Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.523 productos)
- Apoptosis(5.792 productos)
- Ciclo celular / Checkpoint(4.449 productos)
- Cromatina / Epigenética(2.238 productos)
- Señalización citoesquelética(1.383 productos)
- Daño al ADN / Reparación del ADN(2.825 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.526 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.202 productos)
- Transportador de membrana / canal de iones(2.790 productos)
- Metabolismo(9.448 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.926 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.016 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66641 productos de "Inhibidores"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
JNJ-2408068
CAS:<p>JNJ-2408068 inhibits RSV with EC50 of 2.1 nM; blocks fusion (EC50=0.9 nM) by targeting F protein.</p>Fórmula:C22H30N6OPureza:98%Forma y color:SolidPeso molecular:394.51Influenza A virus-IN-5
CAS:<p>Influenza A virus-IN-5 (16e) is a potent, oral anti-IAV with 1.29 μM IC50, inhibiting viral RNA transcription/replication with low cytotoxicity.</p>Fórmula:C24H23N5OForma y color:SolidPeso molecular:397.47UbcH5c-IN-1
CAS:<p>UbcH5c-IN-1 is a selective small-molecule Ubiquitin-conjugating enzyme UbcH5c inhibitor (Kd: 283 nM for E2 UbcH5c-IN-1 by covalent binding with Cys85).</p>Fórmula:C22H21BrO3Pureza:98%Forma y color:SolidPeso molecular:413.3ZINC32540717
CAS:<p>ZINC32540717 is a potent ebolavirus (EBOV) inhibitor.</p>Fórmula:C23H26N4O3Forma y color:SolidPeso molecular:406.48ANA-773
CAS:<p>ANA773, an oral prodrug, activates TLR7 to stimulate immune cells and cytokine release, enhancing innate immunity.</p>Forma y color:SolidTolytoxin
CAS:<p>Tolytoxin: a cytostatic, antifungal macrolide from Scytonema algae, reversibly inhibits mammalian cell cytokinesis.</p>Fórmula:C46H75NO13Forma y color:SolidPeso molecular:850.09Fosravuconazole
CAS:<p>Fosravuconazole is a ravuconazole prodrug. It has antifungal activity.</p>Fórmula:C23H20F2N5O5PSPureza:98%Forma y color:SolidPeso molecular:547.47GBR-13069 dimethanesulfonate
CAS:<p>GBR-13069 dimethanesulfonate is a dopamine reuptake inhibitor.</p>Fórmula:C30H38F2N2O7S2Forma y color:SolidPeso molecular:640.76CAY10487
CAS:<p>CAY10487 reduces aortic fatty streaks in high-cholesterol rabbits by 37.4% and inhibits LDL oxidation by 75% at 2μM, without altering lipids or ACAT activity.</p>Fórmula:C13H15NO5Forma y color:SolidPeso molecular:265.26Azidopine
CAS:<p>Azidopine is a photoactive dihydropyridine channel blocker which may also act as a multidrug resistant (MDR) modulator.</p>Fórmula:C27H26F3N5O5Forma y color:SolidPeso molecular:557.52AMP-PNP tetralithium
CAS:<p>AMP analog that blocks Kir6 channels, inhibits axonal transport, and stabilizes organelle-microtubule interactions.</p>Fórmula:C10H13Li4N6O12P3Forma y color:SolidPeso molecular:529.93D 15413
CAS:<p>D 15413 is an inhibitor of estrogen-dependent mammary tumors.</p>Fórmula:C16H12Cl3NO2Pureza:98%Forma y color:SolidPeso molecular:356.63LY 215891
CAS:<p>LY 215891 is a compound that exhibits potent Gram-negative and Gram-positive antibacterial activity.</p>Fórmula:C12H10ClN5O5S2Pureza:98%Forma y color:SolidPeso molecular:403.82PABA/NO
CAS:<p>PABA/NO, a GST-activated NO donor, hampers hepatocellular carcinoma growth and survival by disrupting PI3K/AKT/mTOR and MEK/ERK.</p>Fórmula:C16H16N6O8Forma y color:SolidPeso molecular:420.33Allyxycarb
