Chromatine/Épigénétique
Les inhibiteurs de la chromatine/épigénétique sont des composés qui modulent la structure et la fonction de la chromatine ou interfèrent avec les modifications épigénétiques, telles que la méthylation de l'ADN et la modification des histones. Ces inhibiteurs sont des outils essentiels pour étudier la régulation de l'expression génique et le rôle de l'épigénétique dans des maladies telles que le cancer, les troubles neurologiques et les anomalies du développement. En ciblant les processus épigénétiques, ces inhibiteurs peuvent modifier les schémas d'expression génique et offrir de nouvelles perspectives thérapeutiques. Chez CymitQuimica, nous offrons une large sélection d'inhibiteurs de la chromatine/épigénétique de haute qualité pour soutenir vos recherches en biologie moléculaire, génétique et épigénétique.
Sous-catégories appartenant à la catégorie "Chromatine/Épigénétique"
2612 produits trouvés pour "Chromatine/Épigénétique"
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EML 425
CAS :EML 425 is a potent and selective inhibitor of CREB binding protein (CBP)/p300 (IC50s: 2.9 and 1.1 μM, respectively).Formule :C27H24N2O4Degré de pureté :97.6%Couleur et forme :SolidMasse moléculaire :440.49Ref: TM-T15216
5mg42,00€10mg67,00€25mg129,00€50mg187,00€100mg276,00€200mg391,00€1mL*10mM (DMSO)46,00€Citric acid trilithium salt tetrahydrate
CAS :Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) , the active component of Lithium, is a medicine used in the therapy ofFormule :C6H13Li3O11Degré de pureté :99.88%Couleur et forme :White Crystalline PowderMasse moléculaire :281.98Brepocitinib P-Tosylate
CAS :Brepocitinib P-Tosylate (PF-06700841 P-Tosylate) is a potent dual inhibitor of Janus kinase 1 (JAK1) and TYK2 (IC50s of 17 nM and 23 nM, respectively).Formule :C25H29F2N7O4SDegré de pureté :99.82% - 99.97%Couleur et forme :SolidMasse moléculaire :561.6BVT948
CAS :BVT948 is a protein tyrosine phosphatase (PTP) inhibitor.It can also inhibit lysine methyltransferase SETD8 (KMT5A) and several cytochrome P450 (P450) isoforms.Formule :C14H11NO3Degré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :241.24Ref: TM-T14841
1mg38,00€2mg49,00€5mg80,00€10mg104,00€25mg157,00€50mg210,00€100mg338,00€1mL*10mM (DMSO)88,00€Hydroxycitric acid tripotassium hydrate
CAS :Hydroxycitric acid tripotassium hydrate (Potassium citrate monohydrate) effectively inhibits HIF, has antioxidation, anti-inflammation, and anti-tumor effects.Formule :C6H7K3O8Degré de pureté :99.85%Couleur et forme :White Solid CrystallineMasse moléculaire :324.41Deferoxamine Mesylate
CAS :Deferoxamine Mesylate (DFOM) is an iron chelator and iron death inhibitor.Formule :C26H52N6O11SDegré de pureté :94.68% - 99.8%Couleur et forme :SolidMasse moléculaire :656.79Diflunisal
CAS :Diflunisal (Dolobid) is a cyclooxygenase (COX) Inhibitor, used as an anti-inflammatory analgesic.Formule :C13H8F2O3Degré de pureté :98.92% - 99.42%Couleur et forme :SolidMasse moléculaire :250.20Tulmimetostat
CAS :Tulmimetostat (CPI-0209) is an orally active EZH1/EZH2 inhibitor.Tulmimetostat has antitumor activity and is used in the study of ovarian cancer and advancedFormule :C28H36ClN3O5SDegré de pureté :98.04% - 99.872%Couleur et forme :SolidMasse moléculaire :562.12Albendazole
CAS :Albendazole (SKF-62979) is used as a drug indicated for the treatment of a variety of worm infestations.Formule :C12H15N3O2SDegré de pureté :98.21% - 98.76%Couleur et forme :Colorless Crystals SolidMasse moléculaire :265.33mTOR/HDAC-IN-1 HCl
mTOR/HDAC-IN-1 HCl，a dual inhibitor of mTOR and HDAC with potential anti-inflammatory, anti-proliferative, autophagic and apoptosis-inducing effects for cancerFormule :C23H24ClN11O3Degré de pureté :99.56%Couleur et forme :SoildMasse moléculaire :537.96Niraparib (R-enantiomer)
CAS :Niraparib R-enantiomer (MK 4827 R-enantiomer) is an inhibitor of PARP1(IC50 of 2.4 nM).
