
Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.542 productos)
- Apoptosis(5.816 productos)
- Ciclo celular / Checkpoint(4.466 productos)
- Cromatina / Epigenética(2.252 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.830 productos)
- Endocrinología / Hormonas(3.518 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.362 productos)
- Inmunología e inflamación(3.540 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(405 productos)
- Señalización MAPK(1.201 productos)
- Transportador de membrana / canal de iones(2.809 productos)
- Metabolismo(9.462 productos)
- Microbiología / Virología(7.003 productos)
- Neurociencia(9.942 productos)
- Otros inhibidores(37.827 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.598 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.012 productos)
- Ubiquitinación(1.651 productos)
Mostrar 16 subcategorías más
Se han encontrado 66618 productos de "Inhibidores"
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(Rac)-Etavopivat
CAS:<p>(Rac)-Etavopivat, an oral PKR activator, targets sickle cell disease and haemoglobinopathies.</p>Fórmula:C22H23N3O6SForma y color:SolidPeso molecular:457.5Meturedepa
CAS:<p>Meturedepa is an antineoplastic agent.</p>Fórmula:C11H22N3O3PPureza:98%Forma y color:SolidPeso molecular:275.28Benzcyclane
CAS:<p>Benzcyclane (Benzcyclan) is an inhibitor of platelet aggregation and also a vasodilator that can be used in a variety of peripheral circulation disorders.</p>Fórmula:C19H31NOPureza:99.75%Forma y color:SolidPeso molecular:289.46SRT3190
CAS:SRT3190 is an antagonist of CXCR2.Fórmula:C18H23F2N5O4S2Pureza:98%Forma y color:SolidPeso molecular:475.53Beloxamide
CAS:<p>Beloxamide is a biochemical.</p>Fórmula:C18H21NO2Forma y color:SolidPeso molecular:283.36DA 1686
CAS:<p>DA 1686, antiarrhythmic drug, outperforms quinidine and procainamide, mitigates aconitine-induced tachycardia.</p>Fórmula:C23H32N2O2Pureza:98%Forma y color:SolidPeso molecular:368.51Gln-AMS TFA (209543-57-7 free base)
<p>Gln-AMS(TFA) inhibits glutaminyl-tRNA synthetase (GlnRS) with a Ki of 1.32 μM. Gln-AMS (TFA) is a type Ia aminoacyl-tRNA synthetase (AARS) inhibitor.</p>Fórmula:C17H23F3N8O10SPureza:98%Forma y color:SolidPeso molecular:588.47AF-013
CAS:<p>AF-013 is a rifamycin derivative -- specifically an O-n-octyloxime of 3-formylrifamycin SV -- which acts as an inhibitor of nucleic acid polymerases.</p>Fórmula:C46H64N2O13Forma y color:SolidPeso molecular:853.01PHCCC(4Me)
CAS:<p>THCCC, a PHCCC analog, is a dual metabotropic glutamate receptor 2/3 negative/positive allosteric modulator.</p>Fórmula:C18H16N2O3Forma y color:SolidPeso molecular:308.33DMI-9523
CAS:<p>DMI-9523 reduces NF-κB activation, lowering interferon-gamma and TNF-alpha in human T cells, thus modulating immune response.</p>Fórmula:C7H10N2O4Pureza:98%Forma y color:SolidPeso molecular:186.17MIF degrader MD13
CAS:<p>MD13, a MIF-degrading PROTAC, disrupts vital protein interactions in cancer and inflammation, showing promise as a therapeutic research tool.</p>Fórmula:C35H35N5O8Forma y color:SolidPeso molecular:653.68CGP52411
CAS:<p>CGP52411 is an orally active, and ATP-competitive inhibitor of EGFR (IC50: 0.3 μM).</p>Fórmula:C20H15N3O2Pureza:99.78%Forma y color:SolidPeso molecular:329.35MitoPBN
