
Chromatine/Épigénétique
Sous-catégories appartenant à la catégorie "Chromatine/Épigénétique"
2616 produits trouvés pour "Chromatine/Épigénétique"
Solcitinib
CAS :Solcitinib (GLPG-0778), a JAK1 inhibitor, may treat psoriasis, ulcerative colitis, and lupus.
Formule :C22H23N5O2Degré de pureté :99.61% - 99.82%Couleur et forme :SolidMasse moléculaire :389.45Dbet57
CAS :dBET57: PROTAC-based BRD4BD1 degrader, DC50/5h at 500 nM, ineffective on BRD4BD2.Formule :C34H31ClN8O5SDegré de pureté :99.36% - 99.52%Couleur et forme :SolidMasse moléculaire :699.18Ref: TM-T5440
1mg47,00€5mg92,00€10mg147,00€1mL*10mM (DMSO)166,00€25mg264,00€50mg409,00€100mg592,00€500mg1.224,00€MAT2A inhibitor 4
CAS :MAT2A Inhibitor 4 acts as an inhibitor targeting the catalytic subunit of methionine S-adenosyltransferase-2 (MAT2A), offering potential utility in cancerFormule :C16H15ClFNDegré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :275.75Ref: TM-T9262
1mg40,00€1mL*10mM (DMSO)89,00€5mg90,00€10mg131,00€25mg220,00€50mg314,00€100mg426,00€200mg575,00€PF-06409577
CAS :PF-06409577 is an effective, orally active, and specific allosteric activator of AMPK (EC50: 7 nM, for α1β1γ1).Formule :C19H16ClNO3Degré de pureté :95.17% - 98.21%Couleur et forme :SolidMasse moléculaire :341.79Ref: TM-T4427
1mg34,00€2mg43,00€5mg63,00€1mL*10mM (DMSO)71,00€10mg100,00€25mg200,00€50mg334,00€100mg537,00€200mg762,00€Mivebresib
CAS :Mivebresib (ABBV-075) is a potent BET inhibitor with antitumor effects, disrupting gene expression and MYC, TMPRSS2-ETS proteins.Formule :C22H19F2N3O4SDegré de pureté :98.74% - 99.32%Couleur et forme :SolidMasse moléculaire :459.47Ref: TM-T3712
1mg55,00€2mg78,00€5mg92,00€1mL*10mM (DMSO)94,00€10mg150,00€25mg244,00€50mg437,00€100mg625,00€PHA-680632
CAS :PHA-680632 is potent inhibitor of Aurora A, Aurora B and Aurora C with IC50 of 27 nM, 135 nM and 120 nM, respectively.Formule :C28H35N7O2Degré de pureté :98.2%Couleur et forme :SolidMasse moléculaire :501.623-Aminobenzamide
CAS :3-Aminobenzamide (PARP-IN-1) is an effective inhibitor of PARP (IC50<50 nM in CHO cells) and a mediator of oxidant-induced myocyte dysfunction duringFormule :C7H8N2ODegré de pureté :98.4% - 99.5%Couleur et forme :White To Off-White PowderMasse moléculaire :136.15ASP4132
CAS :ASP4132 is an orally active AMPK activator (EC50 : 18 nM), has anti-cancer activity.Formule :C46H51F3N6O8S2Degré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :937.06Ref: TM-T8432
1mg50,00€5mg114,00€10mg177,00€1mL*10mM (DMSO)185,00€25mg321,00€50mg482,00€100mg677,00€200mg928,00€SF2523
CAS :SF2523 is a highly selective and potent inhibitor.Formule :C19H17NO5SDegré de pureté :99.1% - 99.51%Couleur et forme :SolidMasse moléculaire :371.41Ref: TM-T3986
1mg34,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg113,00€25mg260,00€50mg409,00€100mg605,00€500mg1.288,00€JNJ-64619178
CAS :JNJ-64619178: selective, oral, pseudo-irreversible PRMT5 inhibitor (IC50: 0.14 nM), effective in lung cancer.Formule :C22H23BrN6O2Degré de pureté :98.86% - 99.98%Couleur et forme :SolidMasse moléculaire :483.36Ref: TM-T15624
1mg84,00€5mg167,00€1mL*10mM (DMSO)172,00€10mg260,00€25mg537,00€50mg893,00€100mg1.571,00€PIN1 inhibitor API-1
CAS :API-1 is a Pin1 inhibitor (IC50: 72.3 nM), enhancing anticancer miRNA biogenesis and inhibiting hepatocellular carcinoma.Formule :C15H13F3N6O2Degré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :366.3Ref: TM-T16538
1mg57,00€5mg120,00€1mL*10mM (DMSO)133,00€10mg222,00€25mg326,00€50mg485,00€100mg612,00€200mg850,00€500mg1.243,00€GeA-69
CAS :GeA-69 (GeA69) is a selective and allosteric PARP14 macrodomain 2 (MD2) inhibitor (Kd: 0.86 μM in ITC assays).Formule :C20H16N2ODegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :300.35CPI-455
CAS :CPI-455 is a specific KDM5 inhibitor.Formule :C16H14N4ODegré de pureté :97.87% - 99.03%Couleur et forme :SolidMasse moléculaire :278.31Ref: TM-T3552
1mg34,00€2mg49,00€5mg70,00€1mL*10mM (DMSO)70,00€10mg105,00€25mg178,00€50mg335,00€100mg505,00€A-769662
CAS :A-769662 is an effective, reversible AMPK activator(EC50=0.8 μM).Formule :C20H12N2O3SDegré de pureté :97.52% - 99.58%Couleur et forme :SolidMasse moléculaire :360.39Ref: TM-T2468
2mg37,00€5mg54,00€1mL*10mM (DMSO)56,00€10mg74,00€25mg135,00€50mg244,00€100mg440,00€500mg964,00€TTK21
CAS :TTK21 is an activator of CBP/p300 histone acetyltransferase activity.Formule :C17H15ClF3NO2Degré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :357.75Ref: TM-T8778
1mg57,00€5mg105,00€1mL*10mM (DMSO)114,00€10mg158,00€25mg308,00€50mg462,00€100mg692,00€500mg1.404,00€Aurora kinase inhibitor-2
CAS :Aurora kinase inhibitor-2 (IUN-70219) is a cell-permeable anilinoquinazoline that inhibit the activity of Aurora A (IC50 = 0.39 M).Formule :C23H20N4O3Degré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :400.43Ref: TM-T9040
1mg63,00€5mg138,00€1mL*10mM (DMSO)150,00€10mg200,00€25mg360,00€50mg532,00€100mg788,00€200mg1.063,00€BAZ1A-IN-1
CAS :BAZ1A-IN-1, a potent inhibitor, KD 0.52 μM against BAZ1A, is effective in high-BAZ1A cancer cells, not in low-BAZ1A ones.Formule :C16H12N4O3SDegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :340.36Ref: TM-T9552
1mg84,00€5mg177,00€1mL*10mM (DMSO)195,00€10mg268,00€25mg537,00€50mg803,00€100mg1.099,00€200mg1.468,00€Amifostine sodium
CAS :Amifostine sodium is a phosphorothioate proposed as a radiation-protective agent. It causes splenic vasodilation and may block autonomic ganglia.Formule :C5H15N2NaO3PSCouleur et forme :SolidMasse moléculaire :237.21I-CBP112
CAS :I-CBP112 is a specific and potent acetyl-lysine competitive protein-protein interaction inhibitor targeting the CBP/p300 bromodomains.Formule :C27H36N2O5Degré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :468.59Ref: TM-T3969
1mg33,00€2mg50,00€5mg92,00€1mL*10mM (DMSO)92,00€10mg161,00€25mg296,00€50mg425,00€100mg583,00€200mg785,00€PX-478
CAS :PX-478 is a HIF-1α inhibitor with selectivity, oral activity, and blood-brain barrier permeability.Formule :C13H20Cl4N2O3Degré de pureté :97% - 99.79%Couleur et forme :SolidMasse moléculaire :394.12Ref: TM-T6961
1mg39,00€5mg84,00€1mL*10mM (DMSO)84,00€10mg130,00€25mg193,00€50mg261,00€100mg411,00€200mg605,00€LW6
CAS :LW6 (HIF-1α inhibitor) is a novel HIF-1 inhibitor.Formule :C26H29NO5Degré de pureté :98.1% - 98.22%Couleur et forme :SolidMasse moléculaire :435.51Ref: TM-T3494
2mg44,00€5mg65,00€1mL*10mM (DMSO)65,00€10mg94,00€25mg173,00€50mg281,00€100mg424,00€500mg888,00€Alobresib
CAS :Alobresib (Vorolanib) is an inhibitor of BET bromodomain,is an antineoplastic drug candidate.Formule :C26H23N5O2Degré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :437.49Ref: TM-T8495
1mg70,00€2mg87,00€5mg137,00€1mL*10mM (DMSO)150,00€10mg260,00€25mg507,00€50mg713,00€100mg982,00€Dehydrocorydaline
CAS :1.Formule :C22H24NO4Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :366.43Ref: TM-T5S2358
1mg49,00€2mg69,00€5mg105,00€1mL*10mM (DMSO)116,00€10mg137,00€25mg197,00€50mg295,00€100mg447,00€Belzutifan
CAS :"Belzutifan (MK-6482) is an oral HIF-2α inhibitor for ccRCC, with enhanced potency (IC50: 9 nM)."Formule :C17H12F3NO4SDegré de pureté :99.34% - 99.88%Couleur et forme :SolidMasse moléculaire :383.34Ref: TM-T16679
