Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.542 productos)
- Apoptosis(5.816 productos)
- Ciclo celular / Checkpoint(4.466 productos)
- Cromatina / Epigenética(2.252 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.830 productos)
- Endocrinología / Hormonas(3.518 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.362 productos)
- Inmunología e inflamación(3.540 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(405 productos)
- Señalización MAPK(1.201 productos)
- Transportador de membrana / canal de iones(2.809 productos)
- Metabolismo(9.462 productos)
- Microbiología / Virología(7.003 productos)
- Neurociencia(9.942 productos)
- Otros inhibidores(37.827 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.598 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.012 productos)
- Ubiquitinación(1.651 productos)
Mostrar 16 subcategorías más
Se han encontrado 66618 productos de "Inhibidores"
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MLN3126
CAS:<p>MLN3126: Oral CCR9 blocker, hinders CCL25-triggered chemotaxis/thymocyte calcium influx, IC50 of 6.3 nM.</p>Fórmula:C21H19ClN2O5SForma y color:SolidPeso molecular:446.9PSB-10211
CAS:<p>PSB-10211 is a potent competitive antagonist and positive modulator of the P2X2 receptor.</p>Fórmula:C23H13Cl2N6NaO5SForma y color:SolidPeso molecular:579.3438Pirbuterol hydrochloride
CAS:<p>Pirbuterol hydrochloride is a bronchodilator.</p>Fórmula:C12H21ClN2O3Forma y color:SolidPeso molecular:276.76Tyrphostin AG17
CAS:<p>Tyrphostin AG17 induces fat cell death, regulates fat tissue growth, may treat obesity, and inhibits cancer cell expansion.</p>Fórmula:C12H10N2OForma y color:SolidPeso molecular:198.22Antiproliferative agent-5
CAS:<p>Compound 4o inhibits gastric cancer growth, blocks G2/M cell cycle, induces ROS, and triggers autophagy. Used in anti-cancer studies.</p>Fórmula:C28H21BrN8OSForma y color:SolidPeso molecular:597.49BBR 2160
CAS:<p>BBR 2160: a calcium-antagonist dihydropyridine derivative, reduces heart tissue contractility and shortens action potentials.</p>Fórmula:C21H25N3O7SForma y color:SolidPeso molecular:463.5(Z)-p-cyano-α-Cyanostilbene
CAS:<p>(Z)-p-cyano-α-Cyanostilbene (compound 11) is a phenantrene derivative that has antiproliferative activity.</p>Fórmula:C16H10N2Forma y color:SolidPeso molecular:230.26Z30529104
CAS:<p>Z30529104 is a Rpn11 inhibitor.</p>Fórmula:C24H28N4O6SForma y color:SolidPeso molecular:500.57HWY-5069 bromide
CAS:<p>HWY-5069 bromide is an isoquinolinium derivative that inhibits the proliferation of wild-type and all mutants of Schizosaccharomyces pombe.</p>Fórmula:C31H45BrFNForma y color:SolidPeso molecular:530.61DOOT-2d
CAS:<p>DOOT-2d is a selective MAO-B inhibitor.</p>Fórmula:C15H13FO3Forma y color:SolidPeso molecular:260.264′-Deoxyphlorizin
CAS:<p>4'-Deoxyphlorizin inhibits glucose transport; Km 0.59 nM, Ki 0.33 nM for phlorizin hydrolase.</p>Fórmula:C21H24O9Forma y color:SolidPeso molecular:420.41IY-80843
CAS:<p>IY-80843 is an H2-receptor antagonist.</p>Fórmula:C19H20N4OForma y color:SolidPeso molecular:320.39Dexefaroxan
CAS:<p>Dexefaroxan is an alpha(2)-adrenoceptor antagonist.</p>Fórmula:C13H16N2OForma y color:SolidPeso molecular:216.28FGFR-IN-9
<p>FGFR-IN-9: oral FGFR inhibitor, IC50: 17.1 nM (FGFR4 WT), 29.6 (FGFR3), 30.7 (V550L), 46.7 (FGFR2), 64.3 nM (FGFR1).</p>Fórmula:C25H28N6O3SForma y color:SolidPeso molecular:492.59JAK1-IN-B61
