C20H24N2O4Pureza:98%Forma y color:SolidPeso molecular:356.42Anticancer agent 86
CAS:<p>Compound 6i, an anticancer agent, exhibits promising activity against breast adenocarcinoma [1].</p>Fórmula:C31H23Cl2N3O5Forma y color:SolidPeso molecular:588.44Fenquinotrione
CAS:<p>Fenquinotrione, a 4-hydroxyphenylpyruvate dioxygenase (HPPD) inhibitor, exhibits IC50 values of 27.2 and 44.7 nM against HPPD from rice and Arabidopsis thaliana</p>Fórmula:C22H17ClN2O5Forma y color:SolidPeso molecular:424.83A 56234
CAS:<p>A 56234 is a high-ceiling diuretic.</p>Fórmula:C16H9ClFKNO4Forma y color:SolidPeso molecular:372.8Gliamilide
CAS:<p>Gliamilide is a high-potency sulfamylurea hypoglycemic agent.</p>Fórmula:C23H33N5O5SForma y color:SolidPeso molecular:491.6WAY-659873
CAS:<p>WAY-659873 is an active molecule.</p>Fórmula:C19H17FN2O4S2Forma y color:SolidPeso molecular:420.48Microtubule Inhibitor 185322
CAS:<p>Microtubule inhibitor 185322 is an inhibitor of microtubule assembly, inducung mitotic arrest and apoptosis of MM cells.</p>Fórmula:C17H15NO3Forma y color:SolidPeso molecular:281.31AZD-9819
CAS:<p>AZD-9819 is an inhibitor of human neutrophil elastase for potential treatment of chronic obstructive pulmonary disease (COPD).</p>Fórmula:C25H19F3N6O2Pureza:99.18%Forma y color:SolidPeso molecular:492.45AS6
CAS:<p>AS6 is an ABA-induced PYL-PP2C interaction antagonist in a dose-dependent manner.</p>Fórmula:C21H32O4SPureza:98%Forma y color:SolidPeso molecular:380.54Elastase LasB-IN-1
CAS:<p>Elastase LasB-IN-1 (Compound 4b), a potent and selective inhibitor of elastase LasB, exhibits antibacterial activity and has been determined to possess an IC50</p>Fórmula:C13H17F3NO4PForma y color:SolidPeso molecular:339.25KFM19
CAS:<p>KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.</p>Fórmula:C16H22N4O3Pureza:98.62%Forma y color:SolidPeso molecular:318.37SGC agonist 1
CAS:<p>SGC agonist 1 is a potent soluble guanylate cyclase (SGC) agonist. SGC agonist 1 is able to increase solubility and has high cell permeability.</p>Fórmula:C22H19F2N7OForma y color:SolidPeso molecular:435.43ICMT-IN-17
CAS:<p>ICMT-IN-17 (compound 52) serves as an ICMT inhibitor, exhibiting an IC50 value of 0.38 μM [1].</p>Fórmula:C22H26F3NOForma y color:SolidPeso molecular:377.44Uplarafenib
CAS:<p>Uplarafenib (B-Raf IN 10), a potent BRAF inhibitor (IC50: 50-100 nM), exhibits antitumor effects on solid cancers.</p>Fórmula:C22H21F3N4O4SPureza:99.85%Forma y color:SolidPeso molecular:494.49JAK-IN-25
CAS:<p>JAK-IN-25 (compound 19), a potent JAK inhibitor, exhibits IC50 values of 6 nM for TYK2, 21 nM for JAK1, 8 nM for JAK2, and 1051 nM for JAK3.</p>Fórmula:C19H17N5O4Pureza:98%Forma y color:SolidPeso molecular:379.37JPI-547 HCl
CAS:<p>JPI-547 (NOV 1402) is an oral anti-cancer drug targeting PARP 1/2 and Tankyrase 1/2, effective alone or with chemo and immunotherapies.</p>Fórmula:C23H26Cl2N6OForma y color:SolidPeso molecular:473.402TRA 418
CAS:<p>TRA 418 is a TP antagonist.</p>Fórmula:C26H27NO4SForma y color:SolidPeso molecular:449.56Nitro-coronene
