Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.523 productos)
- Apoptosis(5.792 productos)
- Ciclo celular / Checkpoint(4.449 productos)
- Cromatina / Epigenética(2.238 productos)
- Señalización citoesquelética(1.383 productos)
- Daño al ADN / Reparación del ADN(2.825 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.526 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.202 productos)
- Transportador de membrana / canal de iones(2.790 productos)
- Metabolismo(9.448 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.926 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.016 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66641 productos de "Inhibidores"
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Azilsartan mopivabil
CAS:<p>Azilsartan mopivabil is the potent antagonist of angiotensin II receptor .</p>Fórmula:C38H36N4O8Forma y color:SolidPeso molecular:676.71Difethialone
CAS:<p>Difethialone is an anticoagulant rodenticide and a vitamin K antagonist.</p>Fórmula:C31H23BrO2SForma y color:SolidPeso molecular:539.48WYE-23
CAS:<p>WYE-23 is an inhibitor of mammalian target of rapamycin (mTOR).</p>Fórmula:C26H32N8O4Forma y color:SolidPeso molecular:520.58AR-13503
CAS:<p>AR-13503, a Netarsudil metabolite, is a ROCK inhibitor, potentially treating glaucoma and lowering eye pressure.</p>Fórmula:C19H19N3O2Forma y color:SolidPeso molecular:321.37F1874-108
CAS:<p>F1874-108 functions as an inhibitor of both brassinosteroid biosynthesis and signal transduction [1].</p>Fórmula:C15H14N4O2SForma y color:SolidPeso molecular:314.36FK-1052
CAS:<p>FK-1052 is a serotonin 3 & 4 dual receptor antagonist.</p>Fórmula:C18H19N3OForma y color:SolidPeso molecular:293.36AC-4
CAS:<p>AC-4 is a blocker of photoswitchable TRPV1 channel.</p>Fórmula:C26H25F3N4O2SForma y color:SolidPeso molecular:514.56Pactimibe
CAS:<p>Pactimibe is a ACAT inhibitor. It has anti-atherosclerotic activity.</p>Fórmula:C25H40N2O3Forma y color:SolidPeso molecular:416.6BIM-46068
CAS:<p>BIM-46068 is a potent inhibitor of human farnesyltransferase with a unique anti-proliferative profile.</p>Fórmula:C21H42N4O3S3Forma y color:SolidPeso molecular:494.78N-Acetylpurinomycin
CAS:<p>N-Acetylpurinomycin is a selective agonist of CB2 receptor.</p>Fórmula:C24H31N7O6Forma y color:SolidPeso molecular:513.55AEW541 HCl
CAS:<p>AEW541 (CAS# 475489-16-8) is a selective IGF-IR kinase inhibitor (IC50: IGF-IR=0.086μM, InsR=2.3μM), blocking IGF-I effects and colony formation.</p>Fórmula:C27H31Cl2N5OForma y color:SolidPeso molecular:512.47NGD9002
CAS:<p>NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.</p>Fórmula:C20H31N5OPureza:98%Forma y color:SolidPeso molecular:357.49RIOK2-IN-1
CAS:<p>RIOK2-IN-1 (com 4) is a selective RIOK2 inhibitor with a Kd of 150 nM, though it demonstrates low cellular activity with an IC50 of 14,600 nM.</p>Fórmula:C18H16N2OForma y color:SolidPeso molecular:276.33Spr 210
CAS:<p>Spr 210 is an aldose reductase (AR) inhibitor with potential uses as a therapeutic agent for preventing and improving some diabetic complications.</p>Fórmula:C18H11F3N2O3S2Forma y color:SolidPeso molecular:424.423β-Hydroxy-lup-20(29)-en-16-one
CAS:<p>3β-Hydroxy-lup-20(29)-en-16-one (compound 9) serves as a dual inhibitor of both AChE and BChE, displaying a preference for BChE with an IC50 of 28.9 μM [1].</p>Fórmula:C30H48O2Forma y color:SolidPeso molecular:440.73-Hydroxyxanthone
