Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.519 productos)
- Apoptosis(5.787 productos)
- Ciclo celular / Checkpoint(4.446 productos)
- Cromatina / Epigenética(2.235 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.824 productos)
- Endocrinología / Hormonas(3.500 productos)
- Enzima(3.639 productos)
- GPCR / proteína G(8.318 productos)
- Inmunología e inflamación(3.516 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.200 productos)
- Transportador de membrana / canal de iones(2.787 productos)
- Metabolismo(9.416 productos)
- Microbiología / Virología(6.968 productos)
- Neurociencia(9.920 productos)
- Otros inhibidores(37.928 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.596 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.649 productos)
Mostrar 16 subcategorías más
Se han encontrado 66627 productos de "Inhibidores"
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DGKα-IN-7
CAS:<p>DGKα-IN-7 is a potent DGKα inhibitor with an IC50 value of 6.225 nM and potential applications in cancer research.</p>Fórmula:C23H17F5N6Forma y color:SolidPeso molecular:472.41NSC756093
CAS:<p>NSC756093 potentially inhibits GBP1:PIM1 interaction. NSC756093 can be used in ovarian cancer studies.</p>Fórmula:C20H19NO4Pureza:99.92%Forma y color:SolidPeso molecular:337.37Acth (1-4)
CAS:<p>Acth (1-4) is the ACTH N-terminal tetrapeptide.</p>Fórmula:C20H30N4O8SPureza:98%Forma y color:SolidPeso molecular:486.54SARS-CoV-2-IN-1
CAS:<p>SARS-CoV-2-IN-1 is a potent inhibitor of Mpro(SARS-CoV-2 Mpro, SARS-CoV Mpro and MERS-CoV Mpro with IC50s of 0.67, 0.90 and 0.58 μM, respectively).</p>Fórmula:C31H39N5O7Pureza:98%Forma y color:SolidPeso molecular:593.67GSK-2262167 sodium
CAS:<p>GSK-2262167 is a potent S1P1 agonist, as effective as fingolimod in collagen-induced arthritis models, and shows good preclinical pharmacokinetic properties.</p>Fórmula:C25H26N4NaO4Forma y color:SolidPeso molecular:469.497TNIK&MAP4K4-IN-1
CAS:<p>TNIK&MAP4K4-IN-1 (compound A-39) is a potent dual inhibitor targeting TNIK and MAP4K4/HGK, exhibiting IC50 values of 1.29 nM and <10 nM, respectively, in human</p>Fórmula:C25H23FN4O3Forma y color:SolidPeso molecular:446.47BAY-60-5521
CAS:<p>BAY-60-5521 is an effective cholesterol ester transfer protein (CETP) inhibitor.</p>Fórmula:C30H37F4NOForma y color:SolidPeso molecular:503.61SARS-CoV-2-IN-43
CAS:<p>Compound 8h, also known as SARS-CoV-2-IN-43, is a powerful inhibitor effective in obstructing the replication of SARS-CoV-2, exhibiting significant antiviral</p>Fórmula:C16H12O3Pureza:98%Forma y color:SolidPeso molecular:252.26C.I. Vat Black 27
CAS:<p>C.I. Vat Black 27 is a black dye.</p>Fórmula:C42H23N3O6Forma y color:SolidPeso molecular:665.65Inflachromene
CAS:<p>Inflachromene (ICM) is an inhibitor of HMGB1 and HMGB expression with anti-inflammatory activity.Inflachromene is used in the study of epilepsy.</p>Fórmula:C21H19N3O4Pureza:97.36% - 99.88%Forma y color:SolidPeso molecular:377.39Zndm19
CAS:<p>Zndm19 is an inhibitor of New Delhi Metallo-β-lactamase-1 (NDM-1), utilized in researching drug-resistant bacterial infections [1].</p>Fórmula:C13H13N3OS2Forma y color:SolidPeso molecular:291.39YM348
CAS:<p>YM348 is an effective and orally active 5-HT2C receptor agonist. YM348 also shows a high affinity for the cloned human 5-HT2C receptor (Ki: 0.89 nM).</p>Fórmula:C14H17N3OPureza:98%Forma y color:SolidPeso molecular:243.3Verzistobart
CAS:<p>Verzistobart, an IgG1κ antibody, specifically targets the hepatitis A virus cellular receptor, HAVCR2.</p>Forma y color:LiquidBenzoadenosine
CAS:<p>Benzoadenosine suppresses kinase activity slightly less than does adenosine.</p>Fórmula:C14H15N5O4Pureza:98%Forma y color:SolidPeso molecular:317.3(R)-FT671
