Endocrinologie/Hormones
Les inhibiteurs en endocrinologie/hormonaux sont des composés qui bloquent l'action des hormones ou interfèrent avec les voies de signalisation hormonales. Ces inhibiteurs sont essentiels pour étudier la régulation des systèmes endocriniens et pour développer des traitements pour les maladies liées aux hormones, telles que le diabète, les troubles de la thyroïde et les cancers hormonodépendants. En modulant l'activité hormonale, ces inhibiteurs peuvent aider à élucider les interactions complexes au sein du système endocrinien. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité en endocrinologie/hormonaux pour soutenir vos recherches en endocrinologie, pharmacologie et sciences médicales.
Sous-catégories appartenant à la catégorie "Endocrinologie/Hormones"
- Récepteur des androgènes(209 produits)
- Annexine A(11 produits)
- Aromatase(20 produits)
- Récepteur d'œstrogène/progestatif(49 produits)
- GPR(1 produits)
- Récepteur des glucocorticoïdes(153 produits)
- LHRH(1 produits)
- Récepteur opioïde(297 produits)
- Récepteur de prostaglandine(120 produits)
- RAAS(87 produits)
- Réductase(52 produits)
- Somatostatine(49 produits)
- Récepteur des hormones thyroïdiennes (THR)(26 produits)
- Récepteur de la vasopressine(44 produits)
Affichez 6 plus de sous-catégories
3183 produits trouvés pour "Endocrinologie/Hormones"
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PROTAC ERRα Degrader-3
CAS :<p>PROTAC ERRα Degrader-3 is a highly effective and selective von Hippel-Lindau-based ligand that efficiently degrades the ERRα protein.</p>Formule :C47H50F6N6O7SCouleur et forme :SolidMasse moléculaire :957.0AKR1C3-IN-10
<p>AKR1C3-IN-10 (compound 5r), a selective inhibitor of AKR1C3 with an IC50 of 51 nM, demonstrates efficacy in a prostate cancer xenograft model [1].</p>Formule :C24H20N4O3Couleur et forme :SolidMasse moléculaire :412.44(E)-4-Hydroxytamoxifen
CAS :<p>(E)-4-Hydroxytamoxifen is a less active isomer of (Z)-4-hydroxytamoxifen and also is an estrogen receptor modulator.</p>Formule :C26H29NO2Couleur et forme :SolidMasse moléculaire :387.51Betamethasone Acetate (Standard)
CAS :Betamethasone Acetate (Standard) is the standard substance of Betamethasone Acetate, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Betamethasone acetate, the 21-acetate ester of betamethasone, is a synthetic glucocorticoid corticosteroid and a corticosteroid ester.Formule :C24H31FO6Masse moléculaire :434.50SCO-267
CAS :<p>SCO-267 is a full agonist of GPR40/FFAR1， stimulating insulin secretion and GLP-1 release in diabetic rats, improving glucose tolerance,type 2 diabetes.</p>Formule :C36H46N4O5Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :614.77Valsartan-d9
CAS :<p>Valsartan D9: deuterium-labeled, angiotensin II receptor antagonist, treats hypertension & heart failure.</p>Formule :C24H29N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :444.57Valsartan Ethyl Ester
CAS :<p>Valsartan Ethyl Ester, an impurity in Valsartan, treats hypertension and heart failure by blocking angiotensin II receptors.</p>Formule :C26H33N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :463.57ML334
CAS :<p>ML334 (LH601A) is an NRF2 activator that inhibits cardiac fibroblast activation and proliferation ameliorating myocardial infarction-induced cardiac fibrosis.</p>Formule :C26H26N2O5Degré de pureté :98.06% - 98.06%Couleur et forme :SolidMasse moléculaire :446.49Azilsartan-d5
CAS :<p>Azilsartan (TAK-536) D5 is the deuterium-labeled Azilsartan. Azilsartan is a specific antagonist of the angiotensin II type 1 receptor.</p>Formule :C25H20N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.485β-Dihydroprogesterone
CAS :<p>5β-Dihydroprogesterone (5β-DHP) is a progesterone receptor agonist and metabolite of progesterone .1,2It is formed from progesterone by 5β-reductase.25β-DHP</p>Formule :C21H32O2Couleur et forme :SolidMasse moléculaire :316.485NQO1 substrate
CAS :<p>NQO1 substrate is a highly potent NQO1 substrate with potential antitumor activity for leukemia research.</p>Formule :C13H2F2N4ODegré de pureté :98.02% - 98.02%Couleur et forme :SolidMasse moléculaire :268.18Hydrocortisone cypionate
CAS :<p>Hydrocortisone cypionate is a corticosteroid ester and synthetic glucocorticoid corticosteroid.</p>Formule :C29H42O6Couleur et forme :SolidMasse moléculaire :486.64GW-1100
CAS :<p>GW-1100 is a selective GPR40 and FFAR1 antagonist for the study of diabetes and metabolic diseases.</p>Formule :C27H25FN4O4SDegré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :520.58(Rac)-PF-998425
CAS :<p>(Rac)-PF-998425: nonsteroidal AR antagonist, potent & selective, IC50: 26 nM (binding), 90 nM (cellular), potential for androgenetic alopecia study.</p>Formule :C14H14F3NOCouleur et forme :SolidMasse moléculaire :269.267AVE 0991 sodium salt
CAS :AVE 0991, a nonpeptide, oral Mas agonist, binds [125I]-Ang-(1-7) with IC50 of 21±35 nM.Formule :C29H31N4NaO5S2Couleur et forme :SolidMasse moléculaire :602.7AMG7703
CAS :<p>AMG7703 is a bioactive chemical.</p>Formule :C14H15ClN2OSCouleur et forme :SolidMasse moléculaire :294.8Olmesartan lactone impurity
CAS :<p>Olmesartan lactone impurity, a cyclic ester from Olmesartan, aids in hypertension research as an AT1R blocker.</p>Formule :C24H24N6O2Couleur et forme :SolidMasse moléculaire :428.496Desoxycorticosterone pivalate
CAS :<p>DOCP, a mineralocorticoid, treats dogs with adrenal insufficiency.</p>Formule :C26H38O4Couleur et forme :SolidMasse moléculaire :414.58Betamethasone acetate
