Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.519 productos)
- Apoptosis(5.787 productos)
- Ciclo celular / Checkpoint(4.446 productos)
- Cromatina / Epigenética(2.235 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.824 productos)
- Endocrinología / Hormonas(3.500 productos)
- Enzima(3.639 productos)
- GPCR / proteína G(8.317 productos)
- Inmunología e inflamación(3.516 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.200 productos)
- Transportador de membrana / canal de iones(2.787 productos)
- Metabolismo(9.416 productos)
- Microbiología / Virología(6.968 productos)
- Neurociencia(9.919 productos)
- Otros inhibidores(37.928 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.596 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.649 productos)
Mostrar 16 subcategorías más
Se han encontrado 66626 productos de "Inhibidores"
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BTM-3566
CAS:<p>BTM-3566 triggers ISR via OMA1, induces apoptosis in cancer cells, and is used to research DLBCL.</p>Fórmula:C24H23F4N3O2S2Pureza:99.95%Forma y color:SolidPeso molecular:525.58Zika virus-IN-3
CAS:<p>Zika virus-IN-3 (Compd 7) is a Zika virus inhibitor, with an EC 50 of 3.4 μM [1].</p>Fórmula:C23H20ClN3OForma y color:SolidPeso molecular:389.88CM-10-18
CAS:<p>CM-10-18: potent ER α-glucosidase inhibitor, strong antiviral against hemorrhagic fever viruses, protects mice from dengue fatality.</p>Fórmula:C17H35NO5Forma y color:SolidPeso molecular:333.46Niraxostat
CAS:<p>Niraxostat (Y-700) is one of the isocytosine derivatives as xanthine oxidase inhibitors.</p>Fórmula:C16H17N3O3Pureza:98.13%Forma y color:SolidPeso molecular:299.32WAY-639299
CAS:<p>WAY-639299 is an investigational compound targeting amyloid disorders and synucleinopathies for research purposes.</p>Fórmula:C19H19N3O2S2Forma y color:SolidPeso molecular:385.5CA-170
CAS:<p>PD-1-IN-1 is a programmed cell dealth-1inhibitor. PD-1-IN-1 can be used as an immune modulator.</p>Fórmula:C12H20N6O7Pureza:98%Forma y color:SolidPeso molecular:360.32L-CCG-lll
CAS:<p>inhibitor of both glial and neuronal uptake of glutamate, aspartate and cysteate.</p>Fórmula:C6H9NO4Pureza:98%Forma y color:SolidPeso molecular:159.14Difelikefalin HCl
CAS:<p>Difelikefalin: KOR agonist, EC50=0.16 nM in humans, >1 µM for MOR. Lowers pain/itch in mice, ED50=0.07 mg/kg.</p>Fórmula:C36H53N7O6·xHClForma y color:SolidPeso molecular:789.237LY 53857
CAS:<p>LY 53857 is a potent and selective antagonist of 5-HT2 serotonin receptor.</p>Fórmula:C27H36N2O7Forma y color:SolidPeso molecular:500.592Nrf2-IN-1
CAS:<p>Nrf2-IN-1 is an nuclear factor-erythroid 2-related factor 2 (Nrf2) inhibitor. Nrf2-IN-1 is developed for the research of acute myeloid leukemia (AML).</p>Fórmula:C21H22ClN3O2Pureza:95.00% - 99.68%Forma y color:SolidPeso molecular:383.87Bromodomain inhibitor-12 (edisylate)
CAS:<p>Bromodomain Inhibitor-12 Edisylate (example 303) serves as a bromodomain inhibitor applicable to autoimmune and inflammatory disease research [1].</p>Fórmula:C30H44N4O11S2Pureza:98%Forma y color:SolidPeso molecular:700.82HM5023507
CAS:<p>HM5023507 is an oral dual inhibitor of PI3Kδ/γ with >100-fold selectivity over PI3Kα/β and high specificity in human immune cells.</p>Fórmula:C21H18ClN7O2Forma y color:SolidPeso molecular:435.87α7β1 integrin modulator-1
CAS:<p>α7β1 Integrin Modulator-1 is a potent modulator with research potential for muscular dystrophy [1].</p>Fórmula:C23H29N3O6SPureza:98%Forma y color:SolidPeso molecular:475.56MS-444