CAS:<p>(R)-FT671 is the R-isomer of FT671. FT671 is a potent, non-covalent and selective inhibitor of USP7 (IC50 of 52 nM)</p>Fórmula:C24H23F4N7O3Pureza:98%Forma y color:SolidPeso molecular:533.48Indole-C2-amide-C2-NH2
CAS:<p>Indole-C2-amide-C2-NH2 serves as a potent linker [1].</p>Fórmula:C13H17N3OForma y color:SolidPeso molecular:231.29Oloctinebart
CAS:<p>Oloctinebart, a humanized immunoglobulin G4-kappa (IgG4-κ) monoclonal antibody targeting LGALS3, is utilized to decrease the formation of amyloid beta oligomers</p>Forma y color:Liquid2,7-Bis(alloxycarbonylamino)-9-chloroacridine
CAS:<p>2,7-Bis(alloxycarbonylamino)-9-chloroacridine serves as a fluorescent label.</p>Fórmula:C21H18ClN3O4Forma y color:SolidPeso molecular:411.84Avarol
CAS:<p>Avarol triggers cell death in pancreatic cancer and is a non-toxic, neuroprotective AChE inhibitor for Alzheimer's.</p>Fórmula:C21H30O2Forma y color:SolidPeso molecular:314.46Tamgiblimab
CAS:<p>Tamgiblimab (IBI939) is a fully human monoclonal antibody that targets the T-cell immunoreceptor with immunoglobulin and ITIM domains (TIGIT), exhibiting</p>Forma y color:LiquidAntifungal agent 26
CAS:<p>Pradimicin A derivative 26 exhibits antifungal, antiviral, and antiparasitic properties by attaching to d-mannose (Man)-rich glycans in pathogenic organisms [1</p>Fórmula:C40H45N3O18Forma y color:SolidPeso molecular:855.79CUR61414
CAS:<p>CUR61414 is a cell-permeable inhibitor of Hedgehog signaling pathway (IC50 =100-200 nM) and selectively binds to smoothened (Ki = 44 nM).</p>Fórmula:C31H42N4O5Pureza:97.34% - 98%Forma y color:SolidPeso molecular:550.69SRX 251
CAS:<p>SRX 251, a vasopressin V1a receptor antagonist, is used potentially for the treatment of primary dysmenorrhea.</p>Fórmula:C43H48F3N5O5Forma y color:SolidPeso molecular:771.87Ogremorphin
CAS:<p>Ogremorphin (GPR68-IN-1) is a potent inhibitor of GPR68, exhibiting an EC50 of 170 nM.it is utilized in the study of autoimmune chronic inflammatory diseases [1</p>Fórmula:C21H17N3OSPureza:99.65% - 99.65%Forma y color:SolidPeso molecular:359.44MK-0736 hydrochloride
CAS:<p>MK-0736 hydrochloride is a potent and selective 11β-HSD-1 inhibitor.</p>Fórmula:C23H31ClF3N3O2SForma y color:SolidPeso molecular:506.03Gentisuric acid
CAS:<p>Gentisuric acid, an Aspirin metabolite and a substrate of α-amidating monooxygenase (PAM), mitigates DNA damage induced by Mitomycin C. [1] [2]</p>Fórmula:C9H9NO5Pureza:98%Forma y color:SolidPeso molecular:211.17PIN1 inhibitor 2
CAS:<p>PIN1 inhibitor 2, compound 12, impedes PIN1, shows promise in breast cancer study, and has IC50 of 9.55 μM in MCF7 cells.</p>Fórmula:C16H21N3S2Forma y color:SolidPeso molecular:319.49Amb123203
CAS:<p>Amb123203 is an inhibitor of the budding of mVP40 and eVP40 VLPs that acts by blocking mVP40-795 Nedd4 protein-protein interaction.</p>Fórmula:C25H27N5OSForma y color:SolidPeso molecular:445.58NEU-1923
<p>NEU-1923 is a potent inhibitor of T. brucei proliferation (EC50= 0.37 μM).</p>Fórmula:C23H20ClN5O3SForma y color:SolidPeso molecular:481.96SID 26681509
CAS:<p>SID 26681509 is a selective, reversible and competitive human cathepsin L inhibitor (IC50 of 56 nM).</p>Fórmula:C27H33N5O5SPureza:98.16%Forma y color:SolidPeso molecular:539.65FK-352
CAS:<p>FK-352 is a pyrazolopyridine derivative and adenosine-1 receptor antagonist.</p>Fórmula:C23H23N3O3Forma y color:SolidPeso molecular:389.45ENT-C225
CAS:<p>ENT-C225 is a potent TrkB neurotrophin receptor (TrkBR) activator with neuroprotective activity for the study of Alzheimer's disease and Parkinson's disease.</p>Fórmula:C26H40N4O5Pureza:99.36% - 99.36%Forma y color:SolidPeso molecular:488.62DDa-1
