Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.811 productos)
- Apoptosis(6.295 productos)
- Ciclo celular / Checkpoint(4.842 productos)
- Cromatina / Epigenética(2.526 productos)
- Señalización citoesquelética(1.550 productos)
- Daño al ADN / Reparación del ADN(2.917 productos)
- Endocrinología / Hormonas(3.708 productos)
- Enzima(3.671 productos)
- GPCR / proteína G(9.024 productos)
- Inmunología e inflamación(3.896 productos)
- Virus de la gripe(302 productos)
- Señalización JAK / STAT(418 productos)
- Señalización MAPK(1.248 productos)
- Transportador de membrana / canal de iones(3.094 productos)
- Metabolismo(10.157 productos)
- Microbiología / Virología(7.623 productos)
- Neurociencia(10.360 productos)
- Otros inhibidores(35.913 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.440 productos)
- Proteasas / Proteasoma(1.711 productos)
- Células madre y Derivados(792 productos)
- Tirosina quinasa / adaptadores(2.013 productos)
- Ubiquitinación(1.722 productos)
Mostrar 16 subcategorías más
Se han encontrado 66619 productos de "Inhibidores"
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Binifibrate
CAS:Binifibrate is a hyperlipemiant drug used for the treatment of hyperlipidemia.Fórmula:C25H23ClN2O7Forma y color:SolidPeso molecular:498.91EMI56
CAS:EMI56, a derivative of EMI1, exhibits enhanced potency against mutant EGFR compared to EMI1. Additionally, EMI56 effectively inhibits EGFR triple mutants[1].Fórmula:C21H20N2O3Forma y color:SolidPeso molecular:348.4Bexin-1
CAS:Bexin-1 blocks Munc13-4 from binding to membranes, targeting its C2 domain and stopping ANF-EGFP release induced by ionomycin.Fórmula:C20H26ClN5OSForma y color:SolidPeso molecular:419.97Sphingofungin B
CAS:Sphingofungin B is a useful organic compound for research related to life sciences. The catalog number is T126215 and the CAS number is 121025-45-4.Fórmula:C20H39NO6Forma y color:SolidPeso molecular:389.533Nb-enantride
CAS:Nb-enantride is a novel chiral trialkylborohydride for the asymmetric reduction of ketones.Fórmula:C26H40BLiOForma y color:SolidPeso molecular:386.36ZK112993
CAS:ZK112993 is an antagonist of human progesterone receptor.Fórmula:C29H32O3Forma y color:SolidPeso molecular:428.56SAMT-247
CAS:SAMT-247 is an HIV inhibitor that acts by modifying the nucleocapsid NCp7 region of Gag in infected cells and blocking Gag processing and reducing infectivity.Fórmula:C12H14N2O3SForma y color:SolidPeso molecular:266.32Dansyllysine
CAS:Dansyllysine aids drug binding studies with albumin and is a template for creating biosensor-recognition MIMs.Fórmula:C18H25N3O4SForma y color:SolidPeso molecular:379.47S 332
CAS:S332 is a beta3-agonist, better at enhancing bladder storage than clenbuterol but weaker in reducing bladder contraction during micturition.Fórmula:C16H17N3O3SForma y color:SolidPeso molecular:331.39Cyclazocine
CAS:Cyclazocine is an analgesic with mixed narcotic agonist-antagonist properties.Fórmula:C18H25NOForma y color:SolidPeso molecular:271.4Lefucoxib
CAS:Lefucoxib is a cyclooxygenase-2 (COX-2) inhibitor.Fórmula:C19H17F3N2O2SForma y color:SolidPeso molecular:394.41DNA-PK-IN-3
CAS:DNA-PK-IN-3 is a potent DNA-PK inhibitor, enhancing radio/chemotherapy and reducing tumors with limited side effects.Fórmula:C19H19N9OForma y color:SolidPeso molecular:389.41Sphaerobioside
