Enzyme
Les inhibiteurs d'enzymes sont des molécules qui se lient aux enzymes et diminuent leur activité. Ces inhibiteurs sont largement utilisés en recherche pour étudier la cinétique enzymatique, la régulation et le rôle spécifique des enzymes dans les voies métaboliques. Les inhibiteurs d'enzymes sont également cruciaux dans le développement de médicaments, car de nombreux agents thérapeutiques agissent en inhibant les enzymes impliquées dans les processus pathologiques. En ciblant les enzymes, ces inhibiteurs peuvent moduler les voies biochimiques et offrir des traitements potentiels pour diverses maladies. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs d'enzymes de haute qualité pour soutenir vos recherches en biochimie, pharmacologie et découverte de médicaments.
Sous-catégories appartenant à la catégorie "Enzyme"
- Anhydrase carbonique(177 produits)
- Hydroxylase(30 produits)
- MPO(2 produits)
- Réductase(52 produits)
- Tyrosinase(67 produits)
3586 produits trouvés pour "Enzyme"
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Carbonic anhydrase inhibitor 30
<p>Carbonic anhydrase inhibitor30 (compound 17) is an inhibitor of carbonic anhydrase with Ki values of 2.13 μM for hCA I and 0.161 μM for hCA II[1].</p>Formule :C23H22FN3O5SCouleur et forme :SolidMasse moléculaire :471.12642α-Amylase (with starch)
CAS :Degré de pureté :≥ 600U/gCouleur et forme :White to beige or pale yellow-brown powderhCAXII-IN-7
<p>hCAXII-IN-7 (compound 6e) functions as an inhibitor of human carbonic anhydrase XII (hCA XII) and possesses blood-brain barrier (BBB) permeability.</p>Formule :C26H25N5O6S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :567.64hCA/VEGFR-2-IN-2
<p>Compound 8g (hCA/VEGFR-2-IN-2) is an indolinonylbenzenesulfonamide identified as a potential dual inhibitor targeting cancer-associated isozymes hCA IX/XII and</p>Formule :C23H26N6O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :498.55hCA/VEGFR-2-IN-4
<p>hCA/VEGFR-2-IN-4 (compound 15b), an indolinylbenzenesulfonamide, serves as a potential dual inhibitor targeting cancer-related human carbonic anhydrases hCA IX/</p>Formule :C22H23FN6O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :502.52hCAIX/XII-IN-14
<p>hCAIX/XII-IN-14 (Compound 1i) is an inhibitor of hCAIX and hCAXII, with Ki values of 9.4 nM for hCAII, 5.6 nM for hCAIX, and 6.3 nM for hCAXII.</p>Formule :C16H14F3N3O4SCouleur et forme :SolidMasse moléculaire :401.36α-Pyrone
CAS :<p>Alpha-Pyrone exhibits inhibitory activity against tyrosinase, carbonic anhydrase 1, and carbonic anhydrase 9</p>Formule :C5H4O2Couleur et forme :SolidMasse moléculaire :96.08Invertase, from Saccharomyces cerevisiae
CAS :Couleur et forme :White to faint-yellow or light-brown powderCarbonic anhydrase
CAS :<p>Carbonic anhydrase, a zinc enzyme in all life forms, converts CO2 to bicarbonate; studied for cancer, glaucoma, obesity, epilepsy.</p>Couleur et forme :SolidCAIX/CAXII-IN-4
<p>CAIX/CAXII-IN-4 (Compound 7h) is an inhibitor of carbonic anhydrase (CA) that binds to CAIX, CA XII, and CAII with Ki values of 1.324 μM, 0.435 μM, and 3.035 μM, respectively. This compound exhibits broad-spectrum anti-tumor activity and inhibits the proliferation of central nervous system tumor cells U251, with a GI50 of 0.361 μM.</p>Formule :C23H21N5O3SCouleur et forme :SolidMasse moléculaire :447.51TSPO/Carbonic Anhydrase Modulator 1
