Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.542 productos)
- Apoptosis(5.816 productos)
- Ciclo celular / Checkpoint(4.466 productos)
- Cromatina / Epigenética(2.252 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.830 productos)
- Endocrinología / Hormonas(3.518 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.362 productos)
- Inmunología e inflamación(3.540 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(405 productos)
- Señalización MAPK(1.201 productos)
- Transportador de membrana / canal de iones(2.809 productos)
- Metabolismo(9.462 productos)
- Microbiología / Virología(7.003 productos)
- Neurociencia(9.942 productos)
- Otros inhibidores(37.827 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.598 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.012 productos)
- Ubiquitinación(1.651 productos)
Mostrar 16 subcategorías más
Se han encontrado 66618 productos de "Inhibidores"
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Decylene glycol
CAS:Decylene glycol, an antimicrobial in cosmetics, alters liposome membrane fluidity.Fórmula:C10H22O2Pureza:98%Forma y color:White Solid Or White Powder And/Or ChunksPeso molecular:174.28Nitroscanate
CAS:<p>Nitroscanate is an anthelmintic found to be effective in certain strains of parasites in canines.</p>Fórmula:C13H8N2O3SForma y color:SolidPeso molecular:272.28QF0301B
CAS:QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.Fórmula:C23H28N2O2Pureza:>99.99%Forma y color:SolidPeso molecular:364.48Litophynin A
CAS:<p>Litophynin A is an insect Growth Inhibitory Diterpenoids from the Soft Coral Litophyton sp.</p>Fórmula:C24H38O3Forma y color:SolidPeso molecular:374.56VUF 8328
CAS:<p>VUF 8328 is an agonist of histamine H(3) receptor.</p>Fórmula:C7H12N4SPureza:98%Forma y color:SolidPeso molecular:184.26SD-36
CAS:SD-36: Potent, selective PROTAC STAT3 degrader, Kd ~50 nM, effective on mutants, IC50=10 nM, strong anti-tumor effects, enables mouse tumor regression.Fórmula:C59H62F2N9O12PPureza:98% - >99.99%Forma y color:SoildPeso molecular:1158.15DMBT
CAS:<p>DMBT is an inhibitor of invasion and metastasis through Akt/GSK-3β/β-catenin pathway in B16BL6 cells.</p>Fórmula:C30H38O17Forma y color:SolidPeso molecular:670.61NPD8716
CAS:<p>NPD8716 is a hepatitis B/D virus entry inhibitor, targeting sodium taurocholate cotransporting polypeptide (NTCP).</p>Fórmula:C23H31NO6SForma y color:SolidPeso molecular:449.56Metitepine
CAS:<p>Metitepine is a serotonin receptor antagonist in the CNS used as an antipsychotic.</p>Fórmula:C20H24N2S2Forma y color:SolidPeso molecular:356.55FKK
CAS:FKK is an indazole derivative and also a novel bronchodilator.Fórmula:C17H17BrN2Pureza:98%Forma y color:SolidPeso molecular:329.23HPK1-IN-26
CAS:<p>HPK1-IN-26, from WO2021254118A1, is a potent dual HPK1/GLK inhibitor for studying animal infections.</p>Fórmula:C19H21N5OSForma y color:SolidPeso molecular:367.47SCH 50911
CAS:<p>SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.</p>Fórmula:C8H15NO3Pureza:98%Forma y color:SolidPeso molecular:173.21Butyrolactone I
CAS:<p>Butyrolactone I (Olomoucin) inhibits CDKs, blocks cdc2 kinases, and shows antitumor activity in lung and prostate cancers.</p>Fórmula:C24H24O7Pureza:98%Forma y color:SolidPeso molecular:424.44(5Z,2E)-CU-3
CAS:<p>(5Z,2E)-CU-3 is a potent and selective inhibitor of DGKα isozyme with an IC50 value of 0.6 μM and inhibition of DGKα by competing ATP with a Km value of 0.48 mM</p>Fórmula:C16H12N2O4S3Pureza:99.02%Forma y color:SolidPeso molecular:392.47DMX-129
