Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.797 productos)
- Apoptosis(6.275 productos)
- Ciclo celular / Checkpoint(4.805 productos)
- Cromatina / Epigenética(2.462 productos)
- Señalización citoesquelética(1.534 productos)
- Daño al ADN / Reparación del ADN(2.959 productos)
- Endocrinología / Hormonas(3.708 productos)
- Enzima(3.670 productos)
- GPCR / proteína G(9.020 productos)
- Inmunología e inflamación(3.884 productos)
- Virus de la gripe(301 productos)
- Señalización JAK / STAT(414 productos)
- Señalización MAPK(1.249 productos)
- Transportador de membrana / canal de iones(3.050 productos)
- Metabolismo(10.206 productos)
- Microbiología / Virología(7.612 productos)
- Neurociencia(10.379 productos)
- Otros inhibidores(36.012 productos)
- Reducción de oxidación(42 productos)
- Señalización PI3K / Akt / mTOR(1.442 productos)
- Proteasas / Proteasoma(1.724 productos)
- Células madre y Derivados(819 productos)
- Tirosina quinasa / adaptadores(2.035 productos)
- Ubiquitinación(1.718 productos)
Mostrar 16 subcategorías más
Se han encontrado 66683 productos de "Inhibidores"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Zotiraciclib HCl
CAS:Zotiraciclib (TG02/SB1317) is a CDK/JAK2/FLT3 inhibitor potentially treating Myc-overexpressing cancers, including glioblastoma.Fórmula:C23H26Cl2N4OForma y color:SolidPeso molecular:445.388KUNB31
CAS:KUNB31 is a potent and selective inhibitor of Hsp90β.Fórmula:C19H18N2O3Forma y color:SolidPeso molecular:322.36D-Ibotenic Acid
CAS:D-Ibotenic Acid: a psychoactive neurotoxin in Amanita mushrooms, mimics glutamate, and is used in brain research.Fórmula:C5H6N2O4Forma y color:SolidPeso molecular:158.11MS437
CAS:MS437 is a potent TSH receptor agonist.Fórmula:C22H24N2OPureza:98%Forma y color:SolidPeso molecular:332.44Carsatrin (free base)
CAS:Carsatrin, a cardiotonic and antiarrhythmic, enhances muscle contraction and AP duration without affecting key cardiac enzymes.Fórmula:C25H26F2N6OSForma y color:SolidPeso molecular:496.58PD 154740
CAS:PD 154740 is an antagonist of tachykinin neurokinin3 (NK3).Fórmula:C32H47N3O5Forma y color:SolidPeso molecular:553.73Sematilide
CAS:Sematilide is a blocker of selective IKr channel.Fórmula:C14H23N3O3SPureza:98%Forma y color:SolidPeso molecular:313.42ProTAME
CAS:ProTAME inhibits APC/CFzr & APC/CCdc20, enhances cell death with doxorubicin/etoposide in primary/MM cells, especially after TOPIIα upregulation.Fórmula:C34H38N4O12SPureza:98%Forma y color:SolidPeso molecular:726.75EGFR-IN-31
CAS:EGFR-IN-31: Potent EGFR inhibitor, targets mutations & overexpression in NSCLC; potential cancer research compound. (WO2021185298A1, 2)Fórmula:C32H36FN7O2Forma y color:SolidPeso molecular:569.67SHS4121705
CAS:SHS4121705, an oral mitochondrial uncoupler, boosts oxygen use in cells at 4.3 μM EC50. Lowers liver fat, triglycerides, and ALT in NASH mice.Fórmula:C11H6F3N5O3Forma y color:SolidPeso molecular:313.19Felypressin acetate
CAS:Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.Fórmula:C48H69N13O13S2Pureza:97.06%Forma y color:SolidPeso molecular:1100.27ABC294735
CAS:ABC294735 is a dual SK1/SK2 inhibitor with potential anticancer activity.Fórmula:C25H28ClNO3Forma y color:SolidPeso molecular:425.95FE-999011
CAS:FE-999011 is a dipeptidyl peptidase IV inhibitor.Fórmula:C11H19N3OForma y color:SolidPeso molecular:209.29MI-223
CAS:MI-223 sensitizes cancer cells to DNA stress by inhibiting Mcl-1-stimulated HR DNA repair.Fórmula:C23H18ClN3O3Forma y color:SolidPeso molecular:419.86ALT-946 HCl