Formule :C19H20N4ODegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :320.39Flufenamic acid
CAS :Flufenamic acid (Arlef) is an anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties.Formule :C14H10F3NO2Degré de pureté :98.68%Couleur et forme :White To Light Yellow Crystalline PowderMasse moléculaire :281.23AES-135
CAS :AES-135 is a potent HDAC inhibitor, inhibits HDAC3, HDAC6, HDAC11 (IC50s: 654, 190, and 636 nM) with anti-tumor activity.Formule :C33H29F6N3O5SDegré de pureté :97.72%Couleur et forme :SolidMasse moléculaire :693.66Ref: TM-T10255
1mg79,00€5mg152,00€10mg250,00€25mg424,00€50mg583,00€100mg803,00€1mL*10mM (DMSO)225,00€Ilginatinib
CAS :Ilginatinib (NS-018) is a highly active and orally bioavailable inhibitor of JAK2.Formule :C21H20FN7Degré de pureté :98.4% - 99.01%Couleur et forme :SolidMasse moléculaire :389.43Ref: TM-T12266
1mg60,00€5mg131,00€10mg177,00€25mg259,00€50mg371,00€100mg532,00€200mg705,00€1mL*10mM (DMSO)126,00€Bufexamac
CAS :Bufexamac (Bufexamic acid) is a COX inhibitor for IFN-α release with anti-inflammatory, analgesic, and antipyretic action.Formule :C12H17NO3Degré de pureté :99.73%Couleur et forme :Acicular CrystalMasse moléculaire :223.27SMARCA-BD ligand 1 for Protac
CAS :SMARCA-BD ligand 1 for Protac is a compound capable of binding to SMARCA2, the BAF ATPase subunit, based on the Protac technology for degrading SMARCA2Formule :C14H17N5ODegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :271.32Nicotinamide riboside
CAS :Nicotinamide riboside increases NAD[+] levels and activates SIRT1 and SIRT3, culminating in enhanced oxidative metabolism and protection against high fat diet-
Formule :C11H15N2O5Degré de pureté :98.82% - 99.58%Couleur et forme :SolidMasse moléculaire :255.25TAK-901
CAS :TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid Metaplasia, and Advanced Solid Tumors, among othersFormule :C28H32N4O3SDegré de pureté :99.02% - 99.59%Couleur et forme :SolidMasse moléculaire :504.64Ref: TM-T2709
1mg35,00€5mg70,00€10mg104,00€25mg202,00€50mg329,00€100mg525,00€200mg748,00€1mL*10mM (DMSO)79,00€Indoprofen
CAS :Indoprofen ((±)-Indoprofe) is a non-steroidal anti-inflammatory drug.Formule :C17H15NO3Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :281.31N-(3-Aminopropyl)cyclohexylamine
CAS :N-(3-Aminopropyl)cyclohexylamine inhibits spermine synthase; used in neuro disease research.Formule :C9H20N2Degré de pureté :98.05% - 98.82%Couleur et forme :Pale Yellow Clear LiquidMasse moléculaire :156.2685Curcumin
CAS :Curcumin (Natural Yellow 3) is a phenolic natural product, an inhibitor of histone acetyltransferase p300/CREB (IC50=25 μM) with specificity.Formule :C21H20O6Degré de pureté :95% - 98.98%Couleur et forme :Orange-Yellow Crystal Powder; Gives Brownish-Red Color With Alkali; Light-Yellow Color With Acids Physical Description Orange-Yellow Needles (Ntp 1992)Masse moléculaire :368.38Delcasertib
CAS :Delcasertib (KAI-9803) is a potent and selective inhibitor of δ-protein kinase C (δPKC).Formule :C120H199N45O34S2Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :2880.28Ref: TM-T11740
