Transporteur membranaire/Canal ionique
Les inhibiteurs des transporteurs membranaires et des canaux ioniques sont des composés qui bloquent la fonction des protéines responsables du transport des ions, des nutriments et d'autres molécules à travers les membranes cellulaires. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie cellulaire, la transduction des signaux et la neurotransmission. Les inhibiteurs des transporteurs membranaires et des canaux ioniques sont également importants pour développer des traitements contre des troubles tels que l'épilepsie, les maladies cardiovasculaires et les syndromes métaboliques. Chez CymitQuimica, nous offrons une sélection diversifiée d'inhibiteurs de haute qualité des transporteurs membranaires et des canaux ioniques pour soutenir vos recherches en physiologie, neurosciences et pharmacologie.
Sous-catégories appartenant à la catégorie "Transporteur membranaire/Canal ionique"
- ABC(3 produits)
- ATPase(101 produits)
- Récepteur de l'adiponectine(5 produits)
- CFTR(65 produits)
- Récepteur CGRP(54 produits)
- Canal calcique(543 produits)
- Canal chlorure(53 produits)
- Récepteur GABA(366 produits)
- Transporteur de monoamine(30 produits)
- Transporteur de monocarboxylate(18 produits)
- NKCC(2 produits)
- NPC1L1(3 produits)
- Cotransporteur Na-K-Cl(10 produits)
- OAT(32 produits)
- OCT(7 produits)
- P-gp(55 produits)
- Canal potassique(280 produits)
- Pompe à protons(42 produits)
- SGLT(31 produits)
- Canal sodique(210 produits)
- Canal TRP/TRPV(96 produits)
Affichez 13 plus de sous-catégories
2534 produits trouvés pour "Transporteur membranaire/Canal ionique"
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Epaminurad
CAS :Epaminurad (UR-1102) is an oral URAT1 inhibitor for gout research with a Ki of 0.057 μM, modestly affects OAT1/3.Formule :C14H10Br2N2O3Couleur et forme :SolidMasse moléculaire :414.05Pilsicainide HCl
CAS :Pilsicainide HCl (SUN 1165) is a pure sodium channel blockerFormule :C17H25ClN2ODegré de pureté :99.01% - 99.80%Couleur et forme :SolidMasse moléculaire :308.85NS 11021
CAS :NS 11021 (NS11021) , a novel opener of large-conductance Ca(2+)-activated K(+) channelsFormule :C16H9BrF6N6SDegré de pureté :97.26%Couleur et forme :SolidMasse moléculaire :511.24Ref: TM-T4294
1mg42,00€5mg88,00€10mg128,00€25mg263,00€50mg447,00€100mg760,00€200mg1.018,00€1mL*10mM (DMSO)89,00€HM-30181 mesylate monohydrate
CAS :HM-30181 mesylate monohydrate is an oral P-glycoprotein (P-gp) inhibitor, used to enhance the oral bioavailability of P-gp substrate drugs.Formule :C39H42N6O11SDegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :802.85Ref: TM-T9173
1mg69,00€2mg88,00€5mg126,00€10mg195,00€25mg325,00€50mg467,00€100mg680,00€200mg882,00€500mg1.320,00€1mL*10mM (DMSO)187,00€JNJ-26990990
CAS :"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."Formule :C9H10N2O2S2Degré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :242.32Ref: TM-T27673
1mg131,00€5mg286,00€10mg424,00€25mg702,00€50mg938,00€100mg1.311,00€1mL*10mM (DMSO)261,00€Revaprazan hydrochloride
CAS :Revaprazan hydrochloride (YH1885) is the hydrochloride salt form of a lipophilic, weak base with potassium-competitive acid blocking (P-CAB) activity.Formule :C22H24ClFN4Degré de pureté :99.62% - 99.91%Couleur et forme :SolidMasse moléculaire :398.9Ipidacrine
CAS :Ipidacrine (NIK‐247) (NIK‐247) is an Antidementia AgentFormule :C12H16N2Degré de pureté :97.73% - 99.99%Couleur et forme :SolidMasse moléculaire :188.27HC-067047
CAS :HC-067047 is a potent and selective TRPV4 antagonist.Also inhibits the endogenous TRPV4-mediated response to 4α-PDH .Formule :C26H28F3N3O2Degré de pureté :99.45% - 99.97%Couleur et forme :SolidMasse moléculaire :471.51Licarbazepine
CAS :<p>Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial</p>Formule :C15H14N2O2Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :254.28Esomeprazole
CAS :Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.Formule :C17H19N3O3SDegré de pureté :97.3%Couleur et forme :SolidMasse moléculaire :345.42UBP710
CAS :UBP710 is an effective and selective NMDA receptor modulator.Formule :C18H14O2Degré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :262.3Ref: TM-T24918
1mg87,00€2mg124,00€5mg187,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€200mg1.159,00€1mL*10mM (DMSO)177,00€Traxoprodil
CAS :Traxoprodil (CP101606) is a selective NMDA antagonist and protects hippocampal neurons (IC50: 10 nM).Formule :C20H25NO3Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :327.42Z944
CAS :Z944 is a T-type calcium channel blocker.Formule :C19H27ClFN3O2Degré de pureté :99.8% - 99.80%Couleur et forme :SolidMasse moléculaire :383.89Ref: TM-T29201
