Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.523 productos)
- Apoptosis(5.792 productos)
- Ciclo celular / Checkpoint(4.449 productos)
- Cromatina / Epigenética(2.238 productos)
- Señalización citoesquelética(1.383 productos)
- Daño al ADN / Reparación del ADN(2.825 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.526 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.202 productos)
- Transportador de membrana / canal de iones(2.790 productos)
- Metabolismo(9.448 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.926 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.016 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66641 productos de "Inhibidores"
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WAY-299375
CAS:<p>WAY-299375 is a research-active molecule targeting amyloid diseases and synucleinopathies.</p>Fórmula:C17H16N2Forma y color:SolidPeso molecular:248.32GW-597901
CAS:<p>GW-597901, an β2 adrenergic receptor agonist, is used potentially for the treatment of asthma and chronic obstructive.</p>Fórmula:C25H38N2O6SForma y color:SolidPeso molecular:494.64AGN-191129
CAS:<p>AGN-191129 (PGF2α-OMe) is a PGF2α analog with C-1 carboxyl replaced by O-methyl; it lowers eye pressure, but its receptors are unclear.</p>Fórmula:C21H38O4Forma y color:SolidPeso molecular:354.52RIPK1-IN-16
CAS:<p>RIPK1-IN-16 is an orally active, potent RIPK1 inhibitor that mitigates excessive inflammation via inhibition of RIPK1-mediated necroptosis in vivo.</p>Fórmula:C20H19N5O2SPureza:98%Forma y color:SolidPeso molecular:393.46Antifungal agent 77
CAS:<p>Antifungal agent 77 (Compound 13h) exhibits not only antifungal properties, but also effective insecticidal activity against Mythimna separata, Helicoverpa</p>Fórmula:C21H18FN5O2Forma y color:SolidPeso molecular:391.4Vadaclidine
CAS:<p>Vadaclidine is an orally acting antinociceptive muscarinic agonist.</p>Fórmula:C13H21N3S2Forma y color:SolidPeso molecular:283.46Cavα2δ1&NET-IN-3
CAS:<p>Cavα2δ1&NET-IN-3 (example 216) is an inhibitor targeting both the α2δ subunit of voltage-gated calcium channels (VGCC) and the noradrenaline transporter (NET).</p>Fórmula:C24H30N6O2SForma y color:SolidPeso molecular:466.6μ opioid receptor agonist 3
CAS:<p>Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.</p>Fórmula:C22H28N2O2Pureza:98%Forma y color:SolidPeso molecular:352.47EG01377
CAS:<p>EG01377 is a NRP1 antagonist with antiangiogenic, antimigratory, and antitumor activity, Kd 1.32 μM, IC50s 609 nM for NRP1-a1/b1, inactive on NRP2.</p>Fórmula:C26H30N6O6S2Pureza:98%Forma y color:SolidPeso molecular:586.68TRA 418
CAS:<p>TRA 418 is a TP antagonist.</p>Fórmula:C26H27NO4SForma y color:SolidPeso molecular:449.56Tubulin/JAK2-IN-1
CAS:<p>Tubulin/JAK2-IN-1 (compound 7g) serves as a potent dual inhibitor targeting both Janus kinase 2 (JAK2) and microtubules, demonstrating significant</p>Fórmula:C22H20N6O3Forma y color:SolidPeso molecular:416.43INU-152
CAS:<p>INU-152: pan-RAF inhibitor with potent anti-tumor effects on BRAFV600E cancers, inhibits MAPK in mutant cells, minimal side effects on RAS-mutant melanoma.</p>Fórmula:C20H13F2N7O3SPureza:98%Forma y color:SolidPeso molecular:469.42Aurora kinase inhibitor-8
CAS:<p>Aurora kinase inhibitor-8 is a highly selective inhibitor of Aurora kinase.</p>Fórmula:C30H29N7O3Forma y color:SolidPeso molecular:535.6Velagliflozin proline hydrate
CAS:<p>Velagliflozin proline hydrate, an oral SGLT2 inhibitor, reduces blood sugar by inhibiting renal glucose reabsorption.</p>Fórmula:C28H36N2O8Forma y color:SolidPeso molecular:528.59ICMT-IN-17
CAS:<p>ICMT-IN-17 (compound 52) serves as an ICMT inhibitor, exhibiting an IC50 value of 0.38 μM [1].</p>Fórmula:C22H26F3NOForma y color:SolidPeso molecular:377.44SP-2-225
