Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.523 productos)
- Apoptosis(5.792 productos)
- Ciclo celular / Checkpoint(4.449 productos)
- Cromatina / Epigenética(2.238 productos)
- Señalización citoesquelética(1.383 productos)
- Daño al ADN / Reparación del ADN(2.825 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.526 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.202 productos)
- Transportador de membrana / canal de iones(2.790 productos)
- Metabolismo(9.448 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.926 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.016 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66641 productos de "Inhibidores"
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Tobevibart
CAS:<p>Tobevibart, an IgG1-lambda humanized monoclonal antibody targeting the hepatitis B virus (HBV) surface envelope protein, exhibits antiviral activity [1].</p>Pureza:98%Forma y color:LiquidPBR28
CAS:<p>PBR28, a TSPO modulator, holds potential for preventative research in Pulmonary Arterial Hypertension (PAH) and is instrumental in brain positron emission</p>Fórmula:C21H20N2O3Pureza:98%Forma y color:SolidPeso molecular:348.4ATX inhibitor 15
CAS:<p>ATX inhibitor 15, an indole-based carbamate, has a 2.17 nM IC50 against ATX, suppresses pro-fibrotic genes, and protects against mouse lung fibrosis.</p>Fórmula:C27H32ClN5O4SForma y color:SolidPeso molecular:558.09PRMT5-IN-25
CAS:<p>PRMT5-IN-25 (compound 503) is a potent inhibitor of PRMT5, exhibiting an inhibition constant (K i) of 0.06 nM and demonstrating antiproliferative properties [1</p>Fórmula:C24H21F3N6OPureza:98%Forma y color:SolidPeso molecular:466.46L-054,522
CAS:<p>L-054,522 is potent, selective agonists of somatostatin receptor.</p>Fórmula:C35H47N7O5Forma y color:SolidPeso molecular:645.79PAN12314
CAS:<p>PAN12314 (Compound 5a) is a 5-HT4R partial agonist with cognition-enhancing effects in animals, lacking a formal name.</p>Fórmula:C21H30N4O2Forma y color:SolidPeso molecular:370.49Cladosporin
CAS:<p>Cladosporin, from Cladosporium cladosporioid fungus, halts dermatophyte growth on agar at 75 μg/mL.</p>Fórmula:C16H20O5Forma y color:SolidPeso molecular:292.33Cyclopentenyl uracil
CAS:<p>Cyclopentenyl uracil 是一种无细胞毒性的尿苷激酶 (uridine kinase) 抑制剂，可有效阻断完整小鼠体内宿主和肿瘤组织对循环尿苷的回收。</p>Fórmula:C10H12N2O5Forma y color:SolidPeso molecular:240.21KDM4-IN-2
CAS:<p>KDM4-IN-2 is a potent and selective KDM4/KDM5 dual inhibitor with Kis of 4 and 7 nM for KDM4A and KDM5B, respectively.</p>Fórmula:C25H26N6OPureza:98%Forma y color:SolidPeso molecular:426.51PPO-IN-2
CAS:<p>PPO-IN-2 is a protoporphyrinogen IX oxidase inhibitor, exhibiting a Ki value of 16 nM [1].</p>Fórmula:C17H15ClFN3O2S2Forma y color:SolidPeso molecular:411.9ERK1/2 inhibitor 5
CAS:<p>ERK1/2 inhibitor 5: potent against ERK1/2, may combat cancer and inflammation.</p>Fórmula:C28H32ClFN6O5Forma y color:SolidPeso molecular:587.04Antitumor agent-49
CAS:<p>Antitumor agent-49 (Compound 10), a harmine derivative-furoxan hybrid featuring nitric oxide (NO) donating properties, exhibits cytotoxic effects against HepG2</p>Fórmula:C42H41BrN4O8SForma y color:SolidPeso molecular:841.77UZH1b
CAS:<p>UZH1b, an enantiomer of UZH1a (a METTL3 inhibitor), exhibits substantially reduced activity against METTL3, with an IC50 value of 28 µM [1].</p>Fórmula:C32H42N6O3Pureza:98%Forma y color:SolidPeso molecular:558.71ASGPR ligand-1
CAS:<p>ASGPR ligand-1 is a compound that targets the asialoglycoprotein receptor (ASGPR) and is utilized in various disease research contexts [1].</p>Fórmula:C61H110N10O27Forma y color:SolidPeso molecular:1415.58DU-125530
