
Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.542 productos)
- Apoptosis(5.816 productos)
- Ciclo celular / Checkpoint(4.466 productos)
- Cromatina / Epigenética(2.252 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.830 productos)
- Endocrinología / Hormonas(3.518 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.362 productos)
- Inmunología e inflamación(3.540 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(405 productos)
- Señalización MAPK(1.201 productos)
- Transportador de membrana / canal de iones(2.809 productos)
- Metabolismo(9.462 productos)
- Microbiología / Virología(7.003 productos)
- Neurociencia(9.942 productos)
- Otros inhibidores(37.827 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.598 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.012 productos)
- Ubiquitinación(1.651 productos)
Mostrar 16 subcategorías más
Se han encontrado 66618 productos de "Inhibidores"
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Metaphit
CAS:<p>Acylator of PCP and σ-receptors</p>Fórmula:C18H24N2SPureza:98%Forma y color:SolidPeso molecular:300.46SNAP 398299
CAS:<p>SNAP 398299 is a Glycopeptide Receptor Type 3 (Gal3) antagonist with anxiolytic and antidepressant-like effects and is used in the study of mood disorders.</p>Fórmula:C27H24F3N3O2Pureza:97.16%Forma y color:SolidPeso molecular:479.49Carbetamide
CAS:Carbetamide (Caswell No. 159B) is a herbicide with a good reproduction of mobility in the soil.Fórmula:C12H16N2O3Pureza:99.88%Forma y color:SolidPeso molecular:236.27CID 5951923
CAS:CID 5951923 is an inhibitor of KLF5 transcription factor with an IC50 of 603 nM.Fórmula:C16H18N2O7SPureza:99.95%Forma y color:SolidPeso molecular:382.39Cyclazosin HCl
CAS:<p>Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.</p>Fórmula:C23H28ClN5O4Pureza:99.10%Forma y color:SolidPeso molecular:473.95MHY908
CAS:MHY908, a novel inhibitor of melanogenesis, potently inhibits mushroom tyrosinase activity in a dose-dependent manner.Fórmula:C17H14ClNO3SPureza:98%Forma y color:SolidPeso molecular:347.8213(R)-HODE cholesteryl ester
CAS:<p>13(R)-HODE cholesteryl ester, found in atherosclerotic lesions, may form enzymatically or by lipid peroxidation, is a standard for chiral HODE analysis.</p>Fórmula:C45H76O3Forma y color:SolidPeso molecular:665.08Homotyrosine, (+)-
CAS:<p>Homotyrosine, (+)- is an amino acid used as a very stable, selective, and renally safe sodium channel blocker.</p>Fórmula:C10H13NO3Pureza:98%Forma y color:SolidPeso molecular:195.22PDE-9 inhibitor
CAS:<p>PDE-9 inhibitor is used for treatment neurodegenerative diseases.</p>Fórmula:C22H27N5O2Pureza:98%Forma y color:SolidPeso molecular:393.48ALDH1A1-IN-2
CAS:<p>ALDH1A1-IN-2 is an aldehyde dehydrogenase 1a1 inhibitor with anticancer activity.ALDH1A1-IN-2 may be used in the study of breast cancer, inflammation or obesity</p>Fórmula:C25H23ClN4O3SPureza:99.48%Forma y color:SolidPeso molecular:494.99Tilapertin
CAS:Tilapertin is an oral glycine transporter type-1 inhibitor.Fórmula:C20H21F3N2O2Pureza:98%Forma y color:SolidPeso molecular:378.39SCH 221510
CAS:<p>SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.</p>Fórmula:C28H31NOPureza:99.54%Forma y color:SolidPeso molecular:397.55Nucleoside-Analog-2
CAS:<p>Nucleoside-Analog-2 is a 4'-Azidocytidine analogue, used to against Hepatitis C virus (HCV) replication.</p>Fórmula:C9H11N5O6Pureza:98%Forma y color:SolidPeso molecular:285.21Dicarbine
