Enzyme
Les inhibiteurs d'enzymes sont des molécules qui se lient aux enzymes et diminuent leur activité. Ces inhibiteurs sont largement utilisés en recherche pour étudier la cinétique enzymatique, la régulation et le rôle spécifique des enzymes dans les voies métaboliques. Les inhibiteurs d'enzymes sont également cruciaux dans le développement de médicaments, car de nombreux agents thérapeutiques agissent en inhibant les enzymes impliquées dans les processus pathologiques. En ciblant les enzymes, ces inhibiteurs peuvent moduler les voies biochimiques et offrir des traitements potentiels pour diverses maladies. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs d'enzymes de haute qualité pour soutenir vos recherches en biochimie, pharmacologie et découverte de médicaments.
Sous-catégories appartenant à la catégorie "Enzyme"
- Anhydrase carbonique(196 produits)
- Hydroxylase(36 produits)
- MPO(2 produits)
- Réductase(51 produits)
- Tyrosinase(71 produits)
3620 produits trouvés pour "Enzyme"
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hCAII-IN-2
CAS :hCAII-IN-2 inhibits human carbonic anhydrases I, II, IX, XII with Ki values of 261.4, 3.8, 19.6, 45.2 nM respectively.Formule :C25H18ClN5O4SCouleur et forme :SolidMasse moléculaire :519.96Clofenamide
CAS :Clofenamide is a low-ceiling sulfonamide diuretic.Formule :C6H7ClN2O4S2Couleur et forme :SolidMasse moléculaire :270.71hCA I-IN-1
CAS :hCA I-IN-1 inhibits hCA I (Ki: 38.3 nM), II (Ki: 716.4 nM), IX (Ki: 940.1 nM), XII (Ki: 192.8 nM).Formule :C27H23N5O4SCouleur et forme :SolidMasse moléculaire :513.57CDK2-IN-12
CAS :CDK2-IN-12 (10b), potent CDK2 inhibitor, IC50: 11.6 μM; inhibits hCA I/II/IX/XII, KI: 3534/638.4/44.3/48.8 nM; anti-cancer properties.Formule :C20H17N9O2SCouleur et forme :SolidMasse moléculaire :447.47hCAIX/XII-IN-2
CAS :Compound 6a: Selective hCAIX/XII inhibitor; Ki: 30 nM (hCAIX), 3.6 nM (hCAXII); >10,000 nM (hCAI/II).Formule :C19H14N2O4Couleur et forme :SolidMasse moléculaire :334.33Phenylthiazolylthiourea
CAS :Phenylthiazolylthiourea ia a dopamine-beta-hydroxylase inhibitor.Formule :C10H9N3S2Couleur et forme :SolidMasse moléculaire :235.33CDK2-IN-11
CAS :CDK2-IN-11 inhibits CDK2 (IC50: 6.4 μM) and targets hCA II, IX, XII (Ki: 23.4-56.3 nM); suited for cancer research.Formule :C18H14ClN7O2SCouleur et forme :SolidMasse moléculaire :427.87CK1 δ/CSNK1D Protein, Human, Recombinant (Baculovirus, His)
Expression system: Baculovirus
Length: 1-415, Full Length
Activity: Not TestedDegré de pureté :85%Couleur et forme :Odour Lyophilized PowderRef: TM-TMPH-03771
1mg8.803,00€5µg947,00€10µg1.598,00€20µg2.712,00€50µg3.520,00€100µg4.337,00€200µg5.358,00€500µg7.113,00€hCAI/II-IN-1
CAS :hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).Formule :C18H29N5O3S3Couleur et forme :SolidMasse moléculaire :459.65hCAIX-IN-11
CAS :hCAIX-IN-11 inhibits carbonic anhydrases IX & XII with Ki of 32.7 nM & 623.5 nM, respectively.Formule :C21H15ClN4O3Couleur et forme :SolidMasse moléculaire :406.82(R)-Nepicastat HCl
CAS :(R)-Nepicastat HCl (RS-25560-198 HCl), R-enantiomer, inhibits bovine/human dopamine-β-hydroxylase (IC50: 25.1/18.3 nM); not affecting other enzymes/receptors.Formule :C14H15F2N3S·HClDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :331.81QPRTase Protein, Human, Recombinant (His)
Nicotinate-Nucleotide Pyrophosphorylase (QPRT) belongs to the nadC/modD family.Couleur et forme :Lyophilized PowderMasse moléculaire :34 KDa (reducing condition)Ref: TM-TMPJ-00473
1mg2.535,00€5µg113,00€10µg178,00€20µg284,00€50µg523,00€100µg759,00€200µg1.103,00€500µg1.765,00€PPIE Protein, Human, Recombinant (His)
Peptidyl-prolyl cis-trans isomerase E, also known as Cyclophilin E, Cyclophilin-33, Rotamase E, CYP33, PPIE, is an enzyme which belongs to the cyclophilin-typeCouleur et forme :Lyophilized PowderMasse moléculaire :34 KDa (reducing condition)Ref: TM-TMPJ-01389
1mg2.535,00€5µg113,00€10µg178,00€20µg284,00€50µg523,00€100µg759,00€200µg1.103,00€500µg1.765,00€WES-1
CAS :WES-1 (Compound 8g), a carbonic anhydrase IX inhibitor (Ki: 55.9 μM), exhibits broad-spectrum antiproliferative activity against various cancer cell lines,Formule :C20H20N4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :396.46L-693612 HCl
CAS :L-693612 HCl is an inhibitor of carbonic anhydrase.Formule :C14H25ClN2O5S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.01AHR-15010
CAS :AHR-15010 is a novel anti-arthritic agent.Formule :C10H16N2O8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :356.37Telotristat besilate
