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Inhibidores

Inhibidores

Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.

Subcategorías de "Inhibidores"

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Se han encontrado 66639 productos de "Inhibidores"

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  • 3'-Deoxy-3'-amino-ATP

    CAS:
    <p>3'-Deoxy-3'-amino-ATP is a competitive ATP inhibitor with a 2.3 μM Ki, used to synthesize tRNA.</p>
    Fórmula:C10H17N6O12P3
    Forma y color:Solid
    Peso molecular:506.197
  • 2-Nitrobenzaldehyde

    CAS:
    <p>2-Nitrobenzaldehyde can be used for fluorescent immunochromatographic strip test</p>
    Fórmula:C7H5NO3
    Forma y color:Pale Yellow Crystalline Powder
    Peso molecular:151.12
  • Estetrol

    CAS:
    <p>Estetrol (Donesta), a fetal liver-synthesized estrogen, selectively modulates estrogen receptors and may ease menopausal symptoms.</p>
    Fórmula:C18H24O4
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:304.38
  • 5'-Deoxy-5-fluoro-N-[(pentyloxy)carbonyl]cytidine 2',3'-diacetate

    CAS:
    <p>5'-Deoxy-5-fluoro-N-[(pentyloxy)carbonyl]cytidine 2',3'-diacetate is an intermediate in the synthesis of capecitabine.</p>
    Fórmula:C19H26FN3O8
    Pureza:99%
    Forma y color:Solid
    Peso molecular:443.42
  • CRM1-IN-1


    <p>CRM1-IN-1 (Compound KL1), a noncovalent inhibitor of CRM1, promotes nuclear degradation of CRM1 with an IC50 of 0.27 μM, inhibits CRM1-mediated nuclear export,</p>
    Fórmula:C29H48N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:504.7
  • Mtb-IN-3


    <p>Mtb-IN-3 (compound 10c), a selective and potent Mycobacterium tuberculosis (Mtb) inhibitor, exhibits strong antimycobacterial activity in vitro without inducing</p>
    Fórmula:C18H12N2O4
    Forma y color:Solid
    Peso molecular:320.3
  • (+)-Geodin

    CAS:
    <p>(+)-Geodin, a fungal metabolite, boosts fibrinolysis in BAECs (50-150 μM) and glucose uptake in rat adipocytes (1-100 μg/ml).</p>
    Fórmula:C17H12Cl2O7
    Forma y color:Solid
    Peso molecular:399.18
  • 9-Methoxycanthin-6-one-N-oxide

    CAS:
    <p>9-Methoxycanthin-6-one-N-oxide shows cytotoxic activity against a panel of cell lines comprising a number of human cancer cell types.</p>
    Fórmula:C15H10N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:266.25
  • NH-bis(PEG3-Boc)

    CAS:
    NH-bis(PEG3-Boc) is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.
    Fórmula:C26H51NO10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:537.68
  • Sarglaroids F


    <p>Sarglaroids F (compound 6), an anti-inflammatory agent extracted from the roots of Grass Coral, suppresses LPS/ATP-induced IL-1β secretion by modulating K+</p>
    Fórmula:C38H44O12
    Pureza:98%
    Forma y color:Solid
    Peso molecular:692.75
  • 3,5-Dihydroxybenzaldehyde

    CAS:
    <p>3,5-Dihydroxybenzaldehyde helps synthesize antileishmanial 2,4-dimethylbenzoylhydrazones with antioxidant properties.</p>
    Fórmula:C7H6O3
    Forma y color:White To Tan To Grey Crystalline Powder
    Peso molecular:138.12
  • PEG2-bis(phosphonic acid diethyl ester)

    CAS:
    <p>PEG2-bis(phosphonic acid diethyl ester) is a PEG derivative used as a linker in PROTACs synthesis.</p>
    Fórmula:C12H28O9P2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:378.29
  • Olean-12-ene-3,11-dione

    CAS:
    <p>Olean-12-ene-3,11-dione is a natural product for research related to life sciences. The catalog number is TN4702 and the CAS number is 2935-32-2.</p>
    Fórmula:C30H46O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:438.69
  • Biotin-amido-PEG4-PFP ester


    <p>Biotin-amido-PEG4-PFP ester is a Polyethylene glycol (PEG)-based PROTAC linker utilized for PROTACs synthesis [1].</p>
    Fórmula:C30H41F5N4O9S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:728.72
  • Bryonamide B

    CAS:
    <p>Bryonamide B is a cucurbitane triterpene that can be extracted from Bryonia aspera.</p>
    Fórmula:C10H13NO4
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:211.21
  • Jacobine

    CAS:
    <p>Jacobine causes dose-dependent DNA interstrand cross-links, catalyzed by guinea pig liver enzymes in vitro.</p>
    Fórmula:C18H25NO6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:351.39
  • BCN-PEG1-Val-Cit-PABC-OH


    <p>BCN-PEG1-Val-Cit-PABC-OH is a cleavable 1-unit PEG linker specifically utilized in the synthesis of antibody-drug conjugates (ADCs)[1].</p>
    Fórmula:C34H50N6O8
    Pureza:98%
    Forma y color:Solid
    Peso molecular:670.8
  • Calcium lactate

    CAS:
    <p>Calcium lactate (Conclyte) fortifies juice with calcium and aids soybean sprout growth and phytic acid breakdown.</p>
    Fórmula:C6H10CaO6
    Pureza:≥98%
    Forma y color:White Crystalline Powder Almost Odourless White Crystalline Powder Or Granules
    Peso molecular:218.22
  • Saikogenin F

    CAS:
    <p>Saikogenin F ((1S,2S,4S,5R,8R,9R,10S,13S,14R,17S,18R)-9-(hydroxymethyl)-4,5,9,13,20,20-hexamethyl-24-oxahexacyclo[15.5.2.01,1?.0?,1?.0?,1?.0?,13]tetracos-15-ene</p>
    Fórmula:C30H48O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:472.7
  • Asebogenin

    CAS:
    <p>Asebogenin is isolated from Salvia miltiorrhiza and has antifungal activity, inhibits platelet reactions and inhibits NET formation.</p>
    Fórmula:C16H16O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:288.3