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Chromatine/Épigénétique

Chromatine/Épigénétique

Les inhibiteurs de la chromatine/épigénétique sont des composés qui modulent la structure et la fonction de la chromatine ou interfèrent avec les modifications épigénétiques, telles que la méthylation de l'ADN et la modification des histones. Ces inhibiteurs sont des outils essentiels pour étudier la régulation de l'expression génique et le rôle de l'épigénétique dans des maladies telles que le cancer, les troubles neurologiques et les anomalies du développement. En ciblant les processus épigénétiques, ces inhibiteurs peuvent modifier les schémas d'expression génique et offrir de nouvelles perspectives thérapeutiques. Chez CymitQuimica, nous offrons une large sélection d'inhibiteurs de la chromatine/épigénétique de haute qualité pour soutenir vos recherches en biologie moléculaire, génétique et épigénétique.

Sous-catégories appartenant à la catégorie "Chromatine/Épigénétique"

2613 produits trouvés pour "Chromatine/Épigénétique"

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produits par page.
  • Amodiaquine dihydrochloride dihydrate

    CAS :
    Amodiaquine dihydrochloride dihydrate (Amodiaquin hydrochloride) is an orally active 4-aminoquinoline derivative with antimalarial and anti-inflammatory effects
    Formule :C20H28Cl3N3O3
    Degré de pureté :99.97%
    Couleur et forme :Solid
    Masse moléculaire :464.82

    Ref: TM-T0381

    100mg
    37,00€
    500mg
    77,00€
    1mL*10mM (DMSO)
    40,00€
  • A-485

    CAS :
    A-485 is a p300/CBP histone acetyltransferase (HAT) inhibitor that inhibits p300 and CBP. A-485 has antitumor effects. Cost effective and quality assured.
    Formule :C25H24F4N4O5
    Degré de pureté :98.01% - 99.98%
    Couleur et forme :Solid
    Masse moléculaire :536.48

    Ref: TM-T14073

    1mg
    88,00€
    5mg
    159,00€
    10mg
    273,00€
    25mg
    339,00€
    50mg
    404,00€
    100mg
    698,00€
    1mL*10mM (DMSO)
    187,00€
  • Niraparib (R-enantiomer)

    CAS :

    Niraparib R-enantiomer (MK 4827 R-enantiomer) is an inhibitor of PARP1(IC50 of 2.4 nM).

    Formule :C19H20N4O
    Degré de pureté :99.83%
    Couleur et forme :Solid
    Masse moléculaire :320.39

    Ref: TM-T12064

    1mg
    37,00€
    5mg
    74,00€
    10mg
    97,00€
    25mg
    135,00€
    50mg
    168,00€
    100mg
    264,00€
  • BRD4 Inhibitor-10

    CAS :
    BRD4 Inhibitor-10 is an inhibitor of BRD4-BD1 (IC50: 8 nM).
    Formule :C25H27N5O2
    Degré de pureté :99.53%
    Couleur et forme :Solid
    Masse moléculaire :429.51

    Ref: TM-T14776

    1mg
    44,00€
    5mg
    92,00€
    10mg
    147,00€
    25mg
    285,00€
    50mg
    414,00€
    100mg
    583,00€
    200mg
    785,00€
    1mL*10mM (DMSO)
    100,00€
  • BVT948

    CAS :
    BVT948 is a protein tyrosine phosphatase (PTP) inhibitor.It can also inhibit lysine methyltransferase SETD8 (KMT5A) and several cytochrome P450 (P450) isoforms.
    Formule :C14H11NO3
    Degré de pureté :98.87%
    Couleur et forme :Solid
    Masse moléculaire :241.24

    Ref: TM-T14841

    1mg
    38,00€
    2mg
    49,00€
    5mg
    80,00€
    10mg
    104,00€
    25mg
    157,00€
    50mg
    210,00€
    100mg
    338,00€
    1mL*10mM (DMSO)
    88,00€
  • Bufexamac

    CAS :
    Bufexamac (Bufexamic acid) is a COX inhibitor for IFN-α release with anti-inflammatory, analgesic, and antipyretic action.
    Formule :C12H17NO3
    Degré de pureté :99.73%
    Couleur et forme :Acicular Crystal
    Masse moléculaire :223.27

    Ref: TM-T0867

    1g
    78,00€
    100mg
    33,00€
    200mg
    43,00€
    500mg
    54,00€
    1mL*10mM (DMSO)
    33,00€
  • Diperodon hydrochloride

    CAS :
    Diperodon hydrochloride (Diperocaine) is a local anesthetic that can be broken down by serolytic enzymes to produce local anesthetic effects.
    Formule :C22H28ClN3O4
    Degré de pureté :99.91%
    Couleur et forme :Solid
    Masse moléculaire :433.93

    Ref: TM-T0325

    1g
    92,00€
    100mg
    33,00€
    200mg
    49,00€
    500mg
    72,00€
  • PT-1

    CAS :
    PT-1 is an AMPKα1 activator that dose-dependently activates AMPK α1394, α1335, and α2398 and enhances AMPK phosphorylation.
    Formule :C23H16ClN3O6S
    Degré de pureté :99.62%
    Couleur et forme :Solid
    Masse moléculaire :497.91

    Ref: TM-T21984

    1mg
    42,00€
    5mg
    99,00€
    10mg
    157,00€
    25mg
    333,00€
    50mg
    539,00€
  • MOZ-IN-2

    CAS :

    MOZ-IN-2 is an protein MOZ inhibitor(IC50 of 125 μM).

    Formule :C17H13FN4O3S
    Degré de pureté :99.17%
    Couleur et forme :Solid
    Masse moléculaire :372.37

    Ref: TM-T12098

    2mg
    37,00€
    5mg
    60,00€
    10mg
    96,00€
    25mg
    188,00€
    50mg
    283,00€
    100mg
    432,00€
    500mg
    938,00€
  • Molidustat

    CAS :
    Molidustat (BAY 85-3934) 是新型HIF-PH 抑制剂,对PHD1(IC50:480 nM)、PHD2(IC50:280 nM)、PHD3(IC50:450 nM)。
    Formule :C13H14N8O2
    Degré de pureté :98.79%
    Couleur et forme :Solid
    Masse moléculaire :314.3

    Ref: TM-T2652

    1mg
    50,00€
    5mg
    92,00€
    10mg
    140,00€
    25mg
    192,00€
    50mg
    295,00€
    1mL*10mM (DMSO)
    101,00€
  • AES-135

    CAS :
    AES-135 is a potent HDAC inhibitor, inhibits HDAC3, HDAC6, HDAC11 (IC50s: 654, 190, and 636 nM) with anti-tumor activity.
    Formule :C33H29F6N3O5S
    Degré de pureté :97.72%
    Couleur et forme :Solid
    Masse moléculaire :693.66

    Ref: TM-T10255

    1mg
    79,00€
    5mg
    152,00€
    10mg
    250,00€
    25mg
    424,00€
    50mg
    583,00€
    100mg
    803,00€
    1mL*10mM (DMSO)
    225,00€
  • Tinengotinib

    CAS :
    Tinengotinib is a multikinase inhibitor that targets a series of kinases , including Aurora kinases A/B, JAK1/2, FGFR1/2/3, VEGFRs, and many other kinases.
    Formule :C20H19ClN6O
    Degré de pureté :99.05%
    Couleur et forme :Solid
    Masse moléculaire :394.86

    Ref: TM-T39718

    1mg
    60,00€
    5mg
    130,00€
    10mg
    200,00€
    25mg
    356,00€
    50mg
    557,00€
    1mL*10mM (DMSO)
    142,00€
  • EHP-101

    CAS :
    EHP-101 is a PPARγ/CB2 dual agonist with anti-inflammatory properties, inhibits fat formation, and combats diet-related obesity.
    Formule :C28H35NO3
    Degré de pureté :98.36%
    Couleur et forme :Solid
    Masse moléculaire :433.58

    Ref: TM-T13289

    1mg
    107,00€
    5mg
    227,00€
    10mg
    378,00€
    25mg
    620,00€
    50mg
    868,00€
    100mg
    1.169,00€
    1mL*10mM (DMSO)
    250,00€
  • PT2399

    CAS :
    PT2399, an oral HIF-2 inhibitor, blocks HIF-2α/1β dimerization, showing strong in vivo antitumor effects.
    Formule :C17H10F5NO4S
    Degré de pureté :98.8% - 99.45%
    Couleur et forme :Solid
    Masse moléculaire :419.32

    Ref: TM-T12675L

    1mg
    88,00€
    5mg
    212,00€
    10mg
    318,00€
    25mg
    575,00€
    50mg
    848,00€
    100mg
    1.189,00€
    1mL*10mM (DMSO)
    233,00€
  • Nicotinamide riboside

    CAS :

    Nicotinamide riboside increases NAD[+] levels and activates SIRT1 and SIRT3, culminating in enhanced oxidative metabolism and protection against high fat diet-

    Formule :C11H15N2O5
    Degré de pureté :98.82% - 99.58%
    Couleur et forme :Solid
    Masse moléculaire :255.25

    Ref: TM-T13795

    5mg
    55,00€
    200mg
    229,00€
  • N6-Cyclohexyladenosine

    CAS :
    N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.
    Formule :C16H23N5O4
    Degré de pureté :99.92% - 99.98%
    Couleur et forme :Solid
    Masse moléculaire :349.38

    Ref: TM-T12160

    10mg
    33,00€
    25mg
    58,00€
    50mg
    99,00€
    100mg
    147,00€
    200mg
    208,00€
    1mL*10mM (DMSO)
    33,00€
  • Phenelzine sulfate

    CAS :
    Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.
    Formule :C8H14N2O4S
    Degré de pureté :98.38% - 99.83%
    Couleur et forme :Solid
    Masse moléculaire :234.27

    Ref: TM-T12441

    1g
    168,00€
    50mg
    39,00€
    100mg
    52,00€
    500mg
    119,00€
    1mL*10mM (DMSO)
    57,00€
  • Acetaminophen

    CAS :
    Acetaminophen: pain reliever, fever reducer; mild anti-inflammatory. Risks: liver, kidney damage, blood cell effects.
    Formule :C8H9NO2
    Degré de pureté :99.85% - 99.99%
    Couleur et forme :Colourless Solid Crystalline
    Masse moléculaire :151.16

    Ref: TM-T0065

    500mg
    46,00€
  • Histone Acetyltransferase Inhibitor II

    CAS :
    Histone Acetyltransferase Inhibitor II is a selective and cell permeable inhibitor of p300 histone acetyltransferase(IC50 : 5 μM).with anti-acetylase activity
    Formule :C20H16Br2O3
    Degré de pureté :97.13%
    Couleur et forme :Solid
    Masse moléculaire :464.15

    Ref: TM-T11563

    1mg
    34,00€
    5mg
    66,00€
    10mg
    92,00€
    25mg
    187,00€
    50mg
    304,00€
    100mg
    487,00€
    1mL*10mM (DMSO)
    69,00€
  • Enarodustat

    CAS :
    Enarodustat (JTZ-951) is an orally active factor inhibitor of prolyl hydroxylase (EC50: 0.22 μM) and has the potential for renal anemia treatment.
    Formule :C17H16N4O4
    Degré de pureté :99.73% - 99.75%
    Couleur et forme :Solid
    Masse moléculaire :340.33

    Ref: TM-T15219

    1mg
    37,00€
    2mg
    52,00€
    5mg
    74,00€
    10mg
    109,00€
    25mg
    178,00€
    50mg
    295,00€
    100mg
    439,00€
    1mL*10mM (DMSO)
    86,00€
  • Roxadustat

    CAS :
    Roxadustat (FG-4592) is an orally bioavailable, hypoxia-inducible factor prolyl hydroxylase inhibitor (HIF-PHI), with potential anti-anemic activity.
    Formule :C19H16N2O5
    Degré de pureté :99% - 99.88%
    Couleur et forme :Solid
    Masse moléculaire :352.34

    Ref: TM-T2515

    5mg
    34,00€
    10mg
    50,00€
    25mg
    70,00€
    50mg
    92,00€
    100mg
    110,00€
    500mg
    259,00€
    1mL*10mM (DMSO)
    50,00€
  • AW68

    CAS :
    AW68 is a potential small molecule BRD4 inhibitor that prevents and treats BRD4-related diseases and can be used in cancer research.
    Formule :C22H21ClN6
    Degré de pureté :98.52% - 98.52%
    Couleur et forme :Soild
    Masse moléculaire :404.89

    Ref: TM-T10638L

    1mg
    175,00€
    5mg
    434,00€
    10mg
    622,00€
    25mg
    973,00€
  • Decitabine

