
Derivados de Quinazolina y Quinolina
Las quinazolinas y quinolinas son compuestos heterocíclicos nitrogenados con estructuras aromáticas que desempeñan un papel clave en la síntesis de fármacos con actividad anticancerígena, antimicrobiana y antiinflamatoria. Sus derivados presentan modificaciones estructurales que optimizan su biodisponibilidad y selectividad, lo que permite el desarrollo de nuevos principios activos para diversas aplicaciones terapéuticas. Estos compuestos se utilizan en la fabricación de APIs destinados al tratamiento de cáncer, infecciones, enfermedades neurodegenerativas y cardiovasculares. Además, los derivados de quinazolina y quinolina son esenciales en la investigación de inhibidores enzimáticos y en el diseño de moléculas bioactivas innovadoras. En CymitQuimica disponemos de derivados de quinazolina y quinolina de alta pureza para aplicaciones en síntesis química, desarrollo farmacéutico y biotecnología.
Se han encontrado 65630 productos de "Derivados de Quinazolina y Quinolina"
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2-[5-(3-bromophenyl)-1H-pyrazol-3-yl]-5-methylphenol
CAS:Pureza:95.0%Peso molecular:329.19699096679693-Phenoxyphenylacetonitrile
CAS:Producto controlado<p>Applications 3-PHENOXYPHENYLACETONITRILE (cas# 51632-29-2) is a useful research chemical.<br></p>Fórmula:C14H11NOForma y color:NeatPeso molecular:209.24Propylthiouracil
CAS:Producto controlado<p>Applications Antihyperthyroid. Has been used to promote fattening. This substance is reasonably anticipated to be a human carcinogen.<br>References Aboul-Enein, H.Y., et al.: Anal. Profiles Drug Subs., 6, 457 (1977), Cooper, D.S., et al.: N. Engl. J. Med., 311, 1353 (1984),<br></p>Fórmula:C7H10N2OSForma y color:White To Off-WhitePeso molecular:170.23rac-erythro Methylphenidate Hydrochloride
CAS:Producto controlado<p>Applications The erythro isomers have been shown to exhibit very little therapeutic effect and contribute mainly to the toxic hypertensive effects of this drug.Controlled substance.<br>References Greenblatt, E.N., et al.: J. Pharmacol. Exp. Ther., 131, 115 (1961), Padmanabhan, G.R., et al.: Anal. Profiles Drug Subs., 10, 473 (1981), Kuczenski, R., et al.: J. Pharmacol. Exp. Ther., 296, 876 (2001), Pelham, W.E., et al.: J. Consult. Clin. Psychol., 61, 506 (1993), Srinivas, N.R., et al.: Pharm. Res., 10, 14 (1993),<br></p>Fórmula:C14H19NO2·ClHForma y color:NeatPeso molecular:269.77Telmisartan-d4
CAS:Producto controlado<p>Applications Telmisartan-d4 is deuterium labelled Telmisartan (T017000). Telmisartan is an angiotensin II receptor antagonist.<br>References Wienen, W. et al.: Br. J. Pharmacol., 110, 245 (1993); Neutel, J.M. et al: Adv. Therap., 15, 206 (1998)<br></p>Fórmula:C33D4H26N4O2Forma y color:NeatPeso molecular:518.643-(Trifluoromethyl)-6,7-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-8(5H)-one
CAS:Producto controladoFórmula:C6H5F3N4OForma y color:Off White To Light GreyPeso molecular:206.13N’-Cyano-N,N-dimethylguanidine