1mg66,00€5mg144,00€1mL*10mM (DMSO)158,00€10mg205,00€25mg389,00€50mg625,00€100mg888,00€200mg1.198,00€I-BET151
CAS :I-BET151 (GSK1210151A) (GSK1210151A) is a specific BET inhibitor for BRD2/3/4 (IC50: 0.5/0.25/0.79 μM, in cell-free assays).Formule :C23H21N5O3Degré de pureté :97.34% - 99.63%Couleur et forme :SolidMasse moléculaire :415.44Ref: TM-T2120
1mg48,00€2mg65,00€5mg96,00€1mL*10mM (DMSO)105,00€10mg115,00€25mg202,00€50mg339,00€100mg507,00€500mg1.130,00€MI-503
CAS :MI-503 is an efficient and selective Menin-MLL inhibitor. MI-503 has a significant inhibitory effect on human MLL leukemia cell line. Cost-effective and quality-assured.Formule :C28H27F3N8SDegré de pureté :99.87% - 99.99%Couleur et forme :SolidMasse moléculaire :564.63Ref: TM-TQ0069
1mg50,00€5mg114,00€1mL*10mM (DMSO)141,00€10mg178,00€25mg334,00€50mg557,00€100mg888,00€Buformin hydrochloride
CAS :Buformin hydrochloride, an oral biguanide antidiabetic, activates AMPK, enhances insulin sensitivity, and inhibits hepatic glucose production.Formule :C6H16ClN5Degré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :193.68AZD1208
CAS :AZD1208 is a novel, orally bioavailable, highly selective PIM kinase inhibitor with single nanomolar potency against all three PIM kinases.Formule :C21H21N3O2SDegré de pureté :97.24% - 99.83%Couleur et forme :SolidMasse moléculaire :379.48Ref: TM-T2300
2mg35,00€5mg49,00€1mL*10mM (DMSO)54,00€10mg71,00€25mg112,00€50mg202,00€100mg358,00€200mg470,00€500mg750,00€Niraparib hydrochloride
CAS :Niraparib hydrochloride (MK-4827) is a PARP inhibitor with potential cancer treatment effects, causing DNA damage and apoptosis.Formule :C19H21ClN4ODegré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :356.85B2
CAS :B2 (Linazolamide intermediate B impurity 2) promotes inclusion formation in cellular models of Huntington's disease and Parkinson's diseaseFormule :C20H17ClN4O3Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :396.83C-7280948
CAS :C-7280948 is a PRMT1 inhibitor.Formule :C14H16N2O2SDegré de pureté :99.55% - ≥95%Couleur et forme :SolidMasse moléculaire :276.35Ref: TM-T2097
5mg46,00€1mL*10mM (DMSO)49,00€10mg66,00€25mg109,00€50mg178,00€100mg268,00€200mg414,00€500mg667,00€Veliparib
CAS :Veliparib (ABT-888) (ABT-888) is an orally bioavailable inhibitor of PARP (Kis: 5.2/2.9 nM for PARP1/2). It enhances apoptosis and autophagy.Formule :C13H16N4ODegré de pureté :98.66% - 99%Couleur et forme :SolidMasse moléculaire :244.29Ref: TM-T2591
5mg54,00€1mL*10mM (DMSO)60,00€10mg77,00€25mg120,00€50mg195,00€100mg314,00€200mg512,00€500mg807,00€BI-847325
CAS :BI-847325 is a selective dual inhibitor of MEK and aurora kinases (AK) with IC50 values of 4 and 15 nM for human MEK2 and AK-C, respectively.Formule :C29H28N4O2Degré de pureté :97.13% - 97.54%Couleur et forme :SolidMasse moléculaire :464.56Tranylcypromine hemisulfate
CAS :Tranylcypromine hemisulfate (Tranylcypromine Sulfate) is an inhibitor of monoamine oxidase (MAO) and lysine-specific demethylase 1 (LSD1) with a rapid onset ofFormule :C9H11N1H2SO4Degré de pureté :98% - 99.96%Couleur et forme :SolidMasse moléculaire :182.23I-CBP112 hydrochloride
CAS :I-CBP112 selectively inhibits CBP/p300 bromodomains, with minimal effect on others, and reduces leukemia cell growth, enhancing JQ1 and doxorubicin's effects.Formule :C27H37ClN2O5Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :505.05Ref: TM-T4247
1mg86,00€2mg138,00€5mg225,00€10mg424,00€1mL*10mM (DMSO)424,00€25mg695,00€50mg973,00€100mg1.314,00€SGI-1027
CAS :SGI-1027 (DNA Methyltransferase Inhibitor II) is an effective and selective inhibitor of DNA methyltransferase (DNMT).Formule :C27H23N7ODegré de pureté :99.45% - 99.78%Couleur et forme :SolidMasse moléculaire :461.52Ref: TM-T1904
5mg58,00€1mL*10mM (DMSO)74,00€10mg94,00€25mg163,00€50mg296,00€100mg467,00€500mg1.035,00€GSK467
CAS :GSK467 is a potent and selective inhibitor of KDM5 (JARID1)(Ki : 10 nM).Formule :C17H13N5O2Degré de pureté :99.55% - 99.85%Couleur et forme :SolidMasse moléculaire :319.32Quercetagetin
CAS :Quercetagetin, a flavonoid from Citrus unshiu, inhibits pim-1 kinase (IC50: 0.34 μM), cell-permeable.Formule :C15H10O8Degré de pureté :99.65% - 99.91%Couleur et forme :SolidMasse moléculaire :318.24Ref: TM-T8114
1mg94,00€5mg192,00€1mL*10mM (DMSO)202,00€10mg286,00€25mg482,00€50mg695,00€100mg945,00€500mg1.882,00€MG 149
CAS :MG 149 (Tip60 HAT inhibitor) is a selective and potent Tip60 inhibitor with IC50 of 74 uM, similar potentcy for MOF(IC50= 47 uM).Formule :C22H28O3Degré de pureté :98.69% - 99.86%Couleur et forme :SolidMasse moléculaire :340.46Ref: TM-T6584
1mg50,00€2mg71,00€5mg90,00€1mL*10mM (DMSO)108,00€10mg167,00€25mg308,00€50mg492,00€100mg708,00€UNC3866
CAS :UNC3866 is a potent antagonist of the CBX7-H3 interaction as determined by AlphaScreen.Formule :C43H66N6O8Degré de pureté :88.06% - 99.62%Couleur et forme :SolidMasse moléculaire :795.02YKL-06-061
CAS :YKL-06-061 is a selective salt-inducible kinase (SIK) inhibitor with IC50 values of 6.56 nM/1.77 nM/20.5 nM for SIK1/2/3, respectively.Formule :C30H37N7O2Degré de pureté :99.52% - 99.79%Couleur et forme :SolidMasse moléculaire :527.66Birabresib
CAS :Birabresib (MK-8628) is a synthetic, small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family of bromodomain-containing proteins 2, 3 and 4Formule :C25H22ClN5O2SDegré de pureté :98.3% - 99.36%Couleur et forme :SolidMasse moléculaire :491.99Ref: TM-T6032
2mg46,00€5mg70,00€1mL*10mM (DMSO)74,00€10mg90,00€25mg142,00€50mg222,00€100mg375,00€200mg560,00€500mg893,00€GW779439X
CAS :GW779439X is an inhibitor of CDK.Formule :C22H21F3N8Degré de pureté :97.87%Couleur et forme :SolidMasse moléculaire :454.45Ref: TM-T8866
1mg58,00€2mg82,00€5mg113,00€1mL*10mM (DMSO)124,00€10mg178,00€25mg404,00€50mg592,00€100mg845,00€CCT241736
CAS :CCT241736 is an orally bioavailable dual FLT3/Aurora kinase inhibitor that also inhibits clinically relevant FLT3-resistant mutants including FLT3-ITD and FLT3Formule :C22H23Cl2N7Degré de pureté :96.2% - 99.81%Couleur et forme :SolidMasse moléculaire :456.37ACBI1
CAS :ACBI1 is a potent PROTAC degrader of BAF ATPase subunits SMARCA2 and SMARCA4, also degrades the polybromo-associated BAF (PBAF) complex member PBRM1, with DC50sFormule :C49H58FN9O7SDegré de pureté :97.54% - 98.15%Couleur et forme :SolidMasse moléculaire :936.1Amodiaquine
CAS :Amodiaquine is a synthetic aminoquinoline, used to treat malaria.Formule :C20H22ClN3ODegré de pureté :99.78% - 99.99%Couleur et forme :Crystals From Absolute Ethanol SolidMasse moléculaire :355.86Ref: TM-T8381
1mg49,00€2mg66,00€5mg90,00€1mL*10mM (DMSO)105,00€10mg170,00€25mg281,00€50mg394,00€100mg550,00€DMOG
CAS :DMOG (Dimethyloxalylglycine), an antagonist of the α-ketoglutarate cofactor, is an inhibitor for HIF prolyl hydroxylase.Formule :C6H9NO5Degré de pureté :80.23% - 99.98%Couleur et forme :SolidMasse moléculaire :175.14G244-LM
CAS :G244-LM is a potent and specific inhibitor of tankyrase 1/2. G244-LM inhibits Wnt signaling.Formule :C18H22N4O3S2Degré de pureté :98.46%Couleur et forme :SolidMasse moléculaire :406.52AMG 900