    CAS :
    Decitabine (Deoxycytidine) is a deoxycytidine analog, a DNA methyltransferase inhibitor with oral activity.
    Formule :C8H12N4O4
    Degré de pureté :98.06% - 99.87%
    Couleur et forme :Physical Description Fine White Crystalline Powder Used As A Drug
    Masse moléculaire :228.21

    Ref: TM-T1508

    1g
    166,00€
    100mg
    39,00€
    500mg
    103,00€
    1mL*10mM (DMSO)
    44,00€
  • HDAC-IN-40

    CAS :
    HDAC-IN-40 is a potent alkoxyamide-based HDAC inhibitor with Ki of 60 nM and 30 nM for HDAC2 and HDAC6, respectively. HDAC-IN-40 had antitumor effects
    Formule :C15H22N2O6
    Degré de pureté :99.04%
    Couleur et forme :Soild
    Masse moléculaire :326.35

    Ref: TM-T60082

    1mg
    34,00€
    5mg
    75,00€
    10mg
    110,00€
    25mg
    245,00€
    50mg
    363,00€
    100mg
    515,00€
  • Tranylcypromine (2-PCPA) hydrochloride

    CAS :
    Tranylcypromine (2-PCPA) HCl, a MAO inhibitor, treats major, dysthymic, and atypical depression.
    Formule :C9H11N·HCl
    Degré de pureté :99.48% - 99.86%
    Couleur et forme :Solid
    Masse moléculaire :169.66

    Ref: TM-T1025

    1g
    104,00€
    200mg
    39,00€
    500mg
    80,00€
    1mL*10mM (DMSO)
    34,00€
  • MK8722

    CAS :
    MK8722 is an effective and systemic activator of pan-AMPK.
    Formule :C24H20ClN3O4
    Degré de pureté :98.08% - 99.8800%
    Couleur et forme :Solid
    Masse moléculaire :449.89

    Ref: TM-T16099

    1mg
    34,00€
    2mg
    49,00€
    5mg
    74,00€
    10mg
    113,00€
    25mg
    215,00€
    50mg
    396,00€
    100mg
    585,00€
    1mL*10mM (DMSO)
    82,00€
  • Ilginatinib maleate

    CAS :

    Ilginatinib maleate (NS-018 maleate) is a highly active and orally bioavailable inhibitor of JAK2.

    Formule :C25H24FN7O4
    Degré de pureté :99.74% - 99.82%
    Couleur et forme :Solid
    Masse moléculaire :505.5

    Ref: TM-T12266L

    1mg
    48,00€
    5mg
    97,00€
    10mg
    135,00€
    25mg
    190,00€
    50mg
    274,00€
    100mg
    393,00€
    200mg
    520,00€
  • MAK683

    CAS :
    MAK683 is an inhibitor of embryonic ectoderm development (EED) (IC50s: 59, 89, 26 nM in EED Alphascreen binding, LC-MS and ELISA assay).
    Formule :C20H17FN6O
    Degré de pureté :98.25% - 99.92%
    Couleur et forme :Solid
    Masse moléculaire :376.39

    Ref: TM-T15201

    1mg
    50,00€
    5mg
    102,00€
    10mg
    178,00€
    25mg
    389,00€
    50mg
    575,00€
    100mg
    802,00€
    500mg
    1.665,00€
    1mL*10mM (DMSO)
    89,00€
  • Levetiracetam

    CAS :
    Levetiracetam (SIB-S1) is a relatively unique anticonvulsant that is typically used in combination with other antiepileptic medications for partial onset
    Formule :C8H14N2O2
    Degré de pureté :99.67% - 99.86%
    Couleur et forme :White Crystalline Powder
    Masse moléculaire :170.21

    Ref: TM-T0192

    10mg
    34,00€
    25mg
    49,00€
    50mg
    60,00€
    100mg
    92,00€
    500mg
    230,00€
    1mL*10mM (DMSO)
    52,00€
  • MS417

    CAS :
    MS417 (GTPL7512) is an inhibitor of BET-specific BRD4(BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively), with weak
    Formule :C20H19ClN4O2S
    Degré de pureté :99.87%
    Couleur et forme :Solid
    Masse moléculaire :414.91

    Ref: TM-T16154

    1mg
    34,00€
    5mg
    66,00€
    10mg
    92,00€
    25mg
    145,00€
    50mg
    215,00€
    100mg
    319,00€
    200mg
    474,00€
  • Diflunisal

    CAS :
    Diflunisal (Dolobid) is a cyclooxygenase (COX) Inhibitor, used as an anti-inflammatory analgesic.
    Formule :C13H8F2O3
    Degré de pureté :98.92% - 99.42%
    Couleur et forme :Solid
    Masse moléculaire :250.20

    Ref: TM-T0808

    25mg
    34,00€
    50mg
    48,00€
    100mg
    63,00€
    200mg
    93,00€
    500mg
    138,00€
    1mL*10mM (DMSO)
    52,00€
  • DC-05

    CAS :
    DC-05 is an inhibitor of DNA methyltransferase 1 (DNMT1) (IC50 and a Kd: 10.3 μM and 1.09 μM, respectively).
    Formule :C25H25N3O
    Degré de pureté :98.95%
    Couleur et forme :Solid
    Masse moléculaire :383.49

    Ref: TM-T15080

    1mg
    66,00€
    5mg
    145,00€
    10mg
    236,00€
    25mg
    515,00€
    50mg
    858,00€
    100mg
    1.251,00€
    200mg
    1.684,00€
    1mL*10mM (DMSO)
    158,00€
  • NU6140

    CAS :
    NU6140 is a selective inhibitor of CDK2-cyclin A (IC50, 0.41 μM).
    Formule :C23H30N6O2
    Degré de pureté :98.33%
    Couleur et forme :Solid
    Masse moléculaire :422.52

    Ref: TM-T16359

    2mg
    39,00€
    5mg
    60,00€
    10mg
    92,00€
    25mg
    177,00€
    50mg
    285,00€
    100mg
    414,00€
    200mg
    580,00€
    1mL*10mM (DMSO)
    67,00€
  • Hydralazine hydrochloride

    CAS :
    Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.
    Formule :C8H9ClN4
    Degré de pureté :99.85% - 99.86%
    Couleur et forme :Yellow Crystals White Crystalline Solid
    Masse moléculaire :196.64

    Ref: TM-T1613

    1g
    99,00€
    200mg
    40,00€
    500mg
    75,00€
  • NI-42

    CAS :
    NI-42, a BRPFs inhibitor: IC50(BRPF1/2/3)=7.9/48/260 nM, Kd(BRPF1/2/3)=40/210/940 nM; selective for class IV BRDs.
    Formule :C18H15N3O3S
    Degré de pureté :99.18%
    Couleur et forme :Solid
    Masse moléculaire :353.39

    Ref: TM-T16321

    5mg
    43,00€
    10mg
    65,00€
    25mg
    119,00€
    50mg
    177,00€
    100mg
    278,00€
    1mL*10mM (DMSO)
    47,00€
  • Gusacitinib

    CAS :
    Gusacitinib (ASN-002) (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 nM).
    Formule :C24H28N8O2
    Degré de pureté :98.06% - 99.94%
    Couleur et forme :Solid
    Masse moléculaire :460.53

    Ref: TM-T14331

    1mg
    39,00€
    5mg
    84,00€
    10mg
    116,00€
    25mg
    178,00€
    50mg
    333,00€
    100mg
    495,00€
    200mg
    710,00€
    1mL*10mM (DMSO)
    110,00€
  • Centrinone

    CAS :
    Centrinone (LCR-263) (LCR-263) is a reversible inhibitor of polo-like kinase 4 (PLK4; Ki:0.16 nM).
    Formule :C26H25F2N7O6S2
    Degré de pureté :98.76%
    Couleur et forme :Solid
    Masse moléculaire :633.65

    Ref: TM-T14927

    1mg
    58,00€
    2mg
    80,00€
    5mg
    111,00€
    10mg
    177,00€
    50mg
    413,00€
    100mg
    605,00€
    1mL*10mM (DMSO)
    156,00€
  • Safingol hydrochloride

    CAS :
    Safingol hydrochloride (L-threo-dihydrosphingosine hydrochloride) is a PKC-specific inhibitor that inhibits PKC and PI3k and induces cancer cell death.
    Formule :C18H40ClNO2
    Degré de pureté :99.39% - 99.71%
    Couleur et forme :Soild
    Masse moléculaire :337.969

    Ref: TM-T83978

    1mg
    175,00€
    5mg
    434,00€
    10mg
    622,00€
    25mg
    973,00€
    50mg
    1.341,00€
    100mg
    1.765,00€
  • Flufenamic acid

    CAS :
    Flufenamic acid (Arlef) is an anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties.
    Formule :C14H10F3NO2
    Degré de pureté :98.68%
    Couleur et forme :White To Light Yellow Crystalline Powder
    Masse moléculaire :281.23

    Ref: TM-T0858

    50mg
    37,00€
    100mg
    49,00€
    200mg
    63,00€
    500mg
    88,00€
    1mL*10mM (DMSO)
    52,00€
  • CG347B

    CAS :
    CG347B is a selective inhibitor of HDAC6.
    Formule :C16H17N3O2
    Degré de pureté :98.34%
    Couleur et forme :Solid
    Masse moléculaire :283.33

    Ref: TM-T10777

    1mg
    33,00€
    5mg
    75,00€
    10mg
    110,00€
    25mg
    190,00€
    50mg
    290,00€
    100mg
    404,00€
    200mg
    568,00€
    1mL*10mM (DMSO)
    81,00€
  • PBIT

    CAS :
    PBIT is a JARID1 inhibitor with IC50: 3 μM for JARID1B, 6 μM for JARID1A, and 4.9 μM for JARID1C.
    Formule :C14H11NOS
    Degré de pureté :99.61% - 99.83%
    Couleur et forme :Solid
    Masse moléculaire :241.31

    Ref: TM-T16435

    1mg
    35,00€
    2mg
    50,00€
    5mg
    75,00€
    10mg
    105,00€
    25mg
    215,00€
    50mg
    340,00€
    100mg
    550,00€
    200mg
    780,00€
    1mL*10mM (DMSO)
    84,00€
  • Nimucitinib

    CAS :
    Nimucitinib is a Janus kinase (JAK) inhibitor that can be used to treat dry eye and promote tear production.
    Formule :C25H26F2N6O2
    Degré de pureté :99.58%
    Couleur et forme :Soild
    Masse moléculaire :480.51

    Ref: TM-T67907

    1mg
    96,00€
    2mg
    139,00€
    5mg
    227,00€
    10mg
    354,00€
    25mg
    653,00€
    50mg
    938,00€
    100mg
    1.454,00€
    500mg
    2.822,00€
  • Glucosamine

    CAS :

    Glucosamine (Chitosamine) is used as a dietary supplement. Glucosamine has pharmacological effects on osteoarthritis cartilage. High-Quality, Low-Cost!

    Formule :C6H13NO5
    Degré de pureté :99.8% - 99.8%
    Couleur et forme :Coa
    Masse moléculaire :179.17

    Ref: TM-T0429

    50mg
    55,00€
  • Pim-1 kinase inhibitor 8

    CAS :
    Pim-1 kinase inhibitor 8 is a Pim-1 kinase inhibitor with anticancer activity that inhibits cell migration and can be studied in breast cancer.
    Formule :C14H17N3O3
    Degré de pureté :99.81%
    Couleur et forme :Soild
    Masse moléculaire :275.3

    Ref: TM-T83627

    1mg
    38,00€
    5mg
    86,00€
    10mg
    124,00€
    25mg
    241,00€
    50mg
    388,00€
    100mg
    610,00€
    200mg
    827,00€
  • Golidocitinib

    CAS :
    Golidocitinib (AZD4205) is a selective JAK1 inhibitor (IC50: 73 nM) and weakly inhibits JAK2/JAK3 (IC50: >14.7, >30 μM).
    Formule :C25H31N9O2
    Degré de pureté :98.87% - 99.88%
    Couleur et forme :Solid
    Masse moléculaire :489.57

    Ref: TM-T10431

    1mg
    47,00€
    5mg
    92,00€
    10mg
    137,00€
    25mg
    234,00€
    50mg
    356,00€
    100mg
    580,00€
    1mL*10mM (DMSO)
    98,00€
  • dAURK-4 hydrochloride


    dAURK-4 hydrochloride, a derivative of Alisertib, functions as a potent and selective degrader of AURKA (Aurora A), exhibiting anticancer properties [1].
    Formule :C52H53Cl2FN8O12
    Degré de pureté :99.44%
    Couleur et forme :Solid
    Masse moléculaire :1071.93

    Ref: TM-T74100

    1mg
    104,00€
  • Valemetostat

    CAS :
    Valemetostat (DS-3201) is a first-in-class EZH1/2 dual inhibitor, which can be used to study T-cell lymphoma.Cost-effective and quality-assured.
    Formule :C26H34ClN3O4
    Degré de pureté :98.38% - 99.83%
    Couleur et forme :Solid
    Masse moléculaire :488.02

    Ref: TM-T13279L

    1mg
    89,00€
    5mg
    177,00€
    10mg
    313,00€
    25mg
    520,00€
    50mg
    742,00€
    100mg
    982,00€
    1mL*10mM (DMSO)
    197,00€
  • A-395

    CAS :
    A-395 blocks PRC2 (EZH2-EED-SUZ12) interactions, strongly inhibiting the complex with an IC50 of 18 nM.
    Formule :C26H35FN4O2S
    Degré de pureté :98.43%
    Couleur et forme :Solid
    Masse moléculaire :486.65

    Ref: TM-T10205

    1mg
    46,00€
    5mg
    93,00€
    10mg
    123,00€
    25mg
    197,00€
    50mg
    À demander
    1mL*10mM (DMSO)
    88,00€
  • Chloramphenicol

    CAS :

    Chloramphenicol (Chloromycetin) is a broad-spectrum antibiotic that inhibits the biosynthesis of bacterial proteins. Cost-effective and quality-assured.

