Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.523 productos)
- Apoptosis(5.792 productos)
- Ciclo celular / Checkpoint(4.449 productos)
- Cromatina / Epigenética(2.238 productos)
- Señalización citoesquelética(1.383 productos)
- Daño al ADN / Reparación del ADN(2.825 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.526 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.202 productos)
- Transportador de membrana / canal de iones(2.790 productos)
- Metabolismo(9.448 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.926 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.016 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66641 productos de "Inhibidores"
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HIV-1 inhibitor-15
CAS:<p>HIV-1 inhibitor-15 (compound 9d): Potent, broad-spectrum, EC50=1.7-9 nM for various strains, good solubility/safety, oral use.</p>Fórmula:C24H20N6Forma y color:SolidPeso molecular:392.46GYKI-13380
CAS:<p>GYKI-13380, also known as LS-79445, is a small molecule with potent bioactivity. Detail information has not been published yet.</p>Fórmula:C16H22N2O3Forma y color:SolidPeso molecular:290.36BI-0282
CAS:<p>BI-0282 (Compound 1) is a potent inhibitor of the MDM2-p53 interaction.</p>Fórmula:C30H23Cl2FN4O4Forma y color:SolidPeso molecular:593.43NW-1772
CAS:<p>NW-1772 is a highly potent and orally active inhibitor of monoamine oxidase B.</p>Fórmula:C19H20ClNO6SPureza:98%Forma y color:SolidPeso molecular:425.88Phentyrin
CAS:<p>Phentyrin is a immunodepressant.</p>Fórmula:C19H22Cl2N2O3Forma y color:SolidPeso molecular:397.3CP-122721
CAS:<p>CP-122721: NK1 receptor blocker, has antidepressant, anti-anxiety, antiemetic effects, and selectively inhibits substance P receptors.</p>Fórmula:C20H23F3N2O2Forma y color:SolidPeso molecular:380.4PA Autoinducer
CAS:<p>PA Autoinducer is a Pseudomonas aeruginosa autoinducer.</p>Fórmula:C16H27NO4Forma y color:SolidPeso molecular:297.39SW203668 (trifluoroacetate salt)
CAS:<p>SW203668: Irreversible stearoyl-CoA desaturase blocker; IC50=54 nM; cytotoxic to CYP4F11-positive cancer cells; IC50=22-116 nM.</p>Fórmula:C24H20F3N3O4SForma y color:SolidPeso molecular:503.49Glisoxepide
CAS:<p>Glisoxepide: sulphonamide, oral K(ATP) blocker, antihyperglycemic, affects heart.</p>Fórmula:C20H27N5O5SPureza:98%Forma y color:SolidPeso molecular:449.52ID110460003
CAS:<p>ID110460003 is a novel μ,δ-Opioid Receptor Dual-Biased Agonist, Overcoming the Limitation of Prior Biased Agonist.</p>Fórmula:C20H25N3O2Forma y color:SolidPeso molecular:339.43CypD-IN-29
CAS:<p>CypD-IN-29 is a non-peptidic inhibitor of cyclophilin D as a neuroprotective agent in Aβ-induced mitochondrial dysfunction.</p>Fórmula:C26H20FN5O2SForma y color:SolidPeso molecular:485.53Acodazole
CAS:<p>Acodazole is a synthetic imidazoquinoline. It has antimicrobial and antineoplastic properties. It also has been shown to treat arrhythmias.</p>Fórmula:C20H19N5OPureza:98%Forma y color:SolidPeso molecular:345.4YM022
CAS:<p>YM022 is a highly effective and selective gastrin/cholecystokinin (CCK)-B receptor antagonist.</p>Fórmula:C32H28N4O3Pureza:98%Forma y color:SolidPeso molecular:516.59BI-RJ 70
CAS:<p>BI-RJ 70, a tritiated azide analog of nevirapine, probes HIV-1 transcriptase binding by labeling enzymes and residues.</p>Fórmula:C15H14N6OForma y color:SolidPeso molecular:294.31CL-216303 HCl
CAS:<p>CL-216303 HCl, a dopamine transporter inhibitor and a 5-HT inhibitor, is used potentially for the treatment of depression.</p>Fórmula:C11H12Cl3NPureza:98%Forma y color:SolidPeso molecular:264.58Neltenexine HCl