CAS :<p>Betamethasone acetate, the 21-acetate ester of betamethasone, is a synthetic glucocorticoid corticosteroid and a corticosteroid ester.</p>Formule :C24H31FO6Couleur et forme :SolidMasse moléculaire :434.50TA 0910 acid-type
CAS :<p>TA 0910 acid-type is a metabolite of TA 0910. TA-0910 is a metabolically stable analog of thyrotropin-releasing hormone.</p>Formule :C17H22N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :406.39Loperamide phenyl
CAS :<p>Loperamide phenyl, an impurity detected in Loperamide, is an opioid receptor agonist.</p>Formule :C35H37ClN2O2Couleur et forme :SolidMasse moléculaire :553.14Vanilpyruvic acid
CAS :<p>Vanillylpyruvic acid is a phenylpyruvic acid derivative applicable in biochemical experiments and drug synthesis research.</p>Formule :C10H10O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :210.18Dienestrol diacetate
CAS :<p>Dienestrol diacetate, a derivative of the synthetic non-steroid phenolic compound, DIENESTROL, exhibits estrogenic activities.</p>Formule :C22H22O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :350.41Fenarimol
CAS :<p>Fenarimol, a pyrimidine-type fungicide, exhibits potent inhibitory activity against BR biosynthesis.</p>Formule :C17H12Cl2N2OCouleur et forme :SolidMasse moléculaire :331.2VTP-27999 Hydrochloride
CAS :<p>VTP-27999 Hcl is an alkyl amine Renin inhibitor; VTP-27999 is useful for Hypertension and End-Organ Diseases.<br><br>IC50 value:<br><br>Target: Renin</p>Formule :C26H42Cl2N4O5Couleur et forme :SolidMasse moléculaire :561.55Losartan (D4 Carboxylic Acid)
CAS :<p>Losartan D4 Carboxylic Acid is the deuterium labeled Losartan, which is an angiotensin II receptor antagonist.</p>Formule :C22H21ClN6O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.92Diflorasone Diacetate
CAS :<p>Diflorasone Diacetate, a topical glucocorticoid, has immunosuppressive and anti-inflammatory properties.</p>Formule :C26H32F2O7Couleur et forme :CrystalsMasse moléculaire :494.53Dihydromunduletone
CAS :<p>Dihydromunduletone (DHM) is an adhesion G protein-coupled receptor (aGPCR) antagonist inhibits GPR56 and GPR114/ADGRG5, which have similar tethered agonists.</p>Formule :C25H28O6Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :424.49Enalaprilat
CAS :<p>Enalaprilat (Enalapril acid) is an ACE inhibitor used in the study of cardiovascular disease.</p>Formule :C18H24N2O5Degré de pureté :97.28%Couleur et forme :SolidMasse moléculaire :348.39Leelamine hydrochloride
CAS :<p>Leelamine hydrochloride, a pine bark extract, inhibits androgen receptor and CB1, reducing lipid synthesis in prostate cancer.</p>Formule :C20H32ClNDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.93Pamoic acid disodium
CAS :<p>Pamoic acid disodium is a GPR35 agonist.</p>Formule :C23H16NaO6Degré de pureté :99.73%Couleur et forme :Yellow PowderMasse moléculaire :411.36DL-Cystine
CAS :<p>DL-Cystine is a cysteine derivative that inhibits endothelial cell proliferation by regulating TGFβ1. a GPR inhibitor and nAChR agonist .</p>Formule :C6H12N2O4S2Couleur et forme :SolidMasse moléculaire :240.32-Bromoestradiol
CAS :<p>2-Bromoestradiol, an estrogen 2-hydroxylase inhibitor, reduces the irreversible binding of radiolabeled estradiol metabolite(s) to microsomal proteins [1].</p>Formule :C18H23BrO2Couleur et forme :SolidMasse moléculaire :351.28AC-186
CAS :<p>AC-186 is an ERβ agonist with neuroprotective activity for the study of Parkinson's disease.</p>Formule :C18H17F3ODegré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :306.32Monomethyl fumarate-d3
CAS :<p>Monomethyl fumarate D3 is a deuterium labeled Monomethyl fumarate.</p>Formule :C5H6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :133.12Trans-Diethyl-1,1,1',1'-Stilbestrol-3,3',5,5'-d8
CAS :<p>Trans-Diethyl-1,1,1',1'-Stilbestrol-3,3',5,5'-d8 is a deuterated compound of Trans-Diethyl-Stilbestrol. Trans-Diethyl-Stilbestrol has a CAS number of 56-53-1. Diethylstilbestrol is used in the treatment of menopausal and postmenopausal disorders.</p>Formule :C18H12D8O2Couleur et forme :SolidMasse moléculaire :276.40MK-0773
CAS :<p>MK-0773 (PF-05314882) is a selective androgen receptor modulator that binds to AR (IC50: 6.6 nM) for the study of diseases caused by endocrine abnormalities.</p>Formule :C27H34FN5O2Degré de pureté :98.38% - 99.14%Couleur et forme :SolidMasse moléculaire :479.59BAN ORL 24 dihydrochloride
CAS :<p>BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that can be used to study neurological diseases.</p>Formule :C27H37Cl2N3O2Degré de pureté :95.03%Couleur et forme :SolidMasse moléculaire :506.51Dehydroepiandrosterone-d2
CAS :<p>Dehydroepiandrosterone-d2 is a deuterated compound of Dehydroepiandrosterone.</p>Formule :C19H26D2O2Couleur et forme :SolidMasse moléculaire :290.44BMS-986121
CAS :<p>BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.</p>Formule :C15H9Cl2N3O2SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :366.22Atosiban
CAS :<p>Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions rapidly.</p>Formule :C43H67N11O12S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :994.19Azilsartan mepixetil
CAS :<p>Azilsartan mepixetil: potent, long-acting angiotensin II blocker, safely lowers blood pressure, protects heart and kidneys.</p>Formule :C36H34N6O8Couleur et forme :SolidMasse moléculaire :678.702(R,S)-Ivosidenib
CAS :(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .Formule :C28H22ClF3N6O3Couleur et forme :SolidMasse moléculaire :582.9617β-Estradiol-2,4-d2