CAS:<p>DDa-1 is a potent (kinase degrader) [1].</p>Fórmula:C60H77Cl2N13O3SForma y color:SoildPeso molecular:1131.31sEH/AChE-IN-3
CAS:<p>sEH/AChE-IN-3 -15: potent dual sEH & AChE inhibitor; crosses BBB; IC50: hsEH 0.4nM, hAChE 1.94nM, hBChE 615nM, msEH 4.3nM, mAChE 2.61nM.</p>Fórmula:C35H39ClF3N5O3Forma y color:SolidPeso molecular:670.16Q-VD(OMe)-OPh
CAS:<p>Q-VD-OPh: broad-spectrum, non-toxic caspase inhibitor; cost-effective, specific for apoptotic inhibition.</p>Fórmula:C27H27F2N3O6Pureza:98%Forma y color:SolidPeso molecular:527.52Disoxaril
CAS:<p>Disoxaril (BRN 3626820, WIN 51711), an anti-picornavirus, blocks enterovirus by targeting VP1; boosts poliovirus inhibition with Ambioxime, Bioxazole.</p>Fórmula:C20H26N2O3Forma y color:SolidPeso molecular:342.43ASP-4000 free base
CAS:<p>ASP-4000 free base is a dipeptidyl peptidase 4 (DPP) inhibitor with antihyperglycemic activity.</p>Fórmula:C12H17N3O2Forma y color:SolidPeso molecular:235.28CL-329167
CAS:<p>CL-329167, a angiotensin type 1 receptor antagonist, is used potentially for the treatment of hypertension.</p>Fórmula:C30H32N6O2Pureza:98%Forma y color:SolidPeso molecular:508.61LG 50643
CAS:<p>LG 50643 is a muscarinic antagonist.</p>Fórmula:C24H34INO2Pureza:98%Forma y color:SolidPeso molecular:495.44NNMT-IN-4
CAS:<p>NNMT-IN-4 (compound 38) is a selective, uncompetitive inhibitor of nicotinamide N-methyltransferase (NNMT) with in vitro biochemical and cell-based assay IC50</p>Fórmula:C9H11N3OForma y color:SolidPeso molecular:177.2CSF1R-IN-5
CAS:<p>CSF1R-IN-5: Potent CSF1R inhibitor, may alter TAM/glioma inflammatory exchanges, potential cancer research tool. (WO2021197276A1, Compound 11)</p>Fórmula:C22H19N7O3Forma y color:SolidPeso molecular:429.43TA-1887
CAS:<p>TA-1887: Selective SGLT2 inhibitor, treats type 2 diabetes, lowers glucose in high-fat diet mice, boosts UGE, has good pharmacokinetics.</p>Fórmula:C24H26FNO5Forma y color:SolidPeso molecular:427.47Mirincamycin HCl
CAS:<p>Mirincamycin HCl is a close analog of the drug clindamycin used for the treatment of Plasmodium falciparum blood stages.</p>Fórmula:C19H36Cl2N2O5SPureza:98%Forma y color:SolidPeso molecular:475.47ATR-IN-18
CAS:<p>ATR-IN-18: oral ATR inhibitor, IC50 0.69 nM; halts LoVo cell growth, IC50 37.34 nM; anti-tumor.</p>Fórmula:C19H22F3N7O5SForma y color:SolidPeso molecular:517.48Firazorexton hydrate
CAS:<p>Firazorexton hydrate (TAK-994) is a brain-penetrant and orally active agonist of the orexin type 2 receptor (OX2R) with a potent EC50 of 19 nM.</p>Fórmula:C22H25F3N2O4SH2OForma y color:SolidPeso molecular:497.53Cenerimod
CAS:<p>Cenerimod (ACT-334441) is an S1P1 agonist used in the study of murine experimental autoimmune encephalomyelitis (EAE) and murine scleroderma.</p>Fórmula:C25H31N3O5Pureza:97.43% - 99.97%Forma y color:SolidPeso molecular:453.53ST 2825
CAS:<p>ST 2825 is a specific MyD88 dimerization inhibitor. ST2825 inhibition of IL-1β-mediated activation of NF-κB transcriptional activity.</p>Fórmula:C27H28Cl2N4O5SPureza:98%Forma y color:SolidPeso molecular:591.51APE1-IN-2
CAS:<p>APE1-IN-2 (AP1), a Pt(IV) proagent, targets APE1 protein, induces DNA damage, and triggers apoptosis with anticancer effects.</p>Fórmula:C9H12Cl2N4O5PtPureza:98%Forma y color:SolidPeso molecular:522.21Z-YVAD-CMK
CAS:<p>Z-YVAD-CMK is an inhibitor of both caspase-1 and caspase-3, as referenced in [1].</p>Fórmula:C30H37ClN4O9Pureza:98%Forma y color:SolidPeso molecular:633.09Formoterol HCl
CAS:<p>Formoterol HCl is a long-acting beta-2 adrenergic agonist (LABA).</p>Fórmula:C19H25ClN2O4Forma y color:SolidPeso molecular:380.869