1mg192,00€5mg485,00€10mg700,00€25mg1.063,00€50mg1.459,00€100mg1.963,00€1mL*10mM (DMSO)1.603,00€T-3775440 hydrochloride
CAS :T-3775440 hydrochloride is an irreversible inhibitor of lysine-specific histone demethylase (LSD1)(IC50 : 2.1 nM).Formule :C18H23ClN4ODegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :346.85Ref: TM-T13055
1mg92,00€2mg118,00€5mg192,00€10mg289,00€25mg485,00€50mg663,00€100mg893,00€1mL*10mM (DMSO)212,00€PT-1
CAS :PT-1 is an AMPKα1 activator that dose-dependently activates AMPK α1394, α1335, and α2398 and enhances AMPK phosphorylation.Formule :C23H16ClN3O6SDegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :497.91MC3482
CAS :MC3482 is a specific inhibitor of sirtuin5 (SIRT5).Formule :C33H38N4O8Degré de pureté :98% - 99.90%Couleur et forme :SoildMasse moléculaire :618.68Ref: TM-T11962
1mg50,00€2mg71,00€5mg105,00€10mg170,00€25mg268,00€50mg423,00€100mg685,00€500mg1.378,00€Abexinostat
CAS :Abexinostat (PCI-24781) is a pan-HDAC inhibitor, strongest on HDAC1; less so on HDACs 2, 3, 6, 10. Very select for HDAC8. In Phase 1/2 trials.Formule :C21H23N3O5Degré de pureté :98.19% - 98.43%Couleur et forme :SolidMasse moléculaire :397.42PKC β pseudosubstrate acetate
PKC β pseudosubstrate acetate (PKC β pseudosubstrate acetate (172308-76-8 Free base)) is a selective cell-permeable inhibitor of PKC.Degré de pureté :95.42%Couleur et forme :SoildYPX-C-05
CAS :YPX-C-05, an isohydroxamic acid derivative, is an HDAC inhibitor with vasodilatory and antihypertensive activity.CAS 번호134608-84-5Formule :C21H19N3O4Degré de pureté :98.09%Couleur et forme :SoildMasse moléculaire :377.39Histone Acetyltransferase Inhibitor II
CAS :Histone Acetyltransferase Inhibitor II is a selective and cell permeable inhibitor of p300 histone acetyltransferase(IC50 : 5 μM).with anti-acetylase activityFormule :C20H16Br2O3Degré de pureté :97.13%Couleur et forme :SolidMasse moléculaire :464.15Cyproheptadine hydrochloride sesquihydrate
CAS :Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formule :C21H24ClNODegré de pureté :99.77% - >99.99%Couleur et forme :White To Slightly Yellowish Crystalline SolidMasse moléculaire :341.88N-Desmethyltamoxifen hydrochloride
CAS :N-Desmethyltamoxifen hydrochloride is the major tamoxifen metabolite in humans.Formule :C25H28ClNODegré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :393.95iso-Azalansta
CAS :(2R,4S)-Azalanstat (Iso-Azalansta) is a selective heme oxygenase (HO) inhibitor that is used in the study of cardiovascular disease.Formule :C22H24ClN3O2SDegré de pureté :99.53% - 99.89%Couleur et forme :SoildMasse moléculaire :429.96PT2399
CAS :PT2399, an oral HIF-2 inhibitor, blocks HIF-2α/1β dimerization, showing strong in vivo antitumor effects.Formule :C17H10F5NO4SDegré de pureté :98.8% - 99.45%Couleur et forme :SolidMasse moléculaire :419.32Ref: TM-T12675L
1mg88,00€5mg212,00€10mg318,00€25mg575,00€50mg848,00€100mg1.189,00€1mL*10mM (DMSO)233,00€(R)-CR8
CAS :(R)-CR8 ((R)-Isomer) is a potent and selective CDK inhibitor.