CAS:Sphaerobioside is a useful organic compound for research related to life sciences. The catalog number is T125786 and the CAS number is 14988-20-6.Fórmula:C27H30O14Forma y color:SolidPeso molecular:578.523JNJ525
JNJ525, a TNFα inhibitor, blocks protein function by hindering TNFα/TNFR1 and TNFα/TNFR2 complexes; IC50s: 1.2 μM (TNFR1), 1.1 μM (TNFR2).Fórmula:C31H30N8Forma y color:SolidPeso molecular:514.64E-4177
CAS:E-4177 is an angiotensin II type 1 receptor (AT1R) antagonist and can be used to study cardiovascular diseases.Fórmula:C24H21N3O2Pureza:98.67% - 99.57%Forma y color:SolidPeso molecular:383.44IMP2-IN-2
CAS:IMP2-IN-2: potent, selective IMP2 inhibitor; IC50s: 120.9 μM (RNA_A), 236.7 μM (RNA_B); used in cancer research.Fórmula:C22H19F3N2O3SForma y color:SolidPeso molecular:448.46Leucinal
CAS:Leucinal inhibits the activity of brain aminopeptidase and potentiates analgesia induced by leu-enkephalen.Fórmula:C6H13NOForma y color:SolidPeso molecular:115.17Rp-cAMPS sodium
CAS:Rp-cAMPS sodium is a phosphorothioate analog of cAMP, a PKA inhibitor and cAMP antagonist that inhibits cAMP-dependent protein kinases.Fórmula:C10H11N5NaO5PSPureza:99.71%Forma y color:SolidPeso molecular:367.25Nicotine lactate
CAS:Nicotine: a stimulant and anxiolytic from nightshades, aids smoking cessation, targets nAChRs excluding α9/α10 subunits.Fórmula:C13H20N2O3Forma y color:SolidPeso molecular:252.31NNGH
CAS:NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.Fórmula:C13H20N2O5SPureza:98.41%Forma y color:SolidPeso molecular:316.37Azetirelin
CAS:Azetirelin, as a TRH analog, has a more potent effect than TRH on the central nervous system.Fórmula:C15H20N6O4Pureza:99.72%Forma y color:SolidPeso molecular:348.36Peraclopone
CAS:Peraclopone, a hypolipidemic drug and 7-Dehydrocholesterol reductase inhibitor, lowers cholesterol and raises provitamin D3 in rats.Fórmula:C20H23Cl2N3O2Forma y color:SolidPeso molecular:408.32Ridazolol
CAS:Ridazolol is a vasodilating and cardioselective beta adrenergic blocker.Fórmula:C15H18Cl2N4O3Pureza:99.05%Forma y color:SolidPeso molecular:373.23FR-900148 sodium dihydrate
CAS:FR-900148 sodium dihydrate is an antibiotic that inhibits cell wall synthesis.Fórmula:C10H16ClN2NaO6Forma y color:SolidPeso molecular:318.69PF-04363467 HCl
CAS:PF-04363467 HCl is a selective dopamine D3/D2 receptor antagonist.Fórmula:C22H30N2O3SForma y color:SolidPeso molecular:402.55(-)-Donepezil
CAS:(-)-Donepezil is an isomer of Donepezil -- a nootropic acting as an inhibitor of acetylcholinesterase.Fórmula:C24H29NO3Forma y color:SolidPeso molecular:379.49BSJ-01-175
CAS:BSJ-01-175: Selective, potent covalent inhibitor of CDK12/13, targets cancer cells, inhibits phosphorylated RNA polymerase II, downregulates CDK12 genes.Fórmula:C30H33ClN6O2Forma y color:SolidPeso molecular:545.08FC9402
CAS:FC9402: selective SQOR inhibitor, lessens heart hypertrophy and LV fibrosis.Fórmula:C19H16N4OForma y color:SolidPeso molecular:316.36L 652813
CAS:L 652813 is one kind of quaternary heterocyclylamino beta-lactam.Fórmula:C24H22N6NaO5S2Forma y color:SolidPeso molecular:561.59MIF-IN-5
CAS:MIF-IN-5: reversible MIF inhibitor, IC50 4.8 μM, Ki 3.3 μM.Fórmula:C18H14FN5O2Forma y color:SolidPeso molecular:351.33ATRA-BA Hybrid
CAS:ATRA-BA, a prodrug, releases ATRA and butyric acid to inhibit MDA-MB-231 and PC3 cancer cells with enhanced potency at 20 μM.Fórmula:C31H40O4Forma y color:SolidPeso molecular:476.65COX-2/5-LOX-IN-2