CAS:<p>MitoPBN: mitochondria-targeted antioxidant, inhibits UCP1-3 at 250 nM, traps hydroxyl & carbon radicals, prevents lipid peroxidation.</p>Fórmula:C33H37BrNO2PForma y color:SolidPeso molecular:590.542Mutated EGFR-IN-3
CAS:<p>Mutated EGFR-IN-3: ATP-competitive, selective dibenzodiazepinone inhibitor for EGFR mutations, IC50 12-13 nM.</p>Fórmula:C31H29FN4O2Pureza:98%Forma y color:SolidPeso molecular:508.59SKF 77434 hydrobromide
CAS:<p>SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.</p>Fórmula:C19H22BrNO2Pureza:98%Forma y color:SolidPeso molecular:376.29Cyclindole
CAS:<p>Cyclindole: unmarketed antipsychotic, tricyclic, D₂ antagonist, displaces spiperone, boosts striatal dopamine.</p>Fórmula:C14H18N2Forma y color:SolidPeso molecular:214.31Nexopamil racemate
CAS:<p>Nexopamil racemate((Rac)-Nexopamil) is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.</p>Fórmula:C24H40N2O3Pureza:98.61%Forma y color:SolidPeso molecular:404.59CAP-53194
CAS:CAP-53194 is a selective Plk1 inhibitor.Fórmula:C21H14N6O5Pureza:98%Forma y color:SolidPeso molecular:430.37K145
CAS:<p>K145: Selective, oral SphK2 inhibitor, IC50 4.3 μM, Ki 6.4 μM, promotes cell apoptosis, strong antitumor effect, inactive against SphK1/other kinases.</p>Fórmula:C18H24N2O3SPureza:98%Forma y color:SolidPeso molecular:348.46NLRP3-IN-20
CAS:<p>NLRP3-IN-20 (compound 11) is an orally administered inhibitor targeting the NLRP3 inflammasome, exhibiting potent inhibition with an IC50 of 25 nM against IL-1β</p>Fórmula:C22H27N3O3SPureza:98%Forma y color:SolidPeso molecular:413.53INSCoV-614(1B)
CAS:<p>INSCoV-614(1B), a potent Mpro inhibitor, may help fight SARS-CoV-2, per patent WO2021219089A1.</p>Fórmula:C23H21ClF3N5O3Forma y color:SolidPeso molecular:507.89N-Arachidonylglycine
CAS:<p>N-Arachidonylglycine, a lipid derived from arachidonic acid, exhibits anti-inflammatory, anti-cancer, anti-diabetic, and antioxidant properties.</p>Fórmula:C22H35NO3Pureza:97.17% - 97.763%Forma y color:SolidPeso molecular:361.52Caprolactam
CAS:<p>Caprolactam is a natural product used in the manufacture of synthetic fibers of the polyamide type.</p>Fórmula:C6H11NOPureza:99.93%Forma y color:White Solid Crystalline Or FlakesPeso molecular:113.16CCD-3693
CAS:<p>CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.</p>Fórmula:C21H31F3O2Pureza:98%Forma y color:SolidPeso molecular:372.46CGP 46381
CAS:<p>CGP 46381 is a GABAB receptor antagonist.</p>Fórmula:C10H22NO2PPureza:98%Forma y color:White SolidPeso molecular:219.26β-L-D4A
CAS:<p>beta-L-D4A inhibits HIV-1 reverse transcriptase, stopping DNA synthesis.</p>Fórmula:C10H11N5O2Pureza:99.45%Forma y color:SolidPeso molecular:233.23PI3Kα/mTOR-IN-1
CAS:<p>PI3Kα/mTOR-IN-1 is a potent dual inhibitor of PI3Kα/mTOR.</p>Fórmula:C16H18N6OPureza:99.89%Forma y color:SolidPeso molecular:310.35NF-κB-IN-2
CAS:<p>NF-κB-IN-2 inhibits canonical NF-κB signaling induced by TNF-α in PC-3 cells.</p>Fórmula:C15H18O3Forma y color:SolidPeso molecular:246.3UR-PI376
CAS:<p>UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.</p>Fórmula:C17H22N6SForma y color:SolidPeso molecular:342.46NPD9948
CAS:<p>NPD9948 is a competitive inhibitor of MTH1.</p>Fórmula:C13H14N6Forma y color:SolidPeso molecular:254.29Ribocitrin
CAS:<p>Ribocitrin is a dextransucrase inhibitor.</p>Fórmula:C22H34O19Forma y color:SolidPeso molecular:602.49FOBISIN101
CAS:<p>FOBISIN101 is a novel inhibitor of all 14-3-3 isoforms in 14-3-3 PPIs.</p>Fórmula:C15H11N3Na3O8PForma y color:SolidPeso molecular:461.2091Genz-669178