<p>TSPO/Carbonic Anhydrase Modulator 1 (Compound 3) acts as a dual modulator of mitochondrial translocator protein and carbonic anhydrase, with a TSPOKi of 1.340 μM and a CAVII KA of 10.7 μM. It enhances neurosteroid production, increases BDNF gene expression, and demonstrates neuroprotective activity.</p>Formule :C35H51N3O3Couleur et forme :SolidMasse moléculaire :561.798Tyrosinase-IN-36
<p>Tyrosinase-IN-36 is a moderately potent inhibitor of tyrosine, exhibiting an inhibition percentage of 42.75% compared to kojic acid at a concentration of 100 μM and possesses antioxidant activity.</p>Couleur et forme :Odour SolidGirentuximab
CAS :<p>Girentuximab (G250) is an anti-carbonic anhydrase IX (CAIX) monoclonal antibody with anti-cancer activity for the study of uroepithelial carcinoma PET (ZiPUP).</p>Couleur et forme :LiquidMasse moléculaire :145.55 kDaTyrosinase-IN-40
<p>Tyrosinase-IN-40 (Compound 9r) is a competitive inhibitor of tyrosinase, boasting an IC50 value of 17.02 µM and a Ki value of 14.87 µM. This compound also exhibits antioxidant activity and can be utilized in studies related to melanin.</p>Formule :C34H29N9O10Couleur et forme :SolidMasse moléculaire :723.648Hyaluronidase
CAS :Degré de pureté :≥ 300U/mgCouleur et forme :White to yellow powderMasse moléculaire :-CAIX Inhibitor S4
CAS :<p>CAIX Inhibitor S4 (S4) is an effective inhibitor of carbonic anhydrase IX/XII with a Ki of 7 nM and 2 nM, respectively.</p>Formule :C15H17N3O4SDegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :335.38hCAII-IN-8
CAS :<p>Compound CDy9 is a highly selective inhibitor of carbonic anhydrase (CA) with an IC50 value of 0.18 μM for hCA II.</p>Formule :C15H16N2O5SDegré de pureté :99.73%Couleur et forme :SoildMasse moléculaire :336.36Carbonic anhydrase inhibitor 32
<p>Carbonic anhydrase inhibitor32 (compound 5B) is an orally active, selective inhibitor of hCA (carbonic anhydrase) II/VII, with Ki values of 6.3 nM for hCA II, 10.1 nM for hCA VII, and 681 nM for hCA I. It shows potential for neuroprotection and anticonvulsant effects by reducing mTOR activation and increasing hippocampal KCC2 levels.</p>Formule :C17H16N6O3SCouleur et forme :SolidMasse moléculaire :384.41Carbonic anhydrase inhibitor 31
<p>Carbonic anhydrase inhibitor31 is an mtCA2 inhibitor (Ki: 5.2 nM) that can be used in antituberculosis research.</p>Formule :C24H20N6O5SCouleur et forme :SolidMasse moléculaire :504.12159hCAIX-IN-17
<p>hCA IX-IN-1 inhibits hCA I/II/IX/XII with Ki of 331.4/28.4/9.4/17.8 nM, has anticancer properties.</p>Formule :C19H18N2O3SCouleur et forme :SolidMasse moléculaire :354.42hCAII/XII-IN-1
<p>hCAII/XII-IN-1 (compound 4l) is a potent inhibitor of hCAXII and hCAII, with Ki values of 8.4 nM and 9.4 nM, respectively. It plays a significant role in cancer research.</p>Formule :C22H20N4O6S2Couleur et forme :SolidMasse moléculaire :500.547CA IX/VEGFR-2-IN-3
<p>CAIX/VEGFR-2-IN-3 (Compound 6i) is an inhibitor of Carbonic Anhydrase IX and VEGFR-2, with IC50 values of 41 and 48 nM, respectively. It exhibits anticancer activity by inhibiting the growth of MCF-7 breast cancer cells (IC50 of 22.33 μM) and mouse fibroblast cell line 3T3, where cell viability is reduced to below 40% at a concentration of 100 μM. This compound is applicable for research in the field of cancer treatment.</p>Formule :C19H16ClN3O5S2Couleur et forme :SolidMasse moléculaire :465.93hCA/VEGFR-2-IN-3
<p>hCA/VEGFR-2-IN-3 (compound 8j) is an indolinonylbenzenesulfonamide with potential as a dual inhibitor of cancer-associated hCA IX/XII and VEGFR-2.</p>Formule :C24H28N6O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :528.58Peroxidase
