
Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.523 productos)
- Apoptosis(5.792 productos)
- Ciclo celular / Checkpoint(4.449 productos)
- Cromatina / Epigenética(2.238 productos)
- Señalización citoesquelética(1.383 productos)
- Daño al ADN / Reparación del ADN(2.825 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.526 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.202 productos)
- Transportador de membrana / canal de iones(2.790 productos)
- Metabolismo(9.448 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.926 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.016 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66641 productos de "Inhibidores"
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Glutaminase-IN-1
CAS:<p>Glutaminase-IN-1 (CB839 derivative), a glutaminase (KGA) inhibitor, has antitumor activity in an aggressive H22 hepatocellular carcinoma xenograft model.</p>Fórmula:C26H24F3N7O3SePureza:98.65% - 98.65%Forma y color:SolidPeso molecular:618.47TOOS
CAS:<p>TOOS is a novel highly water-soluble aniline derivative and is widely used in diagnostic tests and biochemical tests.</p>Fórmula:C12H18NNaO4SPureza:98%Forma y color:White Crystalline PowderPeso molecular:295.335'-Homouridine
<p>5’-Homouridine is a useful organic compound for research related to life sciences and the catalog number is TNU1675.</p>Forma y color:SoildCerulenin
CAS:<p>Cerulenin is a natural inhibitor of fatty acid synthase (FAS). It is produced by the fungus Cephalosporium caeruleus.</p>Fórmula:C12H17NO3Pureza:98% - 99.52%Forma y color:SolidPeso molecular:223.27Vinaginsenoside R3
CAS:<p>Vinaginsenoside R3 is a natural product of Panax, Araliaceae.</p>Fórmula:C48H82O17Pureza:98%Forma y color:SolidPeso molecular:931.167Hoechst 33258 analog 5
CAS:<p>Hoechst 33258 analog 5 is an analog of Hoechst stains which are part of a family of blue fluorescent dyes used to stain DNA.</p>Fórmula:C29H26N6Forma y color:SolidPeso molecular:458.56Buparlisib Hydrochloride
CAS:<p>Buparlisib Hydrochloride is an inhibitor of pan-class I PI3K (IC50: 52 nM/166 nM/116 nM/262 nM for p110α/p110β/p110δ/p110γ, respectively).</p>Fórmula:C18H22ClF3N6O2Pureza:98.94%Forma y color:SolidPeso molecular:446.85NSC-2888
CAS:<p>NSC-2888 is a Novel Rho-Kinase-II Inhibitor with Vasodilatory Activity.</p>Fórmula:C8H18O2S2Forma y color:SolidPeso molecular:210.36Sodium catechol sulfate
CAS:<p>Sodium catechol sulfate is a bioactive chemical.</p>Fórmula:C6H4Na2O8S2Pureza:98%Forma y color:Light Tan PowderPeso molecular:314.20Hinesol
CAS:<p>Hinesol, a sesquiterpenoid from Atractylodes lancea, induces apoptosis in HL-60 cells via JNK pathway.</p>Fórmula:C15H26OPureza:98%Forma y color:SolidPeso molecular:222.37Endothelin 1 (swine, human)
CAS:<p>Endothelin 1, a strong vasoconstrictor, targets ETA/ETB receptors, with a synthetic human/swine peptide sequence.</p>Fórmula:C109H159N25O32S5Forma y color:White PowderPeso molecular:2491.9Quercetin 3,7-di-O-rhamnoside
CAS:<p>Quercetin 3,7-di-O-rhamnoside is a natural product for research related to life sciences. The catalog number is TN6193 and the CAS number is 28638-13-3.</p>Fórmula:C27H30O15Pureza:98%Forma y color:SolidPeso molecular:594.5225-Fluoro-4'-thio-cytidine
<p>Nucleoside Derivatives - Thio-nucleosides; Fluoro-modified nucleosides; 5-Modified pyrimidine nucleosides</p>Forma y color:Soild(R)-GNA-U phosphoramidite
<p>(R)-GNA-U phosphoramidite is a useful organic compound for research related to life sciences and the catalog number is TNU1547.</p>Forma y color:Soild2'-O-Methyl-5-iodouridine
CAS:<p>2'-O-Methyl-5-iodouridine (5-Iodo-2'-O-methyluridine) is a purine nucleoside analog that targets malignant tumors of the inert lymphatic system and possesses a</p>Fórmula:C10H13IN2O6Pureza:99.89%Forma y color:SolidPeso molecular:384.121-(2'-Deoxy-5'-O-DMT-2'-fluoro-b-D-arabinofuranosyl)thymine 3'-CE phosphoramidite