CAS:<p>Neltenexine HCl is the salt form of Neltenexine free base, an elastase inhibitor that may be useful for preventing pulmonary emphysema.</p>Fórmula:C18H21Br2ClN2O2SForma y color:SolidPeso molecular:524.69ML289
CAS:<p>ML289 is a potent CNS-penetrant mGlu3 modulator with IC50 of 0.66 μM, >15-fold selectivity over mGlu2, and inactive against mGlu5.</p>Fórmula:C22H23NO3Pureza:99.54%Forma y color:SolidPeso molecular:349.42Fluroxypyr
CAS:<p>Fluroxypyr is an herbicide in the class of synthetic auxins that is used to control broadleaf weeds and woody brush.</p>Fórmula:C7H5Cl2FN2O3Pureza:99.89%Forma y color:White Powde With The Smell Of SoapPeso molecular:255.03CC260
CAS:<p>CC260 selectively inhibits PI5P4Kα/β (Ki: 40/30 nM), with minimal effect on Plk1/RSK2, useful for metabolic, diabetes, and cancer studies.</p>Fórmula:C24H29Cl2N5O2Forma y color:SolidPeso molecular:490.43Taquidil
CAS:<p>Tocainide hydrochloride: oral antiarrhythmic, sodium channel blocker, akin to lidocaine.</p>Fórmula:C11H17ClN2OForma y color:SolidPeso molecular:228.718JAK-IN-21
CAS:<p>JAK-IN-21 is a selective and potent JAK inhibitor that inhibits JAK1, JAK2, J2V617F and TYK2 with IC50 values of 1.73, 2.04, 109 and 62.9 nM, respectively.</p>Fórmula:C19H16N8OPureza:99.75%Forma y color:SolidPeso molecular:372.38Rentiapril
CAS:<p>Rentiapril is an orally active inhibitor of angiotensin converting enzyme (ACE), with antihypertensive activity.</p>Fórmula:C13H15NO4S2Pureza:98%Forma y color:SolidPeso molecular:313.39Dexverapamil
CAS:<p>Dexverapamil, the R-enantiomer of verapamil, blocks calcium channels and inhibits P-glycoprotein, enhancing antineoplastic drug potency.</p>Fórmula:C27H38N2O4Forma y color:SolidPeso molecular:454.6Metamizol
CAS:<p>Metamizol: anti-thyroid agent, inhibits hormone synthesis; may cause liver toxicity.</p>Fórmula:C13H17N3O4SForma y color:SolidPeso molecular:311.36S 24795
CAS:<p>S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.</p>Fórmula:C14H13BrINOPureza:99.934%Forma y color:SolidPeso molecular:418.07ASP2535
CAS:<p>ASP2535 is a potent, selective, orally bioavailable, brain permeable and centrally-active glycine transporter-1 (GlyT1) inhibitor.ASP2535 can improve cognitive</p>Fórmula:C22H18N6OPureza:98%Forma y color:SolidPeso molecular:382.42LYPLAL1-IN-1
CAS:<p>LYPLAL1-IN-1 is a selective covalent small-molecule inhibitor of Lysophospholipase-like 1 (IC50: 0.006 μM). LYPLAL1-IN-1 also enhances glucose production.</p>Fórmula:C29H29N7O4Pureza:98%Forma y color:SolidPeso molecular:539.59IPR-803
CAS:<p>IPR-803 is an effective inhibitor of the uPAR·uPA protein-protein interaction (PPI) with anti-tumor activity.</p>Fórmula:C27H23N3O4Pureza:95%Forma y color:SolidPeso molecular:453.49BRD9500
CAS:<p>BRD9500 is an oral PDE3 inhibitor, IC50: 10 nM (PDE3A), 27 nM (PDE3B); effective in SK-MEL-3 cancer model.</p>Fórmula:C15H18FN3O2Forma y color:SolidPeso molecular:291.32CAD031
CAS:<p>CAD031, a more active derivative of the Alzheimer's disease (AD) targeting agent J147, exhibits neuroprotective and memory-enhancing properties.</p>Fórmula:C18H14F6N2O2Forma y color:SolidPeso molecular:404.31Etanidazole
CAS:<p>Etanidazole (SR-2508) is a radiosensitizing 2-nitroimidazole that targets glutathione, aiding in cancer imaging and treatment.</p>Fórmula:C7H10N4O4Forma y color:SolidPeso molecular:214.18Azamitosene
CAS:<p>Azamitosene is a DNA cleaving agent exhibiting G and A base specificity. Azamitosene may exhibit a growth inhibitory effect on human gastric cancer cells.</p>Fórmula:C13H13N3O2Forma y color:SolidPeso molecular:243.26Levoleucovorin disodium