CAS:<p>Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.</p>Fórmula:C13H18N2Pureza:98%Forma y color:SolidPeso molecular:202.3Licraside
CAS:<p>Licraside is a tyrosinase inhibitor with an IC50 of 0.072 mM for monophenolase and can be used in studies about antibrowning and depigmenting agents.</p>Fórmula:C26H30O13Pureza:99.75%Forma y color:SolidPeso molecular:550.51Peraclopone
CAS:<p>Peraclopone, a hypolipidemic drug and 7-Dehydrocholesterol reductase inhibitor, lowers cholesterol and raises provitamin D3 in rats.</p>Fórmula:C20H23Cl2N3O2Forma y color:SolidPeso molecular:408.32Ridazolol
CAS:<p>Ridazolol is a vasodilating and cardioselective beta adrenergic blocker.</p>Fórmula:C15H18Cl2N4O3Pureza:99.05%Forma y color:SolidPeso molecular:373.23AKOS024836912
CAS:<p>AKOS024836912 is an inhibitor of EGF-EGFR interactions.</p>Fórmula:C18H23N5O2Forma y color:SolidPeso molecular:341.41BTA-1
CAS:<p>BTA-1 is an uncharged derivative of thioflavin-T that has high affinity for Aβ fibrils and shows very good brain entry and clearance [1].</p>Fórmula:C14H12N2SForma y color:SolidPeso molecular:240.32SC 51089 free base
CAS:<p>SC 51089 free base is a selective antagonist of the prostaglandin E2 EP1 receptor, demonstrating neuroprotective activity.</p>Fórmula:C22H19ClN4O3Forma y color:SolidPeso molecular:422.86Guadecitabine sodium
CAS:<p>Guadecitabine sodium is a inhibitor of second-generation DNA methyltransferases (DNMT) .</p>Fórmula:C18H24N9NaO10PPureza:98%Forma y color:SolidPeso molecular:580.407WEB2347
CAS:<p>WEB2347 is a novel, potent and long acting antagonist of hetrazepinoic PAF.</p>Fórmula:C25H28ClN5OSForma y color:SolidPeso molecular:482.04KRCA-0377
CAS:<p>KRCA-0377 is a potent inhibitor of ALK.</p>Fórmula:C23H26ClN5O3SPureza:98%Forma y color:SolidPeso molecular:488Benzoic acid, m-(2-methyl-5-phenylpyrrol-1-yl)-, compd. with morpholine (1:1)
CAS:<p>Benzoic acid, m-(2-methyl-5-phenylpyrrol-1-yl)-, compd. with morpholine (1:1) is a bioactive chemical.</p>Fórmula:C22H24N2O3Forma y color:SolidPeso molecular:364.44SB26019
CAS:<p>SB26019: Potent anti-neuroinflammation; inhibits NF-κB via α-tubulin monomers preventing p65 translocation.</p>Fórmula:C24H20O4Forma y color:SolidPeso molecular:372.41AH 19437
CAS:<p>AH 19437 is a prostanoid receptor.</p>Fórmula:C24H33NO5Forma y color:SolidPeso molecular:415.52Guanoxabenz
CAS:<p>Guanoxabenz is an α2 adrenergic receptor agonist.</p>Fórmula:C8H8Cl2N4OPureza:98%Forma y color:SolidPeso molecular:247.08UPF-648 sodium salt
CAS:<p>UPF-648 sodium salt is an inhibitor of kynurenine 3-monooxygenase (KMO) and exhibits highly active at 1 uM (81 ± 10% KMO inhibition).</p>Fórmula:C11H8Cl2NaO3Pureza:98%Forma y color:SolidPeso molecular:282.07L 641953
CAS:<p>L 641953 is an antagonist of the thromboxane receptor.</p>Fórmula:C15H9FO3SForma y color:SolidPeso molecular:288.29ML207
CAS:<p>ML207 inhibits lipid storage in Drosophila melanogaster.</p>Fórmula:C26H28N2O3SPureza:98%Forma y color:SolidPeso molecular:448.58Tankyrase Inhibitors (TNKS) 22
<p>Tankyrase Inhibitors 22 is a potent, selective, and orally bioavailable inhibitor of tankyrase (IC50: 0.1nM).</p>Fórmula:C25H25N5O3SPureza:98%Forma y color:SolidPeso molecular:475.56TRK-IN-15
CAS:<p>TRK-IN-15 (X-55): potent TRK kinase inhibitor, aids in TRK-related disease research.</p>Fórmula:C19H20FN5OForma y color:SolidPeso molecular:353.39Mcl1-IN-11