CAS :Telotristat besilate is an inhibitor of tryptophan hydroxylase.Formule :C31H28ClF3N6O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :705.11L 662583
CAS :L 662583 is a topical inhibitor of carbonic anhydrase.Formule :C13H17ClN2O5S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.93L-693612
CAS :L-693612 is an inhibitor of carbonic anhydrase.Formule :C14H24N2O5S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :396.55GV2-20
CAS :GV2-20 is an effective carbonic anhydrase 2 inhibitors.Formule :C15H13N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :331.28L 645151
CAS :L 645151 is an inhibitor of lipophilic CA.Formule :C12H14N2O4S2Couleur et forme :SolidMasse moléculaire :314.38Disulfamide
CAS :Disulfamide: Oral carbonic anhydrase inhibitor, IC50 0.07 μM, diuretic by blocking Na+/HCO3- reabsorption.Formule :C7H9ClN2O4S2Degré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :284.74Fenprinast
CAS :Fenprinast is a tryptophan-like bronchodilator utilized in the study of allergic and exercise-induced asthma. It exhibits oral activity.Formule :C16H16ClN5OCouleur et forme :SolidMasse moléculaire :329.783-Allylphenol
CAS :3-Allylphenol is an inhibitor of dopamine β-hydroxylase (DBH; Ki = 12 mM).Formule :C9H10OCouleur et forme :SolidMasse moléculaire :134.18JM6
CAS :JM6 is a weak kynurenine 3-monooxygenase (KMO) inhibitor that acts on mouse KMO (IC50: 19.85 μM). JM6 can be used to study Alzheimer's disease.Formule :C23H26N4O6S2Couleur et forme :SolidMasse moléculaire :518.61hCAIX-IN-5
CAS :hCAIX-IN-5 was a selective hCAIX inhibitor, inhibiting hCAI, hCAII, hCAIV, and hCAIX with Ki values of >10000, >10000, 130.7, and 829.1 nM, respectively.Formule :C18H12FNO3Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :309.29LP-533401
CAS :LP-533401 is an inhibitor of Tryptophan hydroxylase 1. It is used for regulates serotonin production in the gut.Formule :C27H22F4N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :526.48Invertase
CAS :Invertase is an enzyme that catalyzes the hydrolysis of sucrose to glucose and fructose and can be found in plants and microorganisms
Couleur et forme :Beige PowderTyrosinase-IN-2
CAS :Tyrosinase-IN-2, a potent tyrosinase inhibitor, may help in skin lightening and food preservation research.Formule :C8H8N4O2SDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :224.24Ref: TM-T60278
5mg48,00€10mg71,00€25mg135,00€50mg212,00€100mg340,00€200mg467,00€1mL*10mM (DMSO)49,00€Sultiame
CAS :Sultiame is an inhibitor of carbonic anhydrase. Sultiame can be used in antiepileptic research.Formule :C10H14N2O4S2Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :290.36Transglutaminase from streptoverticillium mobaraense
CAS :selectively deamidates gluten peptides, which results in strongly enhanced T cell-stimulatory activity. It has also been used in a study to improve quantifiable assays to fully characterize the role of transglutaminase in diseases such as Huntington′s disease and Alzheimer′s disease.Couleur et forme :PowderMaltose phosphorylase (from bacteria), ammonium sulphate suspension
CAS :Maltose phosphorylase (systematic name maltose:phosphate 1-beta-D-glucosyltransferase; EC 2.4.1.8) is an enzyme that catalyzes the following reaction: maltose + Pi ⇌ D-glucose + beta-D-glucose 1-phosphate One unit of maltose phosphorylase will produce 1.0 μmole of D-Glucose from maltose per minute at pH 7.0 and 30°C.Degré de pureté :Min. 95%Masse moléculaire :0 g/molLyticase
CAS :Lyticase is a lysing enzyme that is designed to lyse cells in a biological sample. It contains an optimized wild-type guanine nucleotide-binding protein and has been shown to have high enzyme activities. Lyticase has also been shown to be active against opportunistic fungal strains, such as Candida glabrata, by disrupting their cell membranes. Lyticase is classified as a signal peptide with nuclear DNA, which allows it to be used in wastewater treatment applications. The enzyme can also be used for the analysis of the Toll-like receptor (TLR) response of microbes due to its electrochemical impedance spectroscopy properties.Degré de pureté :Min. 95%Endoproteinase Glu-C
CAS :Endoproteinase Glu-C (Glutamyl endopeptidase, V8 protease, GluV8, EC 3.4.21.19) is a protease that hydrolyzes peptide bonds at the carboxylic side of either exclusively Glu, or Glu and Asp residues, depending on the buffer conditions. One unit of endoproteinase Glu-C will generate 1.0 μmole of p-nitroaniline from Z-Phe-Leu-Glu-pNA peptide mimic substrate per minute at pH 7.8 and 25 °C. Z-Phe-Leu-Glu-pNA substrate is available here.molecular weight ~ 27000.