CAS:Producto controlado<p>Impurity Cimetidine EP Impurity G<br>Applications N-Cyano-N',N''-dimethylguanidine (Cimetidine EP Impurity G) is an impurity of Cimetidine (C441650), which acts as a competitive histamine H2-receptor antagonist which inhibits gastric acid secretion and reduces pepsin output (1).<br>References 1. Brimblecombe, R. et al.: J. Int. Med. Res. 1975 Mar:3(2) 86-92<br></p>Fórmula:C4H8N4Forma y color:NeatPeso molecular:112.13Isoniazid-d4
CAS:Producto controlado<p>Applications Labelled Isoniazid. Antibiotic for treatment of Mycobacterium tuberculosis, inhibits mycolic acid biosynthesis. Metabolized by hepatic N-acetyltransferase (NAT) and cytochrome P450 2E1 (CYP2E1) to form hepatotoxins. Selectively induces expression of CYP2E1. Reversibly inhibits CYP2C19 and CYP3A4 activities, and mechanistically inactivates CYP1A2, CYP2A6, CYP2C19 and CYP3A4 at clinically relevant concentrations. Antibacterial (tuberculostatic).<br>References Brewer, G.A., et al.: Anal. Profiles Drug Subs., 6, 183 (1977), Weber, W.W., et al.: Clin. Pharmacokinet., 4, 401 (1979)<br></p>Fórmula:C62H4H3N3OForma y color:White To Light BeigePeso molecular:141.16Brivaracetam-d7
CAS:Producto controlado<p>Applications Brivaracetam-d7, is the labeled analogue of Brivaracetam (B677645), which is a 4-n-propyl analog of levetiracetam (L331500), and a racetam derivative with anticonvulsant properties.<br>References Rosenstiel, P., et al.:Neurotherapeutics, 4 (1), 84 (2007);<br></p>Fórmula:C11H13D7N2O2Forma y color:Off White SolidPeso molecular:219.33Ref: 10-F200680
1gA consultar2gA consultar5gA consultar100mgA consultar250mgA consultar500mgA consultarMethylphenidate Hydrochloride
CAS:Producto controlado<p>Applications Controlled substance (stimulant). CNS stimulant. Four isomers of Methylphenidate are known to exist. One pair of threo isomers and one pair of erythro are distinguished, from which only d-threo-Methylphenidate exhibits the pharmacologically usually desired effects. This compound is a 4:1 mixture of rac-erythro (M325670) and rac-threo (M325671).<br>References Greenblatt, E.N., et al.: J. Pharmacol. Exp. Ther., 131, 115 (1961), Padmanabhan, G.R., Anal. Profiles Drug Subs., 10, 473 (1981), Srinivas, N.R., et al.: Pharm. Res., 10, 14 (1993),<br></p>Fórmula:C14H19NO2·ClHForma y color:White To Off-WhitePeso molecular:269.776-Hydroxy-3,4-dihydro-1H-quinoline-2-one
CAS:Producto controlado<p>Impurity Cilostazol USP Related Compound A<br>Applications A metabolite of Cilostazole.<br>References Gitto, R., et al.: J. Med. Chem., 46, 3758 (2003), Xie, Z., et al.: Bioorg. Med. Chem. Lett., 15, 4803 (2005),<br></p>Fórmula:C9H9NO2Forma y color:NeatPeso molecular:163.172-METHOXY-5-(5-(PYRIDIN-4-YL)-1H-BENZO[D]IMIDAZOL-1-YL)PHENOL
CAS:Pureza:95.0%Peso molecular:317.34799194335942-([1,1'-Biphenyl]-3-yl)-4,6-dichloro-1,3,5-triazine
CAS:Pureza:97.0%Peso molecular:302.1600036621094N-(3-Chloro-4-fluorophenyl)-6-nitro-7-(phenylsulfonyl)quinazolin-4-amine
CAS:Pureza:98+%Peso molecular:458.85000610351563-acetyl-6-fluoro-4-(4-fluorophenyl)quinolin-2(1H)-one
CAS:Pureza:95.0%Peso molecular:299.27700805664063-Amino-5-methylpyridin-2(1H)-one
CAS:Fórmula:C6H8N2OPureza:95.0%Forma y color:SolidPeso molecular:124.143Clidinium Bromide