CAS:<p>JAK1-IN-B61 is a JAK1 inhibitor.</p>Fórmula:C14H17N5O2Forma y color:SolidPeso molecular:287.32ATPase-IN-2
CAS:<p>ATPase-IN-2: ATPase inhibitor (IC50 = 0.9μM), also blocks C. difficile toxin B (AC50 = 30.91μM). Used in ATP research.</p>Fórmula:C22H20N2O4Forma y color:SolidPeso molecular:376.41MAX-40279 hydrochloride
CAS:<p>MAX-40279 HCl: potent FLT3/FGFR inhibitor; potential in AML research.</p>Fórmula:C22H24ClFN6OSForma y color:SolidPeso molecular:474.98Pyrvinium chloride
CAS:<p>Pyrvinium chloride is used in the treatment of pinworm infections</p>Fórmula:C26H28ClN3Forma y color:SolidPeso molecular:417.97GABAA receptor agent 7
CAS:<p>Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.</p>Fórmula:C18H13ClN4OForma y color:SolidPeso molecular:336.77Quoromycin
CAS:<p>Quoromycin, a new antivirulence drug, hinders Vibrio vulnificus by disrupting SmcR in quorum-sensing, reducing virulence in vitro and in vivo.</p>Fórmula:C12H8N2O2SForma y color:SolidPeso molecular:244.27RGB-286147
CAS:<p>RGB-286147 is a potent, selective, ATP-competitive Cdks inhibitor.</p>Fórmula:C23H22Cl2N4O3Pureza:98%Forma y color:SolidPeso molecular:473.35WB403
CAS:<p>WB403 activates TGR5, lowers fasting/postprandial glucose and HbA1c, enhances glucose tolerance, and normalizes pancreatic α/β-cells in diabetic mice.</p>Fórmula:C19H19BrN2OSPureza:98%Forma y color:SolidPeso molecular:403.34FabG1-IN-1
CAS:<p>FabG1-IN-1 (Compound 29) is a potent inhibitor of MabA (FabG1) (IC50: 38 μM).</p>Fórmula:C14H8Cl2INO3Forma y color:SolidPeso molecular:436.03Bourgeonal
CAS:<p>Bourgeonal triggers hOR17-4, boosts sperm calcium levels, acts as chemoattractant, and enhances sperm motility in a dose-dependent way.</p>Fórmula:C13H18OForma y color:SolidPeso molecular:190.28ML-077
CAS:<p>ML-077/VU0255011: Selective KCC2 antagonist, IC50=537 nM, saline soluble, cell permeable, submicromolar potency for in vitro KCC2 research.</p>Fórmula:C17H16N4OS2Forma y color:SolidPeso molecular:356.47Belaperidone
CAS:<p>Belaperidone, an antipsychotic, resembles clozapine, binds D(4) and 5-HT(2A) receptors, minimally extends Q-T without causing arrhythmias.</p>Fórmula:C22H22FN3O2Forma y color:SolidPeso molecular:379.43Dilmapimod tosylate
CAS:<p>Dilmapimod tosylate, a p38 MAPK inhibitor, targets IL-1β, was in phase III trials by GlaxoSmithKline for rheumatoid arthritis and more.</p>Fórmula:C30H27F3N4O6SForma y color:SolidPeso molecular:628.62KUNB31
CAS:<p>KUNB31 is a potent and selective inhibitor of Hsp90β.</p>Fórmula:C19H18N2O3Forma y color:SolidPeso molecular:322.36Ro 04-5595 free base
CAS:<p>"Ro 04-5595: Selective NMDA NR2B antagonist, EC50 186nmol/L; binds EVT-101 site; hierarchy of inhibition affinity observed."</p>Fórmula:C19H22ClNO2Forma y color:SolidPeso molecular:331.84NY0173
CAS:<p>NY0173 is a potent exchange protein activated by cAMP antagonists.</p>Fórmula:C18H15Cl3N4O2Forma y color:SolidPeso molecular:425.7IAA-94
CAS:<p>IAA-94 is an inhibitor of chloride channels, it binds channels in bovine kidney cortex microsomes with a Ki value of 1 µM.</p>Fórmula:C17H18Cl2O4Forma y color:SolidPeso molecular:357.232'-Deoxy-L-guanosine