Formule :C65H98N16O19Masse moléculaire :1,407.56 g/molhCAII-IN-9
CAS :hCAII-IN-9 inhibits hCA II/IX/XII with IC50s of 1.18, 0.17, 2.99 μM; not BBB permeable.
Formule :C15H16ClN3O5S2Degré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :417.89Cocarboxylase hydrochloride
CAS :Cocarboxylase hydrochloride is a coenzyme derivative, which is primarily sourced from thiamine (vitamin B1). It plays a crucial role in biochemical processes by facilitating the enzymatic decarboxylation of alpha-keto acids within the cellular environment. This action is fundamental in energy production as it aids in the conversion of pyruvate to acetyl-CoA, subsequently entering the citric acid cycle. Cocarboxylase hydrochloride’s involvement in carbohydrate metabolism is especially vital for tissues with high metabolic rates, such as the heart and brain.
Formule :C12H19N4O7P2S·ClHClDegré de pureté :Min. 95%Masse moléculaire :497.23 g/molCarbonic anhydrase inhibitor 6
CAS :Carbonic anhydrase inhibitor 6 is an hCA inhibitor that inhibits hCA IX, hCA II, hCA XII, and hCA I. It is used in the study of lupus erythematosus.Formule :C26H25N3O5SDegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :491.56Ref: TM-T63305
1mg164,00€2mg234,00€5mg389,00€10mg532,00€25mg820,00€50mg1.063,00€100mg1.350,00€200mg1.783,00€Glucose dehydrogenase
CAS :Glucose Dehydrogenase is an enzyme, which is typically derived from microbial sources such as bacteria and fungi. It functions by catalyzing the oxidation of glucose to gluconolactone, concurrently reducing a cofactor such as NAD⁺ or PQQ. This biochemical reaction is critical in various analytical applications due to its specificity and efficiency in glucose detection.Glucose Dehydrogenase is widely employed in the development of biosensors and diagnostic assays. Its primary application is in blood glucose monitoring devices, where its ability to accurately quantify glucose levels is crucial for managing diabetes. Additionally, it is utilized in research and development settings for biochemical assays that require precise glucose measurements. The enzyme's rapid and specific action on glucose molecules makes it an indispensable tool in both clinical and laboratory environments, contributing to advancements in biosensing technologies and metabolic studies.Bupicomide
CAS :Bupicomide is a dopamine β-hydroxylase inhibitor with antihypertensive and vasodilatory activity and may be used in the study of hypertension.Formule :C10H14N2ODegré de pureté :99.84% - >99.99%Couleur et forme :SolidMasse moléculaire :178.23Acetylcholinesterase, type VI-S, 200-1,000 units/mg protein
CAS :Acetylcholinesterase is an enzyme that breaks down acetylcholineDegré de pureté :Min. 95%Couleur et forme :PowderEWP 815
CAS :EWP 815, a disulfiram analog, inhibits Ins(1,4)P2, Ins(1,4,5)P3 phosphatases, and dopamine β-hydroxylase.Formule :C12H22N4S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :350.59Lysozyme - Enzyme activity min 40000 FIP/mg
CAS :Lysozyme is a bacteriolytic enzyme, which is primarily derived from hen egg whites. It functions by hydrolyzing the β-1,4-glycosidic linkages in the peptidoglycan layer of bacterial cell walls, particularly in Gram-positive bacteria. This enzymatic activity results in the lysis and subsequent death of the bacterial cells, providing a potent antimicrobial effect.Couleur et forme :PowderProteinase K - from Tritirachium album
CAS :Proteinase K is used for the general digestion of proteins and removal of protein contamination in nucleic acids. Addition of Protease K also stabilizes nucleic acids by degrading any nucleases present. Proteinase K is active in wide range of pH range, in the presence of SDS, urea and Guanidinium chloride at low to moderate concentrations. Proteinase K is also known under names of protease K and endopeptidase K.Butyrylcholinesterase human
CAS :Butyrylcholinesterase is an enzyme made in the liver and found mainly in blood plasma. Butyrylcholinesterase (EC 3.1.1.8), also known as BChE or BuChE, is a nonspecific cholinesterase enzyme that hydrolyses choline-based esters. One unit of Butyrylcholinesterase will hydrolyze 1.0 μmole of butyrylcholine to choline and butyrate per minute at pH 8.0 and 37 °C.