CAS :<p>17β-Estradiol-2,4-d2 is a deuterated compound of 17β-Estradiol. 17β-Estradiol has a CAS number of 50-28-2. Estradiol is an Estrogen. The mechanism of action of estradiol is as an Estrogen Receptor Agonist.</p>Formule :C18H22D2O2Couleur et forme :SolidMasse moléculaire :274.39CGP-42112
CAS :<p>CGP-42112 is an agonist of the Angiotensin-II subtype 2 receptor (AT2 R).</p>Formule :C52H69N13O11Couleur et forme :White SolidMasse moléculaire :1052.18TUG-770
CAS :<p>TUG-770 is a highly potent agonist of free fatty acid receptor 1 (FFA1/GPR40, EC50: 6 nM for hFFA1).</p>Formule :C19H14FNO2Degré de pureté :97.6%Couleur et forme :SolidMasse moléculaire :307.32Alvimopan dihydrate (LY246736 dihydrate)
CAS :<p>Alvimopan dihydrate is a potent, oral μ-opioid receptor blocker (IC50 1.7 nM, Ki 0.47 nM) used in postoperative ileus research.</p>Formule :C25H36N2O6Couleur et forme :SolidMasse moléculaire :460.56YE 120
CAS :<p>YE 120 is a GPR35 agonist.</p>Formule :C16H9Cl2N3ODegré de pureté :99.59% - 99.81%Couleur et forme :SolidMasse moléculaire :330.17GDC-0927
CAS :<p>GDC-0927 is a novel,non-steroidal, potent, orally bioavailable, selective estrogen receptor antagonist.</p>Formule :C28H28FNO4Couleur et forme :SolidMasse moléculaire :461.52Bazedoxifene
CAS :<p>Bazedoxifene is an orally active SERM against ERα and ERβ and inhibits IL-6/GP130, applied in postmenopausal osteoporosis and pancreatic cancer research.</p>Formule :C30H34N2O3Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :470.61ARD-1676
CAS :<p>ARD-1676 is an orally administered androgen receptor (AR) PROTAC degrader that combines an AR ligand with a cereblon ligand.</p>Formule :C44H46ClN7O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :788.33Prednisolone valerate acetate
CAS :<p>Prednisolone valerate acetate is a prodrug anti-inflammatory and immunosuppressive,converted to the active form of Prednisolone and glucocorticoid receptor.</p>Formule :C28H38O7Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :486.6Candesartan-d4
CAS :<p>Candesartan D4 is the deuterium labeled Candesartan. Candesartan is an antagonist of angiotensin II receptor.</p>Formule :C24H20N6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :444.48Olmesartan-d4
CAS :<p>Olmesartan D4 is the deuterium labeled Olmesartan. Olmesartan is an antagonist of angiotensin II receptor (AT1R) used to treat high blood pressure.</p>Formule :C24H26N6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :450.53MS 15203
CAS :<p>MS 15203 is a GPR171 agonist that reduces chronic neuropathic and inflammatory pain in male mice.</p>Formule :C12H11NO5Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :249.22Beclomethasone 17-propionate
CAS :<p>Beclomethasone 17-propionate is the active metabolite of BDP. As a GR agonist, 17-BMP inhibits the production of pro-inflammatory cytokines.</p>Formule :C25H33ClO6Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :464.98Endomorphin 2 TFA
CAS :<p>Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.</p>Formule :C34H38F3N5O7Couleur et forme :SolidMasse moléculaire :685.69Estradiol valerate
CAS :<p>β-estradiol 17-valerate (EV) is a synthetic estrogen. In hormone replacement therapy drugs, it is widely used in combination with other steroid hormones.</p>Formule :C23H32O3Degré de pureté :99.11% - 99.9%Couleur et forme :NaMasse moléculaire :356.51PD 123319 ditrifluoroacetate
CAS :<p>PD 123319 ditrifluoroacetate is a selective non-peptide AT2 receptor antagonist with IC50 of 34 nM.</p>Formule :C35H34F6N4O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :736.66Endoxifen Z-isomer hydrochloride
CAS :<p>Endoxifen Z-isomer hydrochloride (Endoxifen HCl) is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.</p>Formule :C25H28ClNO2Couleur et forme :SolidMasse moléculaire :409.95Taltirelin
CAS :<p>Taltirelin (TA-0910) is at thyrotropin-releasing hormone receptor (TRH-R) superagonist (IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in</p>Formule :C17H23N7O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :405.41Asimadoline
CAS :Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.Formule :C27H30N2O2Couleur et forme :SolidMasse moléculaire :414.54Rezvilutamide
CAS :Rezvilutamide (SHR3680) is an orally available androgen receptor inhibitor that crosses the blood-brain barrier and has antitumor activity.Formule :C22H20F3N3O4SDegré de pureté :99.96% - 99.97%Couleur et forme :SolidMasse moléculaire :479.47Angiotensin II (3-8), human
CAS :<p>Angiotensin II (3-8), human is a less effective agonist at the angiotensin AT1 receptor.</p>Couleur et forme :SolidD4-abiraterone
CAS :<p>D4-abiraterone is the active metabolite of abiraterone.Δ4-Abiraterone is a inhibitor of CYP17A1, 3β-HSD and SRD5A, and an antagonist of the androgen receptor.</p>Formule :C24H29NODegré de pureté :99.75% - 99.8%Couleur et forme :SolidMasse moléculaire :347.49Protirelin
CAS :<p>Protirelin (Thyroliberin) is a tripeptide that stimulates the release of thyrotropin and prolactin.</p>Formule :C16H22N6O4Degré de pureté :99.76%Couleur et forme :White Or Almost White PowderMasse moléculaire :362.38GPR41 agonist-1
CAS :<p>GPR41 agonist-1 is a GPR41 agonist, used for studying metabolic diseases such as diabetes and obesity.</p>Formule :C24H23N3O4Degré de pureté :98.40%Couleur et forme :SolidMasse moléculaire :417.46Apalutamide-13C-d3
<p>Apalutamide-13C-d3 is a 13C and 2H labeled Apalutamide. Apalutamide is an androgen receptor (AR) antagonist, used in research on prostate diseases.</p>Formule :CC20H12F4N5O2SD3Couleur et forme :SolidMasse moléculaire :481.45AZD1979
