Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.519 productos)
- Apoptosis(5.787 productos)
- Ciclo celular / Checkpoint(4.446 productos)
- Cromatina / Epigenética(2.235 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.824 productos)
- Endocrinología / Hormonas(3.500 productos)
- Enzima(3.639 productos)
- GPCR / proteína G(8.317 productos)
- Inmunología e inflamación(3.516 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.200 productos)
- Transportador de membrana / canal de iones(2.787 productos)
- Metabolismo(9.416 productos)
- Microbiología / Virología(6.968 productos)
- Neurociencia(9.919 productos)
- Otros inhibidores(37.928 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.596 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.649 productos)
Mostrar 16 subcategorías más
Se han encontrado 66626 productos de "Inhibidores"
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Antitumor agent-85
<p>Antitumor agent-85 stabilizes G4-DNA with potent anti-tumor effects.</p>Fórmula:C24H33N7Forma y color:SolidPeso molecular:419.57GSK983
CAS:<p>GSK983 inhibits DHODH to halt cell growth and dengue virus replication, acting as a broad-spectrum antiviral.</p>Fórmula:C18H16ClN3OPureza:98%Forma y color:SolidPeso molecular:325.79YW1159
CAS:<p>YW1159 is an inhibitor of Wnt signaling.</p>Fórmula:C19H14FN5OForma y color:SolidPeso molecular:347.35GGsTop
CAS:<p>GGsTop (Nahlsgen) is a GGT inhibitor with anti-aging activity.</p>Fórmula:C13H18NO7PPureza:98.96%Forma y color:SolidPeso molecular:331.26Ici D8731
CAS:<p>Ici D8731 is a nonpeptide angiotensin II antagonist with potential as a treatment for hypertension and heart failure.</p>Fórmula:C25H21N5OForma y color:SolidPeso molecular:407.47Isosalipurposide
CAS:<p>Isosalipurposide, a chalcone compound, exerts a cytoprotective effect against oxidative injury via Nrf2 activation.</p>Fórmula:C21H22O10Forma y color:SolidPeso molecular:434.39Glucosylceramide synthase-IN-2
CAS:<p>T-690: Potent, BBB-permeable, oral GCS inhibitor; human IC50: 15 nM, mouse IC50: 190 nM; non-competitive with C8 ceramide/UDP glucose.</p>Fórmula:C22H20F3N3O4Forma y color:SolidPeso molecular:447.41Cl-HIBO
CAS:<p>desensitising AMPA receptor agonist</p>Fórmula:C6H7ClN2O4Pureza:98%Forma y color:SolidPeso molecular:206.58S107 hydrochloride
CAS:<p>S107 hydrochloride stabilizes RyR2 by improving calstabin2 binding to mutant/PKA-phosphorylated channels.</p>Fórmula:C11H16ClNOSPureza:98%Forma y color:SolidPeso molecular:245.77CEP-14513
CAS:<p>CEP-14513: potent ALK inhibitor; IC50 = 5 nM in vitro, 30 nM in cell assays.</p>Fórmula:C34H36N6O3Forma y color:SolidPeso molecular:576.69Dimethyl-W84 (dibromide)
CAS:<p>Dimethyl-W84, selective M2 muscarinic receptor modulator; slows N-methylscopolamine release, EC50=3 nM.</p>Fórmula:C34H48Br2N4O4Forma y color:SolidPeso molecular:736.59PDE1-IN-3
CAS:<p>PDE1-IN-3 is a selective inhibitor of human phosphodiesterase 1 (PDE1).</p>Fórmula:C18H24N4OPureza:98%Forma y color:SolidPeso molecular:312.41EGFR-IN-49
CAS:<p>EGFR-IN-49 selectively inhibits EGFR mutations T790M (IC50: 65 nM) & T790M/L858R (IC50: 13.6 nM), triggering apoptosis dose-dependently.</p>Fórmula:C22H15N5O2SForma y color:SolidPeso molecular:413.45Viprostol
CAS:<p>Viprostol is an agent of prostaglandin antihypertensive.</p>Fórmula:C23H36O5Pureza:98%Forma y color:SolidPeso molecular:392.53CLK1/2-IN-3