CAS:Producto controlado<p>Applications An anticholinergic. Used as an antispasmodic.<br>References Zhang, L., et al.: Pharm. Res., 25, 1902 (2008), Sanderson, H., et al.: Toxicol Lett., 187, 84 (2009),<br></p>Fórmula:C22H26NO3·BrForma y color:White SolidPeso molecular:432.35Indocyanine Green (~90%)
CAS:Producto controladoFórmula:C43H47N2O6S2·NaPureza:~90%Forma y color:NeatPeso molecular:774.96Diphenylglycoluril
CAS:Producto controlado<p>Applications Diphenylglycoluril is a bicyclic bis-urea derivative. Studies suggest that it has potential anticonvulsant activity.Diphenylglycoluril is also an impurity found in the synthesis of Phenytoin (D491650).<br>References Khlebnikov, A.I. et al.: Pharm. Chem. J., 36, 240 (2002); Babkibayev, A.A. et al.: Pharm. Chem. J., 8, 15 (1994);<br></p>Fórmula:C16H14N4O2Forma y color:NeatPeso molecular:294.31Bupivacaine-d9 Hydrochloride
CAS:Producto controlado<p>Applications Labelled Bupivacaine (B689560). Sodium channel blocker, local anesthetic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Wilson, T.D., et al.: Anal. Profiles Drug Subs., 19, 59 (1990), McClellan, K.J., et al.: Drugs, 56, 355 (1998),<br></p>Fórmula:C182H9H19N2O·ClHForma y color:NeatPeso molecular:333.94Diclazuril 6-Carboxamide
CAS:Producto controlado<p>Applications Diclazuril 6-Carboxamide is an impurity of Diclazuril (D436200), a nucleotide analog with broad-spectrum anticoccidial activity.<br></p>Fórmula:C18H10Cl3N5O3Forma y color:NeatPeso molecular:450.66Trametinib Impurity-I
CAS:Producto controladoFórmula:C26H23FIN5O5Forma y color:NeatPeso molecular:631.394Ethyl 4-(4-chlorophenyl)-2-[2-(4-nitrophenoxy)acetamido]thiophene-3-carboxylate
CAS:Peso molecular:460.89001464843752-Hydroxy Imipramine
CAS:Producto controlado<p>Applications A metabolite of Imipramine.<br>References De Jongh, G.D., et al.: Drug Metab. Dispos., 2, 48 (1981), Suckow, R.F., et al.: J. Pharm. Sci., 73, 1745 (1984), Fraser, A.D., et al.: J. Anal. Toxicol., 11,168 (1987),<br></p>Fórmula:C19H24N2OForma y color:Yellowish SolidPeso molecular:296.414-Phenyl-2-(pyridin-3-yl)thiazole
CAS:Pureza:95.0%Forma y color:Liquid, No data available.Peso molecular:238.309997558593755-[1-(2,3-Dimethylphenyl)ethenyl]-1H-imidazole
CAS:Producto controladoFórmula:C13H14N2Forma y color:NeatPeso molecular:198.261,2,3,4-Tetrahydro-2-[2-(4-hydroxyphenyl)-1-methylethyl]-4,6,8-isoquinolinetriol
CAS:Producto controladoFórmula:C18H21NO4Forma y color:NeatPeso molecular:315.361,1'-Bis(2,4-dinitrophenyl)-4,4'-bipyridinium dichloride
CAS:Pureza:98%Peso molecular:561.2899780273438Demethyl Chlorpromazine Hydrochloride
CAS:Producto controlado<p>Impurity Chlorpromazine EP Impurity D<br>Applications A metabolite of Chlorpromazine (C424750).<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Neuhoff, E., et al.: Archiv. der Pharmazie, 288, 400 (1955), Tomita, M., et al.: Chem. Pharm. Bull., 16, 688 (1968),<br></p>Fórmula:C16H17ClN2S·ClHForma y color:WhitePeso molecular:341.303-Bromomethyl-thiophene-2-carboxylic acid methyl ester