CAS :Degré de pureté :≥ 85units/mg (dry basis)Couleur et forme :Beige to light-brown, reddish brown or dark brown lyophilised powderMasse moléculaire :-hCAII/IX-IN-1
<p>hCAII/IX-IN-1 (compound 4o) is a potent inhibitor of hCAII and hCAIX, with Ki values of 7.4 nM and 7.0 nM, respectively. It plays a significant role in cancer research.</p>Formule :C23H22N4O7S2Couleur et forme :SolidMasse moléculaire :530.573hCA/Wnt/β-catenin-IN-1
<p>hCA/Wnt/β-catenin-IN-1 (Compd 15) serves as an inhibitor with selective affinity for hCA isoforms II, IX, and XII, exhibiting K i values of 33.6, 24.1, and 6.8</p>Couleur et forme :Odour SolidCarbonic anhydrase inhibitor 29
<p>Carbonic anhydrase inhibitor29 (Compound 5d) is an inhibitor targeting carbonic anhydrase IX and XII, with an inhibition constant (Ki) of 26.6 nM for carbonic anhydrase IX and a Ki of 10.9 nM for carbonic anhydrase XII. Carbonic anhydrase inhibitor29 can be used in cancer research.</p>Couleur et forme :Odour SolidPyridine-2-aldoxime methochloride
CAS :Formule :C7H9N2O·ClDegré de pureté :≥ 98.0%Couleur et forme :White to off-white or light yellow crystalline powderMasse moléculaire :172.61CAXII-IN-2
<p>CAXII-IN-2 (compound 3j) is a highly effective inhibitor of CAXII. It demonstrates inhibitory activity against CA IX and CAXII, with Ki values of 27.4 nM and 4.0 nM, respectively.</p>Formule :C16H13FNO4PCouleur et forme :SolidMasse moléculaire :333.05662IOX2-NH2-1
CAS :<p>IOX2-NH2-1 inhibits E. coli EGLN-3 (prolyl hydroxylase) with an IC50 of 0.02–1 μM.</p>Formule :C19H17N3O5Degré de pureté :98.77% - 99.91%Couleur et forme :SoildMasse moléculaire :367.36α-Glycosidase-IN-2
<p>α-Glycosidase-IN-2 (compound 8b) is an inhibitor of α-glycosidase, displaying Ki values of 74.16 nM and 6.09 nM for aldose reductase and α-glycosidase, respectively. This compound is utilized in research related to diabetes.</p>Formule :C25H22N6OS2Couleur et forme :SolidMasse moléculaire :486.61DPP IV/hCA II-IN-1
CAS :<p>DPP IV/hCA II-IN-1: strong DPP IV & CA inhibitor, IC50=0.049μM (DPP IV), Ki=0.0361-3.034μM (CA II-IV).</p>Formule :C17H20N2O5SCouleur et forme :SolidMasse moléculaire :364.42Trypsin, bovine origin
CAS :Degré de pureté :≥ 2000units/mg (USP)Couleur et forme :White or almost white crystalline powderMasse moléculaire :-Phenylsulfamide
CAS :<p>Phenylsulfamide (Compound 10), acting as an inhibitor of human carbonic anhydrase-II (hCA-II), exhibits a dissociation constant (Kd) of 45.50 μM and an</p>Formule :C6H8N2O2SCouleur et forme :SolidMasse moléculaire :172.2hCAIX/XII-IN-11
<p>hCAIX/XII-IN-11 (Compound 6c) is an inhibitor of hCA IX and hCA XII, exhibiting Ki values of 0.7 μM for both isoforms. This compound is applicable in cancer research.</p>Formule :C13H10FN3O4Masse moléculaire :291.06553TPT-004
<p>TPT-004, a TPH inhibitor, exhibits superior pharmacokinetic and pharmacodynamic properties, and demonstrates efficacy in preclinical models for attenuating</p>Couleur et forme :Odour SolidAc-[Nle4,D-Phe7]-α-MSH (4-10)-NH2
CAS :<p>Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effect</p>Formule :C47H64N14O10Couleur et forme :SolidMasse moléculaire :985.1Tyrosinase-IN-14
<p>Tyrosinase-IN-14 (compound 7m), a tyrosinase inhibitor, modulates the enzyme's secondary structure to diminish its catalytic function, exhibits low cytotoxicity</p>Formule :C21H13Br2N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :547.22Peroxidase, from horseradish, approx. 200 U/mg