    Formule :C11H12Cl2N2O5
    Degré de pureté :99.6% - 99.84%
    Couleur et forme :Needles Or Elongated Plates From Water Or Ethylene Dichloride Solid
    Masse moléculaire :323.13

    Ref: TM-T1205

    1g
    52,00€
    5g
    70,00€
    10g
    92,00€
    500mg
    48,00€
  • PROTAC BRD4 ligand-1

    CAS :
    PROTAC BRD4 ligand-1 is a ligand for BRD4 for Protac GNE-987 and an inhibitor of BET.
    Formule :C23H18F2N4O5S
    Degré de pureté :99.28% - 99.93%
    Couleur et forme :Solid
    Masse moléculaire :500.47

    Ref: TM-T12551

    1mg
    116,00€
    5mg
    281,00€
    10mg
    470,00€
    25mg
    888,00€
    50mg
    1.494,00€
    100mg
    2.152,00€
  • YPX-C-05

    CAS :
    YPX-C-05, an isohydroxamic acid derivative, is an HDAC inhibitor with vasodilatory and antihypertensive activity.CAS 번호134608-84-5
    Formule :C21H19N3O4
    Degré de pureté :98.09%
    Couleur et forme :Soild
    Masse moléculaire :377.39

    Ref: TM-T83639

    1mg
    175,00€
    5mg
    434,00€
    10mg
    622,00€
    25mg
    973,00€
    50mg
    1.341,00€
    100mg
    1.773,00€
  • BRD 4354

    CAS :
    BRD 4354 is an inhibitor of HDAC5 and HDAC9. For HDAC5 and HDAC9, the IC50s values are 0.85 and 1.88 μM, respectively.
    Formule :C21H23ClN4O
    Degré de pureté :99.86%
    Couleur et forme :Solid
    Masse moléculaire :382.89

    Ref: TM-T10602L

    1mg
    34,00€
    2mg
    44,00€
    5mg
    66,00€
    10mg
    92,00€
    25mg
    178,00€
    50mg
    308,00€
    100mg
    512,00€
    500mg
    1.071,00€
    1mL*10mM (DMSO)
    73,00€
  • BRD-6929

    CAS :
    BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.
    Formule :C19H17N3O2S
    Degré de pureté :98.01% - 99.05%
    Couleur et forme :Solid
    Masse moléculaire :351.42

    Ref: TM-T10603

    5mg
    48,00€
    10mg
    86,00€
    25mg
    166,00€
    50mg
    289,00€
    100mg
    419,00€
    200mg
    587,00€
    1mL*10mM (DMSO)
    49,00€
  • SNDX-5613

    CAS :
    Revumenib (SNDX-5613) is a potent and selective oral inhibitor of menin-KMT2A interaction.Cost-effective and quality-assured.
    Formule :C32H47FN6O4S
    Degré de pureté :99.12% - 99.74%
    Couleur et forme :Solid
    Masse moléculaire :630.82

    Ref: TM-T12943

    1mg
    73,00€
    2mg
    97,00€
    5mg
    160,00€
    10mg
    274,00€
    25mg
    542,00€
    50mg
    778,00€
    100mg
    1.074,00€
    1mL*10mM (DMSO)
    217,00€
  • Delcasertib

    CAS :
    Delcasertib (KAI-9803) is a potent and selective inhibitor of δ-protein kinase C (δPKC).
    Formule :C120H199N45O34S2
    Degré de pureté :99.96%
    Couleur et forme :Solid
    Masse moléculaire :2880.28

    Ref: TM-T11740

    1mg
    192,00€
    5mg
    485,00€
    10mg
    700,00€
    25mg
    1.063,00€
    50mg
    1.459,00€
    100mg
    1.963,00€
    1mL*10mM (DMSO)
    1.603,00€
  • CBP/p300-IN-3

    CAS :
    CBP/p300-IN-3 (P300/CBP-IN-3) is an inhibitor of p300/CBP histone acetyltransferase.
    Formule :C24H29N7O
    Degré de pureté :97.38% - 98.08%
    Couleur et forme :Solid
    Masse moléculaire :431.53

    Ref: TM-T12345

    1mg
    87,00€
    5mg
    177,00€
    10mg
    295,00€
    25mg
    447,00€
    50mg
    640,00€
    100mg
    893,00€
    500mg
    2.115,00€
    1mL*10mM (DMSO)
    203,00€
  • Miglitol

    CAS :
    Miglitol (BAY1099) is an alpha-Glucosidase Inhibitor with antihyperglycemic activity.
    Formule :C8H17NO5
    Degré de pureté :99.75% - 99.88%
    Couleur et forme :White To Pale-Yellow Powder Solid
    Masse moléculaire :207.22

    Ref: TM-T1529

    1g
    71,00€
    500mg
    47,00€
  • Tulmimetostat

    CAS :
    Tulmimetostat (CPI-0209) is an orally active EZH1/EZH2 inhibitor.Tulmimetostat has antitumor activity and is used in the study of ovarian cancer and advanced
    Formule :C28H36ClN3O5S
    Degré de pureté :98.04% - 99.872%
    Couleur et forme :Solid
    Masse moléculaire :562.12

    Ref: TM-T40199

    1mg
    34,00€
    5mg
    65,00€
    10mg
    92,00€
    25mg
    173,00€
    50mg
    260,00€
    100mg
    515,00€
  • WDR5-IN-6

    CAS :
    WDR5-IN-6 is a WDR5 inhibitor targeting the WBM locus.WDR5-IN-6 is highly synergistic with OICR-9429, a WDR5 inhibitor that targets the WIN locus.WDR5-IN-6
    Formule :C13H8Cl2N2O2S
    Degré de pureté :99.69%
    Couleur et forme :Soild
    Masse moléculaire :327.19

    Ref: TM-T77495

    1mg
    43,00€
    5mg
    93,00€
    10mg
    137,00€
    25mg
    266,00€
    50mg
    430,00€
    100mg
    687,00€
    500mg
    1.395,00€
  • Uzansertib phosphate

    CAS :
    Uzansertib phosphate (INCB053914 phosphate) is an orally active, ATP-competitive inhibitor of pan-PIM kinase, inhibiting PIM1, PIM2 and PIM3.
    Formule :C26H29F3N5O7P
    Degré de pureté :99.75% - 99.79%
    Couleur et forme :Solid
    Masse moléculaire :611.51

    Ref: TM-T12477

    1mg
    93,00€
    5mg
    205,00€
    10mg
    313,00€
    25mg
    562,00€
    50mg
    788,00€
    100mg
    1.099,00€
  • PKC β pseudosubstrate acetate


    PKC β pseudosubstrate acetate (PKC β pseudosubstrate acetate (172308-76-8 Free base)) is a selective cell-permeable inhibitor of PKC.
    Degré de pureté :95.42%
    Couleur et forme :Soild

    Ref: TM-TP1955L

    1mg
    163,00€
    5mg
    353,00€
    10mg
    480,00€
    25mg
    718,00€
    50mg
    945,00€
    100mg
    1.279,00€
    200mg
    1.728,00€
  • TRIM24/BRPF1-IN-2

    CAS :
    TRIM24/BRPF1-IN-2 is a TRIM24/BRPF1 dual inhibitor with anticancer activity that inhibits the proliferation of prostate cancer cells.
    Formule :C20H22N2O4S
    Degré de pureté :98.69% - 99.13%
    Couleur et forme :Soild
    Masse moléculaire :386.47

    Ref: TM-T74271

    1mg
    301,00€
    5mg
    873,00€
    50mg
    À demander
  • (R)​-​CR8

    CAS :

    (R)-CR8 ((R)-Isomer) is a potent and selective CDK inhibitor.

    Formule :C24H29N7O
    Degré de pureté :98.41%
    Couleur et forme :Solid
    Masse moléculaire :431.53

    Ref: TM-T12617L

    1mg
    66,00€
    5mg
    144,00€
    10mg
    210,00€
    25mg
    283,00€
    50mg
    432,00€
    100mg
    612,00€
  • SMARCA-BD ligand 1 for Protac

    CAS :
    SMARCA-BD ligand 1 for Protac is a compound capable of binding to SMARCA2, the BAF ATPase subunit, based on the Protac technology for degrading SMARCA2
    Formule :C14H17N5O
    Degré de pureté :99.93%
    Couleur et forme :Solid
    Masse moléculaire :271.32

    Ref: TM-T13848

    1mg
    63,00€
    5mg
    137,00€
    10mg
    215,00€
    25mg
    364,00€
    50mg
    513,00€
    100mg
    700,00€
    200mg
    954,00€
  • Chitosan oligosaccharide

    CAS :
    Chitosan oligosaccharide (COS) is an oligomer of β-(1→4)-linked D-glucosamine.
    Formule :C12H24N2O9
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :340.327

    Ref: TM-T10789

    1g
    52,00€
  • L-2-Hydroxyglutaric acid disodium

    CAS :
    L-2-Hydroxyglutaric acid disodium may affect epigenetics and contribute to renal cancer, inhibiting Mi-CK (Km 2.52 mM, Ki 11.13 mM).
    Formule :C5H6Na2O5
    Degré de pureté :99.92%
    Couleur et forme :Solid
    Masse moléculaire :192.08

    Ref: TM-T13748

    10mg
    50,00€
    25mg
    86,00€
    50mg
    127,00€
    100mg
    167,00€
  • ZEN-3694

    CAS :
    ZEN-3694 (ZEN 3694) is a bromo-structural domain extra-terminal inhibitor (BETi) with activity in androgen signaling inhibitor (ASI) resistance models and can
    Formule :C19H19N5O
    Degré de pureté :98.94% - 99.76%
    Couleur et forme :Solid
    Masse moléculaire :333.39

    Ref: TM-T29214

    1mg
    63,00€
    5mg
    137,00€
    10mg
    215,00€
    25mg
    394,00€
    50mg
    628,00€
    100mg
    888,00€
    500mg
    1.783,00€
  • ZL0580

    CAS :
    ZL0580 suppresses HIV by blocking Tat activation, halting transcription, and promoting repressive chromatin at the HIV promoter.
    Formule :C25H23F3N4O4S
    Degré de pureté :99.70%
    Couleur et forme :Solid
    Masse moléculaire :532.53

    Ref: TM-T13974

    1mg
    38,00€
    5mg
    80,00€
    10mg
    114,00€
    25mg
    178,00€
    50mg
    269,00€
    100mg
    399,00€
    1mL*10mM (DMSO)
    92,00€
  • TAK-901

    CAS :
    TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid Metaplasia, and Advanced Solid Tumors, among others
    Formule :C28H32N4O3S
    Degré de pureté :99.02% - 99.59%
    Couleur et forme :Solid
    Masse moléculaire :504.64

    Ref: TM-T2709

    1mg
    35,00€
    5mg
    70,00€
    10mg
    104,00€
    25mg
    202,00€
    50mg
    329,00€
    100mg
    525,00€
    200mg
    748,00€
    1mL*10mM (DMSO)
    79,00€
  • Brepocitinib P-Tosylate

    CAS :
    Brepocitinib P-Tosylate (PF-06700841 P-Tosylate) is a potent dual inhibitor of Janus kinase 1 (JAK1) and TYK2 (IC50s of 17 nM and 23 nM, respectively).
    Formule :C25H29F2N7O4S
    Degré de pureté :99.82% - 99.97%
    Couleur et forme :Solid
    Masse moléculaire :561.6