CAS:COX-2/5-LOX-IN-2, a benzothiophen derivative, inhibits COX-1, COX-2, 5-LOX with IC50s of 5.40, 0.01, 1.78 μM. More effective than Celecoxib, Indomethacin.Fórmula:C18H13N3O4S2Forma y color:SolidPeso molecular:399.44Benzoxonium chloride
CAS:Benzoxonium chloride used in Thio-Ben for cutaneous leishmaniasis treatment with cryotherapy.Fórmula:C23H42ClNO2Forma y color:SolidPeso molecular:400.04BMS 180448
CAS:BMS 180448 is a prototype mitochondrial ATP-sensitive K+ (Mitok (ATP)) channel opener with cardioprotective and vasodilating properties.Fórmula:C20H18ClN5O2Forma y color:SolidPeso molecular:395.84APC-3316 hydrochloride
CAS:APC-3316 hydrochloride is a vinyl sulfone cysteine protease inhibitor and selective CCR4 antagonist.Fórmula:C32H39ClN4O4SForma y color:SolidPeso molecular:611.19APC-3316 tosylate
CAS:APC-3316 tosylate is a vinyl sulfone cysteine protease inhibitor and selective CCR4 antagonist.Fórmula:C39H46N4O7S2Forma y color:SolidPeso molecular:746.94GSK730
CAS:GSK730 is an inactive enantiomer of GSK729 (GLXC-09258).Fórmula:C16H16F3N3O2Forma y color:SolidPeso molecular:339.31DNA-PK-IN-5
CAS:DNA-PK-IN-5: potent DNA-PK inhibitor, reduces tumor repair, induces apoptosis, enhances radiotherapy, overcomes resistance.Fórmula:C21H22N8O2Forma y color:SolidPeso molecular:418.45Zelandopam free base
CAS:Zelandopam: dopamine D1 agonist, boosts pancreatic secretion, renal vasodilator, counters renal dysfunction.Fórmula:C15H15NO4Forma y color:SolidPeso molecular:273.28Isoidide mononitrate
CAS:Isoidide mononitrate is a potent mononitrate vasodilator.Fórmula:C6H9NO6Forma y color:SolidPeso molecular:191.14FK-448 methanesulfonate
CAS:FK-448 methanesulfonate is a chymotrypsin inhibitor that has been shown to affect intestinal absorption of insulin in rats and dogs .Fórmula:C25H30N2O3·xCH4O3SForma y color:SolidPeso molecular:502.63Dads-E
CAS:DADT-FA labels Tc99m with DADT at room temp; DADT-E does so in ethanol at high temp, both reduced by stannous.Fórmula:C30H47ClN2O2S2Forma y color:SolidPeso molecular:567.29SV5
CAS:SV5: potent anti-Alzheimer's, protects SHSY-5Y from Aβ1-42 death, stable with optimal pharmacology in plasma, antioxidant, neuroprotective.Fórmula:C21H30N2O4S2Forma y color:SolidPeso molecular:438.6MRS542
CAS:MRS542 acts as an A3AR antagonist and partial agonist; its partial agonism is due to LUF6000.Fórmula:C17H17ClIN5O4Forma y color:SolidPeso molecular:517.71HDAC-IN-43
CAS:HDAC-IN-43: potent HDAC 1/3/6 inhibitor (IC50: 82 nM HDAC1, 45 nM HDAC3, 24 nM HDAC6); weak PI3K/mTOR (IC50: 3.6μM, 3.7μM); anti-proliferative.Fórmula:C22H28N6O4Forma y color:SolidPeso molecular:440.5CBK289001
CAS:CBK289001 inhibits TRAP 5b MV, 5b OX & 5a OX with IC50s: 125μM, 4.21μM, 14.2μM.
Fórmula:C19H20N6O4Forma y color:SolidPeso molecular:396.4Ammonium, (6-(p-triethylammoniophenyl)hexyl)triethyl-, diiodide
CAS:Ammonium, (6-(p-triethylammoniophenyl)hexyl)triethyl-, diiodide is a bioactive chemical.Fórmula:C24H46I2N2Forma y color:SolidPeso molecular:616.44HX-600
CAS:HX-600 is a synthetic agonist for the RXR-Nurr1 heterodimer complex. HX-600 prevents ischemia-induced neuronal damage.Fórmula:C29H30N2O2Forma y color:SolidPeso molecular:438.56Pralidoxime mesylate
CAS:Pralidoxime mesylate is a Cholinesterase ReactivatorFórmula:C8H12N2O4SForma y color:SolidPeso molecular:232.25Debio 0617B
CAS:Debio 0617B inhibits kinases for AML stem cell treatment, targeting JAK, ABL, SRC, and STAT3-related tumours.Fórmula:C28H23ClF3N7O2Forma y color:SolidPeso molecular:581.98