CAS :Degré de pureté :≥ 150U/mgCouleur et forme :Beige to light-brown, reddish brown or dark brown lyophilised powderMasse moléculaire :-Proteinase K
CAS :Degré de pureté :≥ 30units/mg (pH 7.5, 37°C, dried basis)Couleur et forme :White or almost white lyophilized powderMasse moléculaire :-Tyrosinase-IN-34
<p>Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.</p>Formule :C19H14BrClN4OCouleur et forme :SolidMasse moléculaire :429.7Tyrosinase-IN-32
<p>Tyrosinase-IN-32 (compound 11), a hydroxamate-based alkaloid extracted from black pepper (Piper nigrum L.), functions as an inhibitor of mushroom tyrosinase. In addition to its inhibitory properties, it exhibits antioxidant activity.</p>Formule :C15H19NO3Couleur et forme :SolidMasse moléculaire :261.32P-Hydroxybenzoate Hydroxylase
CAS :Couleur et forme :Yellowish lyophilised powderMasse moléculaire :55 ~ 60 kDaLysozyme, from chicken egg white
CAS :Degré de pureté :≥ 20,000U/mgCouleur et forme :White to off-white powderMasse moléculaire :-TrkA Protein, Rabbit, Recombinant (His)
<p>TrkA Protein, Rabbit, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.</p>Couleur et forme :Lyophilized PowderMasse moléculaire :43.4 kDa (predicted)TrkB Protein, Canine, Recombinant (hFc)
<p>TrkB Protein, Canine, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.</p>Couleur et forme :Lyophilized PowderMasse moléculaire :71.2 kDa (predicted)TrkA Protein, Rat, Recombinant (hFc)
<p>TrkA Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.</p>Couleur et forme :Lyophilized PowderMasse moléculaire :69.2 kDa (predicted); 92-102 kDa (reducing conditions)Cuprizone
CAS :<p>Cuprizone is a copper chelator.Cuprizone is used to induce schizophrenia in mice.Cuprizone induces oligodendrocyte death and induces a demyelination response.</p>Formule :C14H22N4O2Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :278.35TrkA Protein, Human, Recombinant (His)
<p>TrkA Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.</p>Degré de pureté :98.7%Couleur et forme :Lyophilized PowderMasse moléculaire :39.5 kDa (predicted); 60-65 kDa (reducing condition, due to glycosylation)HER3/ERBB3 Protein, Cynomolgus/Rhesus macaque, Recombinant (His)
<p>Her3, also called ErbB3, is a type I membrane glycoprotein that is a member of the ErbB family of tyrosine kinase receptors.Her3 is expressed in keratinocytes,</p>Couleur et forme :Lyophilized PowderMasse moléculaire :69.54 kDa (predicted). Due to glycosylation, the protein migrates to 85-105 kDa based on Tris-Bis PAGE result.p38 γ/MAPK12 Protein, Human, Recombinant
<p>p38 gamma/MAPK12 Protein, Human, Recombinant is expressed in Baculovirus insect cells.</p>Couleur et forme :Lyophilized PowderMasse moléculaire :42.1 kDa (predicted); 43 kDa (reducing conditions)Thrombopoietin Protein, Mouse, Recombinant (C-His)
<p>Expression System: HEK293 Cells<br>Length: 22-356, Full Length of Mature Protein<br>Activity: Cell Activity</p>Masse moléculaire :37.20 kDa (Predicted); 75-95 kDa (Due to glycosylation)Carbonic Anhydrase 12 Protein, Human, Recombinant (His) V2
<p>Expression System: HEK293 Cells<br>Length: 25-301, Extracellular Domain<br>Activity: Enzyme Activity</p>Masse moléculaire :32.22 kDa (Predicted); 40-50 kDa (Due to glycosylation)ErbB4 Protein, Rat, Recombinant (His)
<p>ErbB4 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.</p>Couleur et forme :Lyophilized PowderMasse moléculaire :71.3 kDa (predicted); 75-95 kDa (reducing condition, due to glycosylation)TrkB Protein, Human, Recombinant (His), Biotinylated