CAS:<p>DU-125530 is a 5-HT1A receptor antagonist.</p>Fórmula:C23H26ClN3O5SForma y color:SolidPeso molecular:491.99KD-3010
CAS:<p>KD-3010 (Kalypsys) is an orally active potent and selective PPARδ agonist for the study of liver injury.</p>Fórmula:C30H33F3N2O8S2Pureza:99.61%Forma y color:SolidPeso molecular:670.72SARS-CoV-2 3CLpro-IN-15
CAS:<p>SARS-CoV-2 3CLpro-IN-15 (compound a), a beta-nitrostyrene derivative, acts as an inhibitor of the SARS-CoV-2 3CL protease (3CLpro), effectively inhibiting viral</p>Fórmula:C8H6N2O4Pureza:98%Forma y color:SolidPeso molecular:194.14CXJ-2
CAS:<p>CXJ-2, a cyclic peptide, binds EDPs, inhibits PI3K/ERK, and reduces hepatic cell growth/migration, offering antifibrotic effects.</p>Fórmula:C55H87N15O22Pureza:98%Forma y color:SolidPeso molecular:1310.37Moxestrol
CAS:<p>Moxestrol, a synthetic estrogen, treats menopause and menstrual issues in Europe.</p>Fórmula:C21H26O3Pureza:98%Forma y color:SolidPeso molecular:326.43Alclofenac
CAS:<p>Alclofenac (W-7320) aids chronic rheumatism by affecting acute phase proteins and L-tryptophan binding.</p>Fórmula:C11H11ClO3Pureza:99.89%Forma y color:SolidPeso molecular:226.66EGFR-IN-85
CAS:<p>EGFR-IN-85 (Compound 1), an EGFR inhibitor, exhibits potent activity with an IC50 of 0.19 μM against EGFRvⅢ phosphorylation and can suppress intratumoral EGFR</p>Fórmula:C26H30N8O2Pureza:98%Forma y color:SolidPeso molecular:486.57Spectramide
CAS:<p>Spectramide is a dopamine D-2 receptor antagonist.</p>Fórmula:C19H23ClIN3O2Forma y color:SolidPeso molecular:487.76JJH260
CAS:<p>JJH260, a N-hydroxy hydantoin carbamate, inhibits AIG1 and ADTRP with IC50 values of 0.57 μM and 8.5 μM, respectively, and targets ABHD6, LYPLA1/2.</p>Fórmula:C29H34ClN5O5Forma y color:SolidPeso molecular:568.06Ardisin
CAS:<p>Ardisin is a Topoisomerase I and II enzyme inhibitor. Ardisin may have antioxidant effects.</p>Fórmula:C20H32O2Forma y color:SolidPeso molecular:304.475-n-Heptyl-6-hydroxy-4,7-dioxobenzothiazole
CAS:<p>5-n-Heptyl-6-hydroxy-4,7-dioxobenzothiazole acts as a competitive inhibitor at the Qo site of the cytochrome bc1 complex (cytochrome c oxidoreductase) in</p>Fórmula:C14H17NO3SForma y color:SolidPeso molecular:279.36LM-030
CAS:<p>LM-030, also known as BPR277, is a novel inhibitor of kallikrein-related peptidase 7 (KLK7) and epidermal elastase 2 (ELA2).</p>Fórmula:C46H72N8O12Forma y color:SolidPeso molecular:929.11WRN inhibitor 1
CAS:<p>WRN Inhibitor 1 (example 7) is an inhibitor of the Werner Syndrome ATP-dependent helicase enzyme (WRN), selectively targeting its helicase domain.</p>Fórmula:C16H13FN2O4SPureza:98%Forma y color:SolidPeso molecular:348.35Gentisein
CAS:<p>Gentisein (NSC-329491), a primary metabolite of Mangiferin, exhibits significant inhibition of serotonin uptake, demonstrating potency with an IC50 value of 4.7</p>Fórmula:C13H8O5Pureza:96.89%Forma y color:SolidPeso molecular:244.2KCa1.1 channel activator-1
<p>A selective vascular KCa1.1 channel stimulator with CaV1.2 blocking ability and mild myorelaxant effects.</p>Fórmula:C25H16O10Forma y color:SolidPeso molecular:476.39M867
CAS:<p>M867 is a selective, reversible caspase-3 inhibitor, possessing an IC50 of 1.4 nM and a Ki value of 0.7 nM, demonstrating anti-apoptotic activity [1].</p>Fórmula:C27H43N7O6Pureza:98%Forma y color:SolidPeso molecular:561.67pan-KRAS-IN-3
CAS:<p>Pan-KRAS-IN-3 (Example 84) is a pan-KRAS inhibitor suitable for cancer research [1].</p>Fórmula:C33H32F3N5O2Pureza:98%Forma y color:SolidPeso molecular:587.63MC2590
CAS:<p>MC2590 is a histone deacetylase (HDAC) inhibitor that inhibits HDAC1-3, -6, -8, and -10 activities, induces cell cycle arrest, and promotes apoptosis.</p>Fórmula:C20H17N3O3Pureza:99.64%Forma y color:SolidPeso molecular:347.37UBP316
