Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.523 productos)
- Apoptosis(5.792 productos)
- Ciclo celular / Checkpoint(4.449 productos)
- Cromatina / Epigenética(2.238 productos)
- Señalización citoesquelética(1.383 productos)
- Daño al ADN / Reparación del ADN(2.825 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.526 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.202 productos)
- Transportador de membrana / canal de iones(2.790 productos)
- Metabolismo(9.448 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.926 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.016 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66641 productos de "Inhibidores"
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IR-Crizotinib
CAS:<p>IR-Crizotinib is a conjugate of the near-infrared dye IR-786 and Crizotinib, an NF-κB-inducing kinase (NIK) inhibitor, with an IC50 of 3.381 μM for intracranial</p>Fórmula:C53H57Cl2FIN7OPureza:98%Forma y color:SolidPeso molecular:1024.88HPK1-IN-10
CAS:<p>HPK1-IN-10 inhibits HPK1, a MAP4K kinase from progenitor cells, with potential in treating HPK1 diseases, detailed in patent WO2021213317A1.</p>Fórmula:C31H34N6O2Forma y color:SolidPeso molecular:522.64Estrogen receptor modulator 7
CAS:<p>Estrogen Receptor Modulator 7 is a potent modulator of estrogen receptors, utilized in cancer research [1].</p>Fórmula:C30H31BCl2FNO3Pureza:98%Forma y color:SolidPeso molecular:554.29Resorstatin
CAS:<p>Resorstatin is a bioactive chemical.</p>Fórmula:C17H28O2Forma y color:SolidPeso molecular:264.4Activated C Subunit
CAS:<p>Activated C Subunit is utilized in synthesizing exon jumping oligomer conjugates that complement specific target sites within the human anti-muscular atrophy</p>Fórmula:C37H37ClN5O5PForma y color:SolidPeso molecular:698.15ONO 4817
CAS:<p>ONO-4817 suppresses MMPs, limiting plaque progression and aortic hyperplasia in hyperlipidemic rabbits.</p>Fórmula:C22H28N2O6Forma y color:SolidPeso molecular:416.47NAS-181
CAS:<p>NAS-181 is a potent and selective rat 5-hydroxytryptamine 1B (r5-HT1B) antagonist (Ki: 47 nM).NAS-181 enhances the accumulation of 5-HTP in rat brain regions.</p>Fórmula:C20H30N2O7SForma y color:SolidPeso molecular:442.53CP-96021 hydrochloride
CAS:CP-96021 hydrochloride is a potent and orally active antagonist of leukotriene D4 (LTD4)/platelet activating factor receptor (Kis: 34 nM and 37 nM).Fórmula:C29H22ClFN4OSPureza:98%Forma y color:SolidPeso molecular:529.03S1P1 agonist 6 hemicalcium
CAS:<p>Compound I (S1P1 agonist 6 hemicalcium) is an S1P1 agonist that diminishes autoimmune activity by inhibiting lymphocyte trafficking, and serves as an</p>Fórmula:C25H26F3NO3CaPureza:98%Forma y color:SolidPeso molecular:465.51BMS-189664
CAS:<p>BMS-189664 is an inhibitor of thrombin.</p>Fórmula:C22H34N6O4SPureza:98%Forma y color:SolidPeso molecular:478.61KRM-II-81
CAS:<p>KRM-II-81 is a GABAA receptor ligand with enhanced anxiolytic effects in mice and rats.</p>Fórmula:C21H13N5OForma y color:SolidPeso molecular:351.36MF 13
CAS:<p>MF 13 exhibits tumor apoptosis activity.</p>Fórmula:C23H34Cl2N4O4Forma y color:SolidPeso molecular:501.45Targeting the bacterial sliding clamp peptide 46
CAS:<p>Peptide 46 is a short peptide that inhibits SC-dependent DNA synthesis by targeting the bacterial sliding clamp (SC).</p>Fórmula:C47H64N8O11Forma y color:SolidPeso molecular:917.06(R)-JNJ-31020028
CAS:<p>(R)-JNJ-31020028: High-affinity, selective brain-penetrant Y2 receptor antagonist; pIC50: human 8.07, rat 8.22, mouse 8.21.</p>Fórmula:C34H36FN5O2Pureza:98%Forma y color:SolidPeso molecular:565.68BTK-IN-17
<p>BTK-IN-17: selective, oral BTK inhibitor, IC50=13.7 nM, reduces p-BTK Y223/p-PLCγ2 Y1217, anti-inflammatory.</p>Fórmula:C26H23N7O2Forma y color:SolidPeso molecular:465.51BAY-R 1005