CAS:<p>CLK1/2-IN-3 (Cpd-3) is a CLK1 and CLK2 inhibitor with antiproliferative activity that inhibits the activity of CLK and SRPK.</p>Fórmula:C21H21N5O2Pureza:99.04%Forma y color:SolidPeso molecular:375.42CGP 36216 hydrochloride
CAS:<p>CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).</p>Fórmula:C5H14NO2PPureza:98%Forma y color:SolidPeso molecular:151.14γ-secretase modulator 1
CAS:<p>gamma-secretase modulator 1 is a modulator of γ secretase and can be used in studies about the treatment of Alzheimer's disease.</p>Fórmula:C24H24N4OSPureza:99.75% - 99.96%Forma y color:SolidPeso molecular:416.54Andolast
CAS:<p>Andolast (CR-2039) is an anti-allergic for asthma and COPD, inhibiting IgE synthesis and improving airflow.</p>Fórmula:C15H11N9OForma y color:SolidPeso molecular:333.31BI 689648
CAS:<p>BI 689648 is a highly selective inhibitor of aldosterone synthase(CYP11B1 and CYP11B2 with IC50s of 310 and 2.1 nM, respectively).</p>Fórmula:C16H18N4O2Forma y color:SolidPeso molecular:298.34Org30958
CAS:<p>Org30958 is a potent inhibitor of aromatase in vivo.</p>Fórmula:C21H30O2S2Pureza:98%Forma y color:SolidPeso molecular:378.59ICI-170809
CAS:<p>ICI-170809 is a 5-HT2 receptor antagonist.</p>Fórmula:C21H24N2SForma y color:SolidPeso molecular:336.49Capzimin
CAS:<p>Capzimin is a selective inhibitor of proteasome isopeptidase Rpn11.</p>Fórmula:C30H24N6O2S4Pureza:98.31% - 99.32%Forma y color:SolidPeso molecular:628.81Antibacterial agent 64
CAS:<p>Potent antibacterial, YycG inhibitor with 6.1 µM IC50. Synergistic with ampicillin against biofilm bacteria.</p>Fórmula:C29H20ClN3O6S2Forma y color:SolidPeso molecular:606.07HCV-IN-37
CAS:<p>HCV-IN-37: potent HCV inhibitor, stable in rat plasma post-oral dose (15 mg/kg), blocks virus entry phase.</p>Fórmula:C31H35F2N5Forma y color:SolidPeso molecular:515.64KRAS G12D inhibitor 14
CAS:<p>KRAS G12D inhibitor 14 is a potent inhibitor of KRAS G12D that binds KRAS G12D protein (Kd: 33 nM).</p>Fórmula:C20H19F3N4OSPureza:>99.99%Forma y color:SolidPeso molecular:420.45APSR-IN-8
CAS:<p>APSR-IN-8: First-in-class APS reductase inhibitor, key for sulfate use and cysteine biosynthesis.</p>Fórmula:C19H19IN2OForma y color:SolidPeso molecular:418.28YM-1
CAS:<p>YM-1, a stable MKT-077 analog, inhibits Hsp70 orally, kills HeLa cells, and boosts p53 and p21 proteins.</p>Fórmula:C20H20ClN3OS2Forma y color:SolidPeso molecular:417.98FR 110302
CAS:<p>FR 110302 is a potent inhibitor of 5-lipoxygenase.</p>Fórmula:C28H35NO2Pureza:98%Forma y color:SolidPeso molecular:417.58Sirt1/2-IN-1
CAS:<p>Sirt1/2-IN-1 inhibits SIRT1 (IC50: 1.81 μg/mL) and SIRT2 (2.10 μg/mL), less on SIRT3 (20.5 μg/mL), with anticancer properties.</p>Fórmula:C22H13ClN2OS2Forma y color:SolidPeso molecular:420.93ML-309 (hydrochloride)
CAS:<p>ML-309 selectively inhibits mutant IDH1R132H over wild-type, reduces 2-HG in glioblastoma cells. IC50: 96 nM; EC50: 55 nM.</p>Fórmula:C29H30ClFN4O2Forma y color:SolidPeso molecular:521.03Wnt/β-catenin agonist 1
CAS:<p>Wnt/β-catenin agonist 1 is an agonist of Wnt/β-catenin signalling pathway(EC50 of 0.27 μM).</p>Fórmula:C22H25N3O2Pureza:98%Forma y color:SolidPeso molecular:363.45Ifoxetine sulfate
CAS:<p>Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.</p>Fórmula:C13H19NO2H2O4SPureza:98%Forma y color:SolidPeso molecular:270.34TRV0109101
