
Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.524 productos)
- Apoptosis(5.793 productos)
- Ciclo celular / Checkpoint(4.452 productos)
- Cromatina / Epigenética(2.242 productos)
- Señalización citoesquelética(1.382 productos)
- Daño al ADN / Reparación del ADN(2.826 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.527 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.203 productos)
- Transportador de membrana / canal de iones(2.792 productos)
- Metabolismo(9.449 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.921 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66639 productos de "Inhibidores"
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Lipoxamycin
CAS:<p>Lipoxamycin is an inhibitor of serine palmitoyl-transferase.</p>Fórmula:C19H36N2O5Pureza:98%Forma y color:SolidPeso molecular:372.5BN 52111
CAS:<p>BN 52111 is a platelet activating factor antagonist.</p>Fórmula:C33H58BrNO4Pureza:98%Forma y color:SolidPeso molecular:612.734SU-200
CAS:<p>SU-200 is a TRPV1 agonist.</p>Fórmula:C20H26N2O2SPureza:98%Forma y color:SolidPeso molecular:358.5UMB-32
CAS:<p>UMB-32: Potent, selective BRD4 inhibitor, Kd 550 nM, IC50 637 nM, also targets TAF1.</p>Fórmula:C21H23N5OForma y color:SolidPeso molecular:361.44Andolast
CAS:<p>Andolast (CR-2039) is an anti-allergic for asthma and COPD, inhibiting IgE synthesis and improving airflow.</p>Fórmula:C15H11N9OForma y color:SolidPeso molecular:333.31SKF-80723 HBr
CAS:<p>SKF-80723 HBr is a potent D1 agonist enhancing quinpirole-induced circling in 6-OHDA lesioned rats.</p>Fórmula:C16H16BrNO2Pureza:98%Forma y color:SolidPeso molecular:334.21Chlophedianol Hydrochloride
CAS:<p>Chlophedianol hydrochloride: a cough suppressant for dry cough with antihistamine and local anesthetic traits; possibly anticholinergic at high doses.</p>Fórmula:C17H21Cl2NOPureza:98%Forma y color:SolidPeso molecular:326.26N-Phenylacetylphenylalanine
CAS:<p>N-Phenylacetylphenylalanine is a biaromatic agent with properties that make them suitable candidates for the treatment of sickle cell disease.</p>Fórmula:C17H17NO3Forma y color:SolidPeso molecular:283.322-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide
CAS:<p>2-Decenoylaminoethyl cyclohexylethyl sulfide prevents stress ulcers, stabilizes phospholipase A2 and prostaglandin E2.</p>Fórmula:C20H37NOSPureza:98%Forma y color:SolidPeso molecular:339.58CP-64434 hydrate
CAS:<p>CP-64434 hydrate is an antibiotic; anti-proliferative HDAC inhibitor.</p>Fórmula:C37H70N2O12Forma y color:SolidPeso molecular:734.96YM-1
CAS:<p>YM-1, a stable MKT-077 analog, inhibits Hsp70 orally, kills HeLa cells, and boosts p53 and p21 proteins.</p>Fórmula:C20H20ClN3OS2Forma y color:SolidPeso molecular:417.98MEK inhibitor
CAS:<p>MEK inhibitor is a MEK receptor and cell cycle protein/CDK complex inhibitor with antitumor activity that can be used to study tumor cell proliferation.</p>Fórmula:C26H26N4O2Pureza:97.48%Forma y color:SolidPeso molecular:426.51Cgp 55802A
CAS:<p>CGP 55802A is a novel photoaffinity ligand for in-situ labeling of NMDA receptors.</p>Fórmula:C18H24IN5NaO7PForma y color:SolidPeso molecular:603.286Pinoxepin HCl
CAS:<p>Pinoxepin HCl is an antipsychotic.</p>Fórmula:C23H29Cl3N2O2Pureza:98.05%Forma y color:SolidPeso molecular:471.85ML-309 (hydrochloride)