CAS:Pureza:97.0%Forma y color:Solid, Light yellow solidPeso molecular:235.10000610351562N-[1-(1H-1,2,3-Benzotriazol-1-yl)-3-phenylpropyl]pyridine-4-carboxamide
Peso molecular:357.4169921875Rivastigmine N-Oxide (Technical Grade)
CAS:Producto controlado<p>Applications Rivastigmine N-Oxide is an impurity of Rivastigmine (R541000, Tartrate Salt) which is a brain selective acetylcholinesterase inhibitor.<br>References Rosler, M., et al.: Brit. Med. J., 318, 633 (1999), Enz, A., et al.: Prog. Brain Res., 98, 431 (1993)<br></p>Fórmula:C14H22N2O3Forma y color:Light Yellow LiquidPeso molecular:266.34Edoxaban-d6
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications Edoxaban-d6 is the isotope labelled analog of Edoxaban (E555520); an anticoagulant drug which acts as a direct factor Xa inhibitor.<br>References Ruff, C., et al.: Am. Heart J., 160, 635 (2010); Ogata, K., et al.: J. Clin. Pharm., 50, 73 (2010)<br></p>Fórmula:C24H24D6ClN7O4SForma y color:Light Beige To Light BrownPeso molecular:554.09Gleevec-d8 Mesylate (Imatinib-d8 Mesylate)
CAS:Producto controlado<p>Applications A deuterated tyrosine kinase inhibitor. Highly specific for BCR-ABL, the enzyme associated with chronic myelogenous leukemia (CML) and certain forms of acute lymphoblastic leukemia (ALL). It is a COVID19-related research product.<br>References Schindler, T., et al.: Science, 289, 1938 (2000), Drucker, B.J., et al.: N. Engl. J. Med., 344, 1031 (2001),<br></p>Fórmula:C292H8H23N7O·CH4O3SForma y color:NeatPeso molecular:597.761-(4-Methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylic Acid
CAS:Fórmula:C25H24N4O5Forma y color:Light Orange ColourPeso molecular:460.48Roflumilast N-Oxide
CAS:Producto controlado<p>Applications Roflumilast-N-oxide is the active metabolite of Roflumilast (R639700).<br>References Chiba, M., et al.: Drug Metab. Dispos., 25, 1022 (1997), Jarvis, B., et al.: Drugs, 59, 891 (2000),<br></p>Fórmula:C17H14Cl2F2N2O4Forma y color:NeatPeso molecular:419.213-Picoline
CAS:Producto controlado<p>Applications A useful precursor to agrochemicals and antidotes for organophosphate poisoning.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Qiao, L., et al.: Bioorg. Med. Chem. Lett., 19, 6122 (2009), Giri, A., et al.: Food Chem., 120, 621 (2010), Farrer, N., et al.: Chem. Res. Toxicol., 23, 413 (2010),<br></p>Fórmula:C6H7NForma y color:ColourlessPeso molecular:93.134-[4-(4-Chlorophenyl)-3,6-dihydro-1(2H)-pyridinyl]-1-(4-fluorophenyl)-1-butanone
CAS:<p>Applications 4-[4-(4-Chlorophenyl)-3,6-dihydro-1(2H)-pyridinyl]-1-(4-fluorophenyl)-1-butanone is a dehydrated metabolite of haloperidol that can be biotransfomed by humans to Haloperidol pyridinium (HPP+), a potential neurotoxic found in the brain.<br>References Usuki, E., et. al.: Neurotoxicity Res., 4, 51 (2002)<br></p>Fórmula:C21H21ClFNOForma y color:NeatPeso molecular:357.8512-Hydroxy Irinotecan (Mixture of Diastereomers)
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications A metabolite of Irinotecan (I767500) found in human bile and urine.<br>References Lokeic, F. et al.: Clin. Cancer Res., 2, 1943 (1996); Dodds, H.M. et al.: Anti-cancer Drug Des., 16, 239 (2001); Kunimoto, T., et al.: Cancer Res., 47, 5944 (1987); Shimada, Y., et al.: J. Clin. Oncol., 11, 909 (1993);<br></p>Fórmula:C33H38N4O7Forma y color:Off-WhitePeso molecular:602.68Chlorpromazine N-Oxide Maleic Acid Salt
