
Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.542 productos)
- Apoptosis(5.816 productos)
- Ciclo celular / Checkpoint(4.466 productos)
- Cromatina / Epigenética(2.252 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.830 productos)
- Endocrinología / Hormonas(3.518 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.362 productos)
- Inmunología e inflamación(3.540 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(405 productos)
- Señalización MAPK(1.201 productos)
- Transportador de membrana / canal de iones(2.809 productos)
- Metabolismo(9.462 productos)
- Microbiología / Virología(7.003 productos)
- Neurociencia(9.942 productos)
- Otros inhibidores(37.827 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.598 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.012 productos)
- Ubiquitinación(1.651 productos)
Mostrar 16 subcategorías más
Se han encontrado 66618 productos de "Inhibidores"
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Guineesine
CAS:<p>Guineesine is an Acyl-CoA. It acts by inhibiting cholesterol acyltransferase.</p>Fórmula:C24H33NO3Pureza:98%Forma y color:SolidPeso molecular:383.52Indisetron Dihydrochloride
CAS:<p>Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.</p>Fórmula:C17H24ClN5OForma y color:SolidPeso molecular:349.86PM226
CAS:<p>CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.</p>Fórmula:C22H31NO3Forma y color:SolidPeso molecular:357.493'-Chloromethotrexate
CAS:<p>'3'-Chloromethotrexate: cancer/autoimmune treatment, pregnancy termination, chemo, immunosuppressant.</p>Fórmula:C20H21ClN8O5Forma y color:SolidPeso molecular:488.88CAY10773
CAS:<p>CAY10773, a sorafenib derivative, inhibits cancer cells over non-cancerous ones and induces apoptosis or ferroptosis in T24 cells.</p>Fórmula:C22H17Cl2N5OForma y color:SolidPeso molecular:438.31ALR2-IN-3
<p>ALR2-IN-2 inhibits ALR2 strongly (IC50: 22 nM) and ALR1 less (IC50: 116 nM), used in diabetes complication studies.</p>Fórmula:C17H12N2O3S2Forma y color:SolidPeso molecular:356.42Estrone O-sulfamate
CAS:<p>Estrone 3-O-sulfamate, a strong STS inhibitor with IC50 of 18 nM in placenta and 0.83 nM in MCF-7 cells, is used in cancer research.</p>Fórmula:C18H23NO4SPureza:99.86%Forma y color:SolidPeso molecular:349.44S(-)-Bisoprolol
CAS:<p>S(-)-Bisoprolol, a β1-blocker, may aid in researching hypertension and heart diseases.</p>Fórmula:C18H31NO4Forma y color:SolidPeso molecular:325.44CAY10762
CAS:<p>CAY10762, a MAGL inhibitor (IC50=34.1 nM), curbs H2O2-induced LDH in Neuro2a cells and boosts 2-AG in mouse brains at 10 mg/kg.</p>Fórmula:C15H13NOSForma y color:SolidPeso molecular:255.33Helenalin Acetate
CAS:<p>Helenalin Acetate: anti-inflammatory, anti-cancer, hinders C/EBPß and p300 cooperation.</p>Fórmula:C17H20O5Pureza:98%Forma y color:SolidPeso molecular:304.34ZK-90055 hydrochloride
CAS:ZK-90055 hydrochloride is a β2 adrenergic receptor agonist used to study asthma.Fórmula:C16H23ClN2O4Pureza:99.26%Forma y color:SolidPeso molecular:342.82EP1-antagonist-1
CAS:<p>EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).</p>Fórmula:C19H15BrCl2N2O3Pureza:97.06%Forma y color:SolidPeso molecular:470.14Homidium Cl