CAS :AMG 900 is a potent and highly selective pan-Aurora kinases inhibitor for Aurora A/B/C with IC50 of 5 nM/4 nM /1 nM.Formule :C28H21N7OSDegré de pureté :98.4% - 99.51%Couleur et forme :SolidMasse moléculaire :503.58Ref: TM-T6380
1mg49,00€5mg92,00€1mL*10mM (DMSO)100,00€10mg158,00€25mg286,00€50mg442,00€100mg645,00€500mg1.341,00€BGP-15
CAS :BGP-15 (BGP-15 2HCl) is a PARP inhibitor with protecting effect after ischemia-reperfusion injury.Formule :C14H24Cl2N4O2Degré de pureté :98.17% - 99.99%Couleur et forme :SolidMasse moléculaire :351.273-Methoxybenzamide
CAS :3-Methoxybenzamide (3-MBA) is a competitive inhibitor of poly(ADP-ribose) synthetase.Formule :C8H9NO2Degré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :151.16MR837
CAS :MR837 (NSD2-PWWP1 antagonist 3f) is a NSD2-PWWP1 antagonist.Formule :C16H14N2OSDegré de pureté :99.77% - 99.85%Couleur et forme :SolidMasse moléculaire :282.36Ref: TM-T8879
2mg38,00€5mg55,00€1mL*10mM (DMSO)66,00€10mg92,00€25mg138,00€50mg243,00€100mg355,00€200mg502,00€MK-8617
CAS :MK-8617 is an orally available HIF PHD1 3 pan-inhibitor, inhibiting PHD1/2/3 (IC50: 1.0/1.0/14 nM).Formule :C24H21N5O4Degré de pureté :99.38% - >99.99%Couleur et forme :SolidMasse moléculaire :443.45EPZ011989
CAS :EPZ011989: potent, selective oral EZH2 inhibitor, Ki < 3 nM, 15x more selective than EZH1, >3000x over other HMTases.Formule :C35H51N5O4Degré de pureté :98% - 99.45%Couleur et forme :SolidMasse moléculaire :605.81NVP-TNKS656
CAS :NVP-TNKS656 (TNKS656) is a highly potent, selective, and orally active TNKS2 inhibitor.Formule :C27H34N4O5Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :494.58Ref: TM-T3261
1mg43,00€2mg54,00€5mg84,00€1mL*10mM (DMSO)93,00€10mg122,00€25mg248,00€50mg421,00€100mg617,00€RBN012759
CAS :RBN012759 inhibits PARP14 protein and is more than 300-fold selective over all PARP family members.Cost-effective and quality-assured.Formule :C19H23FN2O3SDegré de pureté :98.87% - 99.96%Couleur et forme :SolidMasse moléculaire :378.46Ref: TM-T22414
2mgÀ demander1mg104,00€5mg250,00€1mL*10mM (DMSO)274,00€10mg373,00€25mg645,00€50mg938,00€100mg1.311,00€200mg1.768,00€1,2-Dipalmitoyl-sn-glycerol
CAS :1,2-Dipalmitoyl-sn-glycerol ((S)-1,2-Dipalmitin) is an analog of the PKC-activating second messenger diacylglycerol (DAG). It weakly activates PKC.Formule :C35H68O5Degré de pureté :97.84% - 99.78%Couleur et forme :SolidMasse moléculaire :568.91Amifostine trihydrate
CAS :Amifostine trihydrate (WR2721) is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.Formule :C5H15N2O3PS·3H2ODegré de pureté :99.71% - 99.80%Couleur et forme :SolidMasse moléculaire :268.27Fosifidancitinib
CAS :Fosifidancitinib is a potent inhibitor of JAK 1 and JAK 3.Formule :C21H21FN5O7PDegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :505.39Ref: TM-T38624
1mg93,00€2mg117,00€5mg177,00€10mg269,00€25mg429,00€50mg610,00€100mg820,00€200mg1.099,00€Atractylenolide I
CAS :Atractylenolide-I reduces inflammation, improves sepsis, liver, and kidney function, and enhances EOC cell sensitivity to paclitaxel.Formule :C15H18O2Degré de pureté :97.55% - 99.92%Couleur et forme :SolidMasse moléculaire :230.30PF-CBP1
CAS :PF-CBP1 HCl is a highly selective inhibitor of the bromodomain of CREB-binding protein(CREBBP).Formule :C29H36N4O3Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :488.62MI-463
CAS :MI-463 is a potent and orally bioavailable inhibitor of the menin-mLL interaction (IC50: 15.3 nM).Formule :C24H23F3N6SDegré de pureté :99.18% - >99.99%Couleur et forme :SolidMasse moléculaire :484.54KC7F2
CAS :KC7F2 is a potent HIF-1 pathway inhibitor with potential anti-cancer activity.Formule :C16H16Cl4N2O4S4Degré de pureté :98% - 99.11%Couleur et forme :SolidMasse moléculaire :570.38Bempedoic acid
CAS :Bempedoic acid (ETC1002) is an orally available, once-daily LDL-C lowering small molecule designed to lower elevated levels of LDL-C.Formule :C19H36O5Degré de pureté :99.85% - 99.94%Couleur et forme :SolidMasse moléculaire :344.49Ref: TM-T3625
2mg34,00€5mg50,00€1mL*10mM (DMSO)52,00€10mg70,00€25mg118,00€50mg207,00€100mg333,00€500mg797,00€GLPG0634 analog
CAS :GLPG0634 analog (GLPG0634 analogue) is a specific JAK1 inhibitor with IC50 of 10/28/810/116 nM for JAK1/2/3 and TYK2, respectively.Formule :C23H18N6O2Degré de pureté :99.52% - >99.99%Couleur et forme :SolidMasse moléculaire :410.43Ref: TM-T3076
1mg38,00€2mg50,00€5mg84,00€1mL*10mM (DMSO)93,00€10mg137,00€25mg250,00€50mg442,00€100mg623,00€500mg1.305,00€COH-SR4
CAS :COH-SR4 (COH-SR4 (Mitochondria uncoupler SR4)) is a uncoupler of mitochondrial oxidative phosphorylation.Formule :C13H8Cl4N2ODegré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :350.03WZ4003
CAS :WZ4003, a highly selective NUAK kinase inhibitor, is with IC50 of 20 nM and 100 nM for NUAK1 and NUAK2, respectively.Formule :C25H29ClN6O3Degré de pureté :99.65% - >99.99%Couleur et forme :SolidMasse moléculaire :496.99Ref: TM-T6291
5mg48,00€1mL*10mM (DMSO)50,00€10mg73,00€25mg111,00€50mg166,00€100mg241,00€200mg358,00€500mg590,00€ABBV-744
CAS :ABBV-744 is a BDII-selective BET bromodomain inhibitor that inhibits BRD2/3/4. It is used in the research on inflammatory diseases, cancer, and AIDS.Formule :C28H30FN3O4Degré de pureté :97.03% - >99.99%Couleur et forme :SolidMasse moléculaire :491.55Ref: TM-T4697
1mg44,00€2mg56,00€5mg90,00€1mL*10mM (DMSO)90,00€10mg142,00€25mg284,00€50mg409,00€100mg500,00€200mg718,00€BRD4770
CAS :BRD4770 is a histone methyltransferase G9a inhibitor and induces cell senescence.Formule :C25H23N3O3Degré de pureté :99.53% - 99.82%Couleur et forme :SolidMasse moléculaire :413.47ARV-771
CAS :ARV-771 is an effective BET degrader based on PROTAC technology.Cost-effective and quality-assured.Formule :C49H60ClN9O7S2Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :986.64Ref: TM-T5435
1mg57,00€5mg113,00€10mg177,00€1mL*10mM (DMSO)192,00€25mg354,00€50mg522,00€100mg732,00€200mg973,00€SHR0302
CAS :SHR0302 (ARQ252) is a JAK inhibitor that binds JAK1 with stronger affinity than others (Selectivity for JAK1 is more than 10 times for JAK2, 77 times for JAK3,Formule :C18H22N8O2SDegré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :414.48Ref: TM-T9195
1mg75,00€1mL*10mM (DMSO)164,00€5mg173,00€10mg281,00€25mg485,00€50mg773,00€100mg1.243,00€Oclacitinib maleate
CAS :Oclacitinib maleate is a selective JAK inhibitor (IC50: 10-99 nM; JAK1 cytokines: 36-249 nM), with no effect on 38 non-JAK kinases.Formule :C15H23N5O2S·C4H4O4Degré de pureté :99.17% - 99.92%Couleur et forme :SolidMasse moléculaire :453.51Ref: TM-T6914
1mg37,00€2mg52,00€5mg74,00€1mL*10mM (DMSO)81,00€10mg94,00€25mg166,00€50mg258,00€100mg432,00€Ethyl 3,4-dihydroxybenzoate
CAS :Ethyl 3,4-dihydroxybenzoate (EDHB): a prolyl hydroxylase inhibitor attenuates acute hypobaric hypoxia mediated vascular leakage in brain.Formule :C9H10O4Degré de pureté :99.88%Couleur et forme :White Crystal Or PowderMasse moléculaire :182.17XMD8-92
CAS :XMD8-92 is an effective and specific BMK1/ERK5 inhibitor (Kd: 80 nM).Formule :C26H30N6O3Degré de pureté :98.21%Couleur et forme :SolidMasse moléculaire :474.55JQEZ5
