Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.523 productos)
- Apoptosis(5.792 productos)
- Ciclo celular / Checkpoint(4.449 productos)
- Cromatina / Epigenética(2.238 productos)
- Señalización citoesquelética(1.383 productos)
- Daño al ADN / Reparación del ADN(2.825 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.526 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.202 productos)
- Transportador de membrana / canal de iones(2.790 productos)
- Metabolismo(9.448 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.926 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.016 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66641 productos de "Inhibidores"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
AZD-1386
CAS:<p>AZD1386: oral TRPV1 receptor antagonist. Info from NIH/NCATS and DrugBank.</p>Fórmula:C21H23F2N3OForma y color:SolidPeso molecular:371.42A-371191
CAS:<p>A-371191 is an antagonist of Bcl-XL.</p>Fórmula:C36H47N5O5S2Pureza:98%Forma y color:SolidPeso molecular:693.922-Ethynyl Adenosine
CAS:<p>2-Ethynyl Adenosine, Adenosine derivative, tracks novel polyadenylated transcription, non-radioactive AMPylation reporter.</p>Fórmula:C12H13N5O4Forma y color:SolidPeso molecular:291.26NTRC 0066-0
CAS:<p>NTRC 0066-0 is a TTK inhibitor that can be used in cancer research.</p>Fórmula:C33H39N7O2Pureza:98.30%Forma y color:SolidPeso molecular:565.71FD1024
CAS:<p>FD1024 is a potent PIM inhibitor, displaying inhibitory concentrations (IC50s) of 1.96 nM, 38.9 nM, and 4.17 nM for PIM1, PIM2, and PIM3, respectively.</p>Fórmula:C21H20F2N4O2SPureza:98%Forma y color:SolidPeso molecular:430.47CS-526
CAS:<p>CS-526 is a reversible proton pump inhibitor targeting the K+ site on H+,K+-ATPase, reducing gastric acid secretion and preventing mucosal lesions.</p>Fórmula:C20H22FN3OForma y color:SolidPeso molecular:339.41KCL-286
CAS:<p>KCL-286 is an available and potent retinoic acid receptor beta agonist for the amelioration of spinal cord injury (SCI).</p>Fórmula:C19H14N2O4Pureza:99.93%Forma y color:SolidPeso molecular:334.33Nezulcitinib
CAS:<p>Nezulcitinib (TD-0903) is an inhaled pan-JAK inhibitor targeting COVID-19-related acute lung injury.</p>Fórmula:C30H37N7O2Forma y color:SolidPeso molecular:527.66SIRT-IN-1
CAS:<p>SIRT-IN-1 is a potent SIRT1/2/3 inhibitor(IC50s of 15, 10, 33 μM, respectively).</p>Fórmula:C19H27N5O2SPureza:99.29%Forma y color:SolidPeso molecular:389.52LY 53857
CAS:<p>LY 53857 is a potent and selective antagonist of 5-HT2 serotonin receptor.</p>Fórmula:C27H36N2O7Forma y color:SolidPeso molecular:500.592GRL-8234
CAS:<p>GRL-8234 is a small-molecule BACE1 inhibitor that reverses memory impairments and age-related cognitive decline.</p>Fórmula:C36H42N4O6SForma y color:SolidPeso molecular:658.81Deltakephalin
CAS:<p>Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.</p>Fórmula:C34H48N6O10Pureza:98%Forma y color:SolidPeso molecular:700.78WAY-639872
CAS:<p>WAY-639872 is an active molecule exhibiting (in vivo) efficacy.</p>Fórmula:C21H21N3O3Forma y color:SolidPeso molecular:363.41GSK2646264
CAS:<p>GSK2646264 (Compound 44) inhibits SYK (pIC50=7.1) and kinases like LCK, LRRK2; penetrates skin.</p>Fórmula:C24H26N2O2Forma y color:SolidPeso molecular:374.48RG 14893
CAS:<p>RG 14893 is a antagonist of high-affinity leukotriene B4 receptor.</p>Fórmula:C29H27NO4Pureza:98%Forma y color:SolidPeso molecular:453.53WAY-312491