CAS:<p>Genz-669178 is a wild-type inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH).</p>Fórmula:C17H14N4OSPureza:98%Forma y color:SolidPeso molecular:322.38SOS1 activator 1
CAS:<p>SOS1 activator 1 enhances SOS1's GDP-GTP exchange on Ras (Kd: 44 nM).</p>Fórmula:C26H32ClFN6Forma y color:SolidPeso molecular:483.02WAY 163909
CAS:WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).Fórmula:C14H18N2Pureza:98%Forma y color:SolidPeso molecular:214.31UCD38B HCl
CAS:<p>UCD38B HCl, a cell-permeable uPA inhibitor, induces programmed necrosis in high-grade glioma cells.</p>Fórmula:C15H17Cl2N7O3Pureza:98%Forma y color:SolidPeso molecular:414.25MMP-9-IN-4
CAS:<p>MMP-9-IN-4 inhibits MMP-9 (IC50=7.46nM) and AKT (IC50=8.82nM), induces apoptosis and is used in cancer research.</p>Fórmula:C28H19F3N4O6Forma y color:SolidPeso molecular:564.47MAO-IN-M30 dihydrochloride
CAS:<p>MAO-IN-M30 dihydrochloride: potent, brain-specific MAO-A/B inhibitor, iron chelator with antioxidant effects, counters Parkinson's in mice.</p>Fórmula:C14H16Cl2N2OPureza:99.83%Forma y color:SolidPeso molecular:299.2Fe-Cap folic
CAS:<p>Fe-Cap folic is an encapsulated dosage for use as an iron supplement in pregnancy.</p>Fórmula:C21H22FeN8O12SForma y color:SolidPeso molecular:666.36Ilorasertib hydrochloride
CAS:<p>Ilorasertib hydrochloride (ABT-348 hydrochloride) is an ATP-competitive multitargeted kinase inhibitor, which inhibits Aurora C, Aurora B, and Aurora A (IC50s:</p>Fórmula:C25H22ClFN6O2SPureza:98.45%Forma y color:SolidPeso molecular:525Acodazole hydrochloride
CAS:Acodazole hydrochloride: synthetic imidazoquinoline with antineoplastic activity; disrupts DNA replication by intercalation.Fórmula:C20H20ClN5OPureza:98%Forma y color:SolidPeso molecular:381.86DW-1350
CAS:DW-1350 is an antagonist of LTB4 receptor.Fórmula:C25H31N3O3SPureza:98%Forma y color:SolidPeso molecular:453.6Decamethonium
CAS:<p>Decamethonium (Syncurine) is a depolarizing muscle relaxant or neuromuscular blocking agent, and is used in anesthesia to induce paralysis.</p>Fórmula:C16H38N2Forma y color:SolidPeso molecular:258.49Zofenoprilat arginine
CAS:<p>Zofenoprilat arginine is an antihypertensive.</p>Fórmula:C21H33N5O5S2Pureza:98%Forma y color:SolidPeso molecular:499.65Simmiparib
CAS:<p>Simmiparib (SMOCL-9112) is a PARP1 and PARP2 inhibitor that promotes apoptosis.Simmiparib is used to study Parkinson's disease and melanoma.</p>Fórmula:C23H18F4N6O2Pureza:99.05% - 99.51%Forma y color:SolidPeso molecular:486.42ML263
CAS:<p>ML263 inhibits NF-kB activation induced by B-cell specific antigen receptor.</p>Fórmula:C15H18N2O3Forma y color:SolidPeso molecular:274.32A2AR-antagonist-1
CAS:<p>Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.</p>Fórmula:C27H25N5O2Pureza:98%Forma y color:SolidPeso molecular:451.52G202-0362
CAS:<p>G202-0362 is an antiviral agent against Rift Valley fever virus. It acts by blocking virus budding from the trans Golgi.</p>Fórmula:C29H29N3O5SPureza:98%Forma y color:SolidPeso molecular:531.62Sch 38548
CAS:<p>Sch 38548 is a ligand of D1-dopamine receptor.</p>Fórmula:C17H19ClN2OPureza:98%Forma y color:SolidPeso molecular:302.8KSK213
CAS:<p>KSK213: Strongly inhibits C. trachomatis (EC50=60 nM); non-toxic to commensals/host cells at 25 μM.</p>Fórmula:C28H25N3O2SForma y color:SolidPeso molecular:467.58