CAS:<p>Nitro-coronene-derived carbon dots can serve as lysosome-targeting agents for near-infrared light-induced photothermal cancer therapy research.</p>Fórmula:C24H8N4O8Forma y color:SolidPeso molecular:480.34CGP-49823
CAS:<p>CGP-49823 is a non-peptide tachykinin NK1 receptor antagonist.</p>Fórmula:C31H33N3OForma y color:SolidPeso molecular:463.61PM-43I
CAS:<p>PM-43I is a potent inhibitor of both STAT5- and STAT6-dependent allergic airway disease in mice.</p>Fórmula:C38H50F2N3O10PForma y color:SolidPeso molecular:777.79FPR2 agonist 3
CAS:<p>Compound CMC23, an FPR2 agonist, mitigates lactate dehydrogenase release in LPS-stimulated cultures and reduces pro-inflammatory IL-1β and IL-6 levels.</p>Fórmula:C25H20F2N4O2Forma y color:SolidPeso molecular:446.45S1PL-IN-31
CAS:<p>S1PL-IN-31 is a dual-function chemical compound acting as an inhibitor of sphingosine-1-phosphate (S1P) lyase with an IC50 value of 210 nM and as an antagonist</p>Fórmula:C26H23ClN6Forma y color:SolidPeso molecular:454.95MC-VC-PAB-NH2 TFA
CAS:<p>MC-VC-PAB-NH2 TFA is a cleavable linker for antibody-drug conjugates (ADCs) [1] utilized in their synthesis.</p>Fórmula:C33H47F3N8O10Forma y color:SolidPeso molecular:772.77ICMT-IN-28
CAS:<p>ICMT-IN-28 (compound 65) serves as an inhibitor of ICMT, exhibiting significant potency with an IC50 value of 0.008 μM [1].</p>Fórmula:C22H28FNO2Forma y color:SolidPeso molecular:357.46HDAC-IN-55
CAS:<p>HDAC-IN-55(8j) is a small-molecule inhibitor that enhances E-cadherin expression and suppresses cancer cell proliferation [1].</p>Fórmula:C17H17N3O3Pureza:98%Forma y color:SolidPeso molecular:311.34STING agonist-18
CAS:<p>STING Agonist-18 (Compound 1a) is a precursor for the synthesis of antibody-drug conjugates (ADCs), including Trastuzumab conjugates [1].</p>Fórmula:C38H45N13O6Forma y color:SolidPeso molecular:779.85Vemtoberant
CAS:<p>Vemtoberant is a β3 adrenergic antagonist used in β3-related disorder research like heart failure.</p>Fórmula:C29H37N3O8S2Forma y color:SolidPeso molecular:619.75B 581
CAS:<p>B 581 is an inhibitor that specifically blocks farnesylated.</p>Fórmula:C22H38N4O3S2Pureza:98%Forma y color:SolidPeso molecular:470.69UDM-001651
CAS:<p>UDM-001651: oral PAR4 antagonist, IC50=4 nM, Kd=1.4 nM, antiplatelet IC50=25 nM in γ-thrombin assay.</p>Fórmula:C28H23N3O5SPureza:98%Forma y color:SolidPeso molecular:513.56JBI-589
CAS:<p>JBI-589 is an isoform-selective, non-covalent inhibitor of PAD4 that diminishes CXCR2 expression and impedes neutrophil chemotaxis.</p>Fórmula:C29H28FN5OForma y color:SolidPeso molecular:481.56Paltimatrectinib
CAS:<p>Paltimatrectinib (PBI-200) is a tyrosine kinase inhibitor with anticancer activity, and is used in the study of bladder, breast, and colorectal cancers.</p>Fórmula:C20H15F5N6Pureza:99.96%Forma y color:SolidPeso molecular:434.37ARN-21934
CAS:<p>ARN-21934 inhibits human topoisomerase II α/β; IC50=2μM; stronger than Etoposide (IC50=120μM) in DNA relaxation.</p>Fórmula:C21H24N6Pureza:99.8%Forma y color:SolidPeso molecular:360.46Pazelliptine
CAS:<p>Pazelliptine is a DNA topoisomerase inhibitor and antitumor drug.</p>Fórmula:C22H27N5Forma y color:SolidPeso molecular:361.48