CAS:<p>WAY-312491 is an active compound.</p>Fórmula:C21H24FN3O3SForma y color:SolidPeso molecular:417.5MAC13772
CAS:<p>MAC13772 is a potent inhibitor of the enzyme BioA with an IC50 of 250 nM thereby inhibiting biotin biosynthesis. MAC13772 exhibits antibacterial activity.</p>Fórmula:C8H9N3O3SPureza:98.7%Forma y color:SolidPeso molecular:227.24hMAO-B-IN-32
CAS:<p>hMAO-B-IN-32 is a potent hMAO-B selective inhibitor with an IC50 of 45.52 μM.</p>Fórmula:C16H19NO4Pureza:99.65%Forma y color:SolidPeso molecular:289.33SNJ-1945
CAS:<p>SNJ-1945: Calpain inhibitor, enhances retinal penetration, oral bioavailability, long half-life, protects cells, solubility.</p>Fórmula:C25H37N3O7Forma y color:SolidPeso molecular:491.58Butaprost free acid
CAS:<p>(R)-Butaprost (free acid) is a prostaglandin E2 (PGE2) analog exhibiting high EP2 receptor subtype selectivity, commonly used to delineate EP receptor</p>Fórmula:C23H38O5Forma y color:SolidPeso molecular:394.54O-Benzoylhydroxylamine
CAS:<p>O-Benzoyl hydroxylamine exhibits properties as a dipeptidyl peptidase-IV (DPP-IV) inhibitor and demonstrates antidiabetic effects[1].</p>Fórmula:C7H7NO2Forma y color:SolidPeso molecular:137.14IDH1 Inhibitor 7
CAS:<p>IDH1 Inhibitor 7 is an IDH1 inhibitor with an IC 50 of less than 100 nM .</p>Fórmula:C22H24F3N7OForma y color:SolidPeso molecular:459.47Rohitukine
CAS:<p>Rohitukine: anticancer, modulates apoptosis, antiadipogenic, antidyslipidemic, gastroprotective, antifertility, antileishmanial.</p>Fórmula:C16H19NO5Forma y color:SolidPeso molecular:305.33ABT-255
CAS:<p>ABT-255: novel 2-pyridone antimicrobial for tuberculosis, effective against drug-sensitive/resistant Mycobacterium tuberculosis in vitro/in vivo.</p>Fórmula:C21H24FN3O3Forma y color:SolidPeso molecular:385.43CRF1 receptor antagonist-1
CAS:<p>CRF1 Receptor Antagonist-1 (Compound 2), a CRF1 receptor antagonist, is utilized in research pertaining to congenital adrenal hyperplasia (CAH) [1].</p>Fórmula:C27H28ClFN2O2SPureza:98%Forma y color:SolidPeso molecular:499.04Cgp 6809
CAS:<p>CGP 6809: a methylnitrosoureido-sugar derivative active against various mice/rat tumors; promising for bowel/lung cancer trials.</p>Fórmula:C12H23N3O7Forma y color:SolidPeso molecular:321.33eIF4A i28
CAS:<p>eIF4A i28, an inhibitor of the eukaryotic initiation factor-4A (eIF4A) with an IC50 of 8.60 μM in an eIF4A ATPase assay, effectively reduces the viability of</p>Fórmula:C24H20N2O5Forma y color:SolidPeso molecular:416.43Org 43553
CAS:<p>Org 43553: oral LMW LH-R agonist; targets LH (EC50: 3.7nM) & FSH (EC50: 110nM); useful for endocrine research.</p>Fórmula:C24H30N6O3S2Forma y color:SolidPeso molecular:514.66JNJ-17148066
CAS:<p>JNJ-17148066 is an agonist of estrogen receptor ESR1.</p>Fórmula:C30H31NO5Pureza:98%Forma y color:SolidPeso molecular:485.57Atiprimod (free base)
CAS:<p>Atiprimod: an oral azaspirane inhibiting STAT3, blocking IL-6/VEGF pathways, and promoting apoptosis by downregulating Bcl-2 and Mcl-1.</p>Fórmula:C22H44N2Forma y color:SolidPeso molecular:336.6H3 receptor antagonist 1
CAS:<p>H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.</p>Fórmula:C20H28F2N2OPureza:98%Forma y color:SolidPeso molecular:350.45CBB1007
CAS:<p>CBB1007 is a potent, reversible, and substrate competitive LSD1 inhibitor (IC50: 5.27 μM for hLSD1).</p>Fórmula:C27H34N8O4Pureza:98%Forma y color:SolidPeso molecular:534.61Valyl-glycyl-arginine-4-nitroanilide
CAS:<p>Valyl-glycyl-arginine-4-nitroanilide is a tissue plasminogen activator.</p>Fórmula:C19H30N8O5Forma y color:SolidPeso molecular:450.49FT206