Formule :C24H29N7ODegré de pureté :98.41%Couleur et forme :SolidMasse moléculaire :431.53Chitosan oligosaccharide
CAS :Chitosan oligosaccharide (COS) is an oligomer of β-(1→4)-linked D-glucosamine.Formule :C12H24N2O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :340.327DC-05
CAS :DC-05 is an inhibitor of DNA methyltransferase 1 (DNMT1) (IC50 and a Kd: 10.3 μM and 1.09 μM, respectively).Formule :C25H25N3ODegré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :383.49Ref: TM-T15080
1mg66,00€5mg145,00€10mg236,00€25mg515,00€50mg858,00€100mg1.251,00€200mg1.684,00€1mL*10mM (DMSO)158,00€WDR5-IN-6
CAS :WDR5-IN-6 is a WDR5 inhibitor targeting the WBM locus.WDR5-IN-6 is highly synergistic with OICR-9429, a WDR5 inhibitor that targets the WIN locus.WDR5-IN-6Formule :C13H8Cl2N2O2SDegré de pureté :99.69%Couleur et forme :SoildMasse moléculaire :327.19EHP-101
CAS :EHP-101 is a PPARγ/CB2 dual agonist with anti-inflammatory properties, inhibits fat formation, and combats diet-related obesity.Formule :C28H35NO3Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :433.58Ref: TM-T13289
1mg107,00€5mg227,00€10mg378,00€25mg620,00€50mg868,00€100mg1.169,00€1mL*10mM (DMSO)250,00€Hydralazine hydrochloride
CAS :Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.Formule :C8H9ClN4Degré de pureté :99.85% - 99.86%Couleur et forme :Yellow Crystals White Crystalline SolidMasse moléculaire :196.64Diperodon hydrochloride
CAS :Diperodon hydrochloride (Diperocaine) is a local anesthetic that can be broken down by serolytic enzymes to produce local anesthetic effects.Formule :C22H28ClN3O4Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :433.93Nefiracetam
CAS :Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.Formule :C14H18N2O2Degré de pureté :97.37%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :246.3Miglitol
CAS :Miglitol (BAY1099) is an alpha-Glucosidase Inhibitor with antihyperglycemic activity.Formule :C8H17NO5Degré de pureté :99.75% - 99.88%Couleur et forme :White To Pale-Yellow Powder SolidMasse moléculaire :207.22NI-42
CAS :NI-42, a BRPFs inhibitor: IC50(BRPF1/2/3)=7.9/48/260 nM, Kd(BRPF1/2/3)=40/210/940 nM; selective for class IV BRDs.Formule :C18H15N3O3SDegré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :353.39CBP/p300-IN-3
CAS :CBP/p300-IN-3 (P300/CBP-IN-3) is an inhibitor of p300/CBP histone acetyltransferase.Formule :C24H29N7ODegré de pureté :97.38% - 98.08%Couleur et forme :SolidMasse moléculaire :431.53Ref: TM-T12345
1mg87,00€5mg177,00€10mg295,00€25mg447,00€50mg640,00€100mg893,00€500mg2.115,00€1mL*10mM (DMSO)203,00€Phenelzine sulfate
CAS :Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.Formule :C8H14N2O4SDegré de pureté :98.38% - 99.83%Couleur et forme :SolidMasse moléculaire :234.27MS31 trihydrochloride (2366264-12-0 free base)
MS31 trihydrochloride (2366264-12-0 free base) is a potent, highly affinity and selective fragment-like methyllysine reader protein spindlin 1 (SPIN1) inhibitorFormule :C20H30Cl3N3O2Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :450.83Ref: TM-T12111L
1mg185,00€5mg369,00€10mg542,00€25mg867,00€50mg1.153,00€100mg1.584,00€1mL*10mM (DMSO)379,00€Tinengotinib
CAS :Tinengotinib is a multikinase inhibitor that targets a series of kinases , including Aurora kinases A/B, JAK1/2, FGFR1/2/3, VEGFRs, and many other kinases.Formule :C20H19ClN6ODegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :394.86BRM/BRG1 ATP Inhibitor-1
CAS :BRM/BRG1 ATP Inhibitor-1 is an allosteric dual Brahma homolog (BRM)/SWI/SNF related matrix-associated actin-dependent regulator of chromatin subfamily A memberFormule :C11H9F3N4O2SDegré de pureté :98.17% - 99.84%Couleur et forme :SolidMasse moléculaire :318.27Ref: TM-T10616
1mg167,00€5mg409,00€10mg615,00€25mg1.063,00€50mg1.558,00€100mg2.187,00€1mL*10mM (DMSO)442,00€Safingol hydrochloride