CAS:Producto controlado<p>Applications Chlorpromazine N-Oxide Maleic Acid Salt is an impurity of Chlorpromazine (C424750) which has antiemetic; antipsychotic properties.<br>References Anden, N.-E., et al.: Eur. J. Pharmacol., 11, 303 (1970), Curzon, G., et al.: Trends Pharmacol. Sci., 11, 61 (1990)<br></p>Fórmula:C21H23ClN2O5SForma y color:NeatPeso molecular:450.948-methyl-4-(pyridine-4-carbonyl)-1-oxa-4-azaspiro[4.5]decane-3-carboxylic acid
CAS:Pureza:95.0%Peso molecular:304.346008300781251-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazine
CAS:Producto controlado<p>Applications 1-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazine is an intermediate used to prepare nonracemic γ-bicyclic heteroarylpiperazine- and heteroarylpiperidine-substituted prolinylthiazolidines as selective and orally active dipeptidylpeptidase 4 inhibitors for use as antidiabetic agents.<br>References Yoshida, T., et al.: Bioorg. Med. Chem., 20, 5705 (2012)<br></p>Fórmula:C14H18N4Forma y color:NeatPeso molecular:242.324-(4-Chloro-pyrazol-1-ylmethyl)-phenylamine
CAS:Fórmula:C10H10ClN3Pureza:97%Forma y color:SolidPeso molecular:207.66Febantel
CAS:Producto controlado<p>Applications Used as an anthelmintic.<br>References Thomas, H.: Res. Vet. Sci., 25, 290 (1978), Shmidl, J.A.: Vet. Med. Small Anim. Clin., 73, 775 (1978)<br></p>Fórmula:C20H22N4O6SForma y color:NeatPeso molecular:446.48Isoniazid
CAS:Producto controlado<p>Applications Antibiotic for treatment of Mycobacterium tuberculosis, inhibits mycolic acid biosynthesis. Metabolized by hepatic N-acetyltransferase (NAT) and cytochrome P450 2E1 (CYP2E1) to form hepatotoxins. Selectively induces expression of CYP2E1. Reversibly inhibits CYP2C19 and CYP3A4 activities, and mechanistically inactivates CYP1A2, CYP2A6, CYP2C19 and CYP3A4 at clinically relevant concentrations. Antibacterial (tuberculostatic).<br>References Brewer, G.A., et al.: Anal. Profiles Drug Subs., 6, 183 (1977), Weber, W.W., et al.: Clin. Pharmacokinet., 4, 401 (1979)<br></p>Fórmula:C6H7N3OForma y color:NeatPeso molecular:137.14N-Desmethyl Riociguat
CAS:Producto controlado<p>Applications N-Desmethyl-riociguat, is a complex that is part affiliated with potent oral stimulator for the treatment of pulmonary hypertension.<br>References Mittendorf, J., et al.: ChemMedChem., 4, 853 (2009)<br></p>Fórmula:C19H17FN8O2Forma y color:NeatPeso molecular:408.39N-tert-Butyl-3-(2-hydroxypropan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazole-1-carboxamide
CAS:Producto controlado<p>Stability Light Sensitive<br>Applications N-tert-Butyl-3-(2-hydroxypropan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazole-1-carboxamide is a metabolite of Amicarbazone (A605040); a triazolinone herbicide with a broad spectrum of weed control.<br>References Dayan, F., et al.: Weed Science, 57, 579 (2009); Elmore, M., et al.: Weed Technol., 27, 596 (2013); Dong, M., et al.: J. Sep. Sci., 38, 2245 (2015)<br></p>Fórmula:C10H18N4O3Forma y color:NeatPeso molecular:242.27Everolimus