CAS:<p>DMX-129 is a chemical compound acting as an inhibitor for both ΙΚΚε and TBK-1, demonstrating efficacy with IC50 values of below 30 nM for each [1].</p>Fórmula:C19H17FN8Forma y color:SolidPeso molecular:376.39Cholera autoinducer 1
CAS:<p>Cholera autoinducer 1 is an autoinducer of Vibrio cholerae. Cholera autoinducer 1 influences chemotaxis in C. elegans [1].</p>Fórmula:C13H26O2Forma y color:SolidPeso molecular:214.34OPC-14523 free base
CAS:OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.Fórmula:C23H28ClN3O2Pureza:98%Forma y color:SolidPeso molecular:413.94Obatoclax
CAS:<p>Obatoclax (GX15-070), a pan-BCL-2 inhibitor (Ki 220 nM) induces autophagy, degrades cyclin D1, and has anti-cancer/antiparasitic properties.</p>Fórmula:C20H19N3OPureza:99.44%Forma y color:SolidPeso molecular:317.38BE-16627B
CAS:<p>BE-16627B, a metalloproteinase inhibitor from Streptomyces sp., curbs human stromelysin & 92 kD gelatinase without obvious toxicity, IC50=25 µM pre-trypsin.</p>Fórmula:C16H29N3O7Forma y color:SolidPeso molecular:375.42HMBPP triammonium
CAS:<p>HMBPP triammonium is a stimulator of gamma delta T cells.</p>Fórmula:C5H15NO8P2Forma y color:SolidPeso molecular:279.122Protriptyline
CAS:<p>Protriptyline: Antidepressant, AChE inhibitor (IC50 0.06 mM), prevents Aβ aggregation; potential for depression and Alzheimer's.</p>Fórmula:C19H21NForma y color:SolidPeso molecular:263.3810-DEBC hydrochloride
CAS:<p>10-DEBC hydrochloride, a selective Akt inhibitor demonstrating an IC50 value of 1.28 μM, is identified as a novel anti-tuberculosis compound [1] [2].</p>Fórmula:C20H26Cl2N2OForma y color:SolidPeso molecular:381.34IDO1/TDO-IN-1
CAS:<p>IDO1/TDO-IN-1 (30) inhibits IDO1 (Ki=0.23μM) & TDO (Ki=0.73μM); induces apoptosis via Bcl-2/Bax.</p>Fórmula:C21H16O6Forma y color:SolidPeso molecular:364.358-Aminoinosine
CAS:<p>8-Aminoinosine is an endogenous 8-aminopurine that induces diuresis, natriuresis, and glucosuria by inhibiting purine nucleoside phosphorylase (PNPase).</p>Fórmula:C10H13N5O5Forma y color:SolidPeso molecular:283.24BRD4-Kinases-IN-3
CAS:<p>BRD4-Kinases-IN-3 is a dual BRD4-Kinases inhibitor that can be used as a value-added multi-targeted chemical probe for cancer therapy.</p>Fórmula:C26H34FN7O2SForma y color:SolidPeso molecular:527.66SHP2 inhibitor LY6
CAS:<p>SHP2 inhibitor LY6 (LY6) is a potent and selective SHP2 inhibitor (IC50: 9.8 μM) that blocks SHP2-mediated cell signaling and proliferation.</p>Fórmula:C30H27Cl2N3O4Forma y color:SolidPeso molecular:564.46Tolboxane
CAS:<p>Tolboxane is an alpha-adrenergic blocking drug.</p>Fórmula:C14H21BO2Pureza:98%Forma y color:SolidPeso molecular:232.13LC28
CAS:<p>LC28 is a novel inhibitor of STAT3 signaling, suppressing survival of cisplatin-resistant ovarian cancer cells.</p>Fórmula:C17H13BrClNO2Forma y color:SolidPeso molecular:378.65LK 157
CAS:<p>LK 157 is a tricyclic carbapenem with potent activity against class A and class C beta-lactamases.</p>Fórmula:C14H17NO4Forma y color:SolidPeso molecular:263.293-Phosphoglyceric acid barium
CAS:<p>3-Phosphoglyceric acid barium is a metabolic intermediate in both glycolysis and the Calvin cycle. It is involved in alveolar macrophage epigenetic regulation.</p>Fórmula:C3H9BaO7PPureza:98%Forma y color:SolidPeso molecular:325.3995-HT3 antagonist 3
CAS:<p>5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 receptors in rat brain cortical membranes (Ki: 0.25 nM).</p>Fórmula:C20H21N3OPureza:99.9%Forma y color:SolidPeso molecular:319.43-Methyl-GABA