CAS :JQEZ5 is an inhibitor of EZH2 lysine methyltransferase (IC50 = 11.1 nM).Formule :C30H38N8O2Degré de pureté :98.14% - ≥98%Couleur et forme :SolidMasse moléculaire :542.68BRD9539
CAS :BRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2), also known as G9a, with an IC50 value of 6.3 μMFormule :C24H21N3O3Degré de pureté :98% - 99.57%Couleur et forme :SolidMasse moléculaire :399.44ICG001
CAS :ICG001 antagonizes Wnt signaling, binds CBP with 3 μM IC50, not p300.Formule :C33H32N4O4Degré de pureté :99.06% - 99.95%Couleur et forme :SolidMasse moléculaire :548.63Ref: TM-T2237
1mg34,00€5mg66,00€1mL*10mM (DMSO)81,00€10mg101,00€25mg197,00€50mg341,00€100mg530,00€500mg1.134,00€Bromosporine
CAS :Bromosporine is a broad spectrum inhibitor for bromodomains for BRD2/4/9 and CECR2 (IC50: 0.41/0.29/0.122/0.017 μM), respectively.Formule :C17H20N6O4SDegré de pureté :99.65% - 99.79%Couleur et forme :SolidMasse moléculaire :404.44Ref: TM-T6255
1mg44,00€2mg57,00€1mL*10mM (DMSO)92,00€5mg93,00€10mg133,00€25mg260,00€50mg416,00€100mg665,00€200mg888,00€MLN8054
CAS :MLN8054 is a potent and selective Aurora A kinase inhibitor with an IC50 of 4 nM.Formule :C25H15ClF2N4O2Degré de pureté :98.07% - 98.26%Couleur et forme :SolidMasse moléculaire :476.86Ref: TM-T6315
1mg50,00€2mg67,00€5mg84,00€1mL*10mM (DMSO)88,00€10mg120,00€25mg220,00€50mg356,00€100mg537,00€EED226
CAS :EED226 is a potent, selective, and orally bioavailable embryonic ectoderm development (EED) inhibitor with an IC50 of 22 nM.Formule :C17H15N5O3SDegré de pureté :98.14% - 99.33%Couleur et forme :SolidMasse moléculaire :369.4RK-287107
CAS :RK-287107 is an effective and specific inhibitor of tankyrase (IC50s: 14.3 and 10.6 nM for tankyrase-1 and tankyrase-2, respectively).Formule :C22H26F2N4O2Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :416.46Hispidulin
CAS :Hispidulin, a natural flavone with a broad spectrum of biological activities, is a Pim-1 inhibitor (IC50: 2.71 μM).Formule :C16H12O6Degré de pureté :98.53% - 99.87%Couleur et forme :SolidMasse moléculaire :300.26SGC-SMARCA-BRDVIII
CAS :SGC-SMARCA-BRDVIII is a potent and selective inhibitor of SMARCA2, SMARCA4, PB1(2), PB1(3) and PB1(5) with Kds of 35 nM, 36 nM, 3.7 μM, 2.0 μM and 13 nM,Formule :C19H25N5O3Degré de pureté :99.54% - 99.92%Couleur et forme :SolidMasse moléculaire :371.43Ref: TM-T9568
1mg44,00€1mL*10mM (DMSO)54,00€5mg66,00€10mg101,00€25mg222,00€50mg356,00€100mg530,00€500mg1.153,00€Acetyl Pentapeptide-1 acetate
Acetyl Pentapeptide-1 acetate is an histone deacetylase inhibitor.Formule :C34H55N9O12Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :781.86Fraxinellone
CAS :1.Formule :C14H16O3Degré de pureté :99.35% - 99.92%Couleur et forme :SolidMasse moléculaire :232.27Ref: TM-T6S0071
2mg34,00€5mg50,00€1mL*10mM (DMSO)81,00€10mg84,00€25mg152,00€50mg222,00€100mg334,00€200mg494,00€AZ6102
CAS :AZ6102: Potent TNKS1/2 inhibitor, 100x selective over PARPs, IC50 = 5 nM in DLD-1 Wnt pathway.Formule :C25H28N6ODegré de pureté :97.98% - 99.91%Couleur et forme :SolidMasse moléculaire :428.53ZM-447439
CAS :ZM 447439 selectively inhibits Aurora A/B (IC50: 110/130 nM); 8x less effective on MEK1, Src, Lck; minimal impact on CDK1/2/4, Plk1, Chk1.Formule :C29H31N5O4Degré de pureté :99.11% - 99.59%Couleur et forme :Pale Yellow SolidMasse moléculaire :513.59CPI203
CAS :CPI203 (CPI 203) is an effective BET bromodomain inhibitor (IC50: 37 nM for BRD4).Formule :C19H18ClN5OSDegré de pureté :99.13% - 99.77%Couleur et forme :SolidMasse moléculaire :399.9MM-102 TFA
CAS :MM-102 TFA is a potent WDR5/MLL inhibitor with IC50 of 2.4 nM; it disrupts MLL1-WDR5 interaction, impeding H3K4 HMT activity.Formule :C37H50F5N7O6Degré de pureté :99.4% - 99.78%Couleur et forme :SolidMasse moléculaire :783.83Ref: TM-T8768
1mg37,00€2mg49,00€5mg100,00€1mL*10mM (DMSO)141,00€10mg165,00€25mg269,00€50mg399,00€100mg587,00€OG-L002
CAS :OG-L002 is an effective and selective LSD1 inhibitor (IC50: 20 nM), showing 69- and 36-fold selectivity over MAO-A and MAO-B, respectively.Formule :C15H15NODegré de pureté :97.05% - 98.62%Couleur et forme :SolidMasse moléculaire :225.29AG490
CAS :AG490 inhibits EGFR (0.1 μM IC50), 135x > selective than ErbB2, blocks JAK2, spares Lyn, Lck, Syk, Btk, Src.Formule :C17H14N2O3Degré de pureté :98.6% - 99.85%Couleur et forme :Yellow SolidMasse moléculaire :294.3Fedratinib hydrochloride hydrate
CAS :Fedratinib hydrochloride hydrate (SAR 302503 hydrochloride hydrate) is a potent, selective, ATP-competitive and orally active JAK2 inhibitor.Formule :C27H40Cl2N6O4SDegré de pureté :98.96% - 99.87%Couleur et forme :SolidMasse moléculaire :615.61PARP1-IN-5 dihydrochloride
CAS :PARP1-IN-5 dihydrochloride: oral, potent PARP-1 inhibitor (IC50=14.7 nM), for cancer research.Formule :C25H26Cl2N2O5SDegré de pureté :98.01%Couleur et forme :SolidMasse moléculaire :537.46BMS-911543
CAS :BMS-911543 is a potent and selective inhibitor of JAK2 with IC50 of 1.1 nM, ~350-, 75- and 65-fold selective to JAK1, JAK3 and TYK2, respectively. Phase 1/2.Formule :C23H28N8ODegré de pureté :97.69% - 99.98%Couleur et forme :SolidMasse moléculaire :432.52CCT 137690
CAS :CCT 137690 is a highly specific and oral-available aurora kinase inhibitor, for aurora A(IC50=15 nM ), B(IC50=25 nM) and C(IC50=19 nM).Formule :C26H31BrN8ODegré de pureté :98.51% - 99.89%Couleur et forme :SolidMasse moléculaire :551.48Hinokitiol
CAS :Hinokitiol prevents UVB-caused cell death, boosts antioxidant activity, and hinders breast cancer growth.Formule :C10H12O2Degré de pureté :99.49% - 99.98%Couleur et forme :SolidMasse moléculaire :164.2Tazemetostat hydrobromide
CAS :Tazemetostat hydrobromide: potent, selective EZH2 inhibitor; blocks PRC2/wild-type EZH2 (Ki: 2.5 nM) & EZH1 (IC50: 392 nM).Formule :C34H45BrN4O4Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :653.65Ref: TM-T17002
2mg40,00€5mg57,00€10mg77,00€1mL*10mM (DMSO)79,00€50mg90,00€100mg150,00€200mg219,00€500mg358,00€TAK-632
CAS :TAK-632 is a potent pan-Raf inhibitor.Formule :C27H18F4N4O3SDegré de pureté :98% - 99.5%Couleur et forme :SolidMasse moléculaire :554.52MRTX9768
CAS :MRTX-9768 is a synthetic lethal-based inhibitor designed to bind the PRMT5-MTA complex and selectively target MTAP/CDKN2A-deleted tumors.Formule :C24H17FN6ODegré de pureté :97.02%Couleur et forme :SolidMasse moléculaire :424.43MK-4827 Racemate
CAS :MK-4827 Racemate (Niraparib Racemate) is a selective PARP1 and PARP2 inhibitor with IC50s of 3.8 nM and 2.1 nM, respectively, over 330-fold selectivity forFormule :C19H20N4ODegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :320.39Ref: TM-T22988
1mg50,00€2mg65,00€5mg93,00€1mL*10mM (DMSO)112,00€10mg145,00€25mg268,00€50mg467,00€100mg628,00€FM-381
CAS :FM381, a JAK3 inhibitor with 127 pM IC50, is 410-3600x more selective over JAK1/2/TYK2.Formule :C24H24N6O2Degré de pureté :98.44%Couleur et forme :SolidMasse moléculaire :428.49Ref: TM-T5091
1mg47,00€2mg62,00€5mg92,00€1mL*10mM (DMSO)107,00€10mg128,00€25mg212,00€50mg319,00€100mg485,00€CPI-169 racemate
CAS :CPI-169 racemate (CPI 169) is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively.