CAS:ALT-946 HCl is an inhibitor of advanced glycation that has been shown to improve severe nephropathy in the diabetic transgenic (mREN-2)27 rat.Fórmula:C5H14ClN5OForma y color:SolidPeso molecular:195.65PD 173955-Analog1
CAS:PD 173955-Analog1 is a potent c-Src inhibitor known to have activity against a variety of cancers including colon, lung, head and neck carcinoma.Fórmula:C21H14Cl2N4O3Forma y color:SolidPeso molecular:441.27FR-168888 mesylate
CAS:FR-168888, a new Na+/H+ exchange inhibitor, can protect the heart from arrhythmia and myocardial cell death in ischemic and reperfused situations.Fórmula:C14H18N4O5SPureza:98%Forma y color:SolidPeso molecular:354.38Hyoscyamine hydrobromide
CAS:Hyoscyamine hydrobromide is an agent of anticholinergic.Fórmula:C17H24BrNO3Pureza:98%Forma y color:SolidPeso molecular:370.28Amitifadine free base
CAS:Amitifadine (DOV-21947/EB-1010), an antidepressant SNDRI, curbs binge drinking and negative effects in animals with alcoholism-depression.Fórmula:C11H11Cl2NForma y color:SolidPeso molecular:228.12Z-LLF-CHO
CAS:Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.Fórmula:C29H39N3O5Pureza:98%Forma y color:SolidPeso molecular:509.64Cipamfylline
CAS:Cipamfylline: PDE-4 inhibitor, theophylline analogue; treats atopic dermatitis better than placebo, less so than hydrocortisone-17-butyrate.Fórmula:C13H17N5O2Forma y color:SolidPeso molecular:275.31RTI 336
CAS:RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.Fórmula:C24H26Cl2N2OPureza:98%Forma y color:SolidPeso molecular:429.38ZK93423
CAS:ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.Fórmula:C23H22N2O4Forma y color:SolidPeso molecular:390.43HIV-1 inhibitor-48
CAS:HIV-1 inhibitor-48 is a novel non-nucleoside reverse transcriptase inhibitor (NNRTI) and exhibits anti-HIV-1 activity .Fórmula:C19H16BrN5Forma y color:SolidPeso molecular:394.27ABT-239
CAS:ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.Fórmula:C22H22N2OPureza:99.94%Forma y color:SolidPeso molecular:330.42Ref: TM-T14087
1mg47,00€5mg87,00€10mg140,00€25mg285,00€50mg432,00€100mg628,00€200mg879,00€1mL*10mM (DMSO)96,00€P-2281
CAS:P-2281 is an mTOR inhibitor with anticancer and anti-inflammatory properties.P-2281 inhibits dextran sulfate sodium (DSS)-induced colitis by suppressing T-cellFórmula:C9H8ClN3OPureza:99.98%Forma y color:SolidPeso molecular:209.63Levoprotiline hydrochloride
CAS:Levoprotiline hydrochloride is an antidepressant.Fórmula:C20H24ClNOPureza:98%Forma y color:SolidPeso molecular:329.86Ormetoprim
CAS:Ormetoprim (Ro 5-9754), an antibiotic approved for use in the United States, is used to prevent the spread of disease in freshwater aquaculture.Fórmula:C14H18N4O2Pureza:99.92%Forma y color:SolidPeso molecular:274.32Ref: TM-T20702
5mg48,00€10mg70,00€25mg104,00€50mg153,00€100mg216,00€500mg540,00€1mL*10mM (DMSO)84,00€AT-076
CAS:AT-076: κ-opioid (Ki=1.14 nM) & nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) & δ-opioid (Ki=19.6 nM) competitive antagonist.Fórmula:C26H35N3O3Forma y color:SolidPeso molecular:437.57SNX-7081
CAS:NX-7081 targets Hsp90, inhibits inflammation, cytokines, kinases, and angiogenesis; blocks NF-kappaB, reduces ERK/JNK, NO; aids animal models.Fórmula:C24H31N3O3Forma y color:SolidPeso molecular:409.52HJC0149
CAS:HJC0149 is a potent orally bioavailable signal transducer and activator of transcription 3 inhibitor.Fórmula:C15H10ClNO4SForma y color:SolidPeso molecular:335.76PF-04479745 tartrate