CAS:Producto controlado<p>Impurity Everolimus EP Impurity C<br>Stability Hygroscopic<br>Applications Everolimus Macrolide immunosuppressant; Everolimus is a derivative of Rapamycin. Everolimus inhibits cytokine-mediated lymphocyte proliferation.<br>References Dumont, F.J., et al.: Curr. Opin. Invest. Drugs, 2, 1220 (2001), Kovarik, J. M., et al.: Clin. Pharmacol. Ther., 69, 48 (2001), Nashan, B., et al.: Ther. Drug Monit., 24, 53 (2002),<br></p>Fórmula:C53H83NO14Pureza:~90%Forma y color:NeatPeso molecular:958.224-(4-(3-(1H-Pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-6-yl)phenyl)morpholine
CAS:Pureza:97.0%Peso molecular:346.39401245117192-[2-(pyridin-3-yl)-1H-indol-3-yl]ethan-1-amine hydrochloride
CAS:Pureza:95.0%Peso molecular:273.76000976562510-Oxo Mirtazapine (Mirtazapine Impurity F)
CAS:Producto controlado<p>Impurity Mirtazapine EP Impurity F<br>Applications 10-Oxo Mirtazapine (Mirtazapine Impurity F) is an impurity of Mirtazapine. Mirtazapine EP Impurity F.<br>References De Boer, T., et al.: Neuropharmacol., 27, 399 (1988), Vindevogel, J., et al.: Anal. Chem., 63, 1530 (1991), Wynia, G., et al.: J. Chromatogr., 773, 339 (1997),<br></p>Fórmula:C17H17N3OForma y color:NeatPeso molecular:279.343-(2,4-dimethylphenyl)-2-sulfanylidene-1,2,3,4-tetrahydroquinazolin-4-one
CAS:Pureza:98%Peso molecular:282.35998535156253-Hydroxy Nevirapine
CAS:Producto controlado<p>Applications A metabolite of Nevirapine (N391275).<br>References Rettie, A., et al.: J. Biol. Chem., 263, 13733 (1988), Lamson, M., et al.: Biopharm. Drug Dispos., 20, 285 (1999), Guengerich, F., et al.: Chem. Res. Toxicol., 14, 611 (2001), Lu, W., et al.: Drug Metab. Dispos., 36, 1624 (2008),<br></p>Fórmula:C15H14N4O2Forma y color:NeatPeso molecular:282.30DL-Norepinephrine-d6 Hydrochloride, 85%
CAS:Producto controlado<p>Applications Antagonist of dibutyryl cyclic AMP in the regulation of narcosis. Norepinephrine modulates human dendritic cell activation by altering cytokine release.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Piguet, P., et al.: J. Exp. Med., 173, 673 (1991), Hosoi, J., et al.: Nature, 363, 159 (1993), Elenkov, I., et al.: Pharmacol. Rev., 52, 595 (2000), Kaplan, D., et al.: Immunity, 23, 611 (2005),<br></p>Fórmula:C82H6H5NO3·ClHPureza:85%Forma y color:NeatPeso molecular:211.68Ethyl 2-[6-(formamidomethyl)-3-phenyl-2-pyridyl]acetate
CAS:Pureza:97%Peso molecular:298.3420104980469Ref: 10-F625998
1gA consultar5gA consultar10gA consultar25gA consultar100mgA consultar250mgA consultar500mgA consultar2-Isoniazid
CAS:Producto controlado<p>Applications An impurity of Isoniazid (I821450), which is an antibiotic for treatment of Mycobacterium tuberculosis and inhibits mycolic acid biosynthesis. Intermediate used for the synthesis of analogs of antitumor agent 1-acetyl-2-picolinoylhydrazine.<br>References Brewer, G.A., et al.: Anal. Profiles. Drug. Subs., 6, 183 (1977), Weber, W.W., et al.: Clin. Pharmacokinet., 4, 401 (1979); Rutner, H., et al.: Cancer. Chem. Rep., 58, 803 (1974)<br></p>Fórmula:C6H7N3OForma y color:WhitePeso molecular:137.144-(4-Morpholinyl)-1,2,5-thiadiazol-3(2H)-one 1-Oxide