Formule :C27H36N4O5SDegré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :528.66JW 55
CAS :JW 55 (JW55) is an effective and selective β-catenin signaling pathway inhibitor, works by inhibition of the PARP domain of tankyrase 1 and tankyrase 2 (TNKS1/2Formule :C25H26N2O5Degré de pureté :99.31% - 99.76%Couleur et forme :SolidMasse moléculaire :434.48BMS-P5
CAS :BMS-P5 is a specific and orally active Peptidylarginine Deiminase 4 (PAD4) inhibitor.Formule :C27H33ClN6O2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :509.04Ref: TM-T22277
2mg44,00€5mg86,00€1mL*10mM (DMSO)96,00€10mg136,00€25mg268,00€50mg479,00€100mg760,00€200mg1.018,00€TG101209
CAS :TG101209 is a selective JAK2 inhibitor with IC50 of 6 nM.Formule :C26H35N7O2SDegré de pureté :99% - >99.99%Couleur et forme :SolidMasse moléculaire :509.67TIQ-A
CAS :TIQ-A blocks PARP1 to prevent excessive DNA damage response, implicated in ischemia, asthma, and atherosclerosis.Formule :C11H7NOSDegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :201.24Ref: TM-T50098
1mg52,00€5mg92,00€1mL*10mM (DMSO)96,00€10mg161,00€25mg290,00€50mg414,00€100mg532,00€200mg737,00€BET bromodomain inhibitor
CAS :BET bromodomain inhibitor is a potent BET inhibitor.Formule :C24H20ClN5O2Degré de pureté :98.22% - 99.85%Couleur et forme :SolidMasse moléculaire :445.9Ref: TM-T2072
1mg35,00€2mg50,00€5mg75,00€1mL*10mM (DMSO)84,00€10mg114,00€25mg187,00€50mg264,00€100mg416,00€4-amino-1,8-Naphthalimide
CAS :4-amino-1,8-Naphthalimide (4-ANI) is a PARP inhibitor with IC50 of 180 nMFormule :C12H8N2O2Degré de pureté :95.13%Couleur et forme :Yellow Solid PowderMasse moléculaire :212.2BMS-P5 free base
CAS :BMS-P5 free base is a specific and orally active peptidylarginine deiminase 4 (PAD4) inhibitor.Formule :C27H32N6O2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :472.58AS8351
CAS :AS8351 inhibits histone demethylase, used with various compounds to turn human lung fibroblasts into cardiomyocytes.Formule :C17H13N3O2Degré de pureté :99.54% - 99.72%Couleur et forme :SolidMasse moléculaire :291.3Ref: TM-T4100
5mg48,00€1mL*10mM (DMSO)49,00€10mg66,00€25mg110,00€50mg178,00€100mg333,00€200mg432,00€500mg707,00€PFI-2 hydrochloride
CAS :PFI-2 hydrochloride ((R)-PFI-2 hydrochloride) is a potent, highly selective, and cell-active inhibitor of the methyltransferase activity of SETD7 (IC50: 2 nM),Formule :C23H26ClF4N3O3SDegré de pureté :99.31% - 99.91%Couleur et forme :SolidMasse moléculaire :535.98Ref: TM-T4583
1mg38,00€2mg49,00€5mg80,00€10mg111,00€1mL*10mM (DMSO)122,00€25mg200,00€50mg358,00€100mg523,00€500mg1.108,00€ENMD-2076
CAS :ENMD-2076, a multi-targeted kinase inhibitor, has specific activity against Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, FGFR2, Src, PDGFRα.Formule :C21H25N7Degré de pureté :97.63% - ≥95%Couleur et forme :SolidMasse moléculaire :375.47KDM4D-IN-1
CAS :KDM4D-IN-1 is a KDM4D inhibitor (IC50: 0.41±0.03 μM).Formule :C11H7N5ODegré de pureté :99.51% - >99.99%Couleur et forme :SolidMasse moléculaire :225.21Ref: TM-T4214
1mg73,00€5mg158,00€1mL*10mM (DMSO)168,00€10mg245,00€25mg495,00€50mg795,00€100mg1.161,00€(Z)-SMI-4a
CAS :(Z)-SMI-4a (TCS PIM-1 4a) is a selective ATP-competitive Pim-1 kinase inhibitor with an IC50 of 21 nM.Formule :C11H6F3NO2SDegré de pureté :97.66% - 99.93%Couleur et forme :SolidMasse moléculaire :273.23WDR5-0103 hydrochloride[890190-22-4(free base)]
WDR5-0103 hydrochloride[890190-22-4(free base)] (WD-Repeat Protein 5-0103) is an effective and specific WD repeat-containing protein 5 (WDR5) antagonist (Kd:Formule :C21H26ClN3O4Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :419.96-Bromo-3-methyl-1,4-dihydroquinazolin-2-one
CAS :CHEMBRDG-BB 7118966 is an inhibitor of Bromodomain-containing protein 4 (human).Formule :C9H9BrN2ODegré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :241.08Ref: TM-T8609
1mg58,00€1mL*10mM (DMSO)107,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€Aurora kinase inhibitor-3
CAS :Aurora kinase inhibitor-3 (Aurora Kinase Inhibitor III) is a potent inhibitor of Aurora A kinase (IC50 = 42 nM).1 It is selective for Aurora A over BMX, BTK,Formule :C21H18F3N5ODegré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :413.4Ref: TM-T5524
1mg66,00€2mg89,00€5mg152,00€1mL*10mM (DMSO)167,00€10mg236,00€25mg401,00€50mg580,00€100mg797,00€200mg1.099,00€3-methyl-1,2-dihydroquinolin-2-one
CAS :3-methyl-1,2-dihydroquinolin-2-one is the first known micromolar inhibitors of the ATAD2 bromodomain.Formule :C10H9NODegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :159.18Ref: TM-T50035
1mg35,00€1mL*10mM (DMSO)62,00€5mg77,00€10mg103,00€25mg170,00€50mg250,00€100mg354,00€200mg480,00€TCS PIM-1 1
CAS :TCS PIM-1 1 (SC 204330) is a potent ATP-competitive inhibitor of Pim-1 kinase with an IC50 of 50 nM, selective over MEK1/2 and Pim-2.Formule :C18H11BrN2O2Degré de pureté :97% - 97.98%Couleur et forme :SolidMasse moléculaire :367.2Ref: TM-T2253
1mg34,00€5mg60,00€1mL*10mM (DMSO)92,00€10mg94,00€25mg177,00€50mg269,00€100mg401,00€200mg580,00€Oclacitinib
CAS :Oclacitinib (PF-03394197)(PF03394197) is a potent and selective JAKs inhibitor with IC50 of 10-99 nM; not inhibit a panel of 38 non-JAK kinases (IC50 's > 1000Formule :C15H23N5O2SDegré de pureté :98% - 98.45%Couleur et forme :White To Off-White SolidMasse moléculaire :337.44lutidinic acid
CAS :lutidinic acid (2,4-Dicarboxypyridine) is an in vitro and in cell inhibitor, as well as a known inhibitor of the histone lysine demethylases.