CAS:<p>SP-2-225, a selective inhibitor of HDAC6, augments the production of cancer-associated antigens and enhances macrophage antigen cross-presentation to T cells,</p>Fórmula:C28H34N2O3Pureza:98%Forma y color:SolidPeso molecular:446.58mTOR inhibitor 9a
CAS:<p>mTOR inhibitor 9a inhibited the growth of human LNCap cells with an ic50 of 80 nm.</p>Fórmula:C20H21N5O2SPureza:99.78%Forma y color:SoildPeso molecular:395.48ICMT-IN-43
CAS:<p>ICMT-IN-43 (compound 22) acts as a potent inhibitor of the enzyme ICMT, exhibiting an inhibitory concentration (IC50) value of 0.04 μM [1].</p>Fórmula:C23H31NOForma y color:SolidPeso molecular:337.5Tetrahydro-11-dehydrocorticosterone
CAS:<p>Tetrahydro-11-dehydrocorticosterone is an inhibitor of 11β-hydroxysteroid dehydrogenase [1].</p>Fórmula:C21H32O4Forma y color:SolidPeso molecular:348.48AEG40826
CAS:<p>AEG40826 (HGS1029) is a hydrochloride salt, IAP inhibitor with potential anti-cancer activity, may enhance apoptosis in tumor cells.</p>Fórmula:C58H80N10O8Forma y color:SolidPeso molecular:1045.32Clobutinol hydrochloride
CAS:<p>Clobutinol hydrochloride, an antitussive agent, influences heart rate and blood pressure, and is utilized in cough-related research [1] [2] [3].</p>Fórmula:C14H23Cl2NOPureza:98%Forma y color:SolidPeso molecular:292.25MALT1-IN-9
CAS:<p>MALT1-IN-9: potent MALT1 protease inhibitor, IC50 <500 nM in Raji cells, significant anticancer effects.</p>Fórmula:C16H12ClF3N6OForma y color:SolidPeso molecular:396.75RXFP1 receptor agonist-5
CAS:<p>RXFP1 receptor agonist-5 (Example 98) is an agonist that targets the RXFP1 receptor and demonstrates its bioactivity by inhibiting cAMP production in HEK293</p>Fórmula:C30H23F6N3O7Forma y color:SolidPeso molecular:651.51HJC0152 free base
CAS:<p>HJC0152 (free base) is an orally active, potent STAT3 inhibitor that impedes cell cycle progression, induces apoptosis, and notably reduces MDA-MB-231 xenograft</p>Fórmula:C15H13Cl2N3O4Pureza:98%Forma y color:SolidPeso molecular:370.19Cobimetinib racemate
CAS:<p>Cobimetinib racemate (Cobimetinib (racemate)) (GDC-0973 racemate) is a selective inhibitor of MEK.Cobimetinib racemate is also known as a mitogen-activated</p>Fórmula:C21H21F3IN3O2Pureza:98.00% - 99.71%Forma y color:SolidPeso molecular:531.31TASP0412098
CAS:<p>TASP0412098 is a potent, selective CRTH2 antagonist with oral activity.</p>Fórmula:C27H23ClN2O3Pureza:98%Forma y color:SolidPeso molecular:458.94HA-1004 dihydrochloride
CAS:<p>HA-1004 dihydrochloride is an inhibitor of PKA, PKC, cGKI, MYLK, and calcium channel protein</p>Fórmula:C12H16ClN5O2SPureza:98%Forma y color:White Crystalline SolidPeso molecular:329.81VU0652925
CAS:<p>VU0652925 is a PAR4 antagonist. VU0652925 has a P-sel IC50 of 39.2 pM (-pIC50±SEM: 10.41±0.04) and a PAC1 IC50 of 43.0 pM (-pIC50±SEM: 10.4±0.04).</p>Fórmula:C24H18N4O4S2Forma y color:SolidPeso molecular:490.55H-Gly-Leu-Phe-OH
CAS:<p>GLF (H-Gly-Leu-Phe-OH), a tripeptide isolated from α-lactalbumin with immunostimulatory properties, prevents alopecia, epidermal thickening, and adipocyte layer</p>Fórmula:C17H25N3O4Forma y color:SolidPeso molecular:335.4WAY-658494
CAS:<p>WAY-658494 is an (active) compound.</p>Fórmula:C13H13NO3S2Forma y color:SolidPeso molecular:295.38MS31
CAS:<p>MS31 is a potent and highly affinity inhibitor of spindlin 1 (SPIN1).</p>Fórmula:C20H27N3O2Pureza:98%Forma y color:SolidPeso molecular:341.45TP-1454
CAS:<p>TP-1454 is an activator against PKM2 with a biochemically determined AC50 of 10 Nm. It can regulate tumor immune responses by acting on T regulatory cells.</p>Fórmula:C19H22F4N4O3SForma y color:SolidPeso molecular:462.46LG 83-6-05
