
Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.542 productos)
- Apoptosis(5.816 productos)
- Ciclo celular / Checkpoint(4.466 productos)
- Cromatina / Epigenética(2.252 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.830 productos)
- Endocrinología / Hormonas(3.518 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.362 productos)
- Inmunología e inflamación(3.540 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(405 productos)
- Señalización MAPK(1.201 productos)
- Transportador de membrana / canal de iones(2.809 productos)
- Metabolismo(9.462 productos)
- Microbiología / Virología(7.003 productos)
- Neurociencia(9.942 productos)
- Otros inhibidores(37.827 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.598 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.012 productos)
- Ubiquitinación(1.651 productos)
Mostrar 16 subcategorías más
Se han encontrado 66618 productos de "Inhibidores"
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(±)5-HETE
CAS:<p>(±)5-HETE is one of the six monohydroxy fatty acids produced by the non-enzymatic oxidation of arachidonic acid.</p>Fórmula:C20H32O3Forma y color:SolidPeso molecular:320.47Diacetoxyscirpenol
CAS:<p>Diacetoxyscirpenol: a fungal mycotoxin causing blood disorders in humans/animals.</p>Fórmula:C19H26O7Pureza:98%Forma y color:Solid SolidPeso molecular:366.41Ref: TM-T15111
Producto descatalogadoMitoPY1
CAS:<p>a fluorescent probe for imaging hydrogen peroxide (H2O2) in mitochondria of living cells</p>Fórmula:C52H53BN2O5PPureza:98%Forma y color:SolidPeso molecular:827.77MRS2802
CAS:<p>MRS2802 is a P2Y14 receptor agonist, its EC50 value for P2Y14 receptor is 63 nM.</p>Fórmula:C10H14F2N2O11P2Pureza:98%Forma y color:SolidPeso molecular:438.169HJM-561
CAS:<p>HJM-561 is a potent and selective EGFR PROTAC with oral bioavailability, capable of overcoming osimertinib-resistant EGFR triple mutations and demonstrating</p>Fórmula:C45H51ClN9O5PPureza:98%Forma y color:SolidPeso molecular:864.37Praluzatamab ravtansine
CAS:<p>Sirtratumab vedotin (ASG15-ME) is an antibody-drug conjugate (ADC) that links a SLITRK6-specific human gamma 2 antibody (Igγ2) to the microtubule disruption agent monomethyl auristatin E (MMAE) through a protease-cleavable linker [1].</p>Pureza:99.40%Forma y color:SoildPROTAC BTK Degrader-3
CAS:<p>PROTAC BTK Degrader-3 is a potent degrader of Bruton's tyrosine kinase (BTK), exhibiting a DC50 (median degradation concentration) of 10.9 nM in Mino cells.</p>Fórmula:C41H40N10O5Pureza:98%Forma y color:SolidPeso molecular:752.82STING agonist-9
CAS:<p>STING agonist-9 (Compound 45): potent, EC50 1.2 nM h-STING, 32.82 μM m-STING; antitumor [1].</p>Fórmula:C39H47N13O6SForma y color:SolidPeso molecular:825.94RdRP-IN-3
CAS:<p>RdRP-IN-3, a potential anti-influenza drug candidate, functions by inhibiting the activity of RNA-dependent RNA polymerase (RdRp).</p>Fórmula:C25H21N3O4Forma y color:SolidPeso molecular:427.46Thalidomide-NH-PEG4-Ms
CAS:<p>Thalidomide-NH-PEG4-Ms: cereblon ligand + linker, for PROTAC BCL-XL degrader XZ739.</p>Fórmula:C22H29N3O10SForma y color:SolidPeso molecular:527.55Taragarestrant meglumine
CAS:<p>Taragarestrant (D-0502) is an oral SERD with potent activity against ER+ breast cancer.</p>Fórmula:C32H42Cl2FN3O7Forma y color:SolidPeso molecular:670.60A031
CAS:<p>A031: PROTAC AR degrader, IC50 < 0.25 μM, inhibits prostate cancer growth in zebrafish.</p>Fórmula:C50H61ClN10O7SForma y color:SolidPeso molecular:981.6Yimitasvir
CAS:<p>Yimitasvir, an oral NS5A inhibitor, treats chronic hepatitis C. Used for research.</p>Fórmula:C49H58N8O6Forma y color:SolidPeso molecular:855.03Azido-PEG12-t-butyl ester