CAS:<p>BAY-R 1005, a synthetic glycolipid analogue (GLA) with immunoenhancing properties, is designed to modulate antibody synthesis [1].</p>Fórmula:C44H87N3O8Forma y color:SolidPeso molecular:786.18KRAS G12C inhibitor 21
CAS:<p>KRAS G12C inhibitor 21 is a KRAS G12C inhibitor.</p>Fórmula:C34H30ClN3O4Forma y color:SolidPeso molecular:580.07Lanabecestat HCl
CAS:<p>Lanabecestat (AZD3293/LY3314814) is a potent oral BACE1 inhibitor that crosses the BBB and reduces Aβ levels.</p>Fórmula:C26H29ClN4OForma y color:SolidPeso molecular:448.995Activated T Subunit
CAS:<p>Activated T Subunit is employed in synthesizing exon-jumping oligomer conjugates that target specific sites within the human anti-muscular atrophy protein gene</p>Fórmula:C31H34ClN4O5PForma y color:SolidPeso molecular:609.05INT-767
CAS:<p>INT-767 is a highly potent farneson X receptor (FXR)/TGR5 dual agonist that prevents NASH and promotes visceral fat brown lipogenesis and mitochondrial function</p>Fórmula:C25H43NaO6SPureza:98%Forma y color:SolidPeso molecular:494.66Estrogen receptor modulator 10
CAS:<p>Compound G-5b, an estrogen receptor modulator 10, functions as an estrogen receptor (ER) antagonist (IC50=6.7 nM) and degrader (DC50=0.4 nM).</p>Fórmula:C32H37F9N4O3SPureza:98%Forma y color:SolidPeso molecular:728.71LY3104607
CAS:<p>LY3104607 is an oral GPCR 40 agonist for type 2 diabetes, aimed at reducing glucose.</p>Fórmula:C27H25N3O3Pureza:98%Forma y color:SolidPeso molecular:439.51Ro 5-5453
CAS:<p>Ro 5-5453 is an inhibitor of monoamine oxidase.</p>Fórmula:C9H17NPureza:98%Forma y color:SolidPeso molecular:139.24Isopropyl dodec-11-enylfluorophosphonate
CAS:<p>Isopropyl dodec-11-enylfluorophosphonate (IDEFP) is an organophosphorus ester functioning as a central cannabinoid receptor (CB1) antagonist and exhibits</p>Fórmula:C15H30FO2PPureza:98%Forma y color:SolidPeso molecular:292.37(1α,1'S,4β)-Lanabecestat
CAS:<p>(1α,1'S,4β)-Lanabecestat is a Beta site APP Cleaving Enzymel (BACE1) inhibitor, and has IC50s of 2.2 nM (TR-FRET assay) and 0.28 nM (sAPPp release assay),</p>Fórmula:C26H28N4OForma y color:SolidPeso molecular:412.53RPE65-IN-1
CAS:<p>RPE65-IN-1 (Compound 16e) serves as a potent inhibitor of RPE65, applicable in studies related to retinopathy [1].</p>Fórmula:C17H27NO2Forma y color:SolidPeso molecular:277.4CR-6086
CAS:<p>CR6086: potent EP4 antagonist with DMARD effects, low Ki (16.6 nM), and specific anti-inflammatory action.</p>Fórmula:C26H27F3N2O3Forma y color:SolidPeso molecular:472.5Stafib-2
CAS:<p>Stafib-2 is a potent and selective inhibitor of the transcription factor STAT5b.Stafib-2 inhibits STAT5b and STAT5a with IC50 values of 82 nM and 1.7 μM,</p>Fórmula:C28H26N2O12P2Pureza:98.48%Forma y color:SolidPeso molecular:644.46HIV-1 protease-IN-8
CAS:<p>HIV-1 protease-IN-8 (compound 34b) is a potent inhibitor of the HIV-1 protease enzyme, exhibiting an IC50 of 0.32 nM.</p>Fórmula:C25H35N3O5SPureza:98%Forma y color:SolidPeso molecular:489.63BF738735
CAS:<p>BF738735 is a selective inhibitor of phosphatidylinositol 4-kinase III beta (PI4KIIIβ, IC50 = 5.7 nM) showing higher activity over α(IC50 = 1.7 μM).</p>Fórmula:C21H19FN4O3SPureza:90%Forma y color:SolidPeso molecular:426.46SC 34301
CAS:<p>SC 34301 (Enisoprost), a strong oral PGE1 analog, decreases bacterial translocation and increases burned mice survival.</p>Fórmula:C22H36O5Forma y color:SolidPeso molecular:380.52PAT-505
CAS:<p>PAT-505 is an autologous epidermal growth factor inhibitor.</p>Fórmula:C23H18ClF2N3O2SPureza:98.84%Forma y color:SolidPeso molecular:473.92Nazartinib S-enantiomer