CAS:<p>LG 83-6-05 is a novel kind of sodium channel blocking agent.</p>Fórmula:C21H30ClNO3SForma y color:SolidPeso molecular:411.99RP 70676
CAS:<p>RP 70676 is a potent ACAT inhibitor(rat and rabbit ACAT with IC50 of 25 and 44 nM ).</p>Fórmula:C25H28N4SPureza:99.92%Forma y color:SolidPeso molecular:416.58Cyclohexyl [3,5-bis(methylthio)-4-isothiazolyl]carbamate
CAS:<p>Cyclohexyl [3,5-bis(methylthio)-4-isothiazolyl]carbamate is a chemical agent capable of modulating the lifespan of eukaryotic organisms [1].</p>Fórmula:C12H18N2O2S3Forma y color:SolidPeso molecular:318.48XR9051 Hydrochloride
CAS:<p>XR9051 Hydrochloride, a potent modulator of P-glycoprotein-mediated multidrug resistance (MDR), inhibits the binding of cytotoxics to P-glycoprotein.</p>Fórmula:C39H39ClN4O5Forma y color:SolidPeso molecular:679.21Casein kinase 1δ-IN-4
CAS:<p>"Casein kinase 1δ-IN-4 (compound 567) is a potent inhibitor of casein kinase 1δ with potential application in Alzheimer's disease research [1]."</p>Fórmula:C16H12N6SPureza:98%Forma y color:SolidPeso molecular:320.37T521
CAS:<p>T521 is a selective inhibitor of the PBD of Plk1 and shows no inhibitory effect on Plk2 and Plk3.</p>Fórmula:C17H14FNO5S2Pureza:99.67%Forma y color:SolidPeso molecular:395.43MET kinase-IN-3
CAS:<p>MET kinase-IN-3 is a potent, orally active MET inhibitor (IC50: 9.8 nM) that exhibits good broad-spectrum anti-proliferative effects on cancer cells.</p>Fórmula:C25H16ClF2N5O2Forma y color:SolidPeso molecular:491.88Caspase-3 activator 1
<p>Caspase-3 activator 1 (compound 4b), a Ru(III) metal complex, effectively inhibits gastric tumor growth and metastasis by mediating caspase-3 cleavage.</p>Fórmula:C28H27N6O2RuS2Pureza:98%Forma y color:SolidPeso molecular:644.75(rel)-Tivantinib
CAS:<p>(rel)-Tivantinib is a potent, highly selective inhibitor of the receptor tyrosine kinase c-MET and has additional novel targets, GSK3α and GSK3β, that are</p>Fórmula:C23H19N3O2Forma y color:SolidPeso molecular:369.42NTE-122
CAS:<p>NTE-122 is a competitive Acyl-CoA:cholesterol acyltransferase (ACAT) inhibitor.</p>Fórmula:C38H59ClN6O2Pureza:98%Forma y color:SolidPeso molecular:667.38SB1-F-78
CAS:<p>SB1-F-78 is an USP30 inhibitor.</p>Fórmula:C17H16N6OSForma y color:SolidPeso molecular:352.41CH-5137291
CAS:<p>CH-5137291 is a pure AR antagonist with AR nuclear translocation inhibition activity. It suppresses castration and prevents the growth of prostate cancer cells.</p>Fórmula:C18H14F3N5O3S2Forma y color:SolidPeso molecular:469.46Cy-FBP/SBPase-IN-1
CAS:<p>Cy-FBP/SBPase-IN-1 (compound S5) serves as an inhibitor of the key regulatory enzyme Cy-FBP/SBPase in cyanobacterial photosynthesis, impeding the Calvin cycle</p>Fórmula:C18H14Cl2N4O2S3Forma y color:SolidPeso molecular:485.43CBB1007
CAS:<p>CBB1007 is a potent, reversible, and substrate competitive LSD1 inhibitor (IC50: 5.27 μM for hLSD1).</p>Fórmula:C27H34N8O4Pureza:98%Forma y color:SolidPeso molecular:534.61A 77003
CAS:<p>A 77003 is a HIV-1 protease inhibitor. A77003 impairs HIV-1 protease-mediated Gag processing.</p>Fórmula:C44H58N8O6Forma y color:SolidPeso molecular:794.98p-NH2-CHX-A"-DTPA
CAS:<p>p-NH2-CHX-A"-DTPA is a bifunctional chelating agent [1].</p>Fórmula:C25H36N4O10Forma y color:SolidPeso molecular:552.576CEPN
CAS:<p>6CEPN is a Cyclooxygenase-1 inhibitor that acts by suppressing colorectal cancer growth.</p>Fórmula:C23H18O5Forma y color:SolidPeso molecular:374.39sEH/AChE-IN-4
CAS:<p>sEH/AChE-IN-4-15 is a dual sEH and AChE inhibitor crossing the BBB, with IC50s: 3.1 nM (hsEH), 1660 nM (hAChE), 179 nM (hBChE), 14.5 nM (msEH), 102 nM (mAChE).</p>Fórmula:C35H39ClF3N5O3Forma y color:SolidPeso molecular:670.16
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