CAS :Safingol hydrochloride (L-threo-dihydrosphingosine hydrochloride) is a PKC-specific inhibitor that inhibits PKC and PI3k and induces cancer cell death.Formule :C18H40ClNO2Degré de pureté :99.39% - 99.71%Couleur et forme :SoildMasse moléculaire :337.969Acetaminophen
CAS :Acetaminophen: pain reliever, fever reducer; mild anti-inflammatory. Risks: liver, kidney damage, blood cell effects.Formule :C8H9NO2Degré de pureté :99.85% - 99.99%Couleur et forme :Colourless Solid CrystallineMasse moléculaire :151.16BMS-986158
CAS :BMS-986158: BET inhibitor, IC50 of 6.6 nM in SCLC, 5 nM in TNBC cells.Formule :C30H33N5O2Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :495.62Ref: TM-T14685
1mg87,00€5mg259,00€10mg465,00€25mg745,00€50mg1.026,00€100mg1.388,00€1mL*10mM (DMSO)283,00€BRD-6929
CAS :BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.Formule :C19H17N3O2SDegré de pureté :98.01% - 99.05%Couleur et forme :SolidMasse moléculaire :351.42Ref: TM-T10603
5mg48,00€10mg86,00€25mg166,00€50mg289,00€100mg419,00€200mg587,00€1mL*10mM (DMSO)49,00€LIN28 inhibitor LI71
CAS :LIN28 inhibitor LI71 is a potent and cell-permeable LIN28 inhibitor, which abolishes LIN28-mediated oligouridylation with an IC50 of 7 uM.Formule :C21H21NO3Degré de pureté :95.88%Couleur et forme :SolidMasse moléculaire :335.4Ref: TM-T11850
1mg107,00€5mg255,00€10mg414,00€25mg745,00€50mg1.063,00€100mg1.459,00€1mL*10mM (DMSO)341,00€BRD 4354
CAS :BRD 4354 is an inhibitor of HDAC5 and HDAC9. For HDAC5 and HDAC9, the IC50s values are 0.85 and 1.88 μM, respectively.Formule :C21H23ClN4ODegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :382.89Ref: TM-T10602L
1mg34,00€2mg44,00€5mg66,00€10mg92,00€25mg178,00€50mg308,00€100mg512,00€500mg1.071,00€1mL*10mM (DMSO)73,00€ODM-207
CAS :ODM-207 (BET-IN-4) is a potent BRD4 inhibitor.Formule :C22H21N3O3Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :375.42Ref: TM-T10521
1mg44,00€5mg92,00€10mg133,00€25mg235,00€50mg339,00€100mg480,00€200mg660,00€1mL*10mM (DMSO)90,00€Fenbendazole
CAS :Fenbendazole (Fenbendazol) is an antinematodal benzimidazole used in veterinary medicine.Formule :C15H13N3O2SDegré de pureté :99.74%Couleur et forme :White To Yellowish PowderMasse moléculaire :299.351-Naphthohydroxamic acid
CAS :1-Naphthohydroxamic acid (Compound 2) is a potent and selective HDAC8 inhibitor with an IC50 of 14 μM, and it is more selectively for HDAC8 than class I HDAC1Formule :C11H9NO2Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :187.19Ref: TM-T13996
5mg33,00€10mg60,00€25mg108,00€50mg200,00€100mg299,00€200mg430,00€1mL*10mM (DMSO)38,00€SIRT-IN-2
CAS :SIRT-IN-2 is a potent SIRT1/2/3 inhibitor(IC50s of 4, 1, 7 μM, respectively).Formule :C15H21N5O3S2Degré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :383.49Ref: TM-T12919
1mg92,00€5mg215,00€10mg344,00€25mg587,00€50mg803,00€100mg1.099,00€200mg1.468,00€1mL*10mM (DMSO)236,00€A-3 hydrochloride
CAS :A-3 hydrochloride: potent, reversible kinase antagonist; permeable; inhibits PKC, CKI, PKA, CKII, MLCK; Ki: 4.3-80 μM.Formule :C12H14Cl2N2O2SDegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :321.22Ref: TM-T14069
1mg34,00€5mg63,00€10mg90,00€25mg161,00€50mg260,00€100mg416,00€500mg888,00€1mL*10mM (DMSO)95,00€CG347B
CAS :CG347B is a selective inhibitor of HDAC6.Formule :C16H17N3O2Degré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :283.33Ref: TM-T10777
1mg33,00€5mg75,00€10mg110,00€25mg190,00€50mg290,00€100mg404,00€200mg568,00€1mL*10mM (DMSO)81,00€HDAC-IN-40
CAS :HDAC-IN-40 is a potent alkoxyamide-based HDAC inhibitor with Ki of 60 nM and 30 nM for HDAC2 and HDAC6, respectively. HDAC-IN-40 had antitumor effectsFormule :C15H22N2O6Degré de pureté :99.04%Couleur et forme :SoildMasse moléculaire :326.35PROTAC BRD4 ligand-1