CAS:PF-04479745 (PF-4479745) is a selective 5-HT2C agonist with EC50 10 nM, effective in canine SUI models, not targeting 5-HT2A/B.Fórmula:C21H28N4O6Forma y color:SolidPeso molecular:432.477D54 naponate
CAS:<p>D54 Naponate is a stored salt form of biologically active phenothiazine, which has good antitumor activity and can be maintained longer in the body.</p>Fórmula:C21H21Cl2N5O6S2Forma y color:SolidPeso molecular:574.46Mps-BAY2b
CAS:Mps-BAY2b is a novel MPS1 inhibitor.Fórmula:C20H23N5OForma y color:SolidPeso molecular:349.43FRAN-12
CAS:FRAN-12 is a histamine and 5-hydroxytryptamine antagonist with pressor properties.Fórmula:C19H21ClN4SForma y color:SolidPeso molecular:372.91Azalanstat mesylate
CAS:Azalanstat, an anti-obesity drug, inhibits cholesterol synthesis by targeting P450 enzyme lanosterol 14α-demethylase; reduces LDL more than HDL in hamsters.Fórmula:C23H28ClN3O5S2Forma y color:SolidPeso molecular:526.063SGK1 inhibitor
CAS:SGK1 inhibitor targets SGK1/2 over SGK3, blocks GSK3β phosphorylation, lowers HCC1954 cell viability with BYL719, and reduces tumor growth in mice.Fórmula:C17H12Cl2N6O2SForma y color:SolidPeso molecular:435.29DA-11004
CAS:DA-11004 inhibits NADP-dependent IDPc (IC50: 1.49 μM), reduces fatty acid synthesis and glucose in obese mice.Fórmula:C11H9NO2Pureza:98%Forma y color:SolidPeso molecular:187.19Atuzaginstat
CAS:Atuzaginstat is a bacterial protease lysine gingipain inhibitor.Fórmula:C19H25F3N2O3Forma y color:SolidPeso molecular:386.41PGP-4008
CAS:PGP-4008 is a selective and potent P-glycoprotein (Pgp) inhibitor that inhibits tumor growth by co-administration with Doxorubicin.Fórmula:C26H23N3OPureza:97.41% - 97.99%Forma y color:SolidPeso molecular:393.48AN11251
CAS:AN11251: oral anti-Wolbachia, treats onchocerciasis & lymphatic filariasis, EC50=1.5nM (LDW1), 15nM (C6/36).Fórmula:C29H38BFO7Pureza:98%Forma y color:SolidPeso molecular:528.42JNK-1-IN-1
CAS:JNK-1-IN-1 is an inhibitor specifically targeting JNK-1, also exhibiting inhibition of MKK7 with an IC50 value of 7.8μM.Fórmula:C24H22N6SForma y color:SolidPeso molecular:426.54KU-0058948
CAS:KU-0058948: PARP inhibitor, triggers cell cycle arrest and apoptosis in myeloid leukemia cells in vitro.Fórmula:C21H21FN4O2Forma y color:SolidPeso molecular:380.42GU-285
CAS:GU-285 is a potent non-selective adenosine receptor antagonist.Fórmula:C14H14N6OSForma y color:SolidPeso molecular:314.37LWG-301
LWG-301, a GLS1 allosteric inhibitor, IC50 7 nM, impedes glutamine metabolism and prompts apoptosis; shows antitumor effects.Fórmula:C28H38N8O3SForma y color:SolidPeso molecular:566.72NS004
CAS:NS004 is a large-conductance K+ channel opener, it inhibits mitochondrial function in glioma cells.Fórmula:C14H8ClF3N2O2Pureza:98%Forma y color:SolidPeso molecular:328.67Bradanicline HCl
CAS:Bradanicline(TC-5619) is the agonist of Alpha-7 Nicotinic Receptor.Fórmula:C22H24ClN3O2Forma y color:SolidPeso molecular:397.9Oxydipentonium chloride
CAS:Oxydipentonium chloride is a cholinesterase inhibitor that was studied as a muscle relaxant.Fórmula:C16H38Cl2N2OForma y color:SolidPeso molecular:345.39SUN-C5174
CAS:"SUN-C5174 is a selective 5-HT2 antagonist with pA2=8.98; inhibits platelet aggregation and reduces thromboembolic death in mice at ≥0.3 mg/kg."Fórmula:C22H29FN4O2Pureza:98%Forma y color:SolidPeso molecular:400.49Loperamide oxide
CAS:Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.Fórmula:C29H33ClN2O3Forma y color:SolidPeso molecular:493.04