    Ref: TM-T12427

    1mg
    34,00€
    5mg
    66,00€
    10mg
    99,00€
    25mg
    205,00€
    50mg
    371,00€
    100mg
    595,00€
    1mL*10mM (DMSO)
    82,00€
  • Bendazol

    CAS :
    Bendazol (Dibazol) is always used as the drug for hypertension and cerebral Angiospasm.
    Formule :C14H12N2
    Degré de pureté :98.7% - 99.87%
    Couleur et forme :White Or Almost White Crystalline Powder
    Masse moléculaire :208.26

    Ref: TM-T1322

    200mg
    33,00€
    1mL*10mM (DMSO)
    33,00€
  • Albendazole

    CAS :
    Albendazole (SKF-62979) is used as a drug indicated for the treatment of a variety of worm infestations.
    Formule :C12H15N3O2S
    Degré de pureté :98.21% - 98.76%
    Couleur et forme :Colorless Crystals Solid
    Masse moléculaire :265.33

    Ref: TM-T1152

    1g
    84,00€
    50mg
    43,00€
    100mg
    50,00€
    500mg
    58,00€
    1mL*10mM (DMSO)
    44,00€
  • Delgocitinib

    CAS :
    Delgocitinib is a potent JAK inhibitor (IC50: 2.8-58 nM), treats inflammatory diseases, and is the first topical drug for atopic dermatitis.
    Formule :C16H18N6O
    Degré de pureté :99.95%
    Couleur et forme :Solid
    Masse moléculaire :310.35

    Ref: TM-T15096

    1mg
    160,00€
    5mg
    295,00€
    10mg
    462,00€
    25mg
    879,00€
    50mg
    1.341,00€
    100mg
    1.953,00€
    200mg
    2.628,00€
    1mL*10mM (DMSO)
    330,00€
  • 5-Azacytidine

    CAS :
    5-Azacytidine (Ladakamycin) is a cytidine nucleoside analog, a DNA methylation inhibitor with specificity.
    Formule :C8H12N4O5
    Degré de pureté :98% - 99.79%
    Couleur et forme :Crystals From Methanol Physical Description White Crystalline Powder (Ntp 1992)
    Masse moléculaire :244.2

    Ref: TM-T1339

    50mg
    37,00€
    100mg
    50,00€
    200mg
    62,00€
    500mg
    94,00€
    1mL*10mM (DMSO)
    52,00€
  • mTOR/HDAC-IN-1 HCl


    mTOR/HDAC-IN-1 HCl,a dual inhibitor of mTOR and HDAC with potential anti-inflammatory, anti-proliferative, autophagic and apoptosis-inducing effects for cancer
    Formule :C23H24ClN11O3
    Degré de pureté :99.56%
    Couleur et forme :Soild
    Masse moléculaire :537.96

    Ref: TM-T63399L

    1mg
    175,00€
    5mg
    434,00€
    10mg
    622,00€
    25mg
    973,00€
    50mg
    1.481,00€
  • EML 425

    CAS :
    EML 425 is a potent and selective inhibitor of CREB binding protein (CBP)/p300 (IC50s: 2.9 and 1.1 μM, respectively).
    Formule :C27H24N2O4
    Degré de pureté :97.6%
    Couleur et forme :Solid
    Masse moléculaire :440.49

    Ref: TM-T15216

    5mg
    42,00€
    10mg
    67,00€
    25mg
    129,00€
    50mg
    187,00€
    100mg
    276,00€
    200mg
    391,00€
    1mL*10mM (DMSO)
    46,00€
  • BRM/BRG1 ATP Inhibitor-1

    CAS :
    BRM/BRG1 ATP Inhibitor-1 is an allosteric dual Brahma homolog (BRM)/SWI/SNF related matrix-associated actin-dependent regulator of chromatin subfamily A member
    Formule :C11H9F3N4O2S
    Degré de pureté :98.17% - 99.84%
    Couleur et forme :Solid
    Masse moléculaire :318.27

    Ref: TM-T10616

    1mg
    167,00€
    5mg
    409,00€
    10mg
    615,00€
    25mg
    1.063,00€
    50mg
    1.558,00€
    100mg
    2.187,00€
    1mL*10mM (DMSO)
    442,00€
  • L002

    CAS :
    L002 is a potent inhibitor of acetyltransferase p300 with an IC50 of 1.98 μM, blocking histone and p53 acetylation, and may treat cardiac hypertrophy.
    Formule :C15H15NO5S
    Degré de pureté :98.59%
    Couleur et forme :Solid
    Masse moléculaire :321.35

    Ref: TM-T11807

    2mg
    38,00€
    5mg
    56,00€
    10mg
    84,00€
    25mg
    167,00€
    50mg
    309,00€
    100mg
    510,00€
    1mL*10mM (DMSO)
    63,00€
  • MC3482

    CAS :
    MC3482 is a specific inhibitor of sirtuin5 (SIRT5).
    Formule :C33H38N4O8
    Degré de pureté :98% - 99.90%
    Couleur et forme :Soild
    Masse moléculaire :618.68

    Ref: TM-T11962

    1mg
    50,00€
    2mg
    71,00€
    5mg
    105,00€
    10mg
    170,00€
    25mg
    268,00€
    50mg
    423,00€
    100mg
    685,00€
    500mg
    1.378,00€
  • Abexinostat

    CAS :
    Abexinostat (PCI-24781) is a pan-HDAC inhibitor, strongest on HDAC1; less so on HDACs 2, 3, 6, 10. Very select for HDAC8. In Phase 1/2 trials.
    Formule :C21H23N3O5
    Degré de pureté :98.19% - 98.43%
    Couleur et forme :Solid
    Masse moléculaire :397.42

    Ref: TM-T0431

    1mg
    37,00€
    5mg
    66,00€
    10mg
    102,00€
    25mg
    172,00€
    50mg
    309,00€
    100mg
    485,00€
  • SIRT-IN-2

    CAS :
    SIRT-IN-2 is a potent SIRT1/2/3 inhibitor(IC50s of 4, 1, 7 μM, respectively).
    Formule :C15H21N5O3S2
    Degré de pureté :98.26%
    Couleur et forme :Solid
    Masse moléculaire :383.49

    Ref: TM-T12919

    1mg
    92,00€
    5mg
    215,00€
    10mg
    344,00€
    25mg
    587,00€
    50mg
    803,00€
    100mg
    1.099,00€
    200mg
    1.468,00€
    1mL*10mM (DMSO)
    236,00€
  • A-3 hydrochloride

    CAS :
    A-3 hydrochloride: potent, reversible kinase antagonist; permeable; inhibits PKC, CKI, PKA, CKII, MLCK; Ki: 4.3-80 μM.
    Formule :C12H14Cl2N2O2S
    Degré de pureté :99.32%
    Couleur et forme :Solid
    Masse moléculaire :321.22

    Ref: TM-T14069

    1mg
    34,00€
    5mg
    63,00€
    10mg
    90,00€
    25mg
    161,00€
    50mg
    260,00€
    100mg
    416,00€
    500mg
    888,00€
    1mL*10mM (DMSO)
    95,00€
  • Cyproheptadine hydrochloride sesquihydrate

    CAS :
    Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.
    Formule :C21H24ClNO
    Degré de pureté :99.77% - >99.99%
    Couleur et forme :White To Slightly Yellowish Crystalline Solid
    Masse moléculaire :341.88

    Ref: TM-T0174

    500mg
    33,00€
  • Citric acid trilithium salt tetrahydrate

    CAS :
    Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) , the active component of Lithium, is a medicine used in the therapy of
    Formule :C6H13Li3O11
    Degré de pureté :99.88%
    Couleur et forme :White Crystalline Powder
    Masse moléculaire :281.98

    Ref: TM-T0256

    1g
    33,00€
  • SYP-5

    CAS :
    SYP-5 is a novel inhibitor of HIF-1, suppresses tumor cells invasion and angiogenesis.
    Formule :C18H16O3S
    Degré de pureté :98.31%
    Couleur et forme :Solid
    Masse moléculaire :312.38

    Ref: TM-T13050

    1mg
    34,00€
    5mg
    63,00€
    10mg
    94,00€
    25mg
    178,00€
    50mg
    286,00€
    100mg
    444,00€
    1mL*10mM (DMSO)
    71,00€
  • M-89

    CAS :

    M-89, a potent menin inhibitor (Kd 1.4 nM), disrupts Menin-MLL interaction, offering possible MLL leukemia treatment.

    Formule :C37H47N5O4S
    Degré de pureté :98.38%
    Couleur et forme :Solid
    Masse moléculaire :657.87

    Ref: TM-T11925

    1mg
    166,00€
    5mg
    406,00€
    10mg
    562,00€
    25mg
    825,00€
    50mg
    1.121,00€
    100mg
    1.549,00€
  • Dehydrocorydaline chloride

    CAS :
    Dehydrocorydaline chloride (13-Methylpalmatine chloride) is an alkaloid with anti-inflammatory and anti-cancer activity. Can improve the activation of p38 MAPK.
    Formule :C22H24ClNO4
    Degré de pureté :99.53%
    Couleur et forme :Solid
    Masse moléculaire :401.88

    Ref: TM-T10990

    1mg
    55,00€
    5mg
    105,00€
    10mg
    152,00€
    25mg
    250,00€
    50mg
    375,00€
    100mg
    533,00€
    1mL*10mM (DMSO)
    117,00€
  • RBN-2397

    CAS :
    RBN-2397 is a potent, selective and orally active accross species NAD+ competitive PARP7 inhibitor with IC50 less than 3 nM.
    Formule :C20H23F6N7O3
    Degré de pureté :98.48% - 99.8%
    Couleur et forme :Solid
    Masse moléculaire :523.43

    Ref: TM-T12695

    1mg
    90,00€
    2mg
    132,00€
    5mg
    215,00€
    10mg
    349,00€
    25mg
    708,00€
    50mg
    888,00€
    100mg
    1.224,00€
    200mg
    1.648,00€
    1mL*10mM (DMSO)
    248,00€
  • FIDAS-3

    CAS :
    FIDAS-3, a stilbene derivative and potent Wnt inhibitor with an IC50 of 4.9 μM for methionine S-adenosyltransferase 2A (MAT2A), exhibits anticancer activities
    Formule :C16H15F2N
    Degré de pureté :97.75%
    Couleur et forme :Solid
    Masse moléculaire :259.29

    Ref: TM-T11284

    5mg
    49,00€
    10mg
    73,00€
    25mg
    127,00€
    50mg
    182,00€
    100mg
    264,00€
    200mg
    354,00€
    1mL*10mM (DMSO)
    48,00€
  • Inobrodib

    CAS :
    Inobrodib (CBP-IN-1) is a potent inhibitor of p300/CBP bromodomain.
    Formule :C30H32F2N4O3
    Degré de pureté :98.91% - 99.18%
    Couleur et forme :Solid
    Masse moléculaire :534.6

    Ref: TM-T10717

    1mg
    66,00€
    2mg
    96,00€
    5mg
    144,00€
    10mg
    250,00€
    25mg
    528,00€
    50mg
    755,00€
    100mg
    1.018,00€
    1mL*10mM (DMSO)
    170,00€
  • Dihydro-5-azacytidine FA


    Dihydro-5-azacytidine FA (DHAC) is a pyrimidine analog that has antitumor activity, inhibits cell growth, inhibits DNA methylation, and may be used in the study of malignant mesothelioma.
    Formule :C9H16N4O7
    Degré de pureté :>99.99%
    Couleur et forme :Solid
    Masse moléculaire :292.25

    Ref: TM-T40713L

    1mg
    118,00€
    5mg
    283,00€
    10mg
    405,00€
    25mg
    622,00€
  • N-Desmethyltamoxifen hydrochloride

    CAS :
    N-Desmethyltamoxifen hydrochloride is the major tamoxifen metabolite in humans.
    Formule :C25H28ClNO
    Degré de pureté :99.15%
    Couleur et forme :Solid
    Masse moléculaire :393.95

    Ref: TM-T12148

    5mg
    34,00€
    10mg
    52,00€
    25mg
    92,00€
    50mg
    138,00€
    100mg
    202,00€
    1mL*10mM (DMSO)
    38,00€
  • GNE-781

    CAS :
    GNE-781: potent CBP inhibitor (IC50: 0.94 nM), also targets BRET/BRD4(1) (IC50: 6.2/5100 nM).
    Formule :C27H33F2N7O2
    Degré de pureté :99.25% - 99.64%
    Couleur et forme :Solid
    Masse moléculaire :525.59