<p>Expression system: HEK293 Cells<br>Length: 1-430, Partial<br>Activity: ELISA</p>Couleur et forme :Lyophilized PowderMasse moléculaire :45.66 kDa (predicted); 65.4 kDa (reducing contition, due to glycosylation)DDR2 Protein, Human, Recombinant (His & Avi), Biotinylated
<p>Expression system: HEK293 Cells<br>Length: 1-399, Partial<br>Activity: BLI</p>Couleur et forme :Lyophilized PowderMasse moléculaire :45.84 kDa (predicted); 60.4 kDa (reducing contition)Anti-Tyrosinase/TYR Antibody (7Z445)
<p>Anti-Tyrosinase/TYR Antibody (7Z445) is an antibody targeting Tyrosinase/TYR. Anti-Tyrosinase/TYR Antibody (7Z445) can be used in ELISA, IF.</p>Couleur et forme :Odour LiquidTrkA Protein, Human, Recombinant
<p>TrkA Protein, Human, Recombinant is expressed in HEK293 Cells. The accession number is P04629.</p>Degré de pureté :> 95% as analyzed by SDS-PAGE - > 95% as analyzed by SDS-PAGECouleur et forme :Lyophilized PowderMasse moléculaire :65~85 kDa (Reducing conditions)HER3/ERBB3 Protein, Mouse, Recombinant (His)
<p>HER3/ERBB3 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.</p>Degré de pureté :97.1%Couleur et forme :Lyophilized PowderMasse moléculaire :70 kDa (predicted); 95 kDa (reducing condition, due to glycosylation)TrkA Protein, Cynomolgus, Recombinant (His)
<p>TrkA Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.</p>Couleur et forme :Lyophilized PowderMasse moléculaire :43.95 kDa (predicted); 86 kDa (reducing conditions)HER3/ERBB3 Protein, Mouse, Recombinant (hFc)
<p>HER3/ERBB3 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.</p>Couleur et forme :Lyophilized PowderMasse moléculaire :95.23 kDa (predicted); 117.08 kDa (reducing conditions)p38 γ/MAPK12 Protein, Human, Recombinant (His & GST)
<p>p38 gamma/MAPK12 Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag.</p>Couleur et forme :Lyophilized PowderMasse moléculaire :69.8 kDa (predicted); 65 kDa (reducing conditions)TrkB Protein, Human, Recombinant (His) V2
<p>Expression System: HEK293 Cells<br>Length: 32-430, Extracellular Domain<br>Activity: ELISA</p>Masse moléculaire :45.2 kDa (Predicted); 65-80 kDa (Due to glycosylation)HER3/ERBB3 Protein, Human, Recombinant (His & Avi), FITC-Labeled
<p>Her3, also called ErbB3, is a type I membrane glycoprotein that is a member of the ErbB family of tyrosine kinase receptors.Her3 is expressed in keratinocytes,</p>Couleur et forme :Lyophilized PowderMasse moléculaire :71.6 kDa (predicted). Due to glycosylation, the protein migrates to 72-75 kDa based on Tris-Bis PAGE result.PTP α/PTPRA Protein, Human, Recombinant (aa 174-793, His & GST)
<p>PTPRA is reported to be involved in cancer development and progression through activating the Src family kinase (SFK) signaling pathways.</p>Couleur et forme :Lyophilized PowderMasse moléculaire :99 kDa (predicted); 90 kDa (reducing conditions)Mer Protein, Mouse, Recombinant (hFc)
<p>Mer Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.</p>Couleur et forme :Lyophilized PowderMasse moléculaire :79.3 kDa (predicted); 130 kDa (reducing condition, due to glycosylation)HER3/ERBB3 Protein, Rhesus, Recombinant
<p>HER3/ERBB3 Protein, Rhesus, Recombinant is expressed in HEK293 mammalian cells.</p>Degré de pureté :92.6%Couleur et forme :Lyophilized PowderMasse moléculaire :69.5 kDa (predicted)HER3/ERBB3 Protein, Human, Recombinant (hFc), Biotinylated
<p>HER3/ERBB3 Protein, Human, Recombinant (hFc), Biotinylated is expressed in HEK293 mammalian cells with hFc tag.</p>Couleur et forme :Lyophilized PowderMasse moléculaire :95.4 kDa (predicted)
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