Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.524 productos)
- Apoptosis(5.793 productos)
- Ciclo celular / Checkpoint(4.452 productos)
- Cromatina / Epigenética(2.242 productos)
- Señalización citoesquelética(1.382 productos)
- Daño al ADN / Reparación del ADN(2.826 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.527 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.203 productos)
- Transportador de membrana / canal de iones(2.792 productos)
- Metabolismo(9.449 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.921 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66639 productos de "Inhibidores"
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Galicaftor
CAS:<p>ABBV-2222 is a CFTR corrector which is studied for the treatment of cystic fibrosis (CF).</p>Fórmula:C28H21F4NO7Pureza:98%Forma y color:SolidPeso molecular:559.46MS0017509
CAS:<p>MS0017509 is a DNA damage repair inhibitor.</p>Fórmula:C11H10N4Pureza:98%Forma y color:SolidPeso molecular:198.22Symetine
CAS:<p>Symetine（L 16726） is a small molecule compound with antiparasitic activity that can be used to study amoebic liver abscesses in guinea pigs.</p>Fórmula:C30H48N2O2Pureza:99.79%Forma y color:SolidPeso molecular:468.71Thiazinamium chloride
CAS:<p>Thiazinamium chloride possesses potent anticholinergic and antiallergic activity and inhibits synthesis of TxB2(IC50 value of 0.2 μM).</p>Fórmula:C18H23ClN2SPureza:98%Forma y color:SolidPeso molecular:334.91HSP90-IN-13
CAS:<p>HSP90-IN-13 (5k): potent HSP90 inhibitor, IC50 25.07 nM, targets EGFR/VEGFR-2/Topo-2, blocks MCF-7 G2/M cycle, induces apoptosis.</p>Fórmula:C26H21N5O3SForma y color:SolidPeso molecular:483.54Cinamolol
CAS:<p>Cinamolol is a beta blocker.</p>Fórmula:C16H23NO4Forma y color:SolidPeso molecular:293.36BIM-46174
CAS:<p>BIM-46174 has anticancer activity, inhibits the growth of a large number of human cancer cell lines, and induces caspase-3-dependent cancer cell apoptosis.</p>Fórmula:C22H30N4OSForma y color:SolidPeso molecular:398.57IDO-IN-3
CAS:<p>IDO-IN-3 is a potent indoleamine 2,3-dioxygenase (IDO) inhibitor (IC50: 290 nM).</p>Fórmula:C11H12BrFN6O2Forma y color:SolidPeso molecular:359.15FCE 28654
CAS:<p>FCE 28654 is a water-soluble acyl-CoA inhibitor.</p>Fórmula:C25H35N2O7PForma y color:SolidPeso molecular:506.53AChE-IN-7
CAS:<p>AChE-IN-7 inhibits eeAChE (IC50: 0.045μM), eeBuChE (19.68μM), crosses the blood-brain barrier, safe, with good pharmacokinetics and 55.5% bioavailability.</p>Fórmula:C26H28N2O2Forma y color:SolidPeso molecular:400.51APY0201
CAS:<p>APY0201: potent, specific ATP-competitive PIKfyve inhibitor; IC50=5.2 nM; blocks PtdIns3P to PtdIns(3,5)P2 conversion.</p>Fórmula:C23H23N7OPureza:98% - 99.74%Forma y color:SolidPeso molecular:413.48NS 3763
CAS:<p>NS 3763 is a kainate receptor antagonist.</p>Fórmula:C22H16N2O6Pureza:98%Forma y color:SolidPeso molecular:404.37RS 23597-190 hydrochloride
CAS:<p>RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.</p>Fórmula:C16H24Cl2N2O3Pureza:98%Forma y color:SolidPeso molecular:363.28FD2056
CAS:<p>FD2056 is a potent, orally active PI3K inhibitor, with IC50 values of 0.30, 0.80, 1.10, and 0.42 nM against PI3Kα, PI3Kβ, PI3Kγ, and PI3Kδ, respectively.</p>Fórmula:C23H17ClN6O2SPureza:98%Forma y color:SolidPeso molecular:476.94hMAO-B-IN-2