CAS :<p>AZD1979 is a highly potent MCHR1 (Melanin-concentrating hormone receptor 1) antagonist , CNS exposure and insulin sensitivity in steady-state model assessments,</p>Formule :C25H26N4O5Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :462.5Zearalanone
CAS :<p>Zearalenone is a nonsteroidal estrogenic mycotoxin produced by Fusarium species, which colonizes several grains.</p>Formule :C18H24O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :320.38ERα degrader-2
CAS :<p>ERα degrader-2 is an estrogen receptor (SERD) degrader with anticancer activity that inhibits ERα for the prevention and treatment of HER-positive breast canc</p>Formule :C29H27F3N2O2Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :492.53GPR30 agonist-1
CAS :<p>GPR30 agonist-1 is a compound that acts as an agonist for G protein-coupled receptor 30 (GPR30), inducing vasorelaxation.</p>Formule :C19H17BrFNOCouleur et forme :SolidMasse moléculaire :374.253ZQ-16
CAS :<p>ZQ-16 is a potent GPR84 agonist (EC50=0.213 μM) activating multiple signaling pathways.</p>Formule :C10H16N2O2SDegré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :228.31GPR40 agonist 6
CAS :<p>GPR40 agonist 6 (Compound 7a) is a potent and selective agonist of free fatty acid receptor 1 ( FFAR1 or GPR40 ) with an EC 50 of 0.058 μM against GPR40 [1].</p>Formule :C20H19NO4Couleur et forme :SolidMasse moléculaire :337.37Hydrocortisone buteprate
CAS :<p>Hydrocortisone buteprate is a medium-potent, non-halogenated double-ester of hydrocortisone with a highly favorable benefit-to-risk ratio for inflammatory skin disorders.</p>Formule :C28H40O7Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :488.61Porcine dynorphin A(1-13)
CAS :Porcine dynorphin A (1-13) is a potent κ opioid receptor agonist; it's antinociceptive and raises [Ca2+]i in neurons like NMDA.Formule :C75H126N24O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1603.95Nafoxidine HCl(1845-11-0 Free base)
CAS :<p>Nafoxidine is a partial estrogen antagonist.</p>Formule :C29H32ClNO2Couleur et forme :SolidMasse moléculaire :462.03Harman hydrochloride
CAS :<p>Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.</p>Formule :C12H11ClN2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :218.68Desoximetasone
CAS :<p>Desoximetasone (Topicort) is a topical corticosteroid for treating skin conditions like rashes.</p>Formule :C22H29FO4Degré de pureté :99.06% - 99.89%Couleur et forme :SolidMasse moléculaire :376.46Halobetasol propionate
CAS :<p>Halobetasol propionate (BMY-30056) is the salt of halobetasol, a synthetic corticosteroid with anti-inflammatory, antipruritic, and vasoconstrictor activities.</p>Formule :C25H31ClF2O5Degré de pureté :99.89%Couleur et forme :Distributed As 0 05% OintmentMasse moléculaire :484.96Saralasin acetate(34273-10-4 free base)
CAS :<p>Saralasin acetate is a Non-selective angiotensin II antagonist.</p>Formule :C44H71N13O13Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :990.11A 779 TFA(159432-28-7 free base)
<p>A 779 TFA is a potent antagonist of angiotensin-(1-7) receptor.</p>Formule :C41H61F3N12O13Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :987.01AL 082D06
CAS :<p>AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR.</p>Formule :C23H24ClN3O2Degré de pureté :99.05% - 99.06%Couleur et forme :SolidMasse moléculaire :409.912,4'-Dihydroxybenzophenone
CAS :<p>2,4'-Dihydroxybenzophenone can effectively protect C57BL/6J mice from APAP-induced hepatotoxicity.</p>Formule :C13H10O3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :214.22Novokinin acetate
<p>Novokinin acetate binds AT2 receptor (Ki=7 nM); antihypertensive effect blocked by PD123319.</p>Formule :C41H65N11O9Degré de pureté :99.37%Couleur et forme :SoildMasse moléculaire :856.02Apararenone
CAS :<p>Apararenone (MT-3995) is a receptor antagonist of mineralocorticoid receptor which can be used to treat non-alcoholic steatohepatitis and diabetic nephropathy.</p>Formule :C17H17FN2O4SDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :364.39Elacestrant dihydrochloride
CAS :<p>Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ERα and 870 nM for</p>Formule :C30H40Cl2N2O2Degré de pureté :99.59% - >99.99%Couleur et forme :SolidMasse moléculaire :531.56Eprotirome
CAS :<p>Eprotirome (KB2115), a synthetic thyroid hormone mimetic, is a thyroid hormone receptor agonist.</p>Formule :C18H17Br2NO5Degré de pureté :98.42% - 98.56%Couleur et forme :SolidMasse moléculaire :487.14SNG-1153
CAS :<p>SNG-1153 is a estrogen receptor ER-alpha36 modulator.</p>Formule :C21H17F3O5Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :406.35S-23
CAS :<p>S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (</p>Formule :C18H13ClF4N2O3Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :416.75Abaloparatide TFA
<p>Abaloparatide TFA (BIM 44058 TFA) is a parathyroid hormone-related protein (PTHrP) analog drug used to treat osteoporosis like the related drug teriparatide.</p>Formule :C176H301N56F3O51Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :4074.61Teriparatide acetate
CAS :<p>Teriparatide acetate (Forteo), a synthetic parathyroid hormone, treats osteoporosis by favoring bone growth with a 2 nM IC50.</p>Formule :C183H295N55O53S2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :4177.83Chlorotrianisene
CAS :<p>Chlorotrianisene, a synthetic SERM, is orally active, lipophilic, and has estrogenic and antiestrogenic effects.</p>Formule :C23H21ClO3Degré de pureté :98.88% - 99.03%Couleur et forme :Crystals From Methanol Physical Description Small White Crystals Or White Powder Softens At 226°F Odorless (Ntp 1992)Masse moléculaire :380.86Fevipiprant