CAS:<p>3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.</p>Fórmula:C20H30N2O10S2Pureza:98%Forma y color:SolidPeso molecular:522.59Hsp90-IN-17
CAS:<p>Hsp90-IN-17 (Example 5) is an inhibitor of HSP90, applicable in researching proliferative diseases, including cancer and neurodegenerative conditions.</p>Fórmula:C21H20N4O7Forma y color:SolidPeso molecular:440.4116,17-Dihydroheronamide C
CAS:<p>16,17-Dihydroheronamide C is a probe used for the analysis of the mode of action of heronamide C, which has antifungal properties.</p>Fórmula:C29H41NO3Forma y color:SolidPeso molecular:451.64OHM1
CAS:<p>OHM1, an analog of HIF1α CTAD, effectively inhibits the interaction between HIF1α CTAD and p300/CBP by targeting the CH1 domain with a binding affinity of 0.53</p>Fórmula:C24H42N6O5Forma y color:SolidPeso molecular:494.63Rev 6134
CAS:<p>Rev 6134 is an ACE-inhibitor with non-sulfhydryl containing.</p>Fórmula:C21H32N2O7Pureza:98%Forma y color:SolidPeso molecular:424.49BRD2577
CAS:<p>BRD2577 is an HDAC inhibitor, by suppressing multiple HDAC enzymes and modulating acetylation levels in cells.</p>Fórmula:C15H15N3O3SPureza:98%Forma y color:SolidPeso molecular:317.36Milameline
CAS:<p>Milameline is a muscarinic receptor agonist that improves cognition.</p>Fórmula:C8H14N2OForma y color:SolidPeso molecular:154.21Adaprolol maleate
CAS:<p>Adaprolol maleate: potent beta-blocker with strong antiarrhythmic effects, for glaucoma and eye conditions, impacts heart's electrical activity.</p>Fórmula:C30H43NO8Forma y color:SolidPeso molecular:545.673MK-8133
CAS:<p>MK-8133 is an antagonist of orexin-2 selective receptor with favorable development properties.</p>Fórmula:C23H21N5O2Forma y color:SolidPeso molecular:399.45Azosulfamide
CAS:<p>Azosulfamide is an azo compound with similar antibacterial effect as sulfanilamide.</p>Fórmula:C18H16N4Na2O10S3Forma y color:SolidPeso molecular:590.5Acaprazine
CAS:Acaprazine is an adrenolytic and anxiolytic drug in the class of phenylpiperazine.Fórmula:C15H21Cl2N3OForma y color:SolidPeso molecular:330.25Quinterenol sulfate
CAS:<p>Quinoline sulfate has a bronchiectasis effect on patients with asthma.</p>Fórmula:C14H18N2O2H2O4SForma y color:SolidPeso molecular:295.35Cefcanel daloxate
CAS:<p>Cefcanel daloxate is a pro-drug of KY-087.</p>Fórmula:C27H27N5O9S3Pureza:98%Forma y color:SolidPeso molecular:661.73ST-836
CAS:<p>ST-836 is a dopamine receptor ligand; Antiparkinsonian agent .</p>Fórmula:C23H34N4OSPureza:98%Forma y color:SolidPeso molecular:414.611-Phenylpyrrole
CAS:<p>1-Phenylpyrrole (NSC-16581) is an inhibitor of CYP450 dependant monooxygenase activity in microsomes from rat liver.</p>Fórmula:C10H9NPureza:99.75%Forma y color:Light Beige To Brown Crystalline Powder And LumpsPeso molecular:143.19Antitumor agent-45
CAS:<p>Antitumor agent-45 has an inhibitory effect on c-Met expression and is able to block A549 cells in the G0/G1 and G2/M phases and induce apoptosis.</p>Fórmula:C28H17BrFN5O3Forma y color:SolidPeso molecular:570.37Depramine
CAS:<p>Depramine (GP 31406), a tricyclic antidepressant, exhibits pharmacological activity by inhibiting acetylcholinesterase, Mg^2+-ATPase, and Na^+/K^+ ATPase</p>Fórmula:C19H22N2Forma y color:SolidPeso molecular:278.39iST2-1
CAS:<p>iST2-1 is a first-in-class ST2 inhibitor active in vivo.</p>Fórmula:C22H22N2O4Forma y color:SolidPeso molecular:378.427-Troc-paclitaxel
CAS:<p>7-Troc-paclitaxel is a precursor of paclitaxel which has anti-tumor activity.</p>Fórmula:C50H52Cl3NO16Pureza:99.69%Forma y color:SolidPeso molecular:1029.3