CAS:<p>hMAO-B-IN-2: selective oral hMAO-B inhibitor, crosses BBB, IC50=4 nM, potential for Alzheimer's research, neuroprotective, low toxicity.</p>Fórmula:C18H23NO3Forma y color:SolidPeso molecular:301.38PMPMEase-IN L-28
CAS:<p>PMPMEase-IN L-28 is a novel inhibitor of prenylated methylated protein methylesterase.</p>Fórmula:C17H29FO2S2Pureza:98%Forma y color:SolidPeso molecular:348.54Isobucaine hydrochloride
CAS:<p>Isobucaine hydrochloride is a local anesthetic.</p>Fórmula:C15H24ClNO2Forma y color:SolidPeso molecular:285.81LB-205
CAS:<p>LB-205 is a Zn 2+ dependent pan-inhibitor of class I and class II HDACs. It also has a long half-life in vivo.</p>Fórmula:C18H21N3O2SForma y color:SolidPeso molecular:343.44(4-Acetamidocyclohexyl) nitrate
CAS:<p>(4-Acetamidocyclohexyl) nitrate (BM121307) is an activator of guanylate cyclase.</p>Fórmula:C8H14N2O4Pureza:98%Forma y color:SolidPeso molecular:202.21T761-0184
CAS:<p>T761-0184 is a potent antagonist of α7 nicotinic receptor (nAChR) [1].</p>Fórmula:C16H20FN3OForma y color:SolidPeso molecular:289.359-CP-Ade Mesylate
CAS:<p>9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate cyclase.</p>Fórmula:C11H17N5O3SPureza:99.81%Forma y color:SolidPeso molecular:299.35SARS-CoV-2-IN-32
CAS:<p>SARS-CoV-2-IN-32 inhibits COVID-19 (Mpro; PDB: 6LU7) and has anti-cancer effects; useful for related research.</p>Fórmula:C27H23N5O4Forma y color:SolidPeso molecular:481.5HPK1-IN-24
CAS:<p>HPK1-IN-24 (example 51) has potential to be used in the cancer research which is an inhibitor of hematopoietic progenitor kinase 1 (HPK1) (Ki = 100 nM) [1].</p>Fórmula:C19H14FN5Forma y color:SolidPeso molecular:331.35Premazepam
CAS:<p>Premazepam, a partial benzodiazepine agonist with anxiolytic and sedative effects noted in 1984, was never sold.</p>Fórmula:C15H15N3OForma y color:SolidPeso molecular:253.3PXYC1
CAS:<p>PXYC1 binds Mtb RpsA-CTD (Kd 0.81 μM) & RpsA-CTD Δ438A (Kd 0.31 μM), hindering trans-translation.</p>Fórmula:C9H10N4O3SForma y color:SolidPeso molecular:254.27Hepronicate
CAS:<p>Hepronicate（Megrin） is a small molecule compound with hypolipidemic and vasodilatory activity.</p>Fórmula:C28H31N3O6Pureza:98.41%Forma y color:SolidPeso molecular:505.56CFG920
CAS:<p>CFG920 is an oral CYP17 inhibitor that may reduce androgen production and inhibit growth of androgen-dependent tumors.</p>Fórmula:C14H13ClN4OForma y color:SolidPeso molecular:288.732-Hydroxy atorvastatin calcium salt
CAS:<p>2-Hydroxy atorvastatin calcium salt is a hydroxy metabolite of Atorvastatin calcium salt which is a potent HMG-CoA reductase inhibitor (IC50 = 8 nM).</p>Fórmula:C33H34FN2O60·5CaPureza:97.06%Forma y color:SolidPeso molecular:593.68CAY10727
CAS:<p>CAY10727 selectively inhibits PAD3 (15,600 M^-1min^-1) over PAD1, PAD2, and PAD4.</p>Fórmula:C21H22Cl2N4O2Forma y color:SolidPeso molecular:433.33L-AP5
CAS:<p>L-AP5 is a NMDA antagonist.</p>Fórmula:C5H12NO5PPureza:98%Forma y color:SolidPeso molecular:197.13Oe-9000
CAS:<p>Oe-9000 blocks voltage-gated Na(+) currents in neurons at low µM, affecting both TTX-S and TTX-R types.</p>Fórmula:C21H29NO3Pureza:98%Forma y color:SolidPeso molecular:343.46Lobeglitazone Sulfate