CAS:Producto controlado<p>Impurity Timolol EP Impurity G; Timolol BP Impurity G<br>Stability Moisture Sensitive<br>Applications 4-(4-Morpholinyl)-1,2,5-thiadiazol-3(2H)-one 1-Oxide (Timolol EP Impurity G; Timolol BP Impurity G) is an impurity of Timolol (T4437005), an antihypertensive, an adrenergic blocking agent (1); antiarrhythmic (class II); antianginal; antiglaucoma (2) and antihypertensive (3) agent.<br>References 1. Wasson, B. et al.: J. Med. Chem. 1972 Jun;15(6):651-5.2. Heel, R. et al.: Drugs. 1979 Jan;17(1):38-55.3. Rofman, et al.: Hypertension. 1980 Sep-Oct;2(5):643-8.<br></p>Fórmula:C6H9N3O3SForma y color:WhitePeso molecular:203.22Cyamemazine-d6
CAS:Producto controlado<p>Applications Labelled Cyamemazine is an anxiolytic antipsychotic, which reduces ethanol withdrawal symptoms.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Robinson, et al.: J. Pharm. Pharmacol., 18, 19 (1966), Miller, L., et al.: J. Pharmacol. Exp. Ther., 246, 170 (1988), Podhorna, J., et al.: Curr. Pharm. Des., 8, 23 (2002), Hameg, A., et al.: Biochem. Pharmacol., 65, 435 (2003),<br></p>Fórmula:C19H15D6N3SForma y color:NeatPeso molecular:329.49Maropitant Citrate Salt
CAS:<p>Applications Maropitant is a neurokinin type 1 (NK-1) receptor antagonist. Recent studies show that Maropitant decreased the anesthetic requirements during visceral stimulation of the ovary and ovarian ligament in dogs.<br>References Boscan, P. et al.: Am. J. Vet. Res., 72, 1576 (2011);<br></p>Fórmula:C32H40N2O·C6H8O7Forma y color:Off White SolidPeso molecular:660.8Piperonylic Acid
CAS:Producto controlado<p>Applications Piperonylic Acid is a compound closely mimicking the structure of transcinnamic acid involved in the phenylpropanoid pathway in plant physiology.<br>References Schalk, M. et al.: Plant Physiol., 118, 209 (1998);<br></p>Fórmula:C8H6O4Forma y color:NeatPeso molecular:166.13Rivaroxaban Diol
CAS:Producto controlado<p>Applications A metabolite of Rivaroxaban (R538000).<br>References Kubitza, D., et al.: Clin. Pharmacol. Ther., 78, 412 (2005), Roehrig, S., et al.: J. Med. Chem., 48, 5900 (2005), Biemond, B., et al.: Thromb. Haemost., 97, 471 (2007), Lang, D., et al.: Drug Metab. Dispos., 37, 1046 (2009),<br></p>Fórmula:C19H20ClN3O6SForma y color:White To Off-WhitePeso molecular:453.9Nocodazole
CAS:<p>M05733 - Nocodazole</p>Fórmula:C14H11N3O3SPureza:98%Forma y color:Solid, Beige powderPeso molecular:301.32000732421875Ref: 10-M05733
1gA consultar1mgA consultar10mgA consultar50mgA consultar100mgA consultar250mgA consultarN-(2-Benzylphenyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
CAS:Pureza:98%Peso molecular:354.40899658203125(±)-Rolipram
CAS:Producto controlado<p>Applications (±)-Rolipram is a cAMP-specific phosphodiesterase 4 (PDE4) inhibitor.<br>References Xin, W., et. al.: J. Pharmacol. Exp. Ther., 349, 56 (2014);<br></p>Fórmula:C16H21NO3Forma y color:NeatPeso molecular:275.345-Hydroxy Dantrolene