Formule :C7H5NO4Degré de pureté :98.06%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :167.12UNC 669
CAS :UNC 669 is an effective and specific MBT (malignant brain tumor) inhibitor with IC50 of 4.2/3.1 uM for L3MBTL1/3.Formule :C15H20BrN3ODegré de pureté :97.38%Couleur et forme :SolidMasse moléculaire :338.24XY1
CAS :XY1 is a very close analogue of SGC707 (a potent, selective, and non-competitive inhibitor of PRMT3 with IC50 of 31 nM), It is intended to be used as aFormule :C17H19N3O2Degré de pureté :97.74% - 99%Couleur et forme :SolidMasse moléculaire :297.35AZD5153 6-Hydroxy-2-naphthoic acid
CAS :AZD5153 6-Hydroxy-2-naphthoic acid (AZD5153) is a potent triazolopyridazine-based Bromodomain (BRD4) and Extraterminal (BET) inhibitor used in cancer treatmentsFormule :C25H33N7O3·C11H8O3Degré de pureté :97.26% - ≥95%Couleur et forme :SolidMasse moléculaire :667.75Gusacitinib HCl
CAS :Gusacitinib (ASN-002/EN-3351), a potent SYK/JAK inhibitor, has strong antitumor activity in various cancers.Formule :C24H29ClN8O2Couleur et forme :SolidMasse moléculaire :497RG108
CAS :RG108 (N-Phthalyl-L-tryptophan) is an DNA methyltransferase inhibitor(IC50=115 nM).Formule :C19H14N2O4Degré de pureté :98% - 99.43%Couleur et forme :SolidMasse moléculaire :334.33Ref: TM-T2038
5mg44,00€1mL*10mM (DMSO)52,00€10mg65,00€25mg111,00€50mg195,00€100mg271,00€200mg380,00€500mg618,00€CP21R7
CAS :CP21 is a specific GSK3β inhibitor, used to activate stem cells for differentiation, often paired with BMP4 for mesodermal fate.Formule :C19H15N3O2Degré de pureté :96.14% - 99.16%Couleur et forme :SolidMasse moléculaire :317.34Ref: TM-T3684
1mg38,00€2mg50,00€1mL*10mM (DMSO)77,00€5mg84,00€10mg120,00€25mg236,00€50mg356,00€100mg537,00€HDAC8-IN-1
CAS :MDK-7933 (HDAC8-IN-1) is a HDAC8 inhibitor with an IC50 of 27.2 nM in cancer cell lines.Formule :C22H19NO3Degré de pureté :97.13% - 99.19%Couleur et forme :SolidMasse moléculaire :345.39Ref: TM-T7082
1mg34,00€5mg63,00€1mL*10mM (DMSO)70,00€10mg95,00€25mg172,00€50mg259,00€100mg330,00€200mg467,00€SGC-CBP30
CAS :SGC-CBP30 is an effective CREBBP/EP300 inhibitor (IC50: 21/38 nM).Formule :C28H33ClN4O3Degré de pureté :99.05% - >99.99%Couleur et forme :SolidMasse moléculaire :509.04Ref: TM-T6668
1mg50,00€2mg67,00€5mg84,00€1mL*10mM (DMSO)94,00€10mg113,00€25mg200,00€50mg334,00€100mg500,00€MC1568
CAS :MC1568 is a specific HDAC inhibitor for maize HD1-A (IC50: 100 nM, in a cell-free assay). It is 34-fold more selective for HD1-A than HD1-B.Formule :C17H15FN2O3Degré de pureté :89.82% - ≥95%Couleur et forme :SolidMasse moléculaire :314.31NMS-P118
CAS :NMS-P118 is a potent, selective and orally available Inhibitor of PARP-1 for cancer therapy.Formule :C20H24F3N3O2Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :395.42SGI-1776
CAS :SGI-1776 (Pim-Kinase Inhibitor IX) has been used in trials studying the treatment of Prostate Cancer, Non-Hodgkins Lymphoma, and Relapsed/Refractory Leukemias.Formule :C20H22F3N5ODegré de pureté :99.3% - >99.99%Couleur et forme :SolidMasse moléculaire :405.42Ref: TM-T3078
1mgÀ demander5mg90,00€1mL*10mM (DMSO)94,00€10mg145,00€25mg281,00€50mg409,00€100mg528,00€SRT 1720 dihydrochloride
CAS :SRT 1720 dihydrochloride is a selective activator of SIRT1 (EC1.5: 0.16 μM) and shows less potent activities on SIRT2 (EC1.5: 37 μM) and SIRT3 (EC1.5: 300 μM).Formule :C25H25Cl2N7OSDegré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :542.482-hexyl-4-Pentynoic Acid
CAS :2-hexyl-4-Pentynoic Acid, a valproic acid (VPA) derivatives, is a potent and robust HDACs inhibitor with IC50 value of 13 μM.Formule :C11H18O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :182.26Protein Kinase C 19-31 acetate
PKC 19-31 acetate, a serine-altered PKCa-derived PKC inhibitor, tests PKC activity.Formule :C69H122N26O18Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1603.9PKC-θ inhibitor hcl
CAS :PKC-theta inhibitor hcl is a selective PKC-θinhibitor(IC50:12 nM).Formule :C20H26ClF3N6O3Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :490.91Ref: TM-T5817
1mg88,00€2mg114,00€5mg220,00€10mg356,00€25mg595,00€50mg848,00€100mg1.153,00€500mg2.305,00€SIS17
CAS :SIS17: Potent, selective HDAC11 inhibitor (IC50: 0.83 μM), blocks serine hydroxymethyl transferase 2 demyristoylation, spares other HDACs.Formule :C21H38N2OSDegré de pureté :98.22%Couleur et forme :SolidMasse moléculaire :366.6Darovasertib
CAS :Darovasertib (LXS196) is a potent PKC inhibitor, orally active, with IC50 of 1.9 nM (PKCα), 0.4 nM (PKCθ), 3.1 μM (GSK3β).Formule :C22H23F3N8ODegré de pureté :98.72% - ≥95%Couleur et forme :SolidMasse moléculaire :472.47Remetinostat
CAS :Remetinostat (SHP-141), a hydroxamic acid-based inhibitor of histone deacetylase enzymes, is currently being developed for the treatment of cutaneous T-cellFormule :C16H21NO6Degré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :323.34Thiomyristoyl
CAS :Thiomyristoyl is an effective and selective SIRT2 inhibitor (IC50: 28 nM). It inhibits SIRT1 (IC50: 98 μM) but no effect on SIRT3 even at 200 μM.Formule :C34H51N3O3SDegré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :581.85Ref: TM-T3447
1mg54,00€2mg73,00€5mg92,00€10mg117,00€1mL*10mM (DMSO)117,00€25mg215,00€50mg360,00€100mg537,00€Tucidinostat
CAS :Tucidinostat is an oral HDAC1/2/3/10 inhibitor (IC50: 67-160 nM), weaker on HDAC8/11, inactive on HDAC4/5/6/7/9.Formule :C22H19FN4O2Degré de pureté :97.01% - 99.95%Couleur et forme :SolidMasse moléculaire :390.41Ref: TM-T4481
5mg60,00€1mL*10mM (DMSO)60,00€10mg95,00€25mg159,00€50mg250,00€100mg399,00€200mg558,00€500mg832,00€M344
CAS :M344 (Histone Deacetylase Inhibitor III) is a potent HDAC inhibitor with IC50 of 100 nM and able to induce cell differentiation.Formule :C16H25N3O3Degré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :307.39Daphnetin
CAS :Daphnetin (7,8-Dihydroxycoumarin), a natural coumarin derivative, is a protein kinase inhibitor with inhibitory for EGFR (IC50: 7.67 μM), PKA (IC50: 9.33 μM),
Formule :C9H6O4Degré de pureté :97.47% - 99.8%Couleur et forme :SolidMasse moléculaire :178.14CYC-116
CAS :CYC116 is a potent inhibitor of Aurora A/B with Ki of 8.0 nM/9.2 nM, is less potent to VEGFR2 (Ki of 44 nM), with 50-fold greater potency than CDKs, not activeFormule :C18H20N6OSDegré de pureté :97.36% - 97.59%Couleur et forme :SolidMasse moléculaire :368.46SC-43
CAS :SC-43 is a potent and orally active agonist of SHP-1 (PTPN6).Formule :C21H13ClF3N3O2Degré de pureté :98.44%Couleur et forme :SolidMasse moléculaire :431.8Ruboxistaurin
CAS :Ruboxistaurin (LY333531) is a selective PKC beta inhibitor, Ki 2 nM, inhibits beta I/II (IC50: 4.7/5.9 nM), orally active.Formule :C28H28N4O3Couleur et forme :SolidMasse moléculaire :468.55ORY1001
CAS :ORY1001: Oral LSD1/KDM1A inhibitor, highly selective, IC50 <20 nM.Formule :C15H22N2·2HClDegré de pureté :99.85% - 99.96%Couleur et forme :SolidMasse moléculaire :303.27Ref: TM-T6922
1mg56,00€2mg79,00€5mg127,00€1mL*10mM (DMSO)127,00€10mg221,00€25mg427,00€50mg625,00€100mg889,00€500mg1.783,00€Rucaparib acetate
