Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.523 productos)
- Apoptosis(5.792 productos)
- Ciclo celular / Checkpoint(4.449 productos)
- Cromatina / Epigenética(2.238 productos)
- Señalización citoesquelética(1.383 productos)
- Daño al ADN / Reparación del ADN(2.825 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.526 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.202 productos)
- Transportador de membrana / canal de iones(2.790 productos)
- Metabolismo(9.448 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.926 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.016 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66641 productos de "Inhibidores"
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Lipid peroxidation inhibitor 1
CAS:<p>Lipid peroxidation inhibitor 1 is an inhibitor of lipid peroxidation (IC50: 0.07 μM).</p>Fórmula:C24H32N2OPureza:98%Forma y color:SolidPeso molecular:364.52NB-506 Free Base
CAS:<p>NB-506 Free Base is an indolocarbazole antitumor agent; a DNA topoisomerase I inhibitor.</p>Fórmula:C27H22N4O10Forma y color:SolidPeso molecular:562.48MY-673
CAS:<p>MY-673, a colchicine binding site inhibitor (CBSI), impedes tubulin polymerization and disrupts the ERK signaling pathway, consequently modulating SMAD4 protein</p>Fórmula:C18H14N2O4Forma y color:SolidPeso molecular:322.31WH-10417-099
CAS:<p>WH-10417-099 is a degrader capable of inducing the degradation of an extensive array of unique kinases, exceeding 125 in total [1].</p>Fórmula:C52H62N8O13SPureza:98%Forma y color:SolidPeso molecular:1039.16Bromodomain inhibitor-12 (edisylate)
CAS:<p>Bromodomain Inhibitor-12 Edisylate (example 303) serves as a bromodomain inhibitor applicable to autoimmune and inflammatory disease research [1].</p>Fórmula:C30H44N4O11S2Pureza:98%Forma y color:SolidPeso molecular:700.82Phentolamine Analogue 1
CAS:<p>Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.</p>Fórmula:C17H19N3OPureza:99.96%Forma y color:SolidPeso molecular:281.35LAS191954
CAS:<p>LAS191954 is a selective, potent and orally active PI3Kδ inhibitor for inflammatory diseases treatment(IC50 : 2.6 nM).</p>Fórmula:C20H15N9OPureza:98%Forma y color:SolidPeso molecular:397.39SB-743921 free base
CAS:<p>SB-743921, a kinesin spindle protein (KSP) inhibitor, is used potentially for the treatment of non-Hodgkin's lymphoma (NHL).</p>Fórmula:C31H33ClN2O3Pureza:98%Forma y color:SolidPeso molecular:517.06Testololactone
CAS:<p>Testololactone, an aromatase inhibitor, may be utilized in breast carcinoma research [1].</p>Fórmula:C19H26O3Forma y color:SolidPeso molecular:302.41AM-461
CAS:<p>AM-461 is a DP2 receptor antagonist.</p>Fórmula:C25H33NO5SForma y color:SolidPeso molecular:459.6Casein Kinase II Inhibitor IV
CAS:<p>Casein kinase II inhibitor IV is an effective small molecule inducer, which can be used to induce epidermal keratinocyte differentiation.</p>Fórmula:C24H23N5O3Pureza:99.65% - 99.75%Forma y color:SolidPeso molecular:429.47Angiogenesis inhibitor 4
CAS:<p>Angiogenesis Inhibitor 4 is a potent agent for inhibiting angiogenesis, with potential applications in cancer research [1].</p>Fórmula:C27H30ClN5O5Forma y color:SolidPeso molecular:540.01HDAC6-IN-8
CAS:<p>Compound 12C, with altered cap groups, shows wide-range enzyme inhibition; 9m and 9q target HDAC6 specifically.</p>Fórmula:C23H17BrFN5O3Pureza:98%Forma y color:SolidPeso molecular:510.32ONO 4817
CAS:<p>ONO-4817 suppresses MMPs, limiting plaque progression and aortic hyperplasia in hyperlipidemic rabbits.</p>Fórmula:C22H28N2O6Forma y color:SolidPeso molecular:416.47Osemozotan Free Base