CAS :PROTAC BRD4 ligand-1 is a ligand for BRD4 for Protac GNE-987 and an inhibitor of BET.Formule :C23H18F2N4O5SDegré de pureté :99.28% - 99.93%Couleur et forme :SolidMasse moléculaire :500.47Ilginatinib hydrochloride
CAS :Ilginatinib hydrochloride (NS-018 hydrochloride) is a highly active and orally bioavailable inhibitor of JAK2.Formule :C21H21ClFN7Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :425.89Ref: TM-T12266L2
1mg70,00€5mg150,00€10mg215,00€25mg358,00€50mg517,00€100mg707,00€200mg973,00€1mL*10mM (DMSO)166,00€TRIM24/BRPF1-IN-2
CAS :TRIM24/BRPF1-IN-2 is a TRIM24/BRPF1 dual inhibitor with anticancer activity that inhibits the proliferation of prostate cancer cells.Formule :C20H22N2O4SDegré de pureté :98.69% - 99.13%Couleur et forme :SoildMasse moléculaire :386.47FIDAS-5
CAS :FIDAS-5 is an orally active methionine adenosyltransferase 2A (MAT2A) inhibitor with an IC50 of 2.1 μM. Cost-effective and quality-assured.Formule :C15H13ClFNDegré de pureté :98.3% - 99.17%Couleur et forme :SolidMasse moléculaire :261.72Ref: TM-T11285
1mg56,00€2mg80,00€5mg110,00€10mg177,00€25mg314,00€50mg485,00€100mg700,00€500mg1.341,00€Uzansertib phosphate
CAS :Uzansertib phosphate (INCB053914 phosphate) is an orally active, ATP-competitive inhibitor of pan-PIM kinase, inhibiting PIM1, PIM2 and PIM3.Formule :C26H29F3N5O7PDegré de pureté :99.75% - 99.79%Couleur et forme :SolidMasse moléculaire :611.51Levetiracetam
CAS :Levetiracetam (SIB-S1) is a relatively unique anticonvulsant that is typically used in combination with other antiepileptic medications for partial onsetFormule :C8H14N2O2Degré de pureté :99.67% - 99.86%Couleur et forme :White Crystalline PowderMasse moléculaire :170.21MS402
CAS :MS402 is a novel BD1-selective BET BrD inhibitor.Formule :C20H19ClN2O3Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :370.83Minocycline hydrochloride
CAS :Minocycline HCl: tetracycline antibiotic, treats bacterial infections and acne, may cause acute or chronic hepatitis.Formule :C23H28ClN3O7Degré de pureté :99.28% - >99.99%Couleur et forme :Bright Yellow-Orange Amorphous Solid Crystalline YellowMasse moléculaire :493.94MAK683
CAS :MAK683 is an inhibitor of embryonic ectoderm development (EED) (IC50s: 59, 89, 26 nM in EED Alphascreen binding, LC-MS and ELISA assay).Formule :C20H17FN6ODegré de pureté :98.25% - 99.92%Couleur et forme :SolidMasse moléculaire :376.39Ref: TM-T15201
1mg50,00€5mg102,00€10mg178,00€25mg389,00€50mg575,00€100mg802,00€500mg1.665,00€1mL*10mM (DMSO)89,00€A-485
CAS :A-485 is a p300/CBP histone acetyltransferase (HAT) inhibitor that inhibits p300 and CBP. A-485 has antitumor effects. Cost effective and quality assured.Formule :C25H24F4N4O5Degré de pureté :98.01% - 99.98%Couleur et forme :SolidMasse moléculaire :536.48Ref: TM-T14073
1mg88,00€5mg159,00€10mg273,00€25mg339,00€50mg404,00€100mg698,00€1mL*10mM (DMSO)187,00€Miltefosine
CAS :Miltefosine (HePC), effective oral drug for both visceral and cutaneous leishmaniasis, in clinical trials worldwide.Formule :C21H46NO4PDegré de pureté :98% - 99.94%Couleur et forme :White To Off-White PowderMasse moléculaire :407.57Amifostine
CAS :Amifostine (Ethyol) anhydrous is a cytoprotective agent, acts as a free radical scavenging activity.Formule :C5H15N2O3PSDegré de pureté :99.59%Couleur et forme :White SolidMasse moléculaire :214.22L-2-Hydroxyglutaric acid disodium
CAS :L-2-Hydroxyglutaric acid disodium may affect epigenetics and contribute to renal cancer, inhibiting Mi-CK (Km 2.52 mM, Ki 11.13 mM).Formule :C5H6Na2O5Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :192.08ZEN-3694
CAS :ZEN-3694 (ZEN 3694) is a bromo-structural domain extra-terminal inhibitor (BETi) with activity in androgen signaling inhibitor (ASI) resistance models and canFormule :C19H19N5ODegré de pureté :98.94% - 99.76%Couleur et forme :SolidMasse moléculaire :333.39Oltipraz