CAS:<p>Lobeglitazone Sulfate (CKD-501) is an anti-inflammatory thiazolidinedione that prevents NLRP3 inflammasome activation and is used in T2DM research.</p>Fórmula:C24H26N4O9S2Pureza:98.69%Forma y color:SolidPeso molecular:578.61NSC-636819
CAS:<p>NSC-636819 is a novel inhibitor of KDM4A/KDM4B.</p>Fórmula:C22H12Cl4N2O4Pureza:98%Forma y color:SolidPeso molecular:510.15Abeprazan
CAS:<p>Abeprazan is a potassium-competitive acid blocker targeting acid-related diseases without acid activation.</p>Fórmula:C19H17F3N2O3SPureza:98%Forma y color:SolidPeso molecular:410.41Murayaquinone
CAS:<p>Murayaquinone is a hepatitis C virus proteinase inhibitor and small molecule antagonist of the oncogenic Tcf/β-catenin protein complex.</p>Fórmula:C19H16O5Forma y color:SolidPeso molecular:324.33hA2A/hCA XII modulator 1
CAS:<p>Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.</p>Fórmula:C24H19N7O4SForma y color:SolidPeso molecular:501.52Acetylhydrolase-IN-1
CAS:<p>Acetylhydrolase-IN-1 is an inhibitor of the esterase 1-Alkyl-2-acetylglycerophosphocholine (Alkylacetyl-GPC: acetylhydrolase).</p>Fórmula:C23H48NO7PPureza:98%Forma y color:SolidPeso molecular:481.6Fenclorac
CAS:<p>Fenclorac has anti-inflammatory activity.</p>Fórmula:C14H16Cl2O2Pureza:98%Forma y color:SolidPeso molecular:287.18RIP1 kinase inhibitor 7
CAS:<p>RIP1 Kinase Inhibitor 7 (Compound 41) serves as a potent inhibitory agent for receptor interacting protein 1 kinase (RIP1) with an IC50 of under 100 nM.</p>Fórmula:C20H20FN3OPureza:98%Forma y color:SolidPeso molecular:337.39ZD-0892
CAS:<p>ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).</p>Fórmula:C24H32F3N3O5Pureza:95% - 99.53%Forma y color:SolidPeso molecular:499.52AC710
CAS:<p>AC710 is a potent PDGFR inhibitor (Kds: 0.6, 1, 1.57, 1.3, 1 nM for FLT3, KIT, CSF1R, PDGFRα and PDGFRβ).</p>Fórmula:C31H42N6O4Pureza:99.67%Forma y color:SolidPeso molecular:562.7Febuxostat 67M-4
CAS:<p>Febuxostat 67M-4, a derivative of 67M-1, inhibits xanthine oxidase to lower uric acid and gout/kidney stone risk.</p>Fórmula:C16H14N2O5SForma y color:SolidPeso molecular:346.36Nav1.1-IN-B
CAS:<p>Nav1.1-IN-B is a selective NaV1.1 inhibitor which reduces visceral hypersensitivity.</p>Fórmula:C11H12N4OForma y color:SolidPeso molecular:216.24ACPT-II
CAS:<p>metabotropic receptor antagonist</p>Fórmula:C8H11NO6Pureza:98%Forma y color:SolidPeso molecular:217.18Spirendolol
CAS:<p>Spirendolol is an antagonist of β adrenergic receptor.</p>Fórmula:C21H31NO3Pureza:98%Forma y color:SolidPeso molecular:345.48MPT0L145
CAS:<p>MPT0L145 is a first-in-class PIK3C3/FGFR inhibitor.</p>Fórmula:C25H29Cl3N8O3Forma y color:SolidPeso molecular:595.91L 8412
CAS:<p>L 8412 is an anti-adrenergic agent.</p>Fórmula:C30H42ClNO3Pureza:98%Forma y color:SolidPeso molecular:500.11(R,R)-Glycopyrrolate
CAS:<p>(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.</p>Fórmula:C19H28BrNO3Pureza:98%Forma y color:SolidPeso molecular:398.34(R)-Carvedilol
CAS:<p>(R)-Carvedilol is a non-selective blocker of β/α-1. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).</p>Fórmula:C24H26N2O4Pureza:98%Forma y color:SolidPeso molecular:406.47Nifekalant hydrochloride
CAS:<p>Nifekalant hydrochloride is an IKr potassium channel blocker with an IC50 of 10 µM.</p>Fórmula:C19H28ClN5O5Pureza:99.91%Forma y color:SolidPeso molecular:441.91