CAS:<p>ML-309 selectively inhibits mutant IDH1R132H over wild-type, reduces 2-HG in glioblastoma cells. IC50: 96 nM; EC50: 55 nM.</p>Fórmula:C29H30ClFN4O2Forma y color:SolidPeso molecular:521.03Aha1/Hsp90-IN-1
CAS:<p>Aha1/Hsp90-IN-1 (Compound 17) inhibits Aha1/Hsp90, preventing tau aggregation; IC50 = 3.32 μM.</p>Fórmula:C22H17F3N4O2Forma y color:SolidPeso molecular:426.39Trequinsin hydrochloride
CAS:<p>Azetirelin (YM 14673) is a new thyrotropin-releasing hormone (TRH) analog.</p>Fórmula:C24H28ClN3O3Pureza:99.95%Forma y color:SolidPeso molecular:441.95(S)-MCPG
CAS:<p>(S)-MCPG is the active isomer of (RS)-MCPG, non-selective group I/group II metabotropic glutamate receptor antagonist.</p>Fórmula:C10H11NO4Pureza:98.72%Forma y color:SolidPeso molecular:209.20RL71
CAS:<p>RL71 selectively inhibits SERCA2, binds at a new site, suppresses Ca2+-ATPase, induces apoptosis, and reduces Akt activity.</p>Fórmula:C26H31NO7Forma y color:SolidPeso molecular:469.53AGN 205728
CAS:<p>AGN 205728 is a potent and selective RARγ antagonist (Ki: 3 nM; IC95: 0.6 nM) and has no inhibition on RARα and RARβ.</p>Fórmula:C29H27NO3Pureza:98%Forma y color:SolidPeso molecular:437.53S107 hydrochloride
CAS:<p>S107 hydrochloride stabilizes RyR2 by improving calstabin2 binding to mutant/PKA-phosphorylated channels.</p>Fórmula:C11H16ClNOSPureza:98%Forma y color:SolidPeso molecular:245.77L-733060 hydrochloride
CAS:<p>Potent NK1 antagonist</p>Fórmula:C20H20ClF6NOPureza:98%Forma y color:SolidPeso molecular:439.82DPPY
CAS:<p>DPPY inhibits EGFR, BTK, JAK3 (IC50<10 nM), curbs B-cell lymphoma growth, and may be studied for IPF treatment.</p>Fórmula:C25H26ClN7O3Forma y color:SolidPeso molecular:507.97Thiosildenafil
CAS:<p>Thiosildenafil is a derivative of the phosphodiesterase 5 (PDE5) inhibitor sildenafil.</p>Fórmula:C22H30N6O3S2Forma y color:SolidPeso molecular:490.64Bcl-2/Mcl-1-IN-1
CAS:<p>Bcl-2/Mcl-1-IN-1 is an inhibitor of Bcl-2 (Ki: 4.53 μM) and Mcl-1 (Ki: 1.19 μM).Bcl-2/Mcl-1-IN-1 can be used in cancer research.</p>Fórmula:C28H23NO3Forma y color:SolidPeso molecular:421.49Ceforanide lysine
CAS:<p>Ceforanide lysine is an Anti-Infective.</p>Fórmula:C26H35N9O8S2Pureza:98%Forma y color:SolidPeso molecular:665.74Piperonyl acetone
CAS:<p>Piperonyl acetone (NSC-405365) is a food additive used in edible seasonings.</p>Fórmula:C11H12O3Pureza:99.875%Forma y color:Crystalline PowderPeso molecular:192.21Darenzepine
CAS:<p>Darenzepine is a muscarinic receptor inhibitor.</p>Fórmula:C21H21N3O2Pureza:99.87%Forma y color:SolidPeso molecular:347.41Orf 17910
CAS:<p>Orf 17910 is a histamine H2-receptor antagonist.</p>Fórmula:C18H27N5O2SForma y color:SolidPeso molecular:377.5CLK1/2-IN-3
CAS:<p>CLK1/2-IN-3 (Cpd-3) is a CLK1 and CLK2 inhibitor with antiproliferative activity that inhibits the activity of CLK and SRPK.</p>Fórmula:C21H21N5O2Pureza:99.04%Forma y color:SolidPeso molecular:375.42MDL-72527 free base
CAS:<p>MDL-72527 free base is a polyamine oxidase inactivator.</p>Fórmula:C12H20N2Forma y color:SolidPeso molecular:192.3CGP 36216 hydrochloride
CAS:<p>CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).</p>Fórmula:C5H14NO2PPureza:98%Forma y color:SolidPeso molecular:151.14Phen-DC3
CAS:<p>Phen-DC3 is a G-quadruplex (G4) specific ligand which can inhibit FANCJ and DinG helicases (IC50s of 65±6 and 50±10 nM, respectively).</p>Fórmula:C34H26N6O2Pureza:98%Forma y color:SolidPeso molecular:550.61Hadacidin sodium