CAS:<p>Homidium Chloride, a trypanosomicide and DNA intercalator, is toxic and blocks nicotinic acetylcholine receptors.</p>Fórmula:C21H20ClN3Forma y color:SolidPeso molecular:349.8626'-Iodoresiniferatoxin
CAS:<p>TRPV1 (VR1) vanilloid receptor partial agonist</p>Fórmula:C37H39IO9Pureza:98%Forma y color:SolidPeso molecular:754.6INO5042
CAS:INO5042 is an anti-inflammatory agent.Fórmula:C15H7NO3SForma y color:SolidPeso molecular:281.29MPCI
CAS:<p>MPCI is a selective melanocortin-4 receptor antagonist.</p>Fórmula:C25H32BrFN4O2Pureza:98%Forma y color:SolidPeso molecular:519.45R-82913
CAS:<p>R-82913 blocks RNA-polymerase, lowers mouse DOI-head-shakes, halts 13 HIV-1 strains with 0.15µM IC50, beats AZT-TP by 20x; ineffective on HIV-2.</p>Fórmula:C16H20ClN3SForma y color:SolidPeso molecular:321.87EP2 receptor antagonist-1
CAS:<p>EP2 receptor antagonist-1: reversible, potent, depends on agonist; anti-inflammatory.</p>Fórmula:C24H22N4O5Forma y color:SolidPeso molecular:446.46L-5-BromoTryptophan
CAS:<p>L-5-BromoTryptophan (5-BrW) is an analog of the tryptophan (Trp) effector and inhibits the gelation of hemoglobin S.</p>Fórmula:C11H11BrN2O2Pureza:99.86%Forma y color:SolidPeso molecular:283.12MS437
CAS:<p>MS437 is a potent TSH receptor agonist.</p>Fórmula:C22H24N2OPureza:98%Forma y color:SolidPeso molecular:332.44Laidlomycin butyrate
CAS:<p>Laidlomycin butyrate is a ionophore with enhanced intraruminal activity.</p>Fórmula:C41H68O13Forma y color:SolidPeso molecular:768.97SMM-189
CAS:<p>SMM-189 is a potent and selective CB2 inverse agonist.</p>Fórmula:C19H12Cl2O3Forma y color:SolidPeso molecular:359.2simufilamum
CAS:<p>Simufilam (PTI-125): Low-toxicity, oral drug activating FLNA, correcting its structure, aiding Alzheimer's research.</p>Fórmula:C15H21N3OForma y color:SolidPeso molecular:259.35Sermetacin
CAS:<p>Sermetacin is an anti-inflammatory agent.</p>Fórmula:C22H21ClN2O6Pureza:98%Forma y color:SolidPeso molecular:444.86AMPK activator 11
CAS:<p>AMPK Activator 11 is a nanomolar potent inhibitor of cell proliferation in various colorectal carcinomas (CRCs), acting through the selective activation of AMP-</p>Fórmula:C25H20N4O2Pureza:98%Forma y color:SolidPeso molecular:408.45L-703,664 succinate
CAS:<p>L-703,664 succinate is a 5-HT1D receptor agonist.</p>Fórmula:C20H30N4O6SPureza:98%Forma y color:SolidPeso molecular:454.54ML132
CAS:<p>ML132 is an effective and selective inhibitor of caspase 1 (IC50: 0.316 nM).</p>Fórmula:C22H28ClN5O5Forma y color:SolidPeso molecular:477.94Tankyrase-IN-2
CAS:Tankyrase-IN-2 is a selective, potent and orally active inhibitor of tankyrase with IC50s of 10, 7, and 710 nM for TNKS1, TNKS2 as well as PARP1, respectivelyFórmula:C17H14F2N2O2Pureza:98%Forma y color:SolidPeso molecular:316.3Exp6803
CAS:<p>Exp6803 is an Angiotensin II receptor antagonist.</p>Fórmula:C25H25ClN3NaO5Forma y color:SolidPeso molecular:505.93Aminohexylgeldanamycin
CAS:<p>AHGDM, a Geldanamycin derivative, inhibits HSP90 with strong antiangiogenic and antitumor effects.</p>Fórmula:C34H52N4O8Forma y color:SolidPeso molecular:644.8CJ-17493 (free base)
CAS:<p>CJ-17493 (free base) is a Neurokinin-1 Receptor Antagonist.</p>Fórmula:C24H29F3N2O2Forma y color:SolidPeso molecular:434.49Etamiphylline Camsylate