CAS:<p>1-(2'-Deoxy-5'-O-DMT-2'-fluoro-b-D-arabinofuranosyl)thymine 3'-CE phosphoramidite is a Nucleoside Phosphoramidite.</p>Fórmula:C40H48FN4O8PForma y color:SolidPeso molecular:762.8Esculentoside D
<p>Esculentoside D is a useful organic compound for research related to life sciences and the catalog number is T123975.</p>Fórmula:C37H58O12Forma y color:SolidPeso molecular:694.859Dibutyl phthalate
CAS:<p>Dibutyl phthalate (1,2-benzenedicarboxylic acid) is a plasticizer that modulates the crotonylation of MSH6, thereby disrupting circadian rhythms in cells.</p>Fórmula:C16H22O4Pureza:99.86%Forma y color:Colorless To Faint Yellow Oily Liquid Liquid It Can Easily Penetrate The Soil And Contaminate Groundwater And Nearby Streams It IsPeso molecular:278.34MC-Val-Cit-PAB-MMAF
CAS:<p>MC-Val-Cit-PAB-MMAF: ADC drug-linker with antitumor MMAF, cleaved by cathepsin.</p>Fórmula:C68H103N11O16Pureza:98%Forma y color:SolidPeso molecular:1330.61Fexofenadine-d6
CAS:<p>Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.</p>Fórmula:C32H39NO4Pureza:98%Forma y color:SolidPeso molecular:507.695'-O-(4,4'-Dimethoxytrityl)-N6-Phenoxyacetyl adenosine
CAS:<p>5'-O-(4,4'-Dimethoxytrityl)-N6-Phenoxyacetyl adenosine is a 2/6/8-modified purine nucleoside.</p>Fórmula:C39H37N5O8Forma y color:SolidPeso molecular:703.74Benzeneboronic acid
CAS:<p>Benzeneboronic acid (Phenylboronic acid) is a boronic acid that is used in Mizoroki-Heck and Suzuki-Miyaura coupling reactions.</p>Fórmula:C6H7BO2Pureza:99.83%Forma y color:White To Off-White SolidPeso molecular:121.93Fmoc-D-Cha-OH
CAS:<p>Fmoc-D-Cha-OH (FDCO) is an apoptotic DNase γ inhibitor that inhibits the release of HMGB1.</p>Fórmula:C24H27NO4Pureza:98.62%Forma y color:SolidPeso molecular:393.48PFM39
CAS:<p>PFM39 is a selective MRE11 exonuclease inhibitor and Mirin analog that prolongs mitosis and inhibits HR.</p>Fórmula:C10H9N3OSPureza:98.98%Forma y color:SolidPeso molecular:219.262-Phenylethyl b-D-glucopyranoside
CAS:<p>2-Phenylethyl b-D-glucopyranoside is a useful organic compound for research related to life sciences.</p>Fórmula:C14H20O6Forma y color:SolidPeso molecular:284.3085-Hydroxymethyl-2'-C-methyluridine
CAS:<p>Nucleoside Derivatives - 2’-Modified nucleosides, 5-Modified pyrimidine nucleosides</p>Fórmula:C11H16N2O7Forma y color:SolidPeso molecular:288.25Cromakalim
CAS:<p>Cromakalim (BRL 34915) is an ATP-dependent K(+) channel opener, a smooth muscle relaxant with antiepileptic activity.</p>Fórmula:C16H18N2O3Pureza:99.39%Forma y color:SolidPeso molecular:286.33N1-(1,1,1-Trifluoroethyl)pseudouridine
CAS:<p>Nucleoside Derivatives - C-Nucleosides; N-Alkylated nucleosides; Fluoro-modified nucleosides</p>Fórmula:C11H13F3N2O6Forma y color:SolidPeso molecular:326.23Dienestrol diacetate
CAS:<p>Dienestrol diacetate, a derivative of the synthetic non-steroid phenolic compound, DIENESTROL, exhibits estrogenic activities.</p>Fórmula:C22H22O4Pureza:98%Forma y color:SolidPeso molecular:350.418-Methyaminoadenosine
CAS:<p>8-Methyaminoadenosine is a Nucleoside Derivative - 8-Modified purine nucleoside.</p>Fórmula:C11H16N6O4Forma y color:SolidPeso molecular:296.28DiFMUP
CAS:<p>DiFMUP (6,8-Difluoro-4-methylumbelliferyl phosphate) inhibits protein tyrosine phosphatases (PTPs) and can be used to assay threonine phosphatase activity.</p>Fórmula:C10H7F2O6PPureza:99.25% - >99.99%Forma y color:SolidPeso molecular:292.13C12-Ceramide
CAS:<p>C12-Ceramide (C12 Ceramide (d18:1/12:0)) is a ceramide present in the protective membranes of babies born to women with pre-eclampsia.</p>Fórmula:C30H59NO3Pureza:>99.99%Forma y color:SolidPeso molecular:481.79N4-Benzoyl-7'-OH-N-trityl morpholinocytosine