CAS:<p>MS-444 (BE-34776) is an MLCK and HuR inhibitor with antitumor activity that can be used to study triple-negative breast cancer and colorectal cancer.</p>Fórmula:C13H10O4Pureza:99.45% - 99.45%Forma y color:SolidPeso molecular:230.22BMS-695735
CAS:<p>BMS-695735: benzimidazole, inhibits IGF-1 receptor, broad antitumor effects, affects CYP3A4, low solubility, binds plasma proteins.</p>Fórmula:C26H31ClFN7OForma y color:SolidPeso molecular:512.02Raf inhibitor 3
CAS:<p>Raf inhibitor 3 (Example 30), a potent inhibitor of both B-Raf and C-Raf, exhibits IC50 values below 15 nM. It is applicable in cancer research studies [1].</p>Fórmula:C18H19FN8O2SPureza:98%Forma y color:SolidPeso molecular:430.46GYKI-46903 HCl
CAS:<p>GYKI-46903 is a noncompetitive 5-HT3 receptor antagonist.</p>Fórmula:C17H21ClFNO2Forma y color:SolidPeso molecular:325.814-CPPC
CAS:<p>4-CPPC inhibits MIF-2 (IC50=27μM), not MIF-1; blocks MIF-2/CD74 binding and MIF-2-induced ERK1/2 in fibroblasts.</p>Fórmula:C14H9NO6Pureza:97.50% - 98.03%Forma y color:SolidPeso molecular:287.22Dolutegravir RR Isomer
CAS:<p>Dolutegravir RR Isomer, a second-gen HIV-1 integrase inhibitor, strongly inhibits HIV in various cells.</p>Fórmula:C20H19F2N3O5Forma y color:SolidPeso molecular:419.38WYE-132
CAS:<p>WYE-125132: potent mTOR inhibitor, IC50 0.19 nM, selective over PI3Ks/hSMG1/ATR.</p>Fórmula:C27H33N7O4Pureza:99.16%Forma y color:SolidPeso molecular:519.6MF498
CAS:<p>MF498 is a novel and selective E prostanoid receptor 4 (EP4 receptor) antagonist, displayed a strong binding affinity for the EP4 receptor (Ki: 0.7 nM).</p>Fórmula:C32H33N3O7SPureza:98%Forma y color:SolidPeso molecular:603.69AMG151 HCl
CAS:<p>ARRY-403 (AMG-151) is an oral glucokinase activator for type 2 diabetes with an EC50 of 79 nM and favorable drug properties.</p>Fórmula:C20H20Cl2N6O3S2Forma y color:SolidPeso molecular:527.439SQ 26655
CAS:<p>SQ 26655 is an antagonist of thromboxane A2/prostaglandin H2.</p>Fórmula:C21H34O4Pureza:98%Forma y color:SolidPeso molecular:350.49WAY-612453
CAS:<p>WAY-612453 is an active compound utilized in researching amyloid diseases and synucleinopathies.</p>Fórmula:C9H8Cl2N4SForma y color:SolidPeso molecular:275.16KRAS G12C inhibitor 5
CAS:<p>KRAS G12C inhibitor 5 is a KRas G12C inhibitor.</p>Fórmula:C32H37N7O2Pureza:98%Forma y color:SolidPeso molecular:551.68Plomestane
CAS:<p>Plomestane is a selective inhibitor of aromatization in human breast tissue and may provide a mechanism for controlling estrogen responsive processes.</p>Fórmula:C21H26O2Forma y color:SolidPeso molecular:310.43S 16020-2
CAS:<p>S 16020-2 is an olivacine derivative, and DNA topoisomerase II inhibitor endowed with a remarkable antitumor activity against various experimental tumors.</p>Fórmula:C22H26Cl2N4O2Forma y color:SolidPeso molecular:449.376WAY-324572
CAS:<p>WAY-324572 is an active compound.</p>Fórmula:C20H21FN2OForma y color:SolidPeso molecular:324.39MCT1-IN-2
CAS:<p>SR13800 is a monocarboxylate transporter 1 (MCT1) inhibitor with cell-permeable.</p>Fórmula:C25H29N3O2SForma y color:SolidPeso molecular:435.58XL041
CAS:<p>XL041 (BMS-852927) is an agonist of LXRβ-selective.</p>Fórmula:C29H28Cl2F2N2O4SPureza:98%Forma y color:SolidPeso molecular:609.51CUR61414
CAS:<p>CUR61414 is a cell-permeable inhibitor of Hedgehog signaling pathway (IC50 =100-200 nM) and selectively binds to smoothened (Ki = 44 nM).</p>Fórmula:C31H42N4O5Pureza:97.34% - 98%Forma y color:SolidPeso molecular:550.69NAT6-297775
CAS:<p>NAT6-297775 is a SHP2 inhibitor with IC50 =2.47uM.</p>Fórmula:C25H36N6O2Forma y color:SolidPeso molecular:452.59Immuno modulator-1