    Ref: TM-T15405

    1mg
    131,00€
    5mg
    281,00€
    10mg
    460,00€
    25mg
    765,00€
    50mg
    1.035,00€
    100mg
    1.404,00€
    1mL*10mM (DMSO)
    324,00€
  • Glucosamine hydrochloride

    CAS :
    Glucosamine hydrochloride (Chitosamine hydrochloride) is commonly used as a treatment for osteoarthritis, although its acceptance as a medical therapy varies.
    Formule :C6H13NO5·HCl
    Degré de pureté :99.77%
    Couleur et forme :White Solid Crystalline
    Masse moléculaire :215.63

    Ref: TM-T2941

    1g
    33,00€
    5g
    44,00€
  • Pulrodemstat benzenesulfonate

    CAS :
    Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) is a potent and orally inhibitor of lysine specific demethylase-1 (LSD1) with anticancer effect.
    Formule :C30H29F2N5O5S
    Degré de pureté :97.67%
    Couleur et forme :Solid
    Masse moléculaire :609.64

    Ref: TM-T11882

    1mg
    60,00€
    2mg
    86,00€
    5mg
    124,00€
    10mg
    188,00€
    25mg
    329,00€
    50mg
    490,00€
    100mg
    710,00€
    1mL*10mM (DMSO)
    170,00€
  • Ziftomenib

    CAS :
    Ziftomenib (KO-539) is an inhibitor of menin-MLL interaction with antitumor activity and can be used to study leukemia.
    Formule :C33H42F3N9O2S2
    Degré de pureté :99.65% - 99.99%
    Couleur et forme :Solid
    Masse moléculaire :717.871

    Ref: TM-T39585

    1mg
    107,00€
    5mg
    258,00€
    10mg
    353,00€
    25mg
    578,00€
    50mg
    888,00€
    100mg
    1.314,00€
    200mg
    1.773,00€
  • Lin28-let-7a antagonist 1

    CAS :
    Lin28-let-7a antagonist 1, with an IC50 of 4.03 μM for Lin28A-let-7a-1 interaction,and shows a clear antagonistic effect against the Lin28-let-7a interaction.
    Formule :C31H29N5O7
    Degré de pureté :99.44%
    Couleur et forme :Solid
    Masse moléculaire :583.59

    Ref: TM-T11851

    1mg
    96,00€
    5mg
    205,00€
    10mg
    313,00€
    25mg
    562,00€
    50mg
    845,00€
    100mg
    1.243,00€
    1mL*10mM (DMSO)
    266,00€
  • HIF-2α-IN-2

    CAS :
    HIF-2α-IN-2 is a hypoxia-inducible factor (HIF-2α) inhibitor (IC50: 16 nM in scintillation proximity assay).
    Formule :C17H13F2NO4S
    Degré de pureté :99.24%
    Couleur et forme :Solid
    Masse moléculaire :365.35

    Ref: TM-T11561

    1mg
    52,00€
    5mg
    89,00€
    10mg
    123,00€
    25mg
    205,00€
    50mg
    296,00€
    100mg
    411,00€
    1mL*10mM (DMSO)
    99,00€
  • Tilorone dihydrochloride

    CAS :

    Tilorone dihydrochloride is an orally active interferon inducer, and has antineoplastic and anti-inflammatory actions.

    Formule :C25H36Cl2N2O3
    Degré de pureté :98% - 99.86%
    Couleur et forme :Orange Yellow Crystal Powder
    Masse moléculaire :483.47

    Ref: TM-T0244

    50mg
    40,00€
    100mg
    52,00€
    200mg
    94,00€
  • EBI-2511

    CAS :
    EBI-2511 is a highly potent and orally active inhibitor of EZH2 (IC50: 6 nM in Pfeffiera cell lines).
    Formule :C34H48N4O4
    Degré de pureté :99.74%
    Couleur et forme :Solid
    Masse moléculaire :576.77

    Ref: TM-T15194

    1mg
    57,00€
    5mg
    120,00€
    10mg
    187,00€
    25mg
    354,00€
    50mg
    550,00€
    100mg
    782,00€
    200mg
    1.035,00€
  • Deferoxamine Mesylate

    CAS :
    Deferoxamine Mesylate (DFOM) is an iron chelator and iron death inhibitor.
    Formule :C26H52N6O11S
    Degré de pureté :94.68% - 99.8%
    Couleur et forme :Solid
    Masse moléculaire :656.79

    Ref: TM-T1637

    50mg
    34,00€
    100mg
    50,00€
    500mg
    81,00€
    1mL*10mM (DMSO)
    44,00€
  • Ilginatinib

    CAS :
    Ilginatinib (NS-018) is a highly active and orally bioavailable inhibitor of JAK2.
    Formule :C21H20FN7
    Degré de pureté :98.4% - 99.01%
    Couleur et forme :Solid
    Masse moléculaire :389.43

    Ref: TM-T12266

    1mg
    60,00€
    5mg
    131,00€
    10mg
    177,00€
    25mg
    259,00€
    50mg
    371,00€
    100mg
    532,00€
    200mg
    705,00€
    1mL*10mM (DMSO)
    126,00€
  • BMS-986158

    CAS :
    BMS-986158: BET inhibitor, IC50 of 6.6 nM in SCLC, 5 nM in TNBC cells.
    Formule :C30H33N5O2
    Degré de pureté :98.78%
    Couleur et forme :Solid
    Masse moléculaire :495.62

    Ref: TM-T14685

    1mg
    87,00€
    5mg
    259,00€
    10mg
    465,00€
    25mg
    745,00€
    50mg
    1.026,00€
    100mg
    1.388,00€
    1mL*10mM (DMSO)
    283,00€
  • FIDAS-5

    CAS :
    FIDAS-5 is an orally active methionine adenosyltransferase 2A (MAT2A) inhibitor with an IC50 of 2.1 μM. Cost-effective and quality-assured.
    Formule :C15H13ClFN
    Degré de pureté :98.3% - 99.17%
    Couleur et forme :Solid
    Masse moléculaire :261.72

    Ref: TM-T11285

    1mg
    56,00€
    2mg
    80,00€
    5mg
    110,00€
    10mg
    177,00€
    25mg
    314,00€
    50mg
    485,00€
    100mg
    700,00€
    500mg
    1.341,00€
  • 1-Naphthohydroxamic acid

    CAS :
    1-Naphthohydroxamic acid (Compound 2) is a potent and selective HDAC8 inhibitor with an IC50 of 14 μM, and it is more selectively for HDAC8 than class I HDAC1
    Formule :C11H9NO2
    Degré de pureté :99.19%
    Couleur et forme :Solid
    Masse moléculaire :187.19

    Ref: TM-T13996

    5mg
    33,00€
    10mg
    60,00€
    25mg
    108,00€
    50mg
    200,00€
    100mg
    299,00€
    200mg
    430,00€
    1mL*10mM (DMSO)
    38,00€
  • Hydroxycitric acid tripotassium hydrate

    CAS :
    Hydroxycitric acid tripotassium hydrate (Potassium citrate monohydrate) effectively inhibits HIF, has antioxidation, anti-inflammation, and anti-tumor effects.
    Formule :C6H7K3O8
    Degré de pureté :99.85%
    Couleur et forme :White Solid Crystalline
    Masse moléculaire :324.41

    Ref: TM-T11589

    1g
    46,00€
    5g
    63,00€
    10g
    84,00€
    500mg
    33,00€
  • LIN28 inhibitor LI71

    CAS :
    LIN28 inhibitor LI71 is a potent and cell-permeable LIN28 inhibitor, which abolishes LIN28-mediated oligouridylation with an IC50 of 7 uM.
    Formule :C21H21NO3
    Degré de pureté :95.88%
    Couleur et forme :Solid
    Masse moléculaire :335.4

    Ref: TM-T11850

    1mg
    107,00€
    5mg
    255,00€
    10mg
    414,00€
    25mg
    745,00€
    50mg
    1.063,00€
    100mg
    1.459,00€
    1mL*10mM (DMSO)
    341,00€
  • Fenbendazole

    CAS :
    Fenbendazole (Fenbendazol) is an antinematodal benzimidazole used in veterinary medicine.
    Formule :C15H13N3O2S
    Degré de pureté :99.74%
    Couleur et forme :White To Yellowish Powder
    Masse moléculaire :299.35

    Ref: TM-T1141

    50mg
    37,00€
    100mg
    52,00€
    200mg
    59,00€
    500mg
    85,00€
    1mL*10mM (DMSO)
    52,00€
  • VTP50469

    CAS :
    VTP50469 is a highly selective and orally active small molecule inhibitor of the Menin-MLL protein-protein interaction.Cost-effective and quality-assured.
    Formule :C32H47FN6O4S
    Degré de pureté :98.31% - 99.55%
    Couleur et forme :Solid
    Masse moléculaire :630.82

    Ref: TM-T13336

    1mg
    164,00€
    5mg
    334,00€
    10mg
    401,00€
    25mg
    560,00€
    50mg
    715,00€
    100mg
    964,00€
    1mL*10mM (DMSO)
    465,00€
  • T-3775440 hydrochloride

    CAS :
    T-3775440 hydrochloride is an irreversible inhibitor of lysine-specific histone demethylase (LSD1)(IC50 : 2.1 nM).
    Formule :C18H23ClN4O
    Degré de pureté :99.88%
    Couleur et forme :Solid
    Masse moléculaire :346.85

    Ref: TM-T13055

    1mg
    92,00€
    2mg
    118,00€
    5mg
    192,00€
    10mg
    289,00€
    25mg
    485,00€
    50mg
    663,00€
    100mg
    893,00€
    1mL*10mM (DMSO)
    212,00€
  • ODM-207

    CAS :
    ODM-207 (BET-IN-4) is a potent BRD4 inhibitor.
    Formule :C22H21N3O3
    Degré de pureté :99.75%
    Couleur et forme :Solid
    Masse moléculaire :375.42

    Ref: TM-T10521

    1mg
    44,00€
    5mg
    92,00€
    10mg
    133,00€
    25mg
    235,00€
    50mg
    339,00€
    100mg
    480,00€
    200mg
    660,00€
    1mL*10mM (DMSO)
    90,00€
  • Oltipraz

    CAS :
    Oltipraz (RP 35972) is a synthetic dithiolethione with potential chemopreventive and anti-angiogenic properties.
    Formule :C8H6N2S3
    Degré de pureté :98.79% - 99.77%
    Couleur et forme :Solid
    Masse moléculaire :226.34

    Ref: TM-T0153

    5mg
    34,00€
    10mg
    52,00€
    25mg
    73,00€
    50mg
    93,00€
    100mg
    117,00€
    200mg
    149,00€
    1mL*10mM (DMSO)
    52,00€
  • MS31 trihydrochloride (2366264-12-0 free base)


    MS31 trihydrochloride (2366264-12-0 free base) is a potent, highly affinity and selective fragment-like methyllysine reader protein spindlin 1 (SPIN1) inhibitor
    Formule :C20H30Cl3N3O2
    Degré de pureté :99.69%
    Couleur et forme :Solid
    Masse moléculaire :450.83

    Ref: TM-T12111L

    1mg
    185,00€
    5mg
    369,00€
    10mg
    542,00€
    25mg
    867,00€
    50mg
    1.153,00€
    100mg
    1.584,00€
    1mL*10mM (DMSO)
    379,00€
  • Curcumin

    CAS :
    Curcumin (Natural Yellow 3) is a phenolic natural product, an inhibitor of histone acetyltransferase p300/CREB (IC50=25 μM) with specificity.
    Formule :C21H20O6
    Degré de pureté :95% - 98.98%
    Couleur et forme :Orange-Yellow Crystal Powder; Gives Brownish-Red Color With Alkali; Light-Yellow Color With Acids Physical Description Orange-Yellow Needles (Ntp 1992)
    Masse moléculaire :368.38

    Ref: TM-T1516

    1g
    116,00€
    5g
    187,00€
    50mg
    44,00€
    100mg
    55,00€
    500mg
    94,00€
    1mL*10mM (DMSO)
    55,00€
  • Ilginatinib hydrochloride

    CAS :
    Ilginatinib hydrochloride (NS-018 hydrochloride) is a highly active and orally bioavailable inhibitor of JAK2.
    Formule :C21H21ClFN7
    Degré de pureté :99.55%
    Couleur et forme :Solid
    Masse moléculaire :425.89

    Ref: TM-T12266L2

    1mg
    70,00€
    5mg
    150,00€
    10mg
    215,00€
    25mg
    358,00€
    50mg
    517,00€
    100mg
    707,00€
    200mg
    973,00€
    1mL*10mM (DMSO)
    166,00€
  • N-(3-Aminopropyl)cyclohexylamine