CAS:<p>Etamiphylline Camsylate is used for the treatment of chronic obstructive pulmonary disease (COPD).</p>Fórmula:C23H37N5O6SForma y color:SolidPeso molecular:511.64MDK8228
CAS:<p>MDK8228 is an inhibitor of CBP/p300 and BRD4 bromodomain. MDK8228 downregulates IL-6, IL-ß and IFN-ß in macrophages.</p>Fórmula:C31H41N5O3Forma y color:SolidPeso molecular:531.69Chlordene
CAS:<p>Chlordene, as a polychlorinated flame retardant, has bioaccumulation and biomagnification potentials.</p>Fórmula:C10H6Cl6Forma y color:SolidPeso molecular:338.87Methotrexate-α-alanine
CAS:<p>Methotrexate-alpha-alanine is a prodrug.</p>Fórmula:C23H27N9O6Pureza:98%Forma y color:SolidPeso molecular:525.52Enpp/Carbonic anhydrase-IN-2
<p>Enpp/Carbonic anhydrase-IN-2: A potent inhibitor (IC50: 1.13-0.33 µM) for NPP1-3, CA-IX/XII; anti-cancer, low toxicity, induces apoptosis.</p>Fórmula:C23H24FNO4SForma y color:SolidPeso molecular:429.5S101
CAS:<p>S101 is an inhibitor of proliferating T-cells, rescuing mice from superantigen-induced shock.</p>Fórmula:C24H23N3O3Forma y color:SolidPeso molecular:401.46JX040
CAS:<p>JX040 inhibits enterovirus replication, strong against non-polio strains, weak on polioviruses.</p>Fórmula:C19H17N5OSForma y color:SolidPeso molecular:363.44TC-E 5006
CAS:γ-secretase modulatorFórmula:C29H29F4NO2Pureza:98%Forma y color:SolidPeso molecular:499.54Xanthine oxidase-IN-7
CAS:<p>Xanthine oxidase-IN-7: Potent oral XO inhibitor (IC50=0.36μM), lowers serum uric acid, promising for hyperuricemia/gout research.</p>Fórmula:C16H14N4O2Forma y color:SolidPeso molecular:294.31CA 074
CAS:<p>CA 074 is a potent inhibitor of cathepsin B with a Ki value of 2 to 5 nM.CA 074 inhibits ischemic hippocampal neuronal death in primates and attenuates</p>Fórmula:C18H29N3O6Pureza:97.80%Forma y color:SolidPeso molecular:383.44CCG-4986
CAS:<p>CCG-4986 is the first small molecule RGS inhibitor reported that directly bound to an RGS protein.</p>Fórmula:C13H11ClN2O5S2Forma y color:SolidPeso molecular:374.82GD-131
CAS:<p>GD-131 is an inhibitor of extraneural uptake.</p>Fórmula:C11H22ClNForma y color:SolidPeso molecular:203.75Cgp 55802A
CAS:<p>CGP 55802A is a novel photoaffinity ligand for in-situ labeling of NMDA receptors.</p>Fórmula:C18H24IN5NaO7PForma y color:SolidPeso molecular:603.286CJ 033466
CAS:<p>CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.</p>Fórmula:C19H28ClN5OPureza:99.72%Forma y color:SolidPeso molecular:377.91YM-900
CAS:YM-900, an AMPA receptor antagonist and glutamate receptor antagonist, is used potentially for the treatment of stroke.Fórmula:C11H7N5O4Pureza:98%Forma y color:SolidPeso molecular:273.2Cryosim-3
CAS:<p>Cryosim-3 is a water-soluble, potent, and selective TRPM8 receptor agonist.</p>Fórmula:C15H33OPForma y color:SolidPeso molecular:260.4GSK729
CAS:<p>GSK729 is a novel potent EchA6 inhibitor.</p>Fórmula:C16H16F3N3O2Pureza:98%Forma y color:SolidPeso molecular:339.31BAY1238097
CAS:<p>BAY1238097 is a BET inhibitor with anticancer activity and antiproliferative activity for the study of advanced refractory malignancies.</p>Fórmula:C25H33N5O3Pureza:98.1% - 98.79%Forma y color:SolidPeso molecular:451.56Antibacterial agent 65
CAS:<p>Antibacterial agent 65 is a potential antimicrobial agent and antioxidant agent.</p>Fórmula:C17H16O3Forma y color:SolidPeso molecular:268.31