CAS:<p>Levoleucovorin disodium is the sodium salt of the enantiomerically active form of Folinic Acid.</p>Fórmula:C20H21N7Na2O7Pureza:98%Forma y color:SolidPeso molecular:517.41Kobusine derivative-2
<p>Kobusine derivative-2 halts MDA-MB-231 cancer cell growth in sub-G1 phase.</p>Fórmula:C36H35Cl4NO4Forma y color:SolidPeso molecular:687.48tHGA
CAS:<p>tHGA is a potent inhibitor of lipoxygenase.</p>Fórmula:C18H24O4Pureza:98%Forma y color:SolidPeso molecular:304.38GPR40 agonist 5
CAS:<p>Oral GPR40 agonist 5 (EC50: 47 nM) lowers blood glucose and enhances tolerance, manages type 2 diabetes in mice.</p>Fórmula:C27H24N2O4Forma y color:SolidPeso molecular:440.49GS-9256
CAS:<p>GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].</p>Fórmula:C46H56ClF2N6O8PSPureza:98%Forma y color:SolidPeso molecular:957.46Bentysrepinine
CAS:<p>Bentysrepinine, a novel anti-HBV agent, inhibits DNA-HBV and cccDNA activities for the treatment of hepatitis B virus (HBV)-infected hepatitis.</p>Fórmula:C29H35N3O4Pureza:98%Forma y color:SolidPeso molecular:489.61T-705RTP sodium
CAS:<p>T-705RTP sodium inhibits influenza virus RNA polymerase (IC50: 0.14 μM, Ki: 1.52 μM), displaying strong antiviral effects.</p>Fórmula:C10H15FN3NaO15P3Pureza:98%Forma y color:SolidPeso molecular:552.145HBV-IN-32
CAS:<p>HBV-IN-32 is a strong cccDNA inhibitor with an IC50 of 0.14 µM against HBsAg, also halting cell growth.</p>Fórmula:C22H19ClO5SForma y color:SolidPeso molecular:430.9Azthreonam dipotassium salt
CAS:<p>Azthreonam dipotassium salt is a synthetic monobactam which targets gram-negative bacteria.</p>Fórmula:C13H17KN5O8S2Forma y color:SolidPeso molecular:474.52α-Glucosidase-IN-6
CAS:<p>α-Glucosidase-IN-6 is a competitive inhibitor of α-glucosidase (IC50: 5.69 μM) and exhibits potential for anti-diabetic studies.</p>Fórmula:C24H17ClF3NO3SForma y color:SolidPeso molecular:491.91SKLB0565
CAS:<p>SKLB0565 inhibits tubulin and colorectal cancer growth (IC50: 0.012-0.081 μM), causes G2/M arrest, triggers apoptosis, and prevents HUVEC migration.</p>Fórmula:C20H25ClN6OForma y color:SolidPeso molecular:400.91CD2665
CAS:<p>CD2665 is an orally active antagonist of retinoic acid receptor (RAR). For RARγ and RARβ, the Kis are 110 nM and 306 nM.</p>Fórmula:C31H34O5Pureza:99.71%Forma y color:SolidPeso molecular:486.6IRE1α kinase-IN-9
CAS:<p>IRE1α kinase-IN-9 (compound 2) is a potent inhibitor of IRE-1α, demonstrating an average IC50 value of less than 0.1 μM.</p>Fórmula:C24H24N2O6Pureza:98%Forma y color:SolidPeso molecular:436.46Pelanserin Free Base
CAS:<p>Pelanserin Free Base is an antagonist of the 5-HT2 and α1-adrenergic receptors.</p>Fórmula:C21H24N4O2Forma y color:SolidPeso molecular:364.44Cyclapolin 9
CAS:<p>Cyclapolin 9: Selective PLK1 inhibitor, IC50 500 nM, ATP-competitive, inactive against other kinases.</p>Fórmula:C9H4F3N3O4SPureza:99.5%Forma y color:SolidPeso molecular:307.21COX-2-IN-20
CAS:<p>COX-2-IN-20 (Compound 5d) is a selective and orally active inhibitor of COX-2 (IC 50 = 17.9 nM) with anti-inflammatory activity [1].</p>Fórmula:C11H9ClFN3O2Forma y color:SolidPeso molecular:269.66NMO-IgG blocker A-01
CAS:<p>NMO-IgG blocker A-01 is a idiotype-specific blocker of neuromyelitis opticaimmunoglobulin g (nmo-igg) binding to aquaporin-4 (aqp4)</p>Fórmula:C21H21ClN6OForma y color:SolidPeso molecular:408.88Clofop
CAS:<p>Clofop, an obsolete post-emergence herbicide, was used to control annual grasses in a range of crops.</p>Fórmula:C15H13ClO4Pureza:98%Forma y color:SolidPeso molecular:292.71