    CAS :
    N-(3-Aminopropyl)cyclohexylamine inhibits spermine synthase; used in neuro disease research.
    Formule :C9H20N2
    Degré de pureté :98.05% - 98.82%
    Couleur et forme :Pale Yellow Clear Liquid
    Masse moléculaire :156.2685

    Ref: TM-T35878

    100mg
    47,00€
  • Nefiracetam

    CAS :
    Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.
    Formule :C14H18N2O2
    Degré de pureté :97.37%
    Couleur et forme :White To Off-White Crystalline Powder
    Masse moléculaire :246.3

    Ref: TM-T0169

    100mg
    39,00€
    200mg
    49,00€
    500mg
    79,00€
    1mL*10mM (DMSO)
    33,00€
  • Indoprofen

    CAS :
    Indoprofen ((±)-Indoprofe) is a non-steroidal anti-inflammatory drug.
    Formule :C17H15NO3
    Degré de pureté :99.34%
    Couleur et forme :Solid
    Masse moléculaire :281.31

    Ref: TM-T0321

    5mg
    54,00€
    10mg
    93,00€
    25mg
    166,00€
    50mg
    264,00€
    100mg
    349,00€
    1mL*10mM (DMSO)
    59,00€
  • Minocycline hydrochloride

    CAS :
    Minocycline HCl: tetracycline antibiotic, treats bacterial infections and acne, may cause acute or chronic hepatitis.
    Formule :C23H28ClN3O7
    Degré de pureté :99.28% - >99.99%
    Couleur et forme :Bright Yellow-Orange Amorphous Solid Crystalline Yellow
    Masse moléculaire :493.94

    Ref: TM-T1101

    25mg
    46,00€
    50mg
    55,00€
    100mg
    67,00€
    200mg
    90,00€
    1mL*10mM (DMSO)
    55,00€
  • JAK2 Inhibitor V

    CAS :
    JAK2 Inhibitor V (JAK2 Inhibitor V Z3) is a novel specific inhibitor of Jak2, inhibiting Jak2-V617F and Jak2-WT autophosphorylation in a dose-dependent manner.
    Formule :C23H24N2O
    Degré de pureté :98.36% - 99.15%
    Couleur et forme :Solid
    Masse moléculaire :344.45

    Ref: TM-T3042

    2mg
    37,00€
    5mg
    54,00€
    10mg
    80,00€
    25mg
    148,00€
    50mg
    259,00€
    100mg
    477,00€
    500mg
    1.063,00€
    1mL*10mM (DMSO)
    59,00€
  • MAT2A inhibitor 2

    CAS :
    MAT2A inhibitor 2 is an inhibitor of methionine adenosyltransferase 2A (MAT2A).
    Formule :C18H24ClN3O3
    Degré de pureté :99.52%
    Couleur et forme :Solid
    Masse moléculaire :365.85

    Ref: TM-T11950

    1mg
    34,00€
    5mg
    67,00€
    10mg
    96,00€
    25mg
    170,00€
    50mg
    253,00€
    100mg
    371,00€
    1mL*10mM (DMSO)
    75,00€
  • MS402

    CAS :
    MS402 is a novel BD1-selective BET BrD inhibitor.
    Formule :C20H19ClN2O3
    Degré de pureté :99.72%
    Couleur et forme :Solid
    Masse moléculaire :370.83

    Ref: TM-T12112

    5mg
    39,00€
    10mg
    58,00€
    25mg
    105,00€
    50mg
    172,00€
    100mg
    268,00€
    1mL*10mM (DMSO)
    46,00€
  • iso-Azalansta

    CAS :
    (2R,4S)-Azalanstat (Iso-Azalansta) is a selective heme oxygenase (HO) inhibitor that is used in the study of cardiovascular disease.
    Formule :C22H24ClN3O2S
    Degré de pureté :99.53% - 99.89%
    Couleur et forme :Soild
    Masse moléculaire :429.96

    Ref: TM-T25127L

    1mg
    175,00€
    5mg
    434,00€
    10mg
    622,00€
    25mg
    973,00€
    50mg
    1.341,00€
    100mg
    1.773,00€
    200mg
    2.422,00€
  • Amifostine

    CAS :
    Amifostine (Ethyol) anhydrous is a cytoprotective agent, acts as a free radical scavenging activity.
    Formule :C5H15N2O3PS
    Degré de pureté :99.59%
    Couleur et forme :White Solid
    Masse moléculaire :214.22

    Ref: TM-T3289

    5mg
    34,00€
    10mg
    49,00€
    25mg
    93,00€
    50mg
    117,00€
    100mg
    164,00€
    200mg
    222,00€
  • Miltefosine

    CAS :
    Miltefosine (HePC), effective oral drug for both visceral and cutaneous leishmaniasis, in clinical trials worldwide.
    Formule :C21H46NO4P
    Degré de pureté :98% - 99.94%
    Couleur et forme :White To Off-White Powder
    Masse moléculaire :407.57

    Ref: TM-T0033

    1g
    120,00€
    5g
    325,00€
    50mg
    34,00€
    100mg
    46,00€
    500mg
    93,00€
  • Fluorescein-NAD+


    Fluorescein NAD+ is a non-radioactive PARP assay substrate, enabling direct enzyme measurement by fluorescence. Comes as 81μg in 250μl water.
    Couleur et forme :Solid

    Ref: TM-T36304

    81µg
    1.468,00€
  • (R)-SKBG-1

    CAS :
    (R)-SKBG-1 is an inhibitor of the RNA-binding protein NONO, effectively downregulating androgen receptor expression by targeting both AR-FL mRNA and AR-V7 mRNA
    Formule :C22H26ClN3O6S
    Degré de pureté :97.25%
    Couleur et forme :Solid
    Masse moléculaire :495.98

    Ref: TM-T79156

    1mg
    74,00€
    5mg
    142,00€
    10mg
    254,00€
    25mg
    560,00€
    1mL*10mM (DMSO)
    156,00€
  • SJ10542

    CAS :
    SJ10542: potent JAK2/3-targeting PG-PROTAC; DC50s: JAK2 - 14 nM, JAK3 - 11 nM, JAK2-fusion ALL - 24 nM; CRBN recruiter.
    Formule :C41H46N12O5S
    Couleur et forme :Solid
    Masse moléculaire :818.95

    Ref: TM-T74429

    2mg
    1.288,00€
  • AUR1545

    CAS :
    AUR1545 is a selective KAT2A/KAT2B degradator, inhibitory against AML, SCLC, and NEPC, and suppressing tumour growth in the NCI-H1048 xenograft model.
    Formule :C41H50BrN9O5
    Degré de pureté :98.84%
    Couleur et forme :Solid
    Masse moléculaire :828.8

    Ref: TM-T205224

    1mg
    193,00€
    5mg
    485,00€
    10mg
    782,00€
    25mg
    1.603,00€
    50mg
    2.592,00€
  • FDA-Approved Kinase Inhibitor Library


    A unique collection of 263 kinase inhibitors/regulators for specific targeting of kinases, ready for high-throughput screening and high-content screening.

    Couleur et forme :Liquid

    Ref: TM-L1610

    1mg
    À demander
  • CARM1/IKZF3 ligand 1


    CARM1/IKZF3 ligand 1 functions as an inhibitor of CARM1 and serves as a target protein ligand for the synthesis of PROTAC CARM1/IKZF3 degrader-1.
    Formule :C27H35ClN6O3
    Couleur et forme :Solid
    Masse moléculaire :527.06

    Ref: TM-T205364

    10mg
    À demander
    50mg
    À demander
  • PROTAC BRD4 Degrader-5

    CAS :
    PROTAC BRD4 Degrader-5 is a PROTAC that degrades BRD4 in HER2 positive and negative breast cancer cell lines.
    Formule :C50H62ClN9O8S2
    Couleur et forme :Solid
    Masse moléculaire :1016.67

    Ref: TM-T36242

    1mg
    255,00€
    5mg
    557,00€
    10mg
    893,00€
    25mg
    1.324,00€
    50mg
    1.791,00€
    1mL*10mM (DMSO)
    973,00€
  • TCIP3

    CAS :
    TCIP3 is a bivalent molecular glue (molecular glue) that can simultaneously bind to both p300/CBP and BCL6. It redirects p300 and CBP to activate programmed cell death genes, which are typically repressed by the oncogenic driver BCL6. TCIP3 is useful for studying diffuse large B-cell lymphoma (DLBCL) and is not toxic to untransformed tonsil lymphocytes or fibroblasts.
    Formule :C58H71ClF2N16O7
    Couleur et forme :Solid
    Masse moléculaire :1177.74

    Ref: TM-T206850

    10mg
    À demander
    50mg
    À demander
  • PRMT3-IN-4


    PRMT3-IN-4 (intermediate 15) is an inhibitor of Protein arginine methyltransferase 3 (PRMT3) and serves as the active control for SGC707. It can be utilized in the synthesis of PROTACs targeting PRMT3 and is applicable in research related to leukemia.
    Couleur et forme :Odour Solid

    Ref: TM-T200459

    10mg
    À demander
    50mg
    À demander
  • Protein Kinase C (19-31)

    CAS :
    Protein Kinase C (19-31), a PKC inhibitor derived from PKCa, has a serine at position 25 and tests PKC activity.
    Formule :C67H118N26O16
    Degré de pureté :98%
    Couleur et forme :Lyophilized Powder
    Masse moléculaire :1543.82

    Ref: TM-TP1053

    100mg
    À demander
    500mg
    À demander
  • PROTAC HDAC6 degrader 4


    PROTAC HDAC6 degrader4 (Compound 17c) is a PROTAC that targets and degrades HDAC6, with a DC50 of 14 nM. It exhibits inhibitory activity against HDAC1, HDAC2, HDAC3, and HDAC6, with IC50 values of 2.2, 2.37, 0.61, and 0.295 μM, respectively. [Pink: ligand for target protein HDAC6 ligand-3; Black: linker; Blue: ligand for cereblon E3 ligase]
    Formule :C39H42FN9O7
    Couleur et forme :Solid
    Masse moléculaire :767.81

    Ref: TM-T205547

    10mg
    À demander
    50mg
    À demander
  • PROTAC BRD4 Degrader-10

    CAS :
    Compound 8b, a dual-ligand PROTAC, targets VHL & BRD4, degrades BRD4 in PC3 cells; conjugates with STEAP1/CLL1, DC50: 1.3/18 nM.
    Formule :C59H71F2N9O15S4
    Couleur et forme :Solid
    Masse moléculaire :1312.5

    Ref: TM-T40073

    100mg
    À demander
    500mg
    À demander
  • UNC10142


    UNC10142 (Compound 44) is a small-molecule antagonist of CHD1, with a binding IC50 value of 1.7 μM. It induces a dose-dependent reduction in the viability of PTEN-deficient prostate cancer cells.
    Formule :C33H52N6O3
    Couleur et forme :Solid
    Masse moléculaire :580.8

    Ref: TM-T203332

    10mg
    À demander
    50mg
    À demander
  • CD532 hydrochloride


    CD532 hydrochloride, potent Aurora A inhibitor (IC50=45 nM), hampers MYCN protein, changes AURKA's shape, aids cancer research.
    Couleur et forme :Solid

    Ref: TM-T36932

    5mg
    90,00€
    10mg
    155,00€
    25mg
    291,00€
  • HDAC1-IN-9


    HDAC1-IN-9 (13c) is an HDAC1 inhibitor. It inhibits the HDAC1 enzyme with an IC50 value of 1.07 µM. This compound exhibits the strongest antiproliferative activity against HT-29 (human colon adenocarcinoma cells), with an IC50 of 1.78 μM. In HCT-116 (human colon cancer cells), HDAC1-IN-9 significantly induces apoptosis. Additionally, HDAC1-IN-9 possesses antiangiogenic properties, reducing the expression levels of VEGFR-2 and phosphorylated VEGFR-2 (pVEGFR-2) by approximately 80%.
    Formule :C17H17N3O3
    Couleur et forme :Solid
    Masse moléculaire :311.34

    Ref: TM-T205384

    10mg
    À demander
    50mg
    À demander
  • NP213

    CAS :
    NP213 is a rapidly acting synthetic antimicrobial peptide (AMP).
    Formule :C42H84N28O7
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :1093.3