CAS:<p>3-Hydroxyxanthone (3-Hydroxy-xanthen-9-one), a xanthone derivative, exhibits inhibitory effects on NADPH-catalyzed lipid peroxidation in human umbilical vein</p>Fórmula:C13H8O3Pureza:98%Forma y color:SolidPeso molecular:212.2BD-AcAc 2
CAS:<p>BD-AcAc 2 (Ketone Ester) is a ketone monoester and can be used as a source of oral nutritional ketones.</p>Fórmula:C8H16O4Pureza:99.62%Forma y color:SolidPeso molecular:176.21PHD2/HDACs-IN-1
CAS:<p>PHD2/HDACs-IN-1: strong PHD2/HDAC inhibitor (IC50: 1.15-26.60 μM), low-toxicity, protects kidneys from cisplatin-induced AKI.</p>Fórmula:C18H19N9O4Forma y color:SolidPeso molecular:425.4Cenerimod
CAS:<p>Cenerimod (ACT-334441) is an S1P1 agonist used in the study of murine experimental autoimmune encephalomyelitis (EAE) and murine scleroderma.</p>Fórmula:C25H31N3O5Pureza:97.43% - 99.97%Forma y color:SolidPeso molecular:453.53GSK-2485852
CAS:<p>GSK-2485852, a NS5B inhibitor, is used potentially for treatment of HCV infection.</p>Fórmula:C27H25BF2N2O6SForma y color:SolidPeso molecular:554.37K-8986
CAS:<p>K-8986 is a novel h1-receptor antagonist</p>Fórmula:C32H41N5O7SForma y color:SolidPeso molecular:639.768CD38 inhibitor 2
CAS:<p>CD38 inhibitor 2 is a potent CD38 inhibitor ( IC 50 = 0.01 ~ 0.1 μΜ).</p>Fórmula:C19H24N6O3Forma y color:SolidPeso molecular:384.43SOS1-IN-8
CAS:<p>SOS1-IN-8 is an inhibitor of SOS1 and acts on SOS1-G12D (IC50: 11.6 nM) and SOS1-G12V (IC50: 40.7 nM).</p>Fórmula:C24H26F3N3O4Forma y color:SolidPeso molecular:477.48CT1113
CAS:<p>CT1113, a potent inhibitor of both USP28 and USP25, effectively reduces MYC levels in vivo and demonstrates anti-tumor efficacy in a mouse pancreatic cancer CDX</p>Fórmula:C25H29N5O2SForma y color:SolidPeso molecular:463.6NCQ-469
CAS:<p>NCQ-469 is a metabolite of remoxipride and a dopamine D2 receptor antagonist.</p>Fórmula:C16H23BrN2O4Forma y color:SolidPeso molecular:387.27NC1
CAS:<p>NC1 is a potent allosteric inhibitor of lymphoid-specific PTPN22, a protein tyrosine phosphatase.</p>Fórmula:C29H26N2O7SForma y color:SolidPeso molecular:546.59Sigma-1 receptor antagonist 1
CAS:<p>Sigma-1 receptor antagonist 1 is an effective and selective antagonist of sigma-1 receptor.</p>Fórmula:C19H23Cl2N3OPureza:99.92%Forma y color:SolidPeso molecular:380.31(1R)-Deruxtecan
CAS:<p>Deruxtecan (1R) is a drug-linker conjugate for antibody-drug conjugates (ADC) [1].</p>Fórmula:C52H56FN9O13Forma y color:SolidPeso molecular:1034.05Carbidine dihydrochloride
CAS:<p>Carbidine, a gamma-carboline derivative, is an atypical antipsychotic that modulates dopamine release and tyrosine hydroxylase activity.</p>Fórmula:C13H20Cl2N2Pureza:98.59%Forma y color:SolidPeso molecular:275.217CL-329167
CAS:<p>CL-329167, a angiotensin type 1 receptor antagonist, is used potentially for the treatment of hypertension.</p>Fórmula:C30H32N6O2Pureza:98%Forma y color:SolidPeso molecular:508.61Epimetendiol
CAS:<p>Epimetendiol is an anabolic agent</p>Fórmula:C20H32O2Forma y color:SolidPeso molecular:304.47BMS-932481
CAS:<p>BMS-932481 is a γ-secretase modulator.</p>Fórmula:C24H24FN7OForma y color:SolidPeso molecular:445.49JNJ-40929837
CAS:<p>JNJ-40929837 is an oral inhibitor of LTA4 hydrolase, which catalyzes LTB4 production.</p>Fórmula:C22H24N4O2SForma y color:SolidPeso molecular:408.52N-Formyl-L-histidine