CAS :<p>Fevipiprant (NVP-QAW039) is a selective, potent, reversible competitive CRTh2 antagonist.</p>Formule :C19H17F3N2O4SDegré de pureté :99.32% - 99.59%Couleur et forme :SolidMasse moléculaire :426.41Ciclesonide
CAS :<p>Ciclesonide (Alvesco)(RPR251526) is a glucocorticoid used for the treatment of obstructive airway diseases.</p>Formule :C32H44O7Degré de pureté :99.89% - >99.99%Couleur et forme :SolidMasse moléculaire :540.69EST73502 hydrochloride
CAS :<p>EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.</p>Formule :C19H27ClF2N2O2Couleur et forme :SolidMasse moléculaire :388.88BW-180C
CAS :<p>BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.</p>Formule :C29H39N5O7Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :569.65SNAP 94847 hydrochloride
CAS :<p>SNAP 94847 hydrochloride is a melanin-concentrating hormonereceptor1 (MCHR1) antagonist(Ki= 2.2 nM)</p>Formule :C29H33ClF2N2O2Degré de pureté :99.85% - >99.99%Couleur et forme :SolidMasse moléculaire :515.03VTP-27999 TFA
CAS :<p>VTP-27999 TFA is an inhibitor of Renin (IC50 : 0.47 nM).</p>Formule :C28H42ClF3N4O7Degré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :639.1BigLEN (mouse) acetate
<p>BigLEN (mouse) acetate is a potent and selective agonist of orphan G protein-coupled receptor 171 (GPR171), with a Kd of ∼0.5 nM.</p>Formule :C80H134N24O24Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1816.07PZM21
CAS :<p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>Formule :C19H27N3O2SDegré de pureté :99.93% - >99.99%Couleur et forme :SolidMasse moléculaire :361.5Fasiglifam
CAS :<p>Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.</p>Formule :C29H32O7SDegré de pureté :99.82% - 99.9%Couleur et forme :SolidMasse moléculaire :524.63Beclometasone dipropionate monohydrate
CAS :<p>Beclometasone dipropionate monohydrate, precursor to oral glucocorticoid for inflammation and asthma research.</p>Formule :C28H39ClO8Couleur et forme :SolidMasse moléculaire :539.06Ospemifene
CAS :<p>Ospemifene (FC-1271a) is a new selective non-hormonal estrogen receptor modulator (SERM) that is used for the treatment of moderate to severe dyspareunia, a symptom of vulvar and vaginal atrophy, due to menopause. FDA approved on February 26, 2013.</p>Formule :C24H23ClO2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :378.89Eprosartan Mesylate
CAS :<p>Eprosartan Mesylate (SKF-108566J) is a competitive and reversible Angiotensin II Receptor Blocker.</p>Formule :C23H24N2O4S·CH4O3SDegré de pureté :99.72% - 99.93%Couleur et forme :A White To Off- White PowderMasse moléculaire :520.62Fluorometholone Acetate
CAS :<p>Fluorometholone Acetate (Oxylone acetate) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.</p>Formule :C24H31FO5Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :418.50ADL-5747 (HCl)
CAS :<p>ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.</p>Formule :C24H29ClN2O3Couleur et forme :SolidMasse moléculaire :428.95Deltorphin I
CAS :<p>Deltorphin I is an agonist of δ-opioid receptor.</p>Formule :C37H52N8O10Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :768.86VPC-13566
CAS :<p>VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the</p>Formule :C18H14N2Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :258.32Brilanestrant
CAS :Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM).Formule :C26H20ClFN2O2Degré de pureté :99.07% - 99.17%Couleur et forme :Solid PowderMasse moléculaire :446.9PHTPP
CAS :<p>PHTPP is a selective ERβ antagonist.</p>Formule :C20H11F6N3ODegré de pureté :98.81% - 99.57%Couleur et forme :SolidMasse moléculaire :423.31Broparestrol (E)-
CAS :<p>Broparestrol (E)- has antifertility activity and is a potent inhibitor of rodent mammary tumorigenesis.</p>Formule :C22H19BrDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :363.29Iprodione
CAS :<p>Iprodione is a fungicide. Iprodione is also used in cannabis testing kits as a component of pesticide mixes.</p>Formule :C13H13Cl2N3O3Degré de pureté :98.82%Couleur et forme :Colorless Crystals Cream To Colorless Odorless PowderMasse moléculaire :330.17[Leu5]-Enkephalin TFA(58822-25-6(free bas))
CAS :<p>[Leu5]-Enkephalin TFA(58822-25-6(free bas)) (Leucyl-enkephalin) is the most potent δ-receptor ago</p>Formule :C30H38F3N5O9Degré de pureté :97.03% - 99.78%Couleur et forme :SolidMasse moléculaire :669.64Diflorasone
CAS :<p>Diflorasone is a synthetic glucocorticoid. It has anti-inflammatory and immunosuppressive effects by acting on gene expression.</p>Formule :C22H28F2O5Degré de pureté :99.02% - 99.92%Couleur et forme :SolidMasse moléculaire :410.45BTB06584
CAS :<p>BTB06584: IF1-dependent F1 Fo-ATPase inhibitor; novel AHAS inhibitor targeting MTB.</p>Formule :C19H12ClNO6SDegré de pureté :97.63% - ≥95%Couleur et forme :SolidMasse moléculaire :417.82FH1
CAS :<p>FH1 (NSC-12407) (BRD-K4477), a small molecule, enhances the functions of hepatocytes and promotes differentiation hepatocytes derived by iPS.</p>Formule :C17H18N2O2Degré de pureté :98% - 99.64%Couleur et forme :SolidMasse moléculaire :282.34Angiotensin III, human, mouse
CAS :<p>Angiotensin III, human, mouse (Angiotensin III, human, mouse(3TFA))(3TFA) is an endogenous angiotensin II receptor (AT2R) agonist(IC50s of 0.648 nM).</p>Formule :C46H66N12O9Degré de pureté :98.44%Couleur et forme :SolidMasse moléculaire :931.09BNP (1-32), human
CAS :<p>BNP (1-32), human is a brain natriuretic peptide</p>Formule :C143H244N50O42S4Degré de pureté :98.52%Couleur et forme :White PowderMasse moléculaire :3464.04GW9508