CAS :Rucaparib acetate, an oral PARP-1, -2, -3 inhibitor (Ki 1.4 nM for PARP1), also moderately inhibits H6PD; promising for CRPC research.Formule :C21H22FN3O3Couleur et forme :SolidMasse moléculaire :383.423RGFP966
CAS :RGFP966 is an HDAC3 inhibitor (IC50: 0.08 μM) and does not affect other HDACs at concentrations up to 15 μM.Formule :C21H19FN4ODegré de pureté :99.2% - 99.88%Couleur et forme :SolidMasse moléculaire :362.4Ref: TM-T1762
1mg34,00€2mg49,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg99,00€25mg160,00€50mg245,00€100mg356,00€Ritlecitinib
CAS :Ritlecitinib (PF-06651600) is an orally available, selective JAK3 inhibitor and does not affect the activity of JAK1/2.Cost-effective and quality-assured.Formule :C15H19N5ODegré de pureté :98.82% - 99.92%Couleur et forme :SolidMasse moléculaire :285.34Ref: TM-T5382
2mg37,00€5mg52,00€1mL*10mM (DMSO)73,00€10mg90,00€25mg205,00€50mg290,00€100mg408,00€200mg595,00€AK-1
CAS :AK-1: SIRT2 inhibitor, IC50 12.5 μM, hinders Alzheimer's neurodegeneration, arrests colon cancer cell cycle.Formule :C19H21N3O5SDegré de pureté :98.32% - 99.44%Couleur et forme :SolidMasse moléculaire :403.45Pim1/AKK1-IN-1
CAS :Pim1/AKK1-IN-1: LKB1/AAK1 inhibitor with Kd 35/53/75/380 nM for Pim1/AKK1/MST2/LKB1, also targets MPSK1, TNIK.Formule :C20H13N5ODegré de pureté :97.03% - 98.69%Couleur et forme :SolidMasse moléculaire :339.35Ref: TM-T5093
1mg85,00€2mg124,00€5mg173,00€1mL*10mM (DMSO)192,00€10mg263,00€25mg464,00€50mg672,00€100mg945,00€LMK-235
CAS :LMK-235 is a potent HDAC inhibitor, and is used in cancer research.Formule :C15H22N2O4Degré de pureté :98.18% - 99.68%Couleur et forme :SolidMasse moléculaire :294.35Ref: TM-T6061
1mL*10mM (DMSO)49,00€5mg52,00€10mg74,00€25mg132,00€50mg222,00€100mg403,00€200mg593,00€500mg888,00€Bisindolylmaleimide IV
CAS :Bisindolylmaleimide IV is a protein kinase C (PKC) cell permeable inhibitor( IC50 : 0.10 - 0.55 μM)
Formule :C20H13N3O2Degré de pureté :98.83%Couleur et forme :Dark Red SolidMasse moléculaire :327.34Senaparib
CAS :Senaparib (IMP4297) is a novel highly potent and selective oral PARP1/2 inhibitor with strong antitumor activity.Formule :C24H20F2N6O3Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :478.45Ref: TM-T9593
1mg46,00€2mg59,00€5mg87,00€1mL*10mM (DMSO)96,00€10mg153,00€25mg274,00€50mg432,00€100mg638,00€Pacritinib
CAS :Pacritinib (SB1518) (SB1518) is an effective and specific inhibitor of JAK2 and FLT3 (IC50: 23/22 nM, in cell-free assays).Formule :C28H32N4O3Degré de pureté :99.25% - 99.49%Couleur et forme :SolidMasse moléculaire :472.58XL019
CAS :XL019 is a potent and selective JAK2 inhibitor with IC50 of 2.2 nM, 100 fold selectivity over JAK1.Formule :C25H28N6O2Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :444.53Ref: TM-T3072
2mg43,00€5mg63,00€1mL*10mM (DMSO)78,00€10mg92,00€25mg150,00€50mg215,00€100mg321,00€200mg477,00€G007-LK
CAS :G007-LK is a selective inhibitor of TNKS1 and TNKS2, with IC50s of 46 nM and 25 nM, respectively.Formule :C25H16ClN7O3SDegré de pureté :97.63% - 98.17%Couleur et forme :SolidMasse moléculaire :529.96Ref: TM-T6842
1mg50,00€2mg66,00€5mg94,00€1mL*10mM (DMSO)116,00€10mg158,00€25mg315,00€50mg502,00€100mg707,00€ITSA-1
CAS :ITSA-1 is membrane permeable and specifically suppresses TSA inhibition of HDAC (histone deacetylase), but shows no activity towards other HDAC inhibitors.Formule :C13H7Cl2N3ODegré de pureté :99.78% - 99.89%Couleur et forme :SolidMasse moléculaire :292.12Ref: TM-T3358
10mg34,00€1mL*10mM (DMSO)54,00€25mg66,00€50mg90,00€100mg152,00€200mg219,00€500mg358,00€Danusertib
CAS :Danusertib (PHA-739358) is a small-molecule 3-aminopyrazole derivative with potential antineoplastic activity.Formule :C26H30N6O3Degré de pureté :97.88% - 98.79%Couleur et forme :White PowderMasse moléculaire :474.55AZD-1480
CAS :AZD1480: JAK2 inhibitor, IC50 0.26 nM; selective vs Tyk2, JAK3; less on JAK1. Used in solid tumors, PPV, PMF, ET trials.Formule :C14H14ClFN8Degré de pureté :98.25% - 99.47%Couleur et forme :SolidMasse moléculaire :348.77KW-2449
CAS :KW-2449 is a multiple-targeted inhibitor, mostly for Flt3, modestly effective to Bcr-Abl, FGFR1, and Aurora A; little inhibitory on PDGFRβ, IGF-1R, EGFR.Formule :C20H20N4ODegré de pureté :98.43% - 99.69%Couleur et forme :SolidMasse moléculaire :332.4CXD101
CAS :CXD101 is a novel class I-selective HDACi (HDAC1 (IC50 : 63nM), HDAC2 (IC50 :570nM), HDAC3 (IC50 :550nM)). CXD101(CXD-101) has no activity against HDAC class IIFormule :C24H29N5ODegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :403.52NKL 22
CAS :NKL 22 (Histone Deacetylase Inhibitor IV) is an effective Histone Deacetylase Inhibitor.Formule :C19H23N3O2Degré de pureté :96.16% - 96.24%Couleur et forme :SolidMasse moléculaire :325.4HDAC-IN-7
CAS :HDAC-IN-7 (HBI-8000) (Chidamide impurity) is an impurity of Chidamide.Formule :C22H19FN4O2Degré de pureté :97.64% - 98.45%Couleur et forme :SolidMasse moléculaire :390.41Ref: TM-T2025
1mg58,00€2mg82,00€1mL*10mM (DMSO)111,00€5mg130,00€10mg215,00€25mg429,00€50mg628,00€100mg893,00€BAY 87-2243
CAS :BAY 87-2243 is a potent and selective inhibitor of hypoxia-inducible factor-1 (HIF-1).Formule :C26H26F3N7O2Degré de pureté :98% - 99.95%Couleur et forme :SolidMasse moléculaire :525.53Ref: TM-T2488
1mg34,00€2mg40,00€5mg59,00€1mL*10mM (DMSO)70,00€10mg96,00€25mg200,00€50mg334,00€100mg557,00€Niraparib tosylate monohyrate
CAS :Niraparib (MK-4827), a PARP inhibitor, boosts DNA breaks to trigger genomic instability and apoptosis, offering anti-cancer effects.Formule :C26H30N4O5SDegré de pureté :97.7% - 99.99%Couleur et forme :SolidMasse moléculaire :510.61Ref: TM-T9497
5mg57,00€1mL*10mM (DMSO)66,00€10mg82,00€25mg111,00€50mg137,00€100mg205,00€200mg309,00€500mg515,00€AGK7
CAS :AGK7 is an AGK2 control; it's a less selective SIRT2 inhibitor, with IC50s >5 μM for SIRT3, and >50 μM for SIRT1/2.Formule :C23H13Cl2N3O2Degré de pureté :98.31%Couleur et forme :SolidMasse moléculaire :434.27Nexturastat A
CAS :Nexturastat A is an effective and specific HDAC6 inhibitor (IC50: 5 nM). Its selectivity is >190-fold than other HDACs.Formule :C19H23N3O3Degré de pureté :99.40% - 99.57%Couleur et forme :SolidMasse moléculaire :341.4OSS_128167
CAS :OSS_128167 (SIRT6-IN-1) is a specific SIRT6 inhibitor, and for SIRT6(IC50=89 μM), SIRT1(IC50=1578 μM) and SIRT2(IC50=751 μM).Formule :C19H14N2O6Degré de pureté :97.47% - 98.6%Couleur et forme :SolidMasse moléculaire :366.32CAY10603
CAS :CAY10603 (BML-281) is a potent and selective inhibitor of HDAC6.Formule :C22H30N4O6Degré de pureté :95.75% - 98.1%Couleur et forme :SolidMasse moléculaire :446.5Ref: TM-T1983
1mg59,00€2mg78,00€5mg90,00€1mL*10mM (DMSO)90,00€10mg161,00€25mg290,00€50mg492,00€100mg710,00€TMP195
CAS :TMP195 (TFMO 2) is a selective class IIa histone deacetylase (HDAC) inhibitor.Formule :C23H19F3N4O3Degré de pureté :98.92% - 99.64%Couleur et forme :SolidMasse moléculaire :456.42Ref: TM-T3983
2mg70,00€5mg104,00€1mL*10mM (DMSO)104,00€10mg170,00€25mg341,00€50mg409,00€100mg602,00€200mg857,00€Zebularine
CAS :Zebularine (4-Deoxyuridine) is a DNA methylation inhibitor.Formule :C9H12N2O5Degré de pureté :99.04% - >99.99%Couleur et forme :SolidMasse moléculaire :228.2RG2833