CAS:<p>Allyxycarb is an acetylcholinesterase inhibitor.</p>Fórmula:C16H22N2O2Forma y color:SolidPeso molecular:274.36SA57
CAS:<p>SA57 is a potent, selective inhibitor of FAAH(IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH).</p>Fórmula:C17H23ClN2O3Pureza:98%Forma y color:SolidPeso molecular:338.836α-Fluorotestosterone
CAS:<p>6alpha-Fluorotestosterone: synthetic androgen, nonaromatizable, testosterone analog, activates nuclear receptors, equipotent to testosterone.</p>Fórmula:C19H27FO2Forma y color:SolidPeso molecular:306.41Amicarbalide
CAS:<p>Amicarbalide is an agent for the treatment of anaplasmosis.</p>Fórmula:C15H16N6OForma y color:SolidPeso molecular:296.33MMPX
CAS:<p>calmodulin-sensitive cyclic GMP phosphodiesterase inhibitor</p>Fórmula:C12H18N4O3Pureza:98%Forma y color:SolidPeso molecular:266.3Dunnione
CAS:<p>Dunnione is an antifungal agent exerting its action primarily through initiation of redox cycling.</p>Fórmula:C15H14O3Forma y color:SolidPeso molecular:242.27Antifungal agent 67
CAS:<p>Compound 9 (Antifungal agent 67), an imidazole class antifungal, exhibits efficacy against Candida and possesses a CC50 value of 33.6 μM in neonatal rat</p>Fórmula:C23H25ClN2O3Forma y color:SolidPeso molecular:412.91Parconazole Free Base
CAS:<p>Parconazole Free Base is a broad-spectrum oral antifungal for veterinary use, with no antibacterial properties, inhibiting fungal cytochrome P450.</p>Fórmula:C17H16Cl2N2O3Forma y color:SolidPeso molecular:367.23ERRγ Inverse Agonist 1
CAS:<p>ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].</p>Fórmula:C30H38Cl2N2O2Pureza:98%Forma y color:SolidPeso molecular:529.54BMVC4
CAS:<p>BMVC4 stabilizes G-quadruplexes and induces senescence via DNA damage pathways, separate from telomerase inhibition.</p>Fórmula:C26H23IN5Pureza:98%Forma y color:SolidPeso molecular:532.409FKGK 18
CAS:<p>FKGK 18: GVIA iPLA2 inhibitor, 99.9% at 0.091 fraction, selective, IC50 ~50 nM–3 μM, reduces blood glucose and diabetes in NOD mice.</p>Fórmula:C16H15F3OForma y color:SolidPeso molecular:280.28UK51656
CAS:<p>UK51656 is an antagonist of calcium (IC50: 4 nM).</p>Fórmula:C22H28ClN3O6Pureza:98%Forma y color:SolidPeso molecular:465.93XZH-5
CAS:<p>XZH-5 is an inhibitor of STAT3.</p>Fórmula:C22H25F6N5O4Pureza:98%Forma y color:SolidPeso molecular:537.46AK-106
CAS:<p>AK-106, or AK106-001616, selectively inhibits cPLA2 and has NSAID-like analgesic effects.</p>Fórmula:C26H25N3O3Forma y color:SolidPeso molecular:427.49CPD26
CAS:<p>CPD26 is a novel non-RBD binding modulator to inhibit SARS-CoV-2 by prohibiting the conformational change of the spike (S) protein.</p>Fórmula:C21H23NO2Forma y color:SolidPeso molecular:321.41Carburazepam
CAS:<p>Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.</p>Fórmula:C17H16ClN3O2Pureza:98%Forma y color:SolidPeso molecular:329.78ICI-111075
CAS:<p>ICI-111075 is a methane inhibitor.</p>Fórmula:C11H5Cl5O4Forma y color:SolidPeso molecular:378.42Setastine
CAS:<p>Setastine, a highly selective H1 receptor antagonist, acts as a non-sedative antihistamine.</p>Fórmula:C22H28ClNOForma y color:SolidPeso molecular:357.92BMS 961
CAS:<p>BMS961 is a potent and selective retinoic acid receptor gamma (RARγ) agonist (IC50: 30 nM).</p>Fórmula:C23H26FNO4Pureza:98%Forma y color:SolidPeso molecular:399.46Antifungal agent 35