CAS :<p>GW9508(GW 9508) is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in a glucose-sensitive manner.</p>Formule :C22H21NO3Degré de pureté :97.89% - 99.19%Couleur et forme :SolidMasse moléculaire :347.41MK-6892
CAS :<p>MK-6892 is a selective and full agonist for the high-affinity nicotinic acid receptor GPR109A (Ki: 4 nM; GTPγS EC50: 16 nM).</p>Formule :C19H22N4O5Degré de pureté :99.01% - 99.67%Couleur et forme :SolidMasse moléculaire :386.4β-Estradiol 17-hemisuccinate
CAS :<p>beta-Estradiol 17-hemisuccinate selectively stains estrogen receptor (ER)-rich cells.</p>Formule :C22H28O5Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :372.45L-Thyroxine sodium
CAS :<p>L-Thyroxine sodium (LT4 sodium), the major hormone derived from the thyroid gland, is the agonist of Thyroid hormone receptor alpha and beta.</p>Formule :C15H10I4NO4·NaDegré de pureté :98.74%Couleur et forme :Yellowish To Buff-Colored Amorphous Powder SolidMasse moléculaire :798.85N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Formule :C30H39N5O8Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :597.666-OAU
CAS :<p>6-OAU is a GPR84 agonist, activates it in HEK293 cells with a 105 nM EC50.</p>Formule :C12H21N3O2Degré de pureté :98.14% - 99.01%Couleur et forme :SolidMasse moléculaire :239.31BMS986188
CAS :<p>BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.</p>Formule :C30H31BrO4Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :535.47GR 89696 free base
CAS :<p>GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.</p>Formule :C19H25Cl2N3O3Couleur et forme :SolidMasse moléculaire :414.33Temocapril hydrochloride
CAS :<p>Temocapril hydrochloride (CS-622 HCl), the hydrochloride of Temocapril, is a long-acting ACE inhibitor used for the therapy of hypertension.</p>Formule :C23H28N2O5S2·HClDegré de pureté :99.26% - 99.48%Couleur et forme :White Solid PowderMasse moléculaire :513.07Aviptadil Acetate
CAS :<p>Aviptadil Acetate (Vasoactive Intestinal Peptide acetate salt) induces pulmonary vasodilation and inhibits the proliferation of vascular SMCs.</p>Formule :C147H238N44O42S·C2H4O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :3385.9DIM-C-pPhOCH3
CAS :<p>DIM-C-pPhOCH3 (C-DIM5) is a Nerve Growth Factor-Induced Bα (NGFI-Bα, Nur77) agonist</p>Formule :C24H20N2ODegré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :352.43Naloxegol (NKTR-118)
CAS :<p>Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].</p>Formule :C34H53NO11Couleur et forme :SolidMasse moléculaire :651.78Olmesartan
CAS :<p>Olmesartan (RNH 6270) is an Angiotensin II Type I receptor antagonist.</p>Formule :C24H26N6O3Degré de pureté :91.89% - 99.81%Couleur et forme :White To Beige Solid SolidMasse moléculaire :446.5Propyl pyrazole triol
CAS :<p>PPT is a selective ERα agonist with 410x higher affinity than for ERβ.</p>Formule :C24H22N2O3Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :386.44Isoflupredone Acetate
CAS :<p>Isoflupredone Acetate is a corticosteroid with the activity of topical anti-inflammatory.</p>Formule :C23H29FO6Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :420.47Urotensin II, mouse acetate (9047-55-6 free base)
<p>Urotensin II, mouse acetate (9047-55-6 free base) is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor.</p>Formule :C64H88N14O19S2Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :1421.61Dynorphin A 1-10 acetate(79994-24-4 free base)
<p>Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.</p>Formule :C59H95N19O14Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :1294.53Hemorphin-7 acetate(152685-85-3 free base)
<p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>Formule :C51H68N12O13Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :1057.16WAY-200070
CAS :<p>WAY-200070 is a specific agonist of estrogen receptor β (ERRβ, IC50: 2.3 nM).</p>Formule :C13H8BrNO3Degré de pureté :99.45% - 99.75%Couleur et forme :SolidMasse moléculaire :306.11DPC AJ1951 acetate
<p>DPC-AJ1951 acetate: 14-amino acid peptide, potent PTH/PPR agonist, tested for bone resorption activity ex vivo/in vivo.</p>Formule :C78H131N23O21Degré de pureté :96.63%Couleur et forme :SolidMasse moléculaire :1727.02Orphanin FQ(1-11) acetate(178249-41-7 free base)
<p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>Formule :C51H79N15O16Degré de pureté :95.54%Couleur et forme :SolidMasse moléculaire :1158.26AH-7614
CAS :<p>AH-7614 (AH 7614) is a selective and potent free fatty acid receptor 4 (FFA4/GPR120) antagonist.</p>Formule :C20H17NO3SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :351.42Estradiol hemihydrate
CAS :<p>Estradiol hemihydrate: major female hormone, boosts neural differentiation, studied for cancer and neurodegenerative disease.</p>Formule :C18H26O3Couleur et forme :SolidMasse moléculaire :281.39Alacepril
CAS :<p>Alacepril (DU-1219) is a relatively novel angiotensin-converting enzyme inhibitor, used as an antihypertensive</p>Formule :C20H26N2O5SDegré de pureté :97.78%Couleur et forme :SolidMasse moléculaire :406.5Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Formule :C51H73N15O11Degré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :1072.22[Leu5]-Enkephalin, amide acetate
<p>[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.</p>Formule :C30H42N6O8Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :614.69[D-Ala2]leucine-enkephalin
CAS :<p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>Formule :C29H39N5O7Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :569.65PF3274167