CAS:<p>Osemozotan Free Base is a 5-HT(1A) receptor agonist.</p>Fórmula:C19H21NO5Forma y color:SolidPeso molecular:343.37SQ 26655
CAS:<p>SQ 26655 is an antagonist of thromboxane A2/prostaglandin H2.</p>Fórmula:C21H34O4Pureza:98%Forma y color:SolidPeso molecular:350.49AS-99
<p>AS-99, a potent ASH1L inhibitor with anti-leukemia effects, blocks cell growth and triggers apoptosis. IC50: 0.79µM; Kd: 0.89µM.</p>Fórmula:C27H31ClF3N5O3S2Forma y color:SolidPeso molecular:630.14Pumaprazole
CAS:<p>Pumaprazole (BY-841) is an antagonist of a reversible proton pump.</p>Fórmula:C19H22N4O2Pureza:99.91%Forma y color:SolidPeso molecular:338.4XZ426
CAS:<p>XZ426 is a potent integrase strand transfer inhibitor with anti- HIV activity .</p>Fórmula:C22H24F2N4O4Forma y color:SolidPeso molecular:446.45ZL0420
CAS:<p>ZL0420: Potent, selective BRD4 inhibitor, IC50 27 nM BD1 & 32 nM BD2.</p>Fórmula:C16H16N4O2Pureza:99.38%Forma y color:SolidPeso molecular:296.32PCSK9-IN-3
CAS:<p>PCSK9-IN-3 is a next-generation tricyclic peptide inhibitor of PCSK9, characterized by its novel structure, high potency, and oral bioavailability.</p>Fórmula:C83H105F4N15O17S2Forma y color:SolidPeso molecular:1724.94N-Demethyl Mifepristone
CAS:<p>N-Demethyl Mifepristone (RU 42633), an active metabolite of Mifepristone, exhibits 61% of the affinity for the glucocorticoid receptor relative to Mifepristone'</p>Fórmula:C28H33NO2Pureza:98%Forma y color:SolidPeso molecular:415.57HIV-1 protease-IN-9
CAS:<p>HIV-1 protease-IN-9 (compound 5b), a potent HIV-1 protease inhibitor, exhibits strong antiviral efficacy with a dissociation constant (K_i) of 0.028 nM and a</p>Fórmula:C37H41N7O4SPureza:98%Forma y color:SolidPeso molecular:679.83Tylvalosin
CAS:<p>Tylvalosin (Acetylisovaleryltylosin) is a broad-spectrum macrolide antibiotic with antibacterial and antiviral properties, effective against PRRSV infection.</p>Fórmula:C53H87NO19Pureza:98%Forma y color:SolidPeso molecular:1042.25NAS-181
CAS:<p>NAS-181 is a potent and selective rat 5-hydroxytryptamine 1B (r5-HT1B) antagonist (Ki: 47 nM).NAS-181 enhances the accumulation of 5-HTP in rat brain regions.</p>Fórmula:C20H30N2O7SForma y color:SolidPeso molecular:442.53LM-030
CAS:<p>LM-030, also known as BPR277, is a novel inhibitor of kallikrein-related peptidase 7 (KLK7) and epidermal elastase 2 (ELA2).</p>Fórmula:C46H72N8O12Forma y color:SolidPeso molecular:929.11Voruciclib hydrochloride
CAS:<p>Voruciclib hydrochloride is an orally active and selective inhibitor of CDK (Ki: 0.626 nM-9.1 nM).</p>Fórmula:C22H20Cl2F3NO5Pureza:98%Forma y color:SolidPeso molecular:506.3Androgen receptor antagonist 5
CAS:<p>AR antagonist 5 blocks AR (IC50: 6.17 μM), hinders LNCaP cell growth, and has anti-tumor effects in mouse models.</p>Fórmula:C21H15F4N5O3SForma y color:SolidPeso molecular:493.43TA-270
CAS:<p>TA-720, a 5-lipoxygenase inhibitor, is used potentially for the treatment of asthma.</p>Fórmula:C29H36N2O7Forma y color:SolidPeso molecular:524.61S-2E
CAS:<p>S-2E, an oral inhibitor of HMG-CoA reductase/acetyl-CoA carboxylase, treats hyperlipidemia.</p>Fórmula:C22H25NO4Forma y color:SolidPeso molecular:367.44PA-082
CAS:<p>PA-082: PPARγ partial agonist, boosts coactivator-1α, reduces triglycerides, enhances insulin signaling.</p>Fórmula:C33H38N2O5Forma y color:SolidPeso molecular:542.67IDP-73152 mesylate
CAS:<p>IDP-73152 mesylate is a peptide deformylase inhibitor.</p>Fórmula:C29H45F3N4O7SForma y color:SolidPeso molecular:650.76CJ-12255
CAS:<p>CJ-12255 is a Neurokinin-1 Receptor Antagonist.</p>Fórmula:C32H38N2O3Forma y color:SolidPeso molecular:498.66TLR7/8 agonist 9