CAS :RG2833 (RGFP109) (RGFP109), a brain-penetrant HDAC inhibitor, is with IC50 of 60 nM and 50 nM for HDAC1 and HDAC3, respectively.Formule :C20H25N3O2Degré de pureté :99% - 99.50%Couleur et forme :SolidMasse moléculaire :339.43Tasquinimod
CAS :Tasquinimod (ABR-215050) is an oral antiangiogenic agent and S100A9 inhibitor that binds to the HDAC4Zn2+ binding structural domain with Kd values ranging from 10 to 30 nM.Cost-effective and quality-assured.Formule :C20H17F3N2O4Degré de pureté :99.22% - >99.99%Couleur et forme :SolidMasse moléculaire :406.36Ref: TM-T6695
1mg52,00€2mg67,00€5mg101,00€1mL*10mM (DMSO)110,00€10mg158,00€25mg295,00€50mg484,00€100mg745,00€653-47
CAS :653-47 enhances the effects of 666-15 on inhibiting CREB and is a mild CREB inhibitor itself (IC50: 26.3μM).Formule :C20H19ClN2O3Couleur et forme :SolidMasse moléculaire :370.83NSC 228155
CAS :NSC 228155 is an activator of EGFR, binding to the sEGFR dimerization domain II and modulate EGFR tyrosine phosphorylation.Formule :C11H6N4O4SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :290.25Ref: TM-T6908
2mg34,00€5mg48,00€1mL*10mM (DMSO)50,00€10mg63,00€25mg117,00€50mg178,00€100mg334,00€200mg469,00€YK-3-237
CAS :YK-3-237 (B-[2-Methoxy-5-[(1E)-3-oxo-3-(3,4,5-trimethoxyphenyl)-1-propen-1-yl]phenyl]boronic acid) reduces acetylation of mtp53 and exhibits anti-proliferativeFormule :C19H21BO7Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :372.18Ref: TM-T9320
2mg38,00€5mg57,00€1mL*10mM (DMSO)63,00€10mg93,00€25mg170,00€50mg289,00€100mg507,00€200mg655,00€500mg1.018,00€PI-1840
CAS :PI-1840 is a reversible and selective chymotrypsin-like (CT-L) inhibitor, with little proteasome proteolytic effects on trypsin-like (T-L) and PGPH-L.Formule :C22H26N4O3Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :394.47BI-7273
CAS :BI-7273 is an effective, specific, BRD9 BD Inhibitor, which can infiltrate cell.Formule :C20H23N3O3Degré de pureté :97.37% - 99.57%Couleur et forme :SolidMasse moléculaire :353.41SRT 2104
CAS :SRT 2104 (GSK2245840) is a selective and brain-permeable SIRT1 activator.Formule :C26H24N6O2S2Degré de pureté :98.34% - 99.82%Couleur et forme :SolidMasse moléculaire :516.64Ref: TM-T6679
1mg43,00€5mg93,00€10mg124,00€25mg219,00€50mg358,00€100mg533,00€200mg763,00€500mg1.161,00€1g1.558,00€4-(3-Chlorophenyl)-2(3H)-thiazolone
CAS :4-(3-chlorophenyl)-2,3-dihydro-1,3-thiazol-2-one: a thiazole used to make antifungals, antivirals, and anti-inflammatories.Formule :C9H6ClNOSDegré de pureté :95.311%Couleur et forme :SolidMasse moléculaire :211.67GSK1324726A
CAS :GSK1324726A (I-BET726) is a greatly specific inhibitor of BET family proteins for BRD2(IC50=41 nM), BRD3(IC50=31 nM), and BRD4 (IC50=22 nM).
Formule :C25H23ClN2O3Degré de pureté :98.34% - 99.85%Couleur et forme :SolidMasse moléculaire :434.91PF 477736
CAS :PF 477736 (PF-736,PF-00477736) is a specifc, effective and ATP-competitive Chk1 inhibitor (Ki: 0.49 nM ) and also inhibits FGFR3, Aurora-A, VEGFR2, Flt3, Fms (Formule :C22H25N7O2Degré de pureté :97.58% - 99.94%Couleur et forme :SolidMasse moléculaire :419.48Iadademstat dihydrochloride
CAS :Iadademstat dihydrochloride (ORY-1001(trans)) , a Potent and Selective Covalent KDM1A/LSD1 Inhibitor, for the Treatment of Acute Leukemia.
Formule :C15H24Cl2N2Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :303.27MC2184
CAS :MC2184 is the inhibitor of human recombinant SIRT1.Formule :C11H6N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :214.18Citarinostat
CAS :ACY-241 (Citarinostat), a potent oral HDAC inhibitor, may induce tumor cell death and block growth by altering gene expression.Formule :C24H26ClN5O3Degré de pureté :98.06% - 99.06%Couleur et forme :SolidMasse moléculaire :467.95KA2507 monohydrochloride
KA2507 hydrochloride: potent HDAC6 inhibitor, IC50 = 2.5 nM, non-toxic, with antitumor and immune benefits.Formule :C16H15ClN6O2Couleur et forme :SolidMasse moléculaire :358.78[Ala107]-MBP (104-118) acetate
[Ala107]-MBP (104-118) acetate ([Ala107]-MBP ) is synthetic peptide analog of bovine myelin basic protein (MBP).Formule :C59H108N20O21Degré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :1553.72Resminostat hydrochloride
CAS :Resminostat hydrochloride (RAS2410 hydrochloride) is an effective inhibitor of HDAC1/HDAC3/HDAC6 (IC50: 42.5/50.1/71.8 nM), respectively, and shows less potentFormule :C16H20ClN3O4SDegré de pureté :97.63% - 99.68%Couleur et forme :SolidMasse moléculaire :385.86KA2507
CAS :KA2507 is a potent and selective HDAC6 inibitor with an IC50 of 2.5nM.Formule :C16H14N6O2Degré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :322.32Ref: TM-T9148
1mL*10mM (DMSO)33,00€1mg39,00€5mg84,00€10mg120,00€25mg222,00€50mg334,00€100mg447,00€200mg623,00€CM-272
CAS :CM-272 is a dual G9a/DNA methyltransferases (DNMTs) inhibitor.Formule :C28H38N4O3Degré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :478.63Buformin
CAS :Buformin, a biguanide oral antidiabetic, inhibits liver glucose production and improves insulin sensitivity.Formule :C6H15N5Couleur et forme :SolidMasse moléculaire :157.22Go 6983
CAS :Go 6983 is a PKC inhibitor with IC50 values of 7, 7, 6, 10, and 60 nM for PKCα, PKCβ, PKCγ, PKCδ, and PKCζ, respectively. High-Quality, Low-Cost!Formule :C26H26N4O3Degré de pureté :98.41% - 99.85%Couleur et forme :SolidMasse moléculaire :442.51Ref: TM-T6313
1mg40,00€2mg52,00€5mg79,00€1mL*10mM (DMSO)84,00€10mg119,00€25mg233,00€50mg368,00€100mg533,00€4'-Methoxychalcone
CAS :4'-Methoxychalcone with a variety of pharmacological activities, such as anti-tumor and anti-inflammatory activities.Formule :C16H14O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :238.28NVP-BSK805 trihydrochloride
CAS :NVP-BSK805 trihydrochloride inhibits JAK2 (0.48 nM IC50); also affects JAK1, JAK3, TYK2.Formule :C27H31Cl3F2N6OCouleur et forme :SolidMasse moléculaire :599.937BIO
CAS :7BIO triggers nonapoptotic death, blocks FLT3, DYRK1A/2, Aurora B/C kinases.
Formule :C16H10BrN3O2Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :356.17FG-2216
CAS :FG-2216 (YM-311) is a HIF-prolyl hydroxylase inhibitor for the PDH2 enzyme; orally bioavailable and induced reversible and significant Epo induction in vivo.Formule :C12H9ClN2O4Degré de pureté :97.1% - >99.99%Couleur et forme :SolidMasse moléculaire :280.66Sotrastaurin
CAS :Sotrastaurin (AEB071) is a potent pan-PKC inhibitor (Kis: 0.95/0.64/2.1/3.2/1.8/0.22 nM for PKCα/βI/δ/ε/η/θ).Formule :C25H22N6O2Degré de pureté :98% - 99.70%Couleur et forme :SolidMasse moléculaire :438.48Ref: TM-T6278
1mg44,00€5mg86,00€1mL*10mM (DMSO)94,00€10mg135,00€25mg254,00€50mg423,00€100mg605,00€200mg845,00€AK-7
CAS :AK-7 is a brain-permeable SIRT2 inhibitor and to characterize its cholesterol-reducing properties in neuronal models with an IC50 of 15.5 μM.Formule :C19H21BrN2O3SDegré de pureté :98.43% - 99.34%Couleur et forme :SolidMasse moléculaire :437.35Ref: TM-T5490
1mg34,00€2mg47,00€5mg71,00€1mL*10mM (DMSO)89,00€10mg100,00€25mg177,00€50mg313,00€100mg512,00€