CAS :PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.Formule :C19H19ClFN5O3Degré de pureté :99.67% - 99.88%Couleur et forme :SolidMasse moléculaire :419.84ms48107
CAS :<p>MS48107 enhances GPR68, crosses BBB in mice, and is selective over related proton GPCRs, transporters, and hERG channels.</p>Formule :C23H20FN5O2Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :417.44PW0787
CAS :<p>PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).</p>Formule :C23H20F4N4O2Degré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :460.42Methylnaltrexone bromide
CAS :Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.Formule :C21H26BrNO4Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :436.35DY131
CAS :<p>DY131 (DY-131) is a novel selective agonist of ERRβ and ERRγ.</p>Formule :C18H21N3O2Degré de pureté :98.65% - 99.66%Couleur et forme :SolidMasse moléculaire :311.38G15
CAS :<p>G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)</p>Formule :C19H16BrNO2Degré de pureté :98.46% - 98.59%Couleur et forme :SolidMasse moléculaire :370.24panomifene
CAS :<p>Panomiphene (Gyki-13504, EGIS-5650) is an anti-estrogen drug that is a tamoxifen (TMX) analogue.</p>Formule :C25H24F3NO2Couleur et forme :SolidMasse moléculaire :427.46AMG 837 hemicalcium
CAS :<p>AMG 837 hemicalcium: oral GPR40 agonist, binds human FFA1 (pIC50: 8.13), boosts insulin, lowers glucose in rodents.</p>Formule :C52H40CaF6O6Couleur et forme :SolidMasse moléculaire :914.954MBX-2982
CAS :<p>MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.</p>Formule :C22H24N8OSDegré de pureté :98% - 99.96%Couleur et forme :SolidMasse moléculaire :448.54Pipendoxifene
CAS :<p>Pipendoxifene (ERA-923) is an antiestrogen that blocks ER-alpha and inhibits MCF-7 breast cancer cell growth, effective even when tamoxifen-resistant.</p>Formule :C29H32N2O3Couleur et forme :SolidMasse moléculaire :456.58α-Zearalenol
CAS :<p>α-Zearalenol is one of the major metabolites of Zearalenone.</p>Formule :C18H24O5Degré de pureté :90% - 99.72%Couleur et forme :SolidMasse moléculaire :320.38Deltorphin 2
CAS :<p>Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.</p>Formule :C38H54N8O10Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :782.88Nociceptin
CAS :<p>Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.</p>Formule :C79H129N27O22Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :1809.04Adrenorphin 3TFA(88377-68-8(free base))
<p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Formule :C50H72N15O15SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1326.26EST73502 HCl
CAS :<p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>Formule :C19H27ClF2N2O2Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :388.88Nociceptin (1-7) acetate
<p>Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.</p>Formule :C31H41N7O9Degré de pureté :98.92%Couleur et forme :SoildMasse moléculaire :655.7AR 231453
CAS :<p>Azenosertib (ZN-c3) is an orally active, specific GPR119 agonist. Cost-effective and quality-assured.</p>Formule :C21H24FN7O5SDegré de pureté :99.31% - 99.34%Couleur et forme :SolidMasse moléculaire :505.52MCOPPB
CAS :<p>MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.</p>Formule :C26H40N4Couleur et forme :SolidMasse moléculaire :408.624-CMTB
CAS :<p>4-CMTB is a selective agonist of FFA2 and GPR43.It also is a positive allosteric modulator (pEC50=6.38).</p>Formule :C14H15ClN2OSDegré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :294.8b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Formule :C25H31N3O7Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :485.53DAMGO
CAS :<p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>Formule :C26H35N5O6Degré de pureté :98.83% - 99.92%Couleur et forme :SolidMasse moléculaire :513.59AZD1981
CAS :<p>AZD1981: selective CRTh2 antagonist, IC50 4 nM, 1000x specificity over 340+ enzymes/receptors, tested in asthma and other trials.</p>Formule :C19H17ClN2O3SDegré de pureté :98.87% - 99.67%Couleur et forme :SolidMasse moléculaire :388.87Antide acetate
<p>Antide acetate is an LHRH antagonist and represses LH and FSH release from the pituitary gland. </p>Formule :C84H112ClN17O16Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :1651.34TC-O 9311
CAS :<p>TC-O 9311 (TCO-9311) is an effective agonist of GPR139 (EC50 = 39 nM in CHO-K1 cells expressing human GPR139).</p>Formule :C20H19N3O4Degré de pureté :99.24% - 99.84%Couleur et forme :SolidMasse moléculaire :365.38Bisphenol B
CAS :<p>Bisphenol B has a binding affinity for estrogen receptors.</p>Formule :C16H18O2Degré de pureté :97.35% - 99.62%Couleur et forme :Crystal Or Tan Granules Odorless Slightly Brown SolidMasse moléculaire :242.31H-Val-Pro-Pro-OH
CAS :<p>H-Val-Pro-Pro-OH is an inhibitor of Angiotensin I converting enzyme (ACE)( IC50 : 9 μM).</p>Formule :C15H25N3O4Degré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :311.38VPC-13163
CAS :<p>VPC-13566 inhibits growth in LNCaP, Enzalutamide-resistant MR49F, lowers AR gene, PSA, TMPRSS2 expression, but not in AR-independent PC3 cells.</p>Formule :C16H14N2Degré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :234.3MS21570
CAS :<p>MS21570 as a GPR171 antagonist based on its ability to block,with an IC50 of 220 Nm,that reduces anxiety-like behavior and fear conditioning in mice.</p>Formule :C10H11N3S2Degré de pureté :97.79%Couleur et forme :SolidMasse moléculaire :237.34Apalutamide
CAS :<p>Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.</p>Formule :C21H15F4N5O2SDegré de pureté :99.03% - 99.91%Couleur et forme :SolidMasse moléculaire :477.43Tyr-Gly-Gly-Phe-Met-OH