    Ref: TM-TP2149L

    100mg
    À demander
    500mg
    À demander
  • HDAC6-IN-53


    HDAC6-IN-53 (Compound W28) is an inhibitor targeting histone deacetylase 6 (HDAC6) with an IC50 of 19.65 nM. It reduces the idiopathic pulmonary fibrosis (IPF) phenotype by inhibiting TGF-β1-induced collagen expression and demonstrates therapeutic efficacy in a bleomycin-induced mouse model of pulmonary fibrosis. HDAC6-IN-53 is applicable for research in idiopathic pulmonary fibrosis and related pulmonary fibrotic diseases.
    Couleur et forme :Odour Solid

    Ref: TM-T206842

    10mg
    À demander
    50mg
    À demander
  • SAMS

    CAS :
    SAMS peptide is a specific substrate for the AMP-activated protein kinase (AMPK).
    Formule :C74H131N29O18S2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :1779.15

    Ref: TM-TP1812

    1mg
    494,00€
    5mg
    1.665,00€
    500µg
    259,00€
  • SMD-3236

    CAS :
    SMD-3236 is a PRAOTAC degrader targeting SMARCA2, designed using SMARCA ligand and VHL-1 ligand, and exhibits prolonged anti-tumor activity in vivo. SMARCA2 acts as a synthetic lethal target in cancer cells lacking SMARCA4, with SMD-3236 showing 2000-fold selectivity for SMARCA2 over SMARCA4, having a DC50 of less than 1 nM and a Dmax of over 95%. In the human cancer xenograft models deficient in SMARCA4, notably the H838 model, SMD-3236 effectively induces loss of SMARCA2 in tumor tissue while sparing the SMARCA4 protein, thereby inhibiting tumor growth. The compound consists of a target protein ligand (red part) SMI-1074, a PROTAC linker (black part) (trans-4-Ethynylcyclohexyl)methyl methanesulfonate, and an E3 ligase ligand (blue part) SMARCA2 ligand-14, forming the E3LigaseLigand-linker Conjugate 159.
    Formule :C61H75ClN10O5S
    Couleur et forme :Solid
    Masse moléculaire :1095.83

    Ref: TM-T205371

    10mg
    À demander
    50mg
    À demander
  • ZL0590

    CAS :
    ZL0590 is an effective and selective inhibitor of BD1-BRD4 (IC50 = 90 nM) with anti-inflammatory activities.
    Formule :C23H27F3N4O4S
    Degré de pureté :99.77%
    Couleur et forme :Soild
    Masse moléculaire :512.55

    Ref: TM-T60072

    1mg
    71,00€
    5mg
    152,00€
    10mg
    222,00€
    25mg
    401,00€
    50mg
    602,00€
    100mg
    887,00€
    1mL*10mM (DMSO)
    167,00€
  • KDM1A-IN-29

    CAS :
    KDM1A-IN-29 is a histone demethylase inhibitor.
    Formule :C16H16ClN3O4S
    Couleur et forme :Soild
    Masse moléculaire :381.83

    Ref: TM-T88834

    1mg
    175,00€
    5mg
    434,00€
    10mg
    622,00€
    25mg
    973,00€
    50mg
    1.341,00€
  • 3β,6α,12β-Dammar-E-20(22)-ene-3,6,12,25-tetraol

    CAS :

    3β,6α,12β-Dammar-E-20(22)-ene-3,6,12,25-tetraol is a compound that functions as a SIRT1 activator, effectively enhancing SIRT1 activity.

    Formule :C30H52O4
    Couleur et forme :Solid
    Masse moléculaire :476.742

    Ref: TM-T41125

    100mg
    À demander
    500mg
    À demander
  • DNMT1/HDAC-IN-1


    DNMT1/HDAC-IN-1 (compound (R)-23a), a potent dual inhibitor targeting both DNMT1 and HDAC, exhibits impressive inhibitory effects specifically on HDAC1 (HDAC1:IC50=0.05 μM), a major HDAC isoform that interacts with DNMT1 across multiple protein complexes involved in the transcriptional silencing of TSGs. This compound has been shown to remodel the tumor immune microenvironment and induce tumor regression, effectively reversing cancer-specific epigenetic abnormalities.
    Couleur et forme :Odour Solid

    Ref: TM-T200728

    10mg
    À demander
    50mg
    À demander
  • CBP/p300-IN-8

    CAS :
    CBP/p300-IN-8 strongly inhibits CBP/P300 bromodomains; CBP IC50=0.01-0.1μM, BRD4 IC50=1-1000μM.
    Formule :C27H31N3O4
    Couleur et forme :Solid
    Masse moléculaire :461.562

    Ref: TM-T39826

    5mg
    582,00€
    10mg
    895,00€
    50mg
    2.692,00€
  • Hyp-dBET1


    Hyp-dBET1 is a PROTAC degrader targeting BRD4, with an IC50 value of 3.4 μM in MDA-MB-231 cells. Under hypoxic conditions, Hyp-dBET1 becomes active, recruiting E3 ubiquitin ligase, and facilitates the degradation of BRD4 via the ubiquitin-proteasome system. Hyp-dBET1 is applicable in anti-cancer research.
    Couleur et forme :Odour Solid

    Ref: TM-T206198

    10mg
    À demander
    50mg
    À demander
  • Menin-KMT2A-IN-1


    Menin–KMT2A-IN-1 (Compound 20) is an inhibitor of menin–KMT2A, binding to menin with an IC50 of 8 nM, and disrupting the interaction between menin and lysine methyltransferase 2A (KMT2A). It inhibits hERG channels with an IC50 of 65 μM and suppresses MV4-11 cells with an IC50 of 74 nM. Furthermore, Menin–KMT2A-IN-1 exhibits favorable pharmacokinetic properties in CD-1 mice, with an oral bioavailability of 74%.
    Formule :C28H35FN6O3
    Couleur et forme :Solid
    Masse moléculaire :522.61

    Ref: TM-T205488

    10mg
    À demander
    50mg
    À demander
  • Uzansertib

    CAS :
    Uzansertib (INCB053914) is a potent pan-PIM kinase inhibitor with low IC50s: 0.24, 30, 0.12 nM for PIM1, 2, 3; hinders hematologic tumor growth.
    Formule :C26H26F3N5O3
    Couleur et forme :Solid
    Masse moléculaire :513.51

    Ref: TM-T39090

    25mg
    1.369,00€
  • Pumecitinib

    CAS :

    Pumecitinib is a Janus kinase (JAK) inhibitor. Pumecitinib exhibits anti-inflammatory activity.

    Formule :C17H20N8O2S
    Degré de pureté :99.94%
    Couleur et forme :Soild
    Masse moléculaire :400.46

    Ref: TM-T67758

    5mg
    52,00€
    10mg
    78,00€
    25mg
    128,00€
    50mg
    197,00€
    100mg
    281,00€
  • SMD-3040 TFA


    SMD-3040 TFA is a selective SMARCA2 degrader comprising SMARCA2/4 ligands, a linker, and VHL ligands, utilized in PROTAC drug synthesis.
    Degré de pureté :98%
    Couleur et forme :Odour Solid

    Ref: TM-T81147

    5mg
    À demander
    50mg
    À demander
  • PROTAC BRD4 Degrader-19

    CAS :
    PROTAC BRD4 Degrader-19 (compound 176) is a proteolysis-targeting chimera (PROTAC) designed to specifically degrade the BRD4 protein, offering potential utility
    Formule :C44H38N8O5S2
    Couleur et forme :Solid
    Masse moléculaire :822.95

    Ref: TM-T75149

    5mg
    À demander
    50mg
    À demander
  • GSK040

    CAS :
    GSK040: Potent BET BD2 inhibitor, pIC50 8.3, 5000x selectivity over BD1, for oncology & immunology research.
    Formule :C29H34N4O4
    Couleur et forme :Solid
    Masse moléculaire :502.6

    Ref: TM-T63418

    25mg
    3.615,00€
    50mg
    4.708,00€
    100mg
    5.943,00€
  • GSK8573

    CAS :
    GSK8573 is an inactive control compound for GSK2801. GSK8573 has binding activity to BRD9 (Kd of 1.04 μM).
    Formule :C20H21NO3
    Degré de pureté :99.97%
    Couleur et forme :Solid
    Masse moléculaire :323.39

    Ref: TM-T15441

    5mg
    38,00€
    10mg
    56,00€
    25mg
    95,00€
    50mg
    150,00€
    1mL*10mM (DMSO)
    35,00€
  • Vanicoside A

    CAS :
    Vanicoside A is a protein kinase C( PKC ) inhibitor from Polygonum pensylvanicum [1] .
    Formule :C51H50O21
    Couleur et forme :Solid
    Masse moléculaire :998.93

    Ref: TM-T75565

    5mg
    À demander
    50mg
    À demander
  • MZP-54

    CAS :
    MZP-54 is a selective degrader of BRD3/4 based on PROTAC technology(Kd of 4 nM for Brd4BD2)
    Formule :C55H66ClN7O9S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :1036.67

    Ref: TM-T13785

    5mg
    410,00€
    10mg
    627,00€
    25mg
    1.189,00€
  • HIF-1 α (556-574)

    CAS :
    HIF-1 alpha (556-574) is a 19-mer fragment vital for gene expression in low oxygen; it binds VHL with critical proline 564 for stability.
    Formule :C101H150D2N20O34S2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :2254.6

    Ref: TM-TP1533

    100mg
    À demander
    500mg
    À demander
  • TB22


    TB22 is a non-nucleoside inhibitor of DOT1LR231Q with anticancer activity. It inhibits the malignant phenotype of lung cancer cells harboring the R231Q mutation via the MAPK/ERK signaling pathway, making it useful for lung cancer research.
    Couleur et forme :Odour Solid

    Ref: TM-T200492

    10mg
    À demander
    50mg
    À demander
  • Namoline

    CAS :
    Namoline, a γ-pyrone, inhibits LSD1 with a 51 μM IC50, blocking cell growth and showing potential in prostate cancer studies.
    Formule :C10H3ClF3NO4
    Couleur et forme :Solid
    Masse moléculaire :293.58

    Ref: TM-T40420

    5mg
    873,00€
  • BRD7-IN-1 free base

    CAS :
    BRD7-IN-1, a BI7273 derivative, transforms into PROTAC VZ185 (targets BRD7/9 with 4.5/1.8 nM DC50s) via a VHL linker.
    Formule :C22H26N4O3
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :394.47

    Ref: TM-T17696

    100mg
    À demander
    500mg
    À demander
  • KB02-JQ1

    CAS :
    KB02-JQ1: potent BRD4-degrading PROTAC, stable, specific; doesn't affect BRD2/3, modifies DCAF16 for action.
    Formule :C38H43Cl2N7O6S
    Degré de pureté :98%
    Couleur et forme :Soild
    Masse moléculaire :796.77

    Ref: TM-T18060

    100mg
    À demander
    500mg
    À demander
  • NSC 370284

    CAS :
    NSC 370284 inhibits STAT3/5, reducing AML cell viability with TET1 overexpression in vitro/in vivo.
    Formule :C21H25NO6
    Degré de pureté :99.74%
    Couleur et forme :Solid
    Masse moléculaire :387.43

    Ref: TM-T9949

    5mg
    46,00€
    10mg
    80,00€
    25mg
    156,00€
    50mg
    255,00€
    100mg
    375,00€
    200mg
    532,00€
    1mL*10mM (DMSO)
    49,00€
  • MS9024


    MS9024 is a degrader of DNA methyltransferase 1 (DNMT1), facilitating its degradation in HCT116 cells via the ubiquitin-proteasome pathway, with a DC50 of 35 nM (DC50 values are 254 nM in MDA-MB-468 and 101 nM in H1299). Additionally, MS9024 inhibits DNMT1 with an IC50 of 0.43 μM.
    Couleur et forme :Odour Solid

    Ref: TM-T206183

    10mg
    À demander
    50mg
    À demander
  • CDD-1102 HCl


    CDD-1102 HCl is a novel BRDT-BD4 / BRD2-BD1302 selective inhibitor that shows non-hormonal contraceptive potential in ex vivo experiments.
    Formule :C32H31ClN6O3
    Degré de pureté :98.30%
    Couleur et forme :Soild
    Masse moléculaire :583.08

    Ref: TM-T72058L

    1mg
    315,00€
    5mg
    745,00€
    10mg
    1.018,00€
    25mg
    1.431,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Pim-1 kinase inhibitor 11


    Pim-1 kinase inhibitor 11 (10f) is an inhibitor of PIM-1 with an IC50 value of 0.18 μM. It exhibits anticancer activity by inducing apoptosis and causing cell cycle arrest.
    Couleur et forme :Odour Solid

    Ref: TM-T200676

    10mg
    À demander
    50mg
    À demander
  • PRO-HD3


    PRO-HD3 is a cell-specific, PROTAC-based degrader targeting HDAC6 [1].
    Degré de pureté :98%
    Couleur et forme :Odour Solid