CAS :Oltipraz (RP 35972) is a synthetic dithiolethione with potential chemopreventive and anti-angiogenic properties.Formule :C8H6N2S3Degré de pureté :98.79% - 99.77%Couleur et forme :SolidMasse moléculaire :226.34ZL0580
CAS :ZL0580 suppresses HIV by blocking Tat activation, halting transcription, and promoting repressive chromatin at the HIV promoter.Formule :C25H23F3N4O4SDegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :532.53NU6140
CAS :NU6140 is a selective inhibitor of CDK2-cyclin A (IC50, 0.41 μM).Formule :C23H30N6O2Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :422.52Ref: TM-T16359
2mg39,00€5mg60,00€10mg92,00€25mg177,00€50mg285,00€100mg414,00€200mg580,00€1mL*10mM (DMSO)67,00€VTP50469
CAS :VTP50469 is a highly selective and orally active small molecule inhibitor of the Menin-MLL protein-protein interaction.Cost-effective and quality-assured.Formule :C32H47FN6O4SDegré de pureté :98.31% - 99.55%Couleur et forme :SolidMasse moléculaire :630.82Ref: TM-T13336
1mg164,00€5mg334,00€10mg401,00€25mg560,00€50mg715,00€100mg964,00€1mL*10mM (DMSO)465,00€Glucosamine hydrochloride
CAS :Glucosamine hydrochloride (Chitosamine hydrochloride) is commonly used as a treatment for osteoarthritis, although its acceptance as a medical therapy varies.Formule :C6H13NO5·HClDegré de pureté :99.77%Couleur et forme :White Solid CrystallineMasse moléculaire :215.63N6-Cyclohexyladenosine
CAS :N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.Formule :C16H23N5O4Degré de pureté :99.92% - 99.98%Couleur et forme :SolidMasse moléculaire :349.38GNE-781
CAS :GNE-781: potent CBP inhibitor (IC50: 0.94 nM), also targets BRET/BRD4(1) (IC50: 6.2/5100 nM).Formule :C27H33F2N7O2Degré de pureté :99.25% - 99.64%Couleur et forme :SolidMasse moléculaire :525.59Ref: TM-T15405
1mg131,00€5mg281,00€10mg460,00€25mg765,00€50mg1.035,00€100mg1.404,00€1mL*10mM (DMSO)324,00€SNDX-5613
CAS :Revumenib (SNDX-5613) is a potent and selective oral inhibitor of menin-KMT2A interaction.Cost-effective and quality-assured.Formule :C32H47FN6O4SDegré de pureté :99.12% - 99.74%Couleur et forme :SolidMasse moléculaire :630.82Ref: TM-T12943
1mg73,00€2mg97,00€5mg160,00€10mg274,00€25mg542,00€50mg778,00€100mg1.074,00€1mL*10mM (DMSO)217,00€Tranylcypromine (2-PCPA) hydrochloride
CAS :Tranylcypromine (2-PCPA) HCl, a MAO inhibitor, treats major, dysthymic, and atypical depression.Formule :C9H11N·HClDegré de pureté :99.48% - 99.86%Couleur et forme :SolidMasse moléculaire :169.66Pulrodemstat benzenesulfonate
CAS :Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) is a potent and orally inhibitor of lysine specific demethylase-1 (LSD1) with anticancer effect.Formule :C30H29F2N5O5SDegré de pureté :97.67%Couleur et forme :SolidMasse moléculaire :609.64Ref: TM-T11882
1mg60,00€2mg86,00€5mg124,00€10mg188,00€25mg329,00€50mg490,00€100mg710,00€1mL*10mM (DMSO)170,00€Bendazol
CAS :Bendazol (Dibazol) is always used as the drug for hypertension and cerebral Angiospasm.Formule :C14H12N2Degré de pureté :98.7% - 99.87%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :208.26A-395
CAS :A-395 blocks PRC2 (EZH2-EED-SUZ12) interactions, strongly inhibiting the complex with an IC50 of 18 nM.Formule :C26H35FN4O2SDegré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :486.65Lin28-let-7a antagonist 1
CAS :Lin28-let-7a antagonist 1, with an IC50 of 4.03 μM for Lin28A-let-7a-1 interaction，and shows a clear antagonistic effect against the Lin28-let-7a interaction.Formule :C31H29N5O7Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :583.59Ref: TM-T11851
1mg96,00€5mg205,00€10mg313,00€25mg562,00€50mg845,00€100mg1.243,00€1mL*10mM (DMSO)266,00€Ilginatinib maleate
CAS :Ilginatinib maleate (NS-018 maleate) is a highly active and orally bioavailable inhibitor of JAK2.