CAS:<p>TLR7/8 agonist 9 (Compound 25a), exhibiting EC50 values of 40 nM and 23 nM for hTLR7 and hTLR8 respectively, demonstrates anti-tumor properties and enhances the</p>Fórmula:C20H26N6OForma y color:SolidPeso molecular:366.46Quorum Sensing-IN-2
CAS:<p>Quorum Sensing-IN-2 (compound 23e) is a quorum sensing inhibitor that curtails bacterial pathogenicity without impeding growth.</p>Fórmula:C19H13F2NO3Forma y color:SolidPeso molecular:341.31RPR-106541
CAS:<p>RPR-106541, a GR agonist, is used potentially for the treatment of asthma.</p>Fórmula:C24H34F2O4SForma y color:SolidPeso molecular:456.59Hydroxy Darunavir
CAS:<p>Hydroxy darunavir, a metabolite of the HIV-1 protease inhibitor darunavir, is generated through isobutyl aliphatic hydroxylation of darunavir.</p>Fórmula:C27H37N3O8SForma y color:SolidPeso molecular:563.66BMT-124110
CAS:<p>BMT-124110: AAK1 inhibitor, IC50=0.9 nM, pain relief. BMT-090605: BIKE inhibitor, IC50=17 nM; GAK inhibitor, IC50=99 nM.</p>Fórmula:C21H27N3O3Pureza:98.07%Forma y color:SolidPeso molecular:369.46DW10075
CAS:<p>DW10075, a novel potent and highly selective inhibitor of VEGFR, exhibits antitumor activities both in vitro and in vivo.</p>Fórmula:C29H23N5O3Forma y color:SolidPeso molecular:489.52PCSK9-IN-14
CAS:<p>PCSK9-IN-14, also known as compound Ia-8, is a potent inhibitor of PCSK9 [1].</p>Fórmula:C15H10F6N4O2Forma y color:SolidPeso molecular:392.26TM-N1324
CAS:<p>TM-N1324 is a GPR39 agonist; 280 nM potency without Zn2+, 9 nM with; similar effects on murine GPR39 (EC50s: 180 nM/5 nM).</p>Fórmula:C18H13ClFN7OPureza:99.88%Forma y color:SolidPeso molecular:397.79MSN8C
CAS:<p>MSN8C, a mansonone E analog, acts as a novel catalytic inhibitor of human DNA topoisomerase II, inducing apoptosis in cancer cells and exhibiting considerable</p>Fórmula:C13H10O3Forma y color:SolidPeso molecular:214.22CCT241533
CAS:<p>CCT241533 is an effective and selective ATP competitive inhibitor of CHK2 (Ki: 1.16 nM; IC50: 3 nM).</p>Fórmula:C23H27FN4O4Pureza:98%Forma y color:SolidPeso molecular:442.48MAO-B-IN-13
CAS:<p>MAO-B-IN-13: a potent, reversible MAO-B inhibitor with BBB penetration, neuroprotective effects; used in Parkinson’s research (IC50=10nM).</p>Fórmula:C18H19NO3Forma y color:SolidPeso molecular:297.35HBF-0259
CAS:HBF-0259 is an inhibitors of hepatitis B virus surface antigen (HBsAg) secretion with an EC50 of 11.3 μM and a CC50 value of >50 μM in HepG2.2.15 cells.Fórmula:C16H12Cl2FN5Pureza:98.07% - 99.42%Forma y color:SolidPeso molecular:364.2DGKζ-IN-4
CAS:<p>DGKζ-IN-4 is a DGK-zeta inhibitor employed as an active ingredient in pharmaceutical formulations designed to treat cancers linked to immune cell activation or</p>Fórmula:C23H25ClF3N3O6Forma y color:SolidPeso molecular:531.91RSV L-protein-IN-5
CAS:<p>RSV L-protein-IN-5 (Compound E) serves as a potent inhibitor of the Respiratory Syncytial Virus (RSV), with an EC50 value of 0.1 μM.</p>Fórmula:C31H36N6O4Pureza:98%Forma y color:SolidPeso molecular:556.66Ubiquitination-IN-1
CAS:<p>Ubiquitination-IN-1 is an inhibitor of ubiquitination and Cksl-Skp2 protein-protein interaction (IC50: 0.17 μM).</p>Fórmula:C21H14F3N3O2SPureza:98.396% - 99.88%Forma y color:SolidPeso molecular:429.42Mevociclib
CAS:<p>Mevociclib (SY-1365) is a highly selective covalent inhibitor of CDK7. SY-1365 possesses therapeutic potential in both hematological and solid tumors.</p>Fórmula:C31H35ClN8O2Pureza:98.02% - 98.02%Forma y color:SolidPeso molecular:587.11h15-LOX-2 inhibitor 1
CAS:<p>Compound 105 (h15-LOX-2 inhibitor 1) is a potent inhibitor of human epithelial 15-lipoxygenase-2 (h15-LOX-2), exhibiting an IC50 of 0.34 μM [1].</p>Fórmula:C17H13F3N2SPureza:98%Forma y color:SolidPeso molecular:334.36