CAS:<p>N4-Benzoyl-7'-OH-N-trityl morpholinocytosine is a Morpholino-nucleoside.</p>Fórmula:C35H32N4O4Forma y color:SolidPeso molecular:572.65IMP2-IN-1
CAS:<p>IMP2-IN-1 effectively inhibits IMP2 (IC50: 81.3-127.5 μM), reduces IMP2 in SW480 cells, and hinders Huh7 cell activity.</p>Fórmula:C21H14F3NO4Forma y color:SolidPeso molecular:401.344',5'-Didehydro-5'-deoxyadenosine
CAS:<p>4',5'-Didehydro-5'-deoxyadenosine is a Nucleoside Derivative - 5'-Modified nucleoside.</p>Fórmula:C10H11N5O3Forma y color:SolidPeso molecular:249.23N3-Methylthymidine
CAS:<p>N3-Methylthymidine is a Nucleoside Derivative - N-Methylated nucleoside.</p>Fórmula:C11H16N2O5Forma y color:SolidPeso molecular:256.26Cabralealactone
CAS:<p>Cabralealactone: Antimycobacterial, weakly cytotoxic to BC cells, moderately active vs. NCI-H187 lung cancer.</p>Fórmula:C27H42O3Forma y color:SolidPeso molecular:414.62Ro 41-1049 hydrochloride
CAS:<p>Ro 41-1049 hydrochloride is a reversible and selective inhibitor of monoamine oxidase-A (Kd: 16.5 and 64.4 nM, respectively).</p>Fórmula:C12H13ClFN3OSPureza:98%Forma y color:SolidPeso molecular:301.77FAPI-4
CAS:<p>FAPI-4 is a FAP) inhibitor, a FAPI ligand that shows strong hepatic uptake in PET imaging of the primary liver cancer hepatocellular carcinoma (HCC).</p>Fórmula:C40H54F2N10O10Pureza:98.79%Forma y color:SolidPeso molecular:872.92Propetamphos
CAS:<p>Propetamphos, an organophosphate pesticide, can effectively control cockroaches, flies, mosquitoes, and other pests. It is also effective for cattle lice.</p>Fórmula:C10H20NO4PSPureza:98%Forma y color:SolidPeso molecular:281.316-Chloro-7-deaza-9-(2',3',5'-tri-O-acetyl-b-D-ribofuranosyl)purine
CAS:<p>Nucleoside Derivatives - 7-Deazapurine nucleosides; Halo-nucleosides; Scaffolds and Templates</p>Fórmula:C17H18ClN3O7Forma y color:SolidPeso molecular:411.793'-Azido-3'-deoxy-2-thiouridine
CAS:<p>Nucleoside Derivatives - Azido-nucleosides; Thio-nucleosides; 3’-Modified nucleosides</p>Fórmula:C9H11N5O4SForma y color:SolidPeso molecular:285.28SDZ 220-581 Ammonium salt
CAS:<p>SDZ 220-581 Ammonium salt is a potent, orally active and competitive antagonist of NMDA receptor(pKi : 7.7).</p>Fórmula:C16H20ClN2O5PPureza:98%Forma y color:SolidPeso molecular:386.77Cefoxitin
CAS:<p>Cefoxitin, an oral 2nd-gen cephalosporin antibiotic, combats Gram+/- & anaerobes, for abdominal and gynecological infections.</p>Fórmula:C16H17N3O7S2Pureza:99.8% - 99.89%Forma y color:SolidPeso molecular:427.452'-Chloro-N6-(4-methoxy)benzyl adenosine
CAS:<p>2'-Chloro-N6-(4-methoxy)benzyl adenosine is a Nucleoside Derivative - Halo-nucleoside;2-Modified purine nucleoside; 6-Modified purine nucleoside;.</p>Fórmula:C18H20ClN5O5Forma y color:SolidPeso molecular:421.83N4-Benzoyl-7'-OH-N-DMTr morpholino cytosine
<p>N4-Benzoyl-7'-OH-N-DMTr morpholino cytosine is a Nucleoside Derivative - Morpholino nucleoside.</p>Forma y color:Soild7-Deaza-7-iodoguanosine
CAS:<p>Nucleoside Derivatives - 7-Deaza-purine nucleosides; Halo-nucleosides</p>Fórmula:C11H13IN4O5Forma y color:SolidPeso molecular:408.1511-Oxomogroside III
CAS:<p>11-Oxomogroside III is a natural product from Siraitia grosvenorii Swingle.</p>Fórmula:C48H80O19Pureza:98%Forma y color:SolidPeso molecular:961.143',5'-Bis(O-t-butyldimethylsilyl)-4'-C-hydroxymethyl thymidine
CAS:<p>3',5'-Bis(O-t-butyldimethylsilyl)-4'-C-hydroxymethyl thymidine is a Nucleoside Derivative - 4'-Modified nucleoside; Protected nucleoside w/NH2/OH open.</p>Fórmula:C23H44N2O6Si2Forma y color:SolidPeso molecular:500.786-Methyluridine
CAS:<p>Nucleosides and Reagents - 6-Modified pyrimidine nucleoside</p>Fórmula:C10H14N2O6Forma y color:SolidPeso molecular:258.23