CAS:<p>2'-Deoxy-L-guanosine is a nucleoside that shows antibiotic properties by inhibiting protein synthesis, leading to cell death.</p>Fórmula:C10H13N5O4Forma y color:SolidPeso molecular:267.24FUBP1-IN-2
CAS:<p>FUBP1-IN-2 hinders FUBP1, affects c-Myc and p21 expression, and depletes polyamines.</p>Fórmula:C26H26ClN3O4Forma y color:SolidPeso molecular:479.96Ro 7-0213
CAS:<p>RO 7-0213 is a novel benzodiazepine (RO7-0213) containing a fully positive quaternary ammonium component.</p>Fórmula:C20H23ClN3OForma y color:SolidPeso molecular:356.87ATX inhibitor 16
CAS:<p>ATX inhibitor 16 is a potent inhibitor of ATX (IC50: 0.0021 μM). ATX inhibitor 16 exhibits a significant anti-proliferative effect on breast cancer cells.</p>Fórmula:C28H27F3N6OS2Forma y color:SolidPeso molecular:584.68FAUC-299
CAS:<p>FAUC-299 is a dopamine D4 receptor agonist.</p>Fórmula:C20H20N4Forma y color:SolidPeso molecular:316.4Nampt activator-3
CAS:<p>NAMPT activator-3: a NAT derivative, EC50 of 2.6 μM, KD 132 nM, protects cells, prevents FK866 toxicity, and is neuroprotective in CIPN mice.</p>Fórmula:C19H20N2O3Forma y color:SolidPeso molecular:324.37Lumefantrine Impurity A
CAS:<p>2-(Dibutylamino)-2-(2,7-dichloro-9-(4-chlorobenzylidene)-9H-fluoren-4-yl)ethanol, (RS, Z)- is a bioactive chemical.</p>Fórmula:C30H32Cl3NOForma y color:SolidPeso molecular:528.94Oxyfedrine
CAS:<p>Oxyfedrine: oral β-adrenoreceptor agonist, vasodilator for cardiovascular research.</p>Fórmula:C19H23NO3Forma y color:SolidPeso molecular:313.39JS1310
CAS:<p>JS1310 is a selective PRMT7 inhibitor (IC50: 5 μM against human PRMT7). JS1310 has shown anti-cancer effects on different cancer cells.</p>Fórmula:C23H22FN5O3Forma y color:SolidPeso molecular:435.45N12N
CAS:<p>N12N is a polyamine inverse NMDA receptor agonist.</p>Fórmula:C12H28N2Pureza:98%Forma y color:White SolidPeso molecular:200.36Cgs 11361
CAS:<p>Cgs 11361 is a GABA-A receptor antagonist.</p>Fórmula:C16H11N3O2Forma y color:SolidPeso molecular:277.28GLS1 Inhibitor-3
CAS:<p>GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.</p>Fórmula:C30H32N10O2SForma y color:SolidPeso molecular:596.71RY024
CAS:<p>RY024 is a behavioral alcohol antagonist.</p>Fórmula:C19H19N3O3Forma y color:SolidPeso molecular:337.37AT1R antagonist 1
CAS:<p>AT1R Antagonist 1 (compound 10) serves as a potent, selective ligand for AT1R with considerable affinity, demonstrated by a K i value of 8.5 nM [1].</p>Fórmula:C28H32F3N5O4S2Forma y color:SolidPeso molecular:623.71MCC1189
CAS:<p>MCC1189 is a first-in-class MFS efflux pump CaMdr1p inhibitor.</p>Fórmula:C22H20N2O2Forma y color:SolidPeso molecular:344.41NDJ18
CAS:<p>NDJ18: a potent SIRT2 inhibitor showing anticancer effects on triple-negative breast cancer cells, promising for further study.</p>Fórmula:C21H20N2OForma y color:SolidPeso molecular:316.4EGFR-IN-55
CAS:<p>"EGFR-IN-55 targets EGFRWT (70 nM IC50) & EGFRL858R/T790M (3.9 nM IC50), halts NCI-H1975 cell cycle in G0/G1, showing anticancer properties."</p>Fórmula:C25H25Cl2N7O2Forma y color:SolidPeso molecular:526.42TAK-603
CAS:<p>TAK-603: anti-rheumatic, anti-inflammatory drug; selectively halts Th1 cytokine production, prevents adjuvant arthritis progression.</p>Fórmula:C25H26N4O6Forma y color:SolidPeso molecular:478.5F8-S43-S3
CAS:<p>F8-S43-S3 is a SARS-CoV-2 main protease inhibitor (IC 50 = 9.69 μM) [1].</p>Fórmula:C12H10N4O3SForma y color:SolidPeso molecular:290.3