CAS:<p>TRV0109101 is a G protein-biased agonist of the µ-opioid receptor.</p>Fórmula:C21H28N2OSForma y color:SolidPeso molecular:356.52Ibrutinib-MPEA
CAS:<p>Ibrutinib-MPEA is ibrutinib derivative. Ibrutinib is a covalent and irreversible BTK inhibitor that has been used to treat hematological malignancies.</p>Fórmula:C32H39N9O2Forma y color:SolidPeso molecular:581.71Kgp-IN-1
CAS:<p>Kgp-IN-1 is an arginine-specific gingipain (Rgp) inhibitor.</p>Fórmula:C19H24F4N4O3Pureza:98%Forma y color:SolidPeso molecular:432.41LY2048978
CAS:<p>LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.</p>Fórmula:C19H24N2O2Pureza:98%Forma y color:SolidPeso molecular:312.41(3S,5R)-Pitavastatin calcium
CAS:<p>(3S,5R)-Pitavastatin calcium is the enantiomer of Pitavastatin which is a potent HMG-CoA reductase inhibitor.</p>Fórmula:C25H26CaFNO4Pureza:98%Forma y color:SolidPeso molecular:463.562Glucocerebrosidase-IN-1
CAS:<p>Glucocerebrosidase-IN-1 inhibits GCase with IC50 of 29.3 μM, Ki 18.5 μM, useful for Gaucher's and Parkinson's research.</p>Fórmula:C13H27NO3Forma y color:SolidPeso molecular:245.36SKOG102
CAS:<p>SKOG102, a potent OLIG2 inhibitor, blocks DNA binding for GBM research.</p>Fórmula:C19H25Cl2N7Forma y color:SolidPeso molecular:422.35TG 100572
CAS:<p>TG 100572 is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src kinases(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2</p>Fórmula:C26H26ClN5O2Pureza:98%Forma y color:SolidPeso molecular:475.97LDN-0028574
CAS:<p>LDN-0028574 is a SIRT1 inhibitor that also acts as an inhibitor of the human MDM2-p53 interaction.</p>Fórmula:C21H14N4O4SForma y color:SolidPeso molecular:418.43BR102375
CAS:<p>BR102375 is a non-TZD PPAR γ full agonist (EC50: 0.28 μM) for the treatment of type 2 diabetes.</p>Fórmula:C31H34N6O4Pureza:98%Forma y color:SolidPeso molecular:554.64GSK 189254 HCl
CAS:<p>GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.</p>Fórmula:C21H26ClN3O2Pureza:98%Forma y color:SolidPeso molecular:387.9Ethyl-3,4-dephostatin
CAS:<p>Ethyl-3,4-dephostatin is a novel inhibitor of the interactions of CFTR-associated ligand and PSD-95/Dlg1/ZO-1 domain.</p>Fórmula:C8H10N2O3Forma y color:SolidPeso molecular:182.18Thromboxane B2
CAS:<p>Thromboxane B2 is a prostaglandin derivative that is released during anaphylaxis. Thromboxane B2 induces platelet aggregation and arterial contraction.</p>Fórmula:C20H34O6Forma y color:SolidPeso molecular:370.48JH-XIV-68-3
CAS:<p>JH-XIV-68-3: Selective DYRK1A/B inhibitor; effective in HNSCC cell lines.</p>Fórmula:C21H17F3N8OForma y color:SolidPeso molecular:454.41NFAT:AP-1 inhibitor-10
CAS:<p>NFAT:AP-1 inhibitor-10 blocks NFAT:AP-1:DNA binding on ARRE-2, curbing transcription of Il2 and other key immune cytokine genes.</p>Fórmula:C22H19N5O2SForma y color:SolidPeso molecular:417.48Isometamidium chloride
CAS:<p>Isometamidium chloride is an antiprotozoal agent. It is also used in veterinary medicine.</p>Fórmula:C28H26ClN7Pureza:98%Forma y color:SolidPeso molecular:496.01Elasnin
CAS:<p>Elasnin is a reversible inhibitor of elastase for human granulocyte and pancreatic enzymes with IC50 values of 1.3 and 30 µg/ml, respectively.</p>Fórmula:C24H40O4Forma y color:SolidPeso molecular:392.57SNX2-1-108
CAS:<p>SNX2-1-108 is a selective CDK8 and CDK19 inhibitor.</p>Fórmula:C21H16N4Pureza:98%Forma y color:SolidPeso molecular:324.38