CAS:<p>Antifungal agent 35 is an effective antifungal agent that potentiates the antifungal activity of fluconazole against C. albicans.</p>Fórmula:C26H27BrN4O4Forma y color:SolidPeso molecular:539.42AY 31390
CAS:<p>AY 31390 is a phosphodiesterase (PDE) inhibitor with antithrombotic activity.</p>Fórmula:C11H11Br3N4OForma y color:SolidPeso molecular:454.95PPTN
CAS:<p>PPTN is a high-affinity, competitive and highly selective antagonist of P2Y14 receptor(KB value of 434 pM), with anti-inflammatory and immune activity.</p>Fórmula:C29H24F3NO2Pureza:99.86%Forma y color:SolidPeso molecular:475.5Thiourea, N-(2-phenylethyl)-N'-2-thiazolyl-
CAS:<p>Thiourea, N-(2-phenylethyl)-N'-2-thiazolyl- is a HIV-1 reverse transcriptase inhibitor.</p>Fórmula:C12H13N3S2Forma y color:SolidPeso molecular:263.38MPO-IN-5
CAS:<p>MPO-IN-5: strong, irreversible MPO blocker; IC50s: 0.22 μM for peroxidation, 2.8 μM for hERG.</p>Fórmula:C24H24N6O2Forma y color:SolidPeso molecular:428.496BrCaQ
CAS:<p>6BrCaQ inhibits TRAP1, has antiproliferative effects, and is used in 6BrCaQ-TPP synthesis.</p>Fórmula:C18H15BrN2O3Forma y color:SolidPeso molecular:387.23BMS-688521
CAS:<p>BMS-688521 is an LFA-1/ICAM interaction inhibitor, a small molecule antagonist of LFA-1 with potential anti-inflammatory activity.</p>Fórmula:C26H19Cl2N5O4Pureza:98.87%Forma y color:SolidPeso molecular:536.37FAK-IN-8
CAS:<p>FAK-IN-8 (compound 5h), a FAK inhibitor with an IC50 of 5.32 μM, exhibits potent anti-proliferative activity, making it suitable for use in cancer research [1].</p>Fórmula:C15H9Cl2N3O2SForma y color:SolidPeso molecular:366.22L-858,051 (hydrochloride)
CAS:<p>L-858,051, a forskolin analog, activates adenylate cyclase (EC50 = 3 μM), inhibits glucose transport, and is used in cAMP signaling.</p>Fórmula:C29H50Cl2N2O7Forma y color:SolidPeso molecular:609.63Bismaleimide
CAS:<p>Bismaleimide (XU 292A): heat, oxidation, radiation resistant; for electrical insulation, wear-resistant materials, plastic additives, adhesives.</p>Fórmula:C21H14N2O4Pureza:99.55%Forma y color:Light Yellow Or Light Brown Solid PowderPeso molecular:358.35A-933548
CAS:<p>A-933548: potent calpain inhibitor, selective vs. cathepsins, stable, effective in cell assays.</p>Fórmula:C25H21N5O3Pureza:98%Forma y color:SolidPeso molecular:439.47PLX647(OMe)
CAS:<p>PLX647(OMe) is a slightly less potent inhibitor of FMS than PLX647 but has better aqueous solubility.</p>Fórmula:C22H19F3N4OForma y color:SolidPeso molecular:412.41Revatropate
CAS:<p>Revatropate, a selective muscarinic antagonist, is an antimuscarinic drug.</p>Fórmula:C19H27NO4SForma y color:SolidPeso molecular:365.49HSR-609
CAS:<p>HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.</p>Fórmula:C21H21FN2O3Pureza:98%Forma y color:SolidPeso molecular:368.4MMPSI
CAS:<p>MMPSI (Caspase-3/7 Inhibitor I) is a caspase 3 and caspase 7 inhibitor that inhibits ischemic injury in cardiomyocytes and can be used to study cardioprotection</p>Fórmula:C14H16N2O5SPureza:99.74%Forma y color:SolidPeso molecular:324.35GS 283
CAS:<p>GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.</p>Fórmula:C17H17NO3Forma y color:SolidPeso molecular:283.32WY-135
CAS:<p>WY-135 is a dual inhibitor of ALK and ROS1 (IC50 of 1.4 nM and 1.1 nM, respectively).</p>Fórmula:C28H34ClN9O3SPureza:98%Forma y color:SolidPeso molecular:612.15