CAS:<p>Nazartinib is an EGFR inhibitor. Nazartinib S-enantiomer is the less active S-enantiomer of Nazartinib.</p>Fórmula:C26H31ClN6O2Pureza:98%Forma y color:SolidPeso molecular:495.02TMX-2164
CAS:<p>TMX-2164: strong, irreversible BCL6 inhibitor, IC50=152 nM, long-lasting action, inhibits cell proliferation.</p>Fórmula:C25H24ClFN6O6SForma y color:SolidPeso molecular:591.01Antitumor agent-119
CAS:<p>Antitumor agent-119 (compound 13K), a 2-benzoxazolyl hydrazone derivative, exhibits anticancer capabilities by impeding the proliferation of Burkitt, CCRF-CEM,</p>Fórmula:C18H14N4OForma y color:SolidPeso molecular:302.33MRT-92 HCl salt
CAS:<p>MRT-92 is a potent Smoothened receptor inhibitor with an IC50 of 0.4 nM, affecting Hh pathway and cancer drug target.</p>Fórmula:C33H35ClN4O5Forma y color:SolidPeso molecular:603.12H 142-08
CAS:<p>H 142-08 is a partial beta 1-agonist with adrenoreceptor stimulatory effects.</p>Fórmula:C22H37N3O6Forma y color:SolidPeso molecular:439.55BMS641
CAS:<p>BMS641 (BMS-209641) is a RARβ agonist with affinity for RARβ that synergistically activates RARβ and RARgamma to induce cell maturation.</p>Fórmula:C27H23ClO2Pureza:98.98%Forma y color:SolidPeso molecular:414.92ACHP Hydrochloride
CAS:<p>ACHP Hydrochloride (IKK-2 Inhibitor VIII) is a highly potent and selective IKK-β inhibitor with an IC50 of 8.5 nM.</p>Fórmula:C21H25ClN4O2Pureza:99.83%Forma y color:SolidPeso molecular:400.9Calicheamicin
CAS:<p>Calicheamicin (Calicheamicin γ1) is an antitumor antibiotic and is a DNA synthesis inhibitor. It also is a cytotoxic agent that causes double-strand DNA breaks.</p>Fórmula:C55H74IN3O21S4Pureza:98.22% - 98.78%Forma y color:SolidPeso molecular:1368.35KY386
CAS:<p>KY386 is a potent and selective DHX33 helicase inhibitor with an IC50 value of 19 nM.</p>Fórmula:C21H19N5O2SForma y color:SolidPeso molecular:405.47PLK1/BRD4-IN-1
CAS:<p>PLK1/BRD4-IN-1 (9b) is an orally active dual inhibitor of PLK1 (IC50: 22 nM) and BRD4 (IC50: 109 nM).</p>Fórmula:C31H43N9O2Forma y color:SolidPeso molecular:573.73GCC-4401C free base
CAS:<p>GCC-4401C free base is a factor Xa inhibitor similar to rivaroxaban that is currently under development for venous thromboembolic disease (VTE).</p>Fórmula:C18H18ClN5O3SForma y color:SolidPeso molecular:419.89KRAS G12C inhibitor 58
CAS:<p>KRAS G12C inhibitor 58 is utilized in cancer research as an inhibitor of the KRAS G12C mutation [1].</p>Fórmula:C51H64ClF4N9O8SPureza:98%Forma y color:SolidPeso molecular:1074.62NWP-0476
CAS:<p>NWP-0476 is a modified BCL-2/BCL-xL inhibitor with enhanced specificity for BCL-xL, suitable for research on relapsed T-acute lymphoblastic leukemia (T-ALL) [1</p>Fórmula:C47H53ClN8O8SForma y color:SolidPeso molecular:925.49VGSCs-IN-1
CAS:<p>VGSCs-IN-1, a VGSC inhibitor and Riluzole analog, exhibits good blocking activity on Nav1.4 and can be used to study cellular excitability disorders.</p>Fórmula:C12H12F3N3OSPureza:99.88%Forma y color:SolidPeso molecular:303.3ST-1006
CAS:<p>ST-1006: histamine H4 agonist, pKi 7.94, anti-inflammatory, anti-pruritic, promotes basophil migration.</p>Fórmula:C16H20Cl2N6Pureza:98.87% - 99.96%Forma y color:SolidPeso molecular:367.28LE135
CAS:<p>LE135: RARα/RARβ antagonist (Ki: 1.4 μM/220 nM), favors RARβ, selective vs RARγ/RXRs; also activates TRPV1/TRPA1 (EC50s: 2.5/20 μM).</p>Fórmula:C29H30N2O2Pureza:97.94%Forma y color:SolidPeso molecular:438.56TP-10
CAS:<p>TP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.</p>Fórmula:C26H19F3N4OPureza:99.21%Forma y color:SolidPeso molecular:460.45PXS-6302 hydrochloride
CAS:<p>PXS-6302 hydrochloride is a potent irreversible lysine oxidase (LOX) inhibitor, inhibiting Bovine LOX, rh LOXL1, rh LOXL2, rh LOXL3, and rh LOXL4 with IC50 of 3</p>Fórmula:C10H11ClF3NO2SPureza:99.89%Forma y color:SoildPeso molecular:301.71