CAS :<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Formule :C27H35N5O7SDegré de pureté :≥95%Couleur et forme :White Lyophilised SolidMasse moléculaire :573.662-(pentylsulfanyl)pyrimidine-4,6-diol
CAS :<p>2-(pentylsulfanyl)pyrimidine-4,6-diol 是一种新型 GRP84 激动剂。</p>Formule :C9H14N2O2SDegré de pureté :97.58%Couleur et forme :SolidMasse moléculaire :214.28JTC-801
CAS :<p>JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.</p>Formule :C26H25N3O2·HClDegré de pureté :99.27% - 99.59%Couleur et forme :SolidMasse moléculaire :447.96CVN424
CAS :<p>CVN424 is a selective and novel GPR6 Inverse agonist effective in models of Parkinson Disease.</p>Formule :C24H29F2N5O3Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :473.52Timapiprant
CAS :<p>Timapiprant (OC000459) is a potent and selective D prostanoid receptor 2 (DP2) antagonist (IC50: 13 nM).</p>Formule :C21H17FN2O2Degré de pureté :97.44% - 99.51%Couleur et forme :SolidMasse moléculaire :348.37(Sar¹)-Angiotensin II acetate
<p>(Sar¹)-Angiotensin II acetate, an analogue of Angiotensin II, is a specific agonist of angiotensin AT1 receptor.</p>Formule :C51H75N13O12Degré de pureté :99.89%Couleur et forme :SoildMasse moléculaire :1062.22Kisspeptin-10, human (TFA)(374675-21-5,FREE)
<p>Kisspeptin-10 TFA: vasoconstrictor, inhibits angiogenesis & metastasis; key in kidney development & osteoblast differentiation via GPR54 & NFATc4/BMP2.</p>Formule :C63H83N17O14·C2HF3O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1416.46Norgestrel
CAS :<p>Norgestrel (WY-3707), a synthetic progestin, is used for contraception and hinders LH/FSH, thickens mucus, and slows ova transit.</p>Formule :C21H28O2Degré de pureté :99.71% - 99.72%Couleur et forme :Crystals From Methanol White Crystalline PowderMasse moléculaire :312.45JNJ-63533054
CAS :<p>JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.</p>Formule :C17H17ClN2O2Degré de pureté :99.71% - 99.88%Couleur et forme :SolidMasse moléculaire :316.78Gluten Exorphin C
CAS :<p>Gluten exorphin C is an opioid peptide derived from wheat gluten.</p>Formule :C29H45N5O8Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :591.7Leucylarginylproline
CAS :<p>Leucylarginylproline is an inhibitor of angiotensin-converting enzyme (ACE) (IC50 : 0.27μM).</p>Formule :C17H32N6O4Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :384.47Nafoxidine
CAS :<p>Nafoxidine is an estrogen antagonist that has been used in the treatment of breast cancer.</p>Formule :C29H31NO2Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :425.56Carbetocin acetate
CAS :<p>Carbetocin acetate is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth.</p>Formule :C47H73N11O14SDegré de pureté :98.16% - 99.22%Couleur et forme :SolidMasse moléculaire :1048.22Myristyl nicotinate
CAS :<p>Myristyl nicotinate (Tetradecyl nicotinate) is an ester prodrug being developed for delivery of nicotinic acid (NIC) into the skin for prevention of actinic</p>Formule :C20H33NO2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :319.48DJ-V-159
CAS :<p>DJ-V-159 is a GPRC6A agonist, targeting the G protein-coupled receptor family C group 6 member A (GPRC6A).</p>Formule :C24H12F6N4O2Degré de pureté :99.85% - 99.96%Couleur et forme :SolidMasse moléculaire :502.37AM251
CAS :<p>AM251: potent CB1 blocker (IC50: 8 nM), 306x CB2 selective; GPR55 activator (EC50: 39 nM).</p>Formule :C22H21Cl2IN4ODegré de pureté :97.43% - 98.79%Couleur et forme :A Crystalline SolidMasse moléculaire :555.24PSN 375963
CAS :<p>PSN 375963 (PSN 375963 hydrochloride) hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.</p>Formule :C17H23N3ODegré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :285.38Zaprinast
CAS :<p>Zaprinast is a cGMP-selective phosphodiesterase (PDE) inhibitor and a GPR35 agonist.</p>Formule :C13H13N5O2Degré de pureté :99.73% - 99.77%Couleur et forme :White To Off White PowderMasse moléculaire :271.27Osilodrostat phosphate
CAS :<p>Osilodrostat phosphate is a potent oral 11β-hydroxylase inhibitor.</p>Formule :C13H13FN3O4PCouleur et forme :SolidMasse moléculaire :325.23Sparsentan
CAS :<p>Sparsentan (DARA-a) is a first-in-class orally active and highly potent dual endothelin A and angiotensin II receptor antagonist(Ki of 9.3 and 0.8 nM,</p>Formule :C32H40N4O5SDegré de pureté :97.94% - 98.69%Couleur et forme :SolidMasse moléculaire :592.75Kisspeptin 234 acetate(1145998-81-7 free base)
<p>Kisspeptin receptor (KISS1/GPR54) blocker; analog to kisspeptin-10. Curbs IP activation (IC50=7nM) & GnRH release.</p>Formule :C65H82N18O15Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :1355.46GSK1292263
CAS :<p>GSK1292263 is a GPR119 agonist and has been investigated for the treatment of DIABETES MELLITUS, TYPE 2.</p>Formule :C23H28N4O4SDegré de pureté :98.34% - 99.53%Couleur et forme :SolidMasse moléculaire :456.56Palosuran hydrochloride 540769-28-6(free base)
<p>Palosuran hydrochloride 540769-28-6(free base)(ACT-058362 hydrochloride) is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.</p>Formule :C25H31ClN4O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :454.99Alvimopan monohydrate
CAS :<p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>Formule :C25H34N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :442.55Delapril hydrochloride
CAS :<p>Delapril HCl (indalapril) is a prodrug forming two ACE inhibitors, blocking angiotensin I-II conversion.</p>Formule :C26H33ClN2O5Degré de pureté :97.18% - 97.45%Couleur et forme :White Crystalline PowderMasse moléculaire :489.01
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