CAS:Mcl1-IN-11 (Compound G) is a selective Mcl-1 inhibitor, less potent at Bcl-2, with Kis of 0.06 and 4.2 μM, respectively.Fórmula:C38H41N3O5S2Pureza:98%Forma y color:SolidPeso molecular:683.88Prolyldiketopiperazine B
CAS:<p>Prolyldiketopiperazine B is a proline-based diketopiperazine.</p>Fórmula:C12H20N2O2Forma y color:SolidPeso molecular:224.3Indoleacetyl phenylalanine
CAS:<p>Indoleacetyl phenylalanine is an indole-acetyl-amino acid involved in regulating auxin activity.</p>Fórmula:C19H18N2O3Pureza:98%Forma y color:SolidPeso molecular:322.36Clogestone acetate
CAS:<p>Clogestone acetate is a a new orally effective progestagen.</p>Fórmula:C25H33ClO5Forma y color:SolidPeso molecular:448.98Foscarbidopa
CAS:<p>Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.</p>Fórmula:C10H15N2O7PPureza:96.17% - 97.27%Forma y color:SolidPeso molecular:306.21A-123189
CAS:<p>A-123189 is a potent, alpha1D-selective antagonist.</p>Fórmula:C26H28N4O3SPureza:98%Forma y color:SolidPeso molecular:476.59Trimazosin hydrochloride
CAS:<p>Trimazosin hydrochloride is used in the treatment of hypertensive patients failing to respond to thiazides.</p>Fórmula:C20H32ClN5O7Forma y color:SolidPeso molecular:489.95Vin-F03
CAS:<p>Vin-F03 protects pancreatic β-cells in type 2 diabetes research with an EC50 of 0.27 μM and prevents STZ-induced apoptosis.</p>Fórmula:C22H29N3Forma y color:SolidPeso molecular:335.49JAK-IN-11
CAS:<p>JAK-IN-11 (R-348) is a potent and selective inhibitor of JAK, has the potential for the skin disorders treatment.</p>Fórmula:C23H22FN5O4SPureza:99.75%Forma y color:SolidPeso molecular:483.52Atorvastatin magnesium trihydrate
CAS:<p>Atorvastatin reduces cholesterol and prevents heart disease by blocking HMG-CoA reductase; also treats dyslipidemia.</p>Fórmula:C66H74F2MgN4O13Forma y color:SolidPeso molecular:1193.61Leptospermone
CAS:<p>Leptospermone is an essential oil from Leptospermum scoparium (manuka oil).</p>Fórmula:C15H22O4Forma y color:SolidPeso molecular:266.33CGP-53437
CAS:<p>CGP-53437 is a novel HIV-1 protease inhibitor, also potently inhibiting major aspartyl peptidase 1 (May1), a secreted Cryptococcus neoformans protease.</p>Fórmula:C42H56N4O7Forma y color:SolidPeso molecular:728.92VL-0395
CAS:VL-0395 is an antagonist of CCK1 receptor.Fórmula:C25H21N3O4Pureza:98%Forma y color:SolidPeso molecular:427.45Sotrastaurin acetate
CAS:<p>Sotrastaurin acetate is a pan-protein kinase C inhibitor. It also has potential immunosuppressive and antineoplastic activities.</p>Fórmula:C27H26N6O4Pureza:98%Forma y color:SolidPeso molecular:498.53Brecanavir
CAS:<p>Brecanavir is a tyrosyl-based arylsulfonamide, high affinity, protease inhibitor (PI) for the treatment of human immunodeficiency virus type 1.</p>Fórmula:C33H41N3O10S2Forma y color:SolidPeso molecular:703.82SAR127303
CAS:<p>SAR127303 is an effective covalent inhibitor of MAGL. SAR127303 behaves as a selective and competitive inhibitor of mouse and human MAGL.</p>Fórmula:C16H17ClF6N2O4SPureza:98%Forma y color:SolidPeso molecular:482.83Deltazinone
CAS:<p>Deltazinone selectively inhibits PDEδ with low cytotoxicity, mimicking PDEδ knockdown in human pancreatic cancer cells.</p>Fórmula:C27H31N5O2Pureza:98%Forma y color:SolidPeso molecular:457.57JTV-519 free base
CAS:JTV-519 free base (K201 free base), recognized for its antiarrhythmic and cardioprotective properties, functions as a Ca2+-dependent blocker of sarcoplasmicFórmula:C25H32N2O2SPureza:98%Forma y color:SolidPeso molecular:424.6