    Ref: TM-T81392

    5mg
    À demander
    50mg
    À demander
  • Axl-IN-16


    Axl-IN-16, a dual Axl/HIF inhibitor, promotes Flammulina velutipes fruiting body formation and suppresses hypoxia-inducible factor activity along with receptor
    Formule :C14H19ClO8
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :350.75

    Ref: TM-T79969

    5mg
    À demander
    50mg
    À demander
  • XF067-68

    CAS :
    XF067-68 is a PROTAC for targeted degradation of WD40 repeat domain protein 5 ( WDR5 )[1] .
    Formule :C52H59F4N9O7S
    Couleur et forme :Solid
    Masse moléculaire :1030.14

    Ref: TM-T74889

    5mg
    À demander
    50mg
    À demander
  • JB300

    CAS :
    JB300 is a PROTAC-based compound that serves as a highly selective degrader of Aurora A, with a DC50 of 30 nM. It is utilized in cancer research. JB300 comprises the PROTAC target protein ligand MK-5108 [pink part], E3 ligase ligand Thalidomide-O-COOH [blue part], and PROTAC Linker Boc-NH-PEG2-C2-NH2 [black part]. The conjugate of the E3 ubiquitin ligase ligand and linker is Thalidomide-O-COOH-NH2-C2-PEG2-NH-Boc.
    Formule :C43H45ClFN7O10S
    Couleur et forme :Solid
    Masse moléculaire :906.375

    Ref: TM-T204223

    10mg
    À demander
    50mg
    À demander
  • SNIPER(BRD)-1

    CAS :
    SNIPER(BRD)-1 has LCL-161, (+)-JQ1 linked; degrades BRD4, cIAP1/2, XIAP; IC50s: 6.8, 17, 49nM.
    Formule :C53H66ClN9O8S2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :1056.73

    Ref: TM-T16905

    100mg
    À demander
    500mg
    À demander
  • PROTAC BET degrader-3


    PROTAC BET Degrader-3 is a potent degrader OF BET based on PROTAC.
    Formule :C53H64N12O9S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :1045.22

    Ref: TM-T13850

    5mg
    410,00€
    10mg
    627,00€
    25mg
    1.378,00€
    50mg
    À demander
    100mg
    À demander
  • PROTAC SMARCA2/4-degrader-28

    CAS :
    PROTAC SMARCA2/4-degrader-28 (PROTAC 1) functions as a partial degrader of SMARCA2 and SMARCA4 through the PROTAC-based mechanism.
    Formule :C54H68ClN9O11S2
    Couleur et forme :Solid
    Masse moléculaire :1118.75

    Ref: TM-T200190

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  • PF-04577806

    CAS :
    PF-04577806: potent & selective PKC inhibitor, ATP competitive, blocks PKCα/βI/βII/γ/θ (IC50: 2.4-45.9 nM), may reverse diabetic retinal leakage.
    Formule :C26H37N7O3
    Couleur et forme :Solid
    Masse moléculaire :495.628

    Ref: TM-T38462

    5mg
    873,00€
  • MNK/PIM-IN-1

    CAS :
    MNK/PIM-IN-1 is a novel dual inhibitor targeting both MNK and PIM pathways, characterized by its favorable pharmacokinetic profile.
    Formule :C27H27FN6O2
    Couleur et forme :Solid
    Masse moléculaire :486.551

    Ref: TM-T40092

    5mg
    873,00€
  • HDAC11-IN-1


    HDAC11-IN-1 (Compound 14-NC6OH) is a macrocyclic inhibitor that selectively targets HDAC11 with a Ki of 40 nM. It demonstrates effective cell permeability and suppresses the expression of YAP1 and SOX2.
    Formule :C43H63F3N6O6S2
    Couleur et forme :Solid
    Masse moléculaire :881.12

    Ref: TM-T205328

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  • VinSpinIn

    CAS :
    VinSpinIn is a probe for the Spin family proteins.
    Formule :C42H58N8O4
    Couleur et forme :Solid
    Masse moléculaire :738.98

    Ref: TM-T35060

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  • R 8605

    CAS :
    R 8605 is a third-generation retinoid.
    Formule :C22H27NO4
    Couleur et forme :Solid
    Masse moléculaire :369.45

    Ref: TM-T34239

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  • GSK3735967

    CAS :
    GSK3735967: DNMT1 inhibitor, IC50 40 nM, dicyanopyridine core, binds hemimethylated CpG, interacts with H4K20me3.
    Formule :C25H31N7OS
    Couleur et forme :Solid
    Masse moléculaire :477.62

    Ref: TM-T74887

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  • GNE-987

    CAS :
    GNE-987 is a potent chimeric BET degrader, binding BRD4 BD1/BD2 at IC50: 4.7/4.4 nM & has a DC50: 0.03 nM in EOL-1 AML cells.
    Formule :C56H67F2N9O8S2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :1096.31

    Ref: TM-T11441

    1mg
    444,00€
    5mg
    1.009,00€
    10mg
    1.603,00€
  • ZMF-23


    ZMF-23, a PAK1/HDAC6 dual inhibitor, suppresses PAK1 and HDAC6-mediated aerobic glycolysis and cellular migration while inducing TNF-α-regulated necroptosis and
    Formule :C22H23Cl2N5O3
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :476.36

    Ref: TM-T79369

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  • HDAC6 ligand-3


    HDAC6ligand-3 serves as a ligand for HDAC6 and can be utilized as a target protein ligand in the synthesis of [PROTAC] HDAC6 degrader4.
    Formule :C20H21N3O3
    Couleur et forme :Solid
    Masse moléculaire :351.399

    Ref: TM-T205606

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  • HIV-1 protease-IN-10


    HIV-1 protease-IN-10 (Compound 2), exhibiting HIV-1 latency reversing activity (IC50: 0.22 μM), selectively binds to the PKCδ C1b domain (IC50: 0.69 μM) and
    Formule :C23H40O5
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :396.56

    Ref: TM-T79493

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  • TAT-cyclo-CLLFVY

    CAS :
    Blocks HIF-1α/β dimerization, not HIF-2α; suppresses VEGF, CAIX in cancer cells; antiangiogenic in HUVECs (IC50 = 1.3 μM).
    Formule :C111H188N42O24S2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :2559.1

    Ref: TM-TP2046

    1mg
    1.063,00€
  • Sirtuin modulator 5

    CAS :
    Sirtuin modulator 5 activates SIRT1 (<50 μM DC50), may extend cell lifespan, and could aid in researching various age/stress-related diseases.
    Formule :C24H23N3O4
    Couleur et forme :Solid
    Masse moléculaire :417.46

    Ref: TM-T74672

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  • SR-0813

    CAS :
    SR-0813 is a potent and selective inhibitor of the YEATS domain in ENL/AF9.
    Formule :C25H32N6O3S
    Degré de pureté :98.81%
    Couleur et forme :Solid
    Masse moléculaire :496.62

    Ref: TM-T40229

    1mg
    39,00€
    5mg
    86,00€
    10mg
    124,00€
    25mg
    253,00€
    50mg
    384,00€
    100mg
    532,00€
    200mg
    705,00€
    1mL*10mM (DMSO)
    94,00€
  • MAK-683 hydrochloride

    CAS :
    MAK683 hydrochloride is an inhibitor of embryonic ectoderm development (EED), with IC50 values of 59, 26nM measured in EED Alphascreen, ELISA.Cost-effective and quality-assured.
    Formule :C20H18ClFN6O
    Degré de pureté :97.02% - >99.99%
    Couleur et forme :Solid
    Masse moléculaire :412.85

    Ref: TM-T9681

    1mg
    185,00€
    5mg
    415,00€
    10mg
    622,00€
    25mg
    947,00€
    50mg
    1.359,00€
    100mg
    1.833,00€
  • PROTAC BET Degrader-1

    CAS :
    PROTAC BET Degrader-1 is a potent degrader of BET based on PROTAC.
    Formule :C44H45N11O9
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :871.9

    Ref: TM-T13849

    5mg
    410,00€
    10mg
    627,00€
    25mg
    1.378,00€
    50mg
    À demander
    100mg
    À demander
    1mL*10mM (DMSO)
    447,00€
  • MRS2698

    CAS :
    MRS2698: potent P2Y2 agonist, EC50 8 nM, >300x selectivity over P2Y4/P2Y6.
    Formule :C9H16N3O13P3S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :499.22

    Ref: TM-T16139

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  • HSP90/LSD1-IN-1


    HSP90/LSD1-IN-1 (compound 6) is a dual inhibitor of HSP90 and LSD1. This compound effectively inhibits the proliferation of prostate cancer cell lines PC-3 and DU145, with GI50 values of 0.24 μM and 0.30 μM, respectively.
    Couleur et forme :Odour Solid

    Ref: TM-T200725

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  • Okicenone

    CAS :

    Okicenone is an antibiotic, interferring with HuR RNA binding, HuR trafficking, T-cell activation and cytokine expression.

    Formule :C15H14O4
    Couleur et forme :Solid
    Masse moléculaire :258.27

    Ref: TM-T28228

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  • BAY-184

    CAS :
    BAY-184,KAT6A/B inhibitor (IC50=71/83 nM). Suppresses ERα activity. Impedes breast cancer proliferation.
    Formule :C23H20N2O4S
    Degré de pureté :98.87%
    Couleur et forme :Solid
    Masse moléculaire :420.48

    Ref: TM-T203636

    2mg
    46,00€
    5mg
    66,00€
    10mg
    97,00€
    25mg
    187,00€
    50mg
    303,00€
  • Lyngbyatoxin A

    CAS :

    Lyngbyatoxin A is an indole alkaloid from blue-green alga Lyngbya majuscula Gomont; responsible for dermatitis known as &quot;swimmers' itch&quot; in Hawaii.

    Formule :C27H39N3O2
    Couleur et forme :Solid
    Masse moléculaire :437.62

    Ref: TM-T33033

    25mg
    1.444,00€
  • HIF1-IN-3 

    CAS :
    HIF1-IN-3 (Benzenepropanamide, N-[(8-hydroxy-7-quinolinyl)(4-methoxyphenyl)methyl]-) is an effective inhibitor of HIF-1 (EC50 = 0.9 μM) and can be used in
    Formule :C26H24N2O3
    Degré de pureté :99.59%
    Couleur et forme :Solid
    Masse moléculaire :412.48

    Ref: TM-T9890

    5mg
    43,00€
    10mg
    60,00€
    25mg
    110,00€
    50mg
    200,00€
    100mg
    276,00€
    200mg
    400,00€
    1mL*10mM (DMSO)
    50,00€
  • PROTAC BRD4 Degrader-13

    CAS :
    PROTAC BRD4 Degrader-13 targets VHL and BRD4, degrading BRD4 with DC50 of 0.025/6.0 nM in PC3 cells when linked to STEAP1/CLL1 antibodies.
    Formule :C68H85F2N11O17P2S2
    Couleur et forme :Solid
    Masse moléculaire :1492.55

    Ref: TM-T40075

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  • MS33

    CAS :
    MS33 degrades WDR5 protein, Kd 870 nM (VCB), 120 nM (WDR5); uses VHL ligase, aids acute myeloid leukemia study.
    Formule :C64H84F3N11O7S
    Couleur et forme :Solid
    Masse moléculaire :1208.5

    Ref: TM-T39975

    25mg
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  • MNN-02-155

    CAS :
    MNN-02-155 is a bivalent molecular glue that can simultaneously interact with both p300/CBP and BCL6. It effectively induces the activation of BCL6-targeted reporter genes and promotes cell death. This compound is used in the research of diffuse large B-cell lymphoma (DLBCL).
    Formule :C56H68ClF2N15O7
    Couleur et forme :Solid
    Masse moléculaire :1136.69

    Ref: TM-T206805

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  • DS-103


    DS-103 is an HDAC inhibitor that targets HDAC1, HDAC2, HDAC3, HDAC6, and HDAC8 with IC50 values of 0.029, 0.123, 0.022, 0.367, and 9.26 μM, respectively. It also inhibits the malignant malaria parasite [Plasmodium falciparum 3D7] with an IC50 of 5.08 μM. In A2780 and Cal27 cells, DS-103 exhibits cytotoxicity with IC50 values of 1.48 μM and 1.47 μM, respectively, and reverses cisplatin resistance in these cells with IC50 values of 4.62 μM and 2.23 μM. DS-103 acts synergistically with cisplatin, enhancing apoptosis induced by cisplatin.
    Formule :C28H33N5O3
    Couleur et forme :Solid
    Masse moléculaire :487.59

    Ref: TM-T205596

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