CAS:<p>GluR5-containing kainate receptor antagonist</p>Fórmula:C20H19N3O6SPureza:98%Forma y color:SolidPeso molecular:429.45TPC-144
CAS:<p>TPC-144: Potent, selective reversible LSD1 inhibitor with antitumor effects in AML/SCLC cells and xenografts.</p>Fórmula:C31H31F2N3O2Pureza:98%Forma y color:SolidPeso molecular:515.59AZD1092
CAS:<p>AZD1092 is the glucokinase enzyme activator.</p>Fórmula:C24H26N4O5Pureza:98%Forma y color:SolidPeso molecular:450.49LCB-2853
CAS:<p>LCB-2853 is a potent thromboxane A2/prostaglandin H2 (TXA2/PGH2) receptor antagonist with antiplatelet aggregation, antivasospasm, and antithrombotic effects.</p>Fórmula:C21H24ClNO4SPureza:97.15%Forma y color:SolidPeso molecular:421.94WAY 316606 HCl (915759-45-4 free base)
<p>WAY 316606 HCl is a selective small-molecule inhibitor of secreted frizzled-related protein-1 (EC50: 0.65 μM).</p>Fórmula:C18H19F3N2O4S2·HClPureza:98%Forma y color:SolidPeso molecular:484.94Autotaxin-IN-5
CAS:<p>Autotaxin-IN-5 is an Autotaxin inhibitor. It has the potential to treat idiopathic pulmonary fibrosis.</p>Fórmula:C30H29N9O2Pureza:98%Forma y color:SolidPeso molecular:547.61Asem F-18
CAS:<p>Asem F-18 is a radiolabeled antagonist for imaging the α7-nicotinic acetylcholine receptor with PET .</p>Fórmula:C19H19FN2O2SForma y color:SolidPeso molecular:357.43eIF4A3-IN-9
CAS:<p>eIF4A3-IN-9, a silvestrol analogue, disrupts eIF4F complex assembly; EC50s: 29/450/80 nM (myc/tub-LUC, MB-231 cells); for cancer research.</p>Fórmula:C28H27NO8Forma y color:SolidPeso molecular:505.52PF-06260414
CAS:<p>PF-06260414 is a selective androgen receptor modulator or SARM used to treat muscle weakness.</p>Fórmula:C14H14N4O2SForma y color:SolidPeso molecular:302.35L 670548
CAS:<p>L 670548 is an agonist of muscarinic receptor.</p>Fórmula:C9H13N3OPureza:98%Forma y color:SolidPeso molecular:179.22TMP778
CAS:<p>TMP778 is an effective and selective RORγt inverse agonist (IC50: 7 nM in FRET assay).</p>Fórmula:C31H30N2O4Pureza:98%Forma y color:SolidPeso molecular:494.58AMPK-α1β1γ1 activator 1
CAS:<p>AMPK-α1β1γ1 activator 1 (M1), an acyl glucuronide metabolite derived from an Indole-3-carboxylic Acid-based AMPK activator, selectively activates the β1</p>Fórmula:C25H24ClNO9Pureza:98%Forma y color:SolidPeso molecular:517.91L-368899 free base
CAS:<p>L-368899: non-peptide, oral oxytocin receptor antagonist (IC50: 8.9 nM), 40x more selective than vasopressin V1a/V2.</p>Fórmula:C26H42N4O5S2Pureza:98%Forma y color:SolidPeso molecular:554.77AAK1-IN-5
CAS:<p>AAK1-IN-5: Potent, selective AAK1 inhibitor; CNS-penetrant; oral; IC50: 1.2 nM; Ki: 0.05 nM; cell IC50: 0.5 nM. Useful in neuropathic pain research.</p>Fórmula:C19H23F4N3OForma y color:SolidPeso molecular:385.4ATAC21
CAS:<p>ATAC21 is a linker-immune-stimulatory compound created by conjugating a noncleavable maleimide-PEG4 linker, which includes a succinimide group, with an immune-</p>Fórmula:C38H50N12O21P2Forma y color:SolidPeso molecular:1072.82Mpro 61
CAS:<p>Mpro 61 is a potent non-covalent inhibitor of SARS-CoV-2 main protease.</p>Fórmula:C28H19Cl2FN4O4Forma y color:SolidPeso molecular:565.38Encaleret
CAS:<p>Encaleret( JIT-305) is an antagonist of oral calcium-sensing receptor (CaSR), it is used for the treatment of osteoporosis.</p>Fórmula:C29H33ClFNO4Forma y color:SolidPeso molecular:514.03I-287
CAS:<p>I-287 is a selective, orally active PAR2 inhibitor that functions as a negative allosteric modulator of Gαq and Gα12/13 activity and their downstream effectors.</p>Fórmula:C30H30ClFN4O4Forma y color:SolidPeso molecular:565.04