CAS:<p>N-Formyl-L-histidine demonstrates a binding affinity for histidyl-tRNA synthetase, featuring a K i value of 4.6 μM.</p>Fórmula:C7H9N3O3Forma y color:SolidPeso molecular:183.16Zatosetron
CAS:<p>Zatosetron is a serotonin antagonists.</p>Fórmula:C19H25ClN2O2Forma y color:SolidPeso molecular:348.87Antiparasitic agent-8
CAS:<p>Antiparasitic agent-8 (Compound 9) exhibits potent antiparasitic activity against Hymenolepis nana, while demonstrating low levels of cytotoxicity [1].</p>Fórmula:C17H22FN3O4Forma y color:SolidPeso molecular:351.37L 699333
CAS:<p>L 699333 is an effective inhibitor of 5-lipoxygenase.</p>Fórmula:C36H35ClN2O4SForma y color:SolidPeso molecular:627.19SORT-PGRN interaction inhibitor 2
CAS:<p>SORT-PGRN Interaction Inhibitor 2 is a compound that downregulates SORT1 protein expression and enhances extracellular progranulin (PGRN) secretion in various</p>Fórmula:C19H31NOForma y color:SolidPeso molecular:289.46SSR 69071
CAS:<p>SSR69071: selective neutrophil elastase inhibitor, stronger for humans (Ki=0.0168 nM), may treat COPD, asthma, and reduce heart injury.</p>Fórmula:C27H32N4O7SForma y color:SolidPeso molecular:556.63DC_AC50
CAS:<p>"DC_AC50 inhibits Atox1/CCS to reduce cancer cell growth and prevent chemotherapy resistance."</p>Fórmula:C17H12BrF2N3OSPureza:99.84% - 99.9%Forma y color:SolidPeso molecular:424.26SAR-260301
CAS:<p>SAR-260301 is an orally available and selective inhibitor of PI3Kβ (IC50: 23 nM).</p>Fórmula:C19H22N4O3Pureza:99.74%Forma y color:SolidPeso molecular:354.4RIPK1-IN-16
CAS:<p>RIPK1-IN-16 is an orally active, potent RIPK1 inhibitor that mitigates excessive inflammation via inhibition of RIPK1-mediated necroptosis in vivo.</p>Fórmula:C20H19N5O2SPureza:98%Forma y color:SolidPeso molecular:393.46MC-VA-PAB-Exatecan
CAS:<p>MC-VA-PAB-Exatecan is an agent-linker conjugate designed for Antibody-Drug Conjugate (ADC) applications, comprising the ADC linker (peptide MC-VA-PAB) and the</p>Fórmula:C50H54FN7O11Forma y color:SolidPeso molecular:948.02AMG151 HCl
CAS:<p>ARRY-403 (AMG-151) is an oral glucokinase activator for type 2 diabetes with an EC50 of 79 nM and favorable drug properties.</p>Fórmula:C20H20Cl2N6O3S2Forma y color:SolidPeso molecular:527.439Antiproliferative agent-37
CAS:<p>Antiproliferative agent-37 (compound 10J) inhibits cell proliferation by arresting cells at the G2/M phase of the cell cycle [1].</p>Fórmula:C21H17FN2O2Forma y color:SolidPeso molecular:348.37S 16020-2
CAS:<p>S 16020-2 is an olivacine derivative, and DNA topoisomerase II inhibitor endowed with a remarkable antitumor activity against various experimental tumors.</p>Fórmula:C22H26Cl2N4O2Forma y color:SolidPeso molecular:449.376Cyclic HPMPC
CAS:<p>Cyclic HPMPC: Potent antiviral, raises O2 in mice with lethal vaccinia, lowers guinea pig CMV replication.</p>Fórmula:C8H12N3O5PForma y color:SolidPeso molecular:261.17SPH3127
CAS:<p>SPH3127 is a potent oral direct renin inhibitor, effective at 0.4 nM for human renin, used to study hypertension.</p>Fórmula:C22H32N6O4Forma y color:SolidPeso molecular:444.53DPP-4/GPR119 modulator 2
CAS:<p>DPP-4/GPR119 modulator 2 is an inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 0.22 μM) and an agonist of GPR119 (EC50: 0.95 μM).</p>Fórmula:C30H40N8O3Forma y color:SolidPeso molecular:560.69KP-544
CAS:<p>KP-544 is an agent of neurotrophin potentiator.</p>Fórmula:C18H19ClN4OPureza:98%Forma y color:SolidPeso molecular:342.82