CAS:<p>Immuno modulator-1 (compound 22) effectively suppresses the secretion of TNFα and IL-2 in human peripheral blood mononuclear cells (hPBMC) with IC50 values of 4</p>Fórmula:C32H31FN6O4Forma y color:SolidPeso molecular:582.62Cyclic HPMPC
CAS:<p>Cyclic HPMPC: Potent antiviral, raises O2 in mice with lethal vaccinia, lowers guinea pig CMV replication.</p>Fórmula:C8H12N3O5PForma y color:SolidPeso molecular:261.17NMS-P953
CAS:<p>NMS-P953: JAK2 inhibitor, reduces tumor growth in SET-2 model, confirmed in vivo action, good pharmacokinetics and safety.</p>Fórmula:C16H11ClF3N5OForma y color:SolidPeso molecular:381.74Quorum Sensing-IN-2
CAS:<p>Quorum Sensing-IN-2 (compound 23e) is a quorum sensing inhibitor that curtails bacterial pathogenicity without impeding growth.</p>Fórmula:C19H13F2NO3Forma y color:SolidPeso molecular:341.31Antipsychotic agent 54
CAS:<p>Telomerase-IN-1 is a telomerase inhibitor (IC50: 0.19 μM).</p>Fórmula:C21H23FN2O4Pureza:98.10%Forma y color:SolidPeso molecular:386.42M5N36
CAS:<p>M5N36: selective Cdc25C inhibitor, IC50: 0.15µM A, 0.19µM B, 0.06µM C; halts cell growth, boosts p-CDK1/2.</p>Fórmula:C20H16ClN5O3Forma y color:SolidPeso molecular:409.83PROTAC KRAS G12C degrader-3
CAS:<p>PROTAC KRAS G12C Degrader-3 (Comp 283) serves as a potent degrader of KRAS G12C, utilized in cancer research [1].</p>Fórmula:C63H75ClN14O6Pureza:98%Forma y color:SolidPeso molecular:1159.815'-ODMT cEt N-Bzm5 C Phosphoramidite (Amidite)
CAS:<p>5'-ODMT cEt N-Bzm5 C Phosphoramidite is a strong modified nucleic acid analog for antisense oligos.</p>Fórmula:C49H56N5O9PForma y color:SolidPeso molecular:889.97CI 972 anhydrous
CAS:<p>CI 972 anhydrous is an inhibitor of purine nucleoside phosphorylase (PNP) (Ki: 0.83 μM) used as a T cell-selective immunosuppressive agent.</p>Fórmula:C11H12ClN5OSPureza:98%Forma y color:SolidPeso molecular:297.76Taragarestrant
CAS:<p>Taragarestrant (D-0502), an oral estrogen receptor degrader, combats ER+ breast cancer in research.</p>Fórmula:C25H25Cl2FN2O2Forma y color:SolidPeso molecular:475.38MGS-0039
CAS:<p>MGS-0039: Group II mGluR2/3 antagonist, non-serotonergic antidepressant-like effect, AMPA involvement, regulates dopamine in NAc.</p>Fórmula:C15H14Cl2FNO5Pureza:98%Forma y color:SolidPeso molecular:378.18CCG-63808
CAS:<p>CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins.</p>Fórmula:C25H15FN4O2SPureza:90%Forma y color:SolidPeso molecular:454.48JAK-IN-31
CAS:<p>JAK-IN-31 (Example 75), a JAK inhibitor, demonstrates IC50 values of ≤0.01 µM for JAK1, ≤0.01 µM for JAK2, 0.01-0.1 µM for JAK3, and ≤0.01 µM for Tyk2,</p>Fórmula:C21H19N7O2S2Pureza:98%Forma y color:SolidPeso molecular:465.55NT113
CAS:<p>NT113: ERBB inhibitor, penetrates brain, hinders GBM growth (high EGFR/EGFRvIII), targets ERBB/Akt phosphorylation in vivo/in vitro.</p>Fórmula:C27H25ClFN5O2Forma y color:SolidPeso molecular:505.97L-742001 Hydrochloride
CAS:<p>L-742001 Hydrochloride is an RNA polymerase inhibitor.</p>Fórmula:C23H25Cl2NO4Forma y color:SolidPeso molecular:450.36PCSK9-IN-14
CAS:<p>PCSK9-IN-14, also known as compound Ia-8, is a potent inhibitor of PCSK9 [1].</p>Fórmula:C15H10F6N4O2Forma y color:SolidPeso molecular:392.26p38-α MAPK-IN-1
CAS:<p>p38-α MAPK-IN-1 is a MAPK14 (p38-α) inhibitor with IC50 of 2300 nM and 5500 nM in EFC displacement assay and HTRF assay,respectively.</p>Fórmula:C27H35N5O3Pureza:99.93%Forma y color:SolidPeso molecular:477.6BMS-538203
CAS:<p>BMS-538203 is a novel HIV integrase inhibitor.</p>Fórmula:C12H12FNO5Pureza:98%Forma y color:SolidPeso molecular:269.23