CAS:Producto controladoFórmula:C14H10N4O6Forma y color:YellowPeso molecular:330.25Aprepitant
CAS:Producto controlado<p>Applications Aprepitant is a neurokinin-1 antagonist and an antiemetic agent (1). It is used to prevent chemotherapy-induced nausea and vomiting (CINV) in colorectal cancer patients (2) Aprepitant has also been shown to induce apoptotic cell death and G1 arrest through Akt/p53 axis in pre-B acute lymphoblastic leukemia cells (3).<br>References (1) Takemoto, H., et al.: nt J Clin Oncol (2016) (2) Bayati, S., et al.: Eur J Pharmacol. 791, 274 (2016) (3) Navari, R.M.: Expert Rev Anticancer Ther. 4, 715 (2004)<br></p>Fórmula:C23H21F7N4O3Forma y color:Off-WhitePeso molecular:534.437-Bromo-2-chloro-3-methylquinoline
CAS:Fórmula:C10H7BrClNPureza:97%Forma y color:No data available.Peso molecular:256.53Darunavir-d9
CAS:Producto controlado<p>Applications Second generation HIV-1-protease inhibitor; structurally similar to amprenavir. Antiviral. It is a COVID19-related research product.<br>References Koh, Y., et al.: Antimicrob. Agents Chemother., 47, 3123 (2003), Arasteh, K., et al.: AIDS, 19, 943 (2005), Surleraux, D.L.N.G., et al.: J. Med. Chem., 48, 1813 (2005),<br></p>Fórmula:C272H9H28N3O7SForma y color:Off-White To Light BeigePeso molecular:556.72Loratadine Epoxide
CAS:Producto controladoFórmula:C22H23ClN2O3Forma y color:White To Off-WhitePeso molecular:398.883-[2-[4-(4-Fluoro-2-hydroxybenzoyl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one Hydrochloride
CAS:Producto controlado<p>Applications Risperidone (R525000) metabolite.<br>References Meuldermans, W. et al.; Drug Metab. Dispos. 22, 129 (1994); Mannens, G. et al.; Drug Metab. Dispos. 21, 1134 (1993)<br></p>Fórmula:C23H28FN3O3·HClForma y color:NeatPeso molecular:449.946(2E)-1-{[1,1'-biphenyl]-4-yl}-3-(thiophen-2-yl)prop-2-en-1-one
CAS:Pureza:95.0%Peso molecular:290.3800048828125(R)-Albuterol Hydrochloride
CAS:Producto controlado<p>Applications The R-enantiomer of Albuterol (A514500). A β2-adrenoceptor agonist. Bronchodilator; tocolytic.<br>References Han, et al.: Bioorg. Med. Chem., 14, 6043 (2006), Liyou, H., et al.: Biochem., 46, 1432 (2007), Agrawal, D., et al.: J. Allergy Clin. Immunol., 113, 503 (2004),<br></p>Fórmula:C13H21NO3·ClHForma y color:Off-WhitePeso molecular:275.773-(3-methoxyphenyl)-1-methyl-1{H}-pyrazole-5-carboxylic acid
CAS:Pureza:95.0%Peso molecular:232.23899841308594Nadolol-d9
CAS:Producto controlado<p>Applications Labelled Nadolol (N201052). β-Adrenergic blocker. Antihypertensive; antianginal.<br>References Dreyfuss, J., et al.: J. Clin. Pharmacol., 17, 300 (1977), Sibley, P.L., et al.: Toxicol. Appl. Pharmacol., 44, 379 (1978), Slusarek, L., et al.: Anal. Profiles Drug Subs., 9, 455 (1980),<br></p>Fórmula:C17H18D9NO4Forma y color:NeatPeso molecular:318.46Pamabrom
CAS:Producto controlado<p>Applications A diuretic used to reduce menstrual pains.<br>References Varga, J., et al.: Mol. Immunol., 28, 641 (1991), Marrero-Ponce, Y., et al.: Bioorg. Med. Chem., 13, 2881 (2005), Ibrahim, H., et al.: Drug Discov. Ther., 3, 168 (2009),<br></p>Fórmula:C7H7BrN4O2·C4H11NOForma y color:NeatPeso molecular:348.20