CAS:<p>Hadacidin sodium is an inhibitor of AMP synthesis. Hadacidin and hadacidin analogues have anticancer activity and activity against adenylosuccinate synthetase.</p>Fórmula:C3H4NNaO4Forma y color:SolidPeso molecular:141.06MmpL3-IN-2
CAS:<p>MmpL3-IN-2, an inhibitor targeting MmpL3, exhibits low cytotoxicity and moderate metabolic stability, making it suitable for tuberculosis research [1].</p>Fórmula:C27H30N2Forma y color:SolidPeso molecular:382.54SU-13197
CAS:<p>SU-13197 is an antiarrhythmic drug with oral activity.</p>Fórmula:C20H23Cl2N3Pureza:98%Forma y color:SolidPeso molecular:376.33KRAS G12D inhibitor 14
CAS:<p>KRAS G12D inhibitor 14 is a potent inhibitor of KRAS G12D that binds KRAS G12D protein (Kd: 33 nM).</p>Fórmula:C20H19F3N4OSPureza:>99.99%Forma y color:SolidPeso molecular:420.45Alimadol
CAS:<p>Alimadol is an opioid analgesic.</p>Fórmula:C19H23NOForma y color:SolidPeso molecular:281.39EVT-101 HCl
CAS:<p>EVT-101, a unique GluN2B antagonist, binds differently at GluN1/GluN2B interface with its own subcavity.</p>Fórmula:C16H15Cl2F3N4Forma y color:SolidPeso molecular:391.22AHR-13268D
CAS:<p>AHR-13268D is a new agent of antiallergic/antihistaminic.</p>Fórmula:C28H29F2NNaO4Pureza:98%Forma y color:SolidPeso molecular:504.53MurA-IN-3
CAS:<p>MurA-IN-3, a reversible pyrrolidinedione-based MurA inhibitor, exhibits an IC50 of 4.5 μM against MurA and demonstrates antibacterial activity [1].</p>Fórmula:C27H23ClN2O5SForma y color:SolidPeso molecular:523HSK0935
CAS:<p>HSK0935 is a highly selective and orally available SGLT2 inhibitor (IC50: 1.3 nM). It has antihyperglycemic activities.</p>Fórmula:C22H25ClO7Pureza:98%Forma y color:SolidPeso molecular:436.88P-gp inhibitor 3
<p>P-gp inhibitor 3 boosts Paclitaxel's effect by strongly reversing MDR via P-gp efflux blockade.</p>Fórmula:C48H67N3O6Forma y color:SolidPeso molecular:782.06Antitumor agent-85
<p>Antitumor agent-85 stabilizes G4-DNA with potent anti-tumor effects.</p>Fórmula:C24H33N7Forma y color:SolidPeso molecular:419.57Isosalipurposide
CAS:<p>Isosalipurposide, a chalcone compound, exerts a cytoprotective effect against oxidative injury via Nrf2 activation.</p>Fórmula:C21H22O10Forma y color:SolidPeso molecular:434.39TK05
CAS:<p>TK05 is a potent and selective leukotriene C4 synthase (LTC4S) inhibitor (IC50: 95 nM).</p>Fórmula:C31H25ClN2O5Pureza:98%Forma y color:SolidPeso molecular:540.99AV-1101
CAS:<p>AV-1101, a cytokine production inhibitor, is used potentially for the treatment of HIV infection.</p>Fórmula:C19H20N2O4Pureza:98%Forma y color:SolidPeso molecular:340.37M8891
CAS:<p>M8891: Oral, reversible MetAP-2 inhibitor, brain-penetrant (IC50: 54nM; Ki: 4.33nM), hinders endothelial & tumor cell growth, antiangiogenic & antitumor.</p>Fórmula:C20H17F2N3O3Forma y color:SolidPeso molecular:385.36GPR40 Activator 2
CAS:<p>GPR40 Activator 2 is a highly effective activator of the GPR40 receptor.</p>Fórmula:C28H29NO6S2Pureza:98%Forma y color:SolidPeso molecular:539.66HexylHIBO
CAS:<p>HexylHIBO is a type I mGluR antagonist that inhibits mGlu1a and mGlu5a, with Kb values of 140 and 110 μM, respectively.HexylHIBO decreases sEPSC in rats.</p>Fórmula:C12H20N2O4Pureza:99.55%Forma y color:SolidPeso molecular:256.3