Formule :C25H24FN7O4Degré de pureté :99.74% - 99.82%Couleur et forme :SolidMasse moléculaire :505.5Delgocitinib
CAS :Delgocitinib is a potent JAK inhibitor (IC50: 2.8-58 nM), treats inflammatory diseases, and is the first topical drug for atopic dermatitis.Formule :C16H18N6ODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :310.35Ref: TM-T15096
1mg160,00€5mg295,00€10mg462,00€25mg879,00€50mg1.341,00€100mg1.953,00€200mg2.628,00€1mL*10mM (DMSO)330,00€5-Azacytidine
CAS :5-Azacytidine (Ladakamycin) is a cytidine nucleoside analog, a DNA methylation inhibitor with specificity.Formule :C8H12N4O5Degré de pureté :98% - 99.79%Couleur et forme :Crystals From Methanol Physical Description White Crystalline Powder (Ntp 1992)Masse moléculaire :244.2Gusacitinib
CAS :Gusacitinib (ASN-002) (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 nM).Formule :C24H28N8O2Degré de pureté :98.06% - 99.94%Couleur et forme :SolidMasse moléculaire :460.53Ref: TM-T14331
1mg39,00€5mg84,00€10mg116,00€25mg178,00€50mg333,00€100mg495,00€200mg710,00€1mL*10mM (DMSO)110,00€MAT2A inhibitor 2
CAS :MAT2A inhibitor 2 is an inhibitor of methionine adenosyltransferase 2A (MAT2A).Formule :C18H24ClN3O3Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :365.85Golidocitinib
CAS :Golidocitinib (AZD4205) is a selective JAK1 inhibitor (IC50: 73 nM) and weakly inhibits JAK2/JAK3 (IC50: >14.7, >30 μM).Formule :C25H31N9O2Degré de pureté :98.87% - 99.88%Couleur et forme :SolidMasse moléculaire :489.57Centrinone
CAS :Centrinone (LCR-263) (LCR-263) is a reversible inhibitor of polo-like kinase 4 (PLK4; Ki:0.16 nM).Formule :C26H25F2N7O6S2Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :633.65JAK2 Inhibitor V
CAS :JAK2 Inhibitor V (JAK2 Inhibitor V Z3) is a novel specific inhibitor of Jak2, inhibiting Jak2-V617F and Jak2-WT autophosphorylation in a dose-dependent manner.Formule :C23H24N2ODegré de pureté :98.36% - 99.15%Couleur et forme :SolidMasse moléculaire :344.45Ref: TM-T3042
2mg37,00€5mg54,00€10mg80,00€25mg148,00€50mg259,00€100mg477,00€500mg1.063,00€1mL*10mM (DMSO)59,00€MK8722
CAS :MK8722 is an effective and systemic activator of pan-AMPK.Formule :C24H20ClN3O4Degré de pureté :98.08% - 99.8800%Couleur et forme :SolidMasse moléculaire :449.89Ref: TM-T16099
1mg34,00€2mg49,00€5mg74,00€10mg113,00€25mg215,00€50mg396,00€100mg585,00€1mL*10mM (DMSO)82,00€MS417
CAS :MS417 (GTPL7512) is an inhibitor of BET-specific BRD4(BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively), with weakFormule :C20H19ClN4O2SDegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :414.91L002
CAS :L002 is a potent inhibitor of acetyltransferase p300 with an IC50 of 1.98 μM, blocking histone and p53 acetylation, and may treat cardiac hypertrophy.Formule :C15H15NO5SDegré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :321.35PBIT
CAS :PBIT is a JARID1 inhibitor with IC50: 3 μM for JARID1B, 6 μM for JARID1A, and 4.9 μM for JARID1C.Formule :C14H11NOSDegré de pureté :99.61% - 99.83%Couleur et forme :SolidMasse moléculaire :241.31Ref: TM-T16435
1mg35,00€2mg50,00€5mg75,00€10mg105,00€25mg215,00€50mg340,00€100mg550,00€200mg780,00€1mL*10mM (DMSO)84,00€