CAS:<p>FT206 is a carboxamide inhibitor of ubiquitin-specific protease[1].</p>Fórmula:C25H29N5OSForma y color:SolidPeso molecular:447.6ST8155AA1
CAS:<p>ST8155AA1, a component of antibody-drug conjugates (ADCs), is tethered to an HDAC inhibitor via a linker and exhibits antitumor activity [1].</p>Fórmula:C43H62N8O9SForma y color:SolidPeso molecular:867.07BMS-186511
CAS:<p>BMS-186511: An FT inhibitor targeting malignant cells in NF1, halting growth and spread without affecting related enzymes.</p>Fórmula:C34H60N3O7PSForma y color:SolidPeso molecular:685.89PK68
CAS:<p>PK68 selectively inhibits RIPK1 (IC50=90nM), potentially useful in inflammation and cancer metastasis studies.</p>Fórmula:C22H24N4O3SPureza:98.09% - 99.64%Forma y color:SolidPeso molecular:424.52HDAC-IN-46
CAS:<p>HDAC-IN-46 inhibits HDAC1 & HDAC6, affects p-p38, Bcl-xL & cyclin D1, blocks G2 phase & induces apoptosis in TNBC research.</p>Fórmula:C22H30N8O2Forma y color:SolidPeso molecular:438.53Fenpropidin
CAS:<p>Fenpropidin (Ro-12-3049), a fungicide, is a specific inhibitor of sterol 14-reductase and biosynthesis.</p>Fórmula:C19H31NPureza:98.58% - 99.54%Forma y color:SolidPeso molecular:273.46BI-10N
CAS:<p>BI-10N is an effective Interleukin-2 inducible T-cell kinase antagonist.</p>Fórmula:C26H34N6O2SPureza:98%Forma y color:SolidPeso molecular:494.65hCAIX/XII-IN-8
CAS:<p>hCAIX/XII-IN-8 (compound 3g) is a potent inhibitor of the human carbonic anhydrases (CAs) IX and XII, with inhibition constants (K i) of 8.5 nM for CA IX and 6.</p>Fórmula:C16H13Cl2N5O3SPureza:98%Forma y color:SolidPeso molecular:426.28SCH-39370
CAS:<p>SCH-39370 is a potent and specific neutral metalloendopeptidase (NEP) inhibitor.</p>Fórmula:C22H26N2O6Forma y color:SolidPeso molecular:414.45L 691121
CAS:<p>L 691121 is a class III antiarrhythmic compound. It also blocks potassium currents.</p>Fórmula:C22H25ClN4O5SPureza:98%Forma y color:SolidPeso molecular:492.98CycLuc1
CAS:<p>CycLuc1 is a brain penetrant luciferase substrate.</p>Fórmula:C13H11N3O2S2Pureza:98.38%Forma y color:SolidPeso molecular:305.38NSC 288387
CAS:<p>NSC 288387, a pan-flavivirus MTase inhibitor, binds to the SAM-binding pocket and effectively inhibits Zika virus (ZIKV) with an IC50 of 0.2 μM, also preventing</p>Fórmula:C19H16N4O3Pureza:98%Forma y color:SolidPeso molecular:348.36H 142-08
CAS:<p>H 142-08 is a partial beta 1-agonist with adrenoreceptor stimulatory effects.</p>Fórmula:C22H37N3O6Forma y color:SolidPeso molecular:439.55CR-6086
CAS:<p>CR6086: potent EP4 antagonist with DMARD effects, low Ki (16.6 nM), and specific anti-inflammatory action.</p>Fórmula:C26H27F3N2O3Forma y color:SolidPeso molecular:472.5Oseltamivir acid methyl ester
CAS:<p>Oseltamivir acid methyl ester, a CES1-convertible neuraminidase inhibitor, serves as an antiviral prodrug.</p>Fórmula:C15H26N2O4Pureza:98.78%Forma y color:SolidPeso molecular:298.387-Aminomethyl-10-methyl-11-fluoro camptothecin
CAS:<p>7-Aminomethyl-10-methyl-11-fluoro camptothecin, serving as a cytotoxic component of the antibody-drug conjugate (ADC) MC-AAA-NHCH2OCH2COO-7-aminomethyl-10-</p>Fórmula:C22H20FN3O4Forma y color:SolidPeso molecular:409.41(+)-Apogossypol
CAS:<p>(+)-Apogossypol is an antagonist of pan-BCL-2. (+)-Apogossypol binds to Mcl-1(Bcl-2 and Bcl-xL with EC50s of 2.6, 2.8 and 3.69 μM, respectively).</p>Fórmula:C28H30O6Pureza:98%Forma y color:SolidPeso molecular:462.53