CAS:<p>Azido-PEG12-t-butyl ester, a soluble PEG with azide/reactive t-butyl, forms triazoles via Click Chemistry; deprotectable in acid.</p>Fórmula:C31H62N3O14Forma y color:SolidPeso molecular:700.84BODIPY 576/589
CAS:<p>BODIPY 576/589 is a long wavelength biological labeled dye.</p>Fórmula:C16H14BF2N3O2Forma y color:SolidPeso molecular:329.11Lichenase
CAS:<p>Lichenase, an enzyme, breaks down β-glucans in grains into GOS, aiding polysaccharide degradation in cell walls.</p>Forma y color:SolidDL-Glyceraldehyde-3-phosphate
CAS:<p>DL-Glyceraldehyde-3-phosphate (3-Phosphoglyceraldehyde) inhibits acyltransferases and inhibits the growth of E. coli at high concentrations.</p>Fórmula:C3H7O6PForma y color:SolidPeso molecular:170.06Dabigatran Acyl-β-D-Glucuronide
CAS:<p>Dabigatran acyl-β-D-glucuronide is a major active metabolite of the thrombin inhibitor dabigatran .</p>Fórmula:C31H33N7O9Forma y color:SolidPeso molecular:647.645Glabralide A
CAS:<p>Glabralide A is a natural product from plants</p>Fórmula:C27H32O5Pureza:98%Forma y color:SolidPeso molecular:436.54Ref: TM-TN2407
Producto descatalogadoQuestiomycin A derivatives 20
<p>Questiomycin A derivatives 20 is a Questiomycin A derivative.</p>Fórmula:C15H12N2O4Pureza:99.94%Forma y color:SoildPeso molecular:284.27(D)-PPA 1
CAS:<p>PD-1/PD-L1 binder, Kd 0.51 μM; blocks interaction in flow cytometry at 1 mg/mL; inhibits tumors, extends mouse survival.</p>Fórmula:C70H98N20O21Pureza:98%Forma y color:SolidPeso molecular:1555.67Methyl Green zinc chloride
CAS:<p>Methyl Green zinc chloride: fluorescent DNA dye for cell/gel staining, viability tests; absorbance at 633/677 nm. Store in dark.</p>Fórmula:C27H35N3·Br·xCl2Zn·ClForma y color:SolidPeso molecular:653.23m-Ciaamp
CAS:<p>3-Carboxyphenyl((N-((4-iodophenyl)acetyl)amino)methyl)phosphonate is a bioactive chemical.</p>Fórmula:C16H15INO6PForma y color:SolidPeso molecular:475.175mTORC1-IN-1
<p>mTORC1-IN-1 (T1), a rapamycin homologue (rapalog) and selective inhibitor of mTORC1, controls cell growth and metabolism, with implications in various diseases</p>Pureza:98%Forma y color:Odour SolidPEG2-bis(phosphonic acid)
CAS:<p>PEG2-bis(phosphonic acid) is a PEG Linker.</p>Fórmula:C6H16O8P2Forma y color:SolidPeso molecular:278.13PROTAC BRD4 Degrader-16
CAS:<p>PROTAC BRD4 Degrader-16 is a potent degrader of BRD4, exhibiting IC50 values of 34.58 nM for BRD4 (BD1) and 40.23 nM for BRD4 (BD2).</p>Fórmula:C46H41N7O8Pureza:98%Forma y color:SolidPeso molecular:819.86DAUDA
CAS:<p>DAUDA (11-(dansylamino)undecanoic acid), an environment-sensitive fluorescent fatty acid analogue, exhibits changes in fluorescent emission spectra and</p>Fórmula:C23H34N2O4SForma y color:SolidPeso molecular:434.59FGFR-IN-1
CAS:<p>FGFR-IN-1 targets FGFR1-3 with IC50 <100 nM. (US20130338134A1, ex 219)</p>Fórmula:C26H24F2N4O6SForma y color:SolidPeso molecular:558.55Thalidomide-C2-amido-C2-COOH
CAS:<p>Thalidomide-C2-amido-C2-COOH is a compound that includes a CRBN ligand for the E3 ubiquitin ligase, as well as a linker.</p>Fórmula:C19H20N4O7Pureza:98%Forma y color:SolidPeso molecular:416.38Melarsonyl dipotassium
CAS:<p>Melarsonyl dipotassium, also known as melarsonic acid dipotassium, is a potent anthelmintic agent with the ability to effectively inhibit parasites.</p>Fórmula:C13H13AsK2N6O4S2Forma y color:SolidPeso molecular:534.52Elamipretide acetate
<p>Elamipretide acetate (MTP 131), a small tetrapeptide, targets mitochondria to reduce toxic species and stabilize cardiolipin.</p>Fórmula:C34H53N9O7Pureza:99.76%Forma y color:SoildPeso molecular:699.84ER degrader 3
CAS:<p>ER degrader 3 targets estrogen receptor, key in cell regulation, potential for cancer research.</p>Fórmula:C39H47N5O4Forma y color:SolidPeso molecular:649.82(5R)-Platyphyllone
CAS:<p>(5R)-Platyphyllone has a wide range of applications in life science related research.</p>Fórmula:C19H22O4Pureza:98%Forma y color:SolidPeso molecular:314.381Oroxin A