Couleur et forme :PowderD-Alanine Aminotransferase, Bacilus subtilis, Recombinant
D-Alanine aminotransferase (L-glutamic-pyruvic transaminase; EC 2.6.1.21) is an enzyme that catalyzes the following reaction: D-alanine + α-ketoglutarate ⇌ pyruvate + D-glutamate Please enquire for more information about D-Alanine Aminotransferase, Bacilus subtilis, Recombinant including the price, delivery time and more detailed product information at the technical inquiry form on this page
Degré de pureté :>90% By Sds-Page.β-Galactosidase >100KU/g
CAS :beta-Galactosidase (EC 3.2.1.23, shortly beta-Gal, also know as lactase) catalyses the hydrolysis of beta-d-galactoside in the presence of water to galactose and alcohol, or lactose into glucose and galactose. beta-Gal has a molecular weight of 540,000 and is composed of four identical subunits of MW 135,000, each with an independent active site. The enzyme has divalent metals as cofactors, with chelated Mg2+ ions required to maintain active site conformation. The molecule contains numerous sulfhydryl groups and is glycosylated.Couleur et forme :Powderα-Glucosidase from bacillus stearothermophilus, lyophilized powder, 250 Units
CAS :α-Glucosidase is a glycoside hydrolase enzyme that hydrolyzes α-1,4-linked D-glucose residues to produce α-D-glucose. This enzyme has been isolated from Bacillus stearothermophilus and is used as an industrial catalyst in the production of glucose syrups. One Unit of α-Glucosidase will release 1.0 µmole of p-nitrophenol from the chromogenic substrate mimic 4-nitrophenyl α-D-glucopyranoside per minute under optimum conditions.Couleur et forme :Powderendo-β-1,4-Mannanase
CAS :Endo-β-1,4-Mannanase (other names Mannan endo-1,4-β-mannosidase, endo-β-1,4-mannase, β-mannanase B, β-1, 4-mannan 4-mannanohydrolase, endo-β-mannanase, β-D-mannanase, 1,4-β-D-mannan mannanohydrolase; EC 3.2.1.78) is an enzyme, catalyzing the hydrolysis of -1, 4-mannosidic linkages in mannans, glucomannans and galactomannans. One unit of Endo-β-1,4-Mannanase will release 1.0 µmole of mannose reducing-sugar per minute from a 3mg/ml mannan solution at pH 5.5 and 37degC. Expressed in U/g.hCAI/II-IN-6
CAS :hCAI/II-IN-6 is a selective and orally active inhibitor of human carbonic anhydrase (CA).Formule :C19H24N4O3SDegré de pureté :98.49%Couleur et forme :SolidMasse moléculaire :388.48Nucleoside phosphorylase from microorganisms
CAS :Nucleoside phosphorylase (Purine nucleoside phosphorylase, PNP, PNPase, inosine phosphorylase, inosine-guanosine phosphorylase; EC 2.4.2.1) is an enzyme that catalyzes the following reaction: purine nucleoside + Pi ⇌ purine + alpha-D-ribose 1-phosphate One unit of nucleoside phosphorylase will phosphorylate 1.0 micromole of inosine to hypoxanthine and alpha-D-ribose 1-phosphate per min at pH 7.4 and 25°C.Formule :C5H6ClN3Degré de pureté :Min. 95%Masse moléculaire :143.57 g/mol