CAS:<p>Oroxin A, a partial PPARγ agonist, activates PPARγ, inhibits α-glucosidase, and has antioxidant properties.</p>Fórmula:C21H20O10Pureza:98%Forma y color:SolidPeso molecular:432.38Neuraminic acid
CAS:<p>Neuraminic acid: acidic amino sugar, 9 carbon chain, from pyruvic acid + D-mannosamine, in active mucoproteins.</p>Fórmula:C9H17NO8Forma y color:SolidPeso molecular:267.23TLQP-21 TFA
<p>TLQP-21 TFA is a VGF-derived peptide, C3aR1 agonist (mouse EC50: 10.3μM; human EC50: 68.8μM), that raises intracellular Ca2+ for nociception research.</p>Pureza:98%Forma y color:LiquidPYBG
CAS:<p>PYBG serves as a flexible precursor for facile conjugation with diverse fluorescent dyes using 'Click chemistry' and Sonogashira coupling reactions.</p>Fórmula:C16H15N5O2Forma y color:SolidPeso molecular:309.329(Rac)-IBT6A hydrochloride
CAS:<p>(Rac)-IBT6A HCl: racemic Ibrutinib impurity; for IBT6A dimers/adducts; Ibrutinib is a Btk inhibitor (IC50=0.5nM).</p>Fórmula:C22H23ClN6OForma y color:SolidPeso molecular:422.91N2S2-CBMBC
CAS:<p>N2S2-CBMBC, a bromo-benzyl ether, binds to 99mTc for PD-L1 tumor imaging, offering a real-time alternative to immunohistochemistry.</p>Fórmula:C34H33BrClN3O3S2Forma y color:SolidPeso molecular:711.1318-Hydroxycortisol
CAS:<p>18-Hydroxycortisol: adrenal steroid, cortisol derivative, studied in primary aldosteronism.</p>Fórmula:C21H30O6Forma y color:SolidPeso molecular:378.46Kbz probe 1
CAS:<p>Kbz probe 1, an adaptable probe utilized for examining histone benzoylation and interactions within living cells, showcases extensive versatility.</p>Fórmula:C13H17ClF2N2O3Forma y color:SolidPeso molecular:322.73C12 NBD Sphingomyelin
CAS:<p>C12 NBD sphingomyelin, a fluorescent sphingomyelin derivative, serves as a sphingomyelinase substrate (Ex=470 nm, Em=525 nm).</p>Fórmula:C41H73N6O9PForma y color:SolidPeso molecular:825.03Ref: TM-T75371
Producto descatalogadoGynosaponin V
CAS:<p>Gynosaponin V is a useful organic compound for research related to life sciences. The catalog number is T126218 and the CAS number is 1207861-73-1.</p>Fórmula:C54H92O22Forma y color:SolidPeso molecular:1093.31Coumberone
CAS:<p>Coumberone, a fluorogenic probe, is reduced by AKR1C family to fluorescent coumberol; vital for AKR1C research.</p>Fórmula:C22H19NO3Forma y color:SolidPeso molecular:345.398HX103
CAS:<p>HX103: Fluorogenic EGFR-TKI probe; inhibits various EGFR mutations; predicts NSCLC treatment response. IC50: 1.3-977 nM.</p>Fórmula:C26H25ClFN7O5SForma y color:SolidPeso molecular:602.04Ref: TM-T75015
Producto descatalogadoCap-dependent endonuclease-IN-22
CAS:<p>Cap-dependent endonuclease-IN-22 is a powerful inhibitor of cap-dependent endonuclease (CEN) [1].</p>Fórmula:C37H37ClF2N6O7S2Forma y color:SolidPeso molecular:815.31(3,4-Dihydroxy-5-methoxybenzoyl)taraxerol
CAS:<p>(3,4-Dihydroxy-5-methoxybenzoyl)taraxerol is a natural products from plants</p>Fórmula:C38H56O5Pureza:98%Forma y color:SolidPeso molecular:592.85Ref: TM-TN2397
Producto descatalogado2-Cyclohexen-1-one, 5-(1,5-dimethyl-4-hexen-1-yl)-4-hydroxy-2-methyl-
CAS:<p>1-Hydroxybisabola-2,10-dien-4-one is a natural product for research related to life sciences. The catalog number is TN5398 and the CAS number is 124898-71-1.</p>Fórmula:C15H24O2Pureza:98%Forma y color:SolidPeso molecular:236.35Microcystin-LF
CAS:<p>Microcystin-LF, a phenylalanine variant of Microcystin-LR, is a bacterial metabolite that exhibits cellular toxicity in Caco-2 cells [1] [2].</p>Pureza:98%HDAC3/6-IN-2
CAS:<p>HDAC3/6-IN-2 inhibits HDAC6/3 with IC50s 0.368/0.635 μM; promotes cancer cell apoptosis and histone acetylation.</p>Fórmula:C49H67N5O6Forma y color:SolidPeso molecular:822.09