1mg52,00€5mg111,00€10mg180,00€25mg359,00€50mg530,00€100mg758,00€200mg1.035,00€1mL*10mM (DMSO)124,00€Talniflumate
CAS :<p>Talniflumate (Somalgen) is a calcium-activated chloride channel (hCLCA1/mCLCA3) blocker that reduces mucin synthesis and releases in animal models and cell</p>Formule :C21H13F3N2O4Degré de pureté :98% - 99.81%Couleur et forme :White To Pale Yellow Crystalline PowderMasse moléculaire :414.33SKF89976A hydrochloride
CAS :SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) andFormule :C22H26ClNO2Degré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :371.9Ref: TM-T12930
1mg35,00€5mg69,00€10mg95,00€25mg170,00€50mg279,00€100mg432,00€200mg622,00€1mL*10mM (DMSO)74,00€DNQX disodium salt
CAS :DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptorFormule :C8H2N4Na2O6Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :296.1Ref: TM-T8459
1mg62,00€5mg123,00€10mg180,00€25mg298,00€50mg419,00€100mg567,00€200mg752,00€1mL*10mM (DMSO)123,00€Enflurane
CAS :Enflurane (Efrane), a volatile anaesthetic, inhibits Ca2+-activated K+ channels and is used to gauge anesthesia levels in gas chromatography.Formule :C3H2ClF5ODegré de pureté :99.64%Couleur et forme :Clear Colorless Liquid Ordinary Temperature And Pressure Bp 56 8°C Density 1 50 G Cm-3 At Room Temperature Used As AnMasse moléculaire :184.49ZL006
CAS :ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.Formule :C14H11Cl2NO4Degré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :328.15Ref: TM-T17293
5mg50,00€10mg66,00€25mg117,00€50mg180,00€100mg306,00€200mg444,00€1mL*10mM (DMSO)52,00€Mirogabalin besylate
CAS :Mirogabalin besylate is an oral α2δ ligand for voltage-gated calcium channels, with Kd values of 13.5-47.6 nM across species.Formule :C18H25NO5SCouleur et forme :SolidMasse moléculaire :367.46Tezacaftor
CAS :Tezacaftor (VX661) is a small molecule that can be used as a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) gene function.Formule :C26H27F3N2O6Degré de pureté :98.84% - >99.99%Couleur et forme :SolidMasse moléculaire :520.5Ref: TM-T2263
1mg40,00€2mg52,00€5mg82,00€10mg123,00€25mg212,00€50mg343,00€100mg505,00€1mL*10mM (DMSO)88,00€Mitiglinide Calcium
CAS :Mitiglinide Calcium (KAD-1229) is a blood glucose-lowering drugs, stimulating insulin secretion by closing the ATP-sensitive K+ channels in pancreatic beta-Formule :(C19H24NO3)2·CaDegré de pureté :99.83%Couleur et forme :White Crystal PosderMasse moléculaire :668.88Tariquidar
CAS :Tariquidar (XR9576)(Kd=5.1 nM) is a specific and effective non-competitive inhibitor of P-glycoprotein. It can reverse drug resistance in MDR cell Lines.Formule :C38H38N4O6Degré de pureté :98.07% - 99.45%Couleur et forme :SolidMasse moléculaire :646.73Neramexane Free Base
CAS :Neramexane is a memantine-related, NMDA-blocking, neuroprotective drug, potentially treating tinnitus, Alzheimer's, addiction, and pain.Formule :C11H23NCouleur et forme :SolidMasse moléculaire :169.31Memantine
CAS :Memantine treats moderate to severe Alzheimer's; it's an amantadine derivative blocking NMDA receptors.Formule :C12H21NDegré de pureté :≥98%Couleur et forme :White PowderMasse moléculaire :179.3Trans-ACBD
CAS :Trans-ACBD (Trans-1-aminocyclobutane-1,3-dicarboxylic acid) is an effective and specific N-methyl-D-aspartate receptor agonist.Formule :C6H9NO4Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :159.14Pipequaline hydrochloride
CAS :Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.Formule :C22H25ClN2Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :352.9Fatostatin hydrobromide
CAS :<p>Fatostatin hydrobromide (Fatostatin A HBr), an inhibitor of sterol regulatory element binding protein (SREBP), impairs the activation of SREBP-1 and SREBP-2.</p>Formule :C18H18N2S·HBrDegré de pureté :98.62% - 99.91%Couleur et forme :SolidMasse moléculaire :375.33Disopyramide HCl
CAS :Disopyramide HCl, a Class 1a antiarrhythmic, treats ventricular tachycardia, blocks sodium channels, and has anticholinergic effects.Formule :C21H30ClN3OCouleur et forme :SolidMasse moléculaire :375.94Aminooxyacetic acid hemihydrochloride
CAS :Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFormule :C2H5NO3·5HClDegré de pureté :98.03%Couleur et forme :Light Beige Crystalline PowderMasse moléculaire :109.3SB 452533
CAS :SB 452533 is an antagonist of the vanilloid receptor 1(pKb: 7.8).Formule :C18H22BrN3ODegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :376.29Ref: TM-T23322
2mg39,00€5mg60,00€10mg92,00€25mg173,00€50mg269,00€100mg389,00€200mg555,00€1mL*10mM (DMSO)73,00€(S)-(-)-5-Fluorowillardiine hydrochloride
CAS :(S)-(-)-5-Fluorowillardiine hydrochloride is a potent and specific agonist of AMPAR.Formule :C7H9ClFN3O4Couleur et forme :SolidMasse moléculaire :253.62AMG 333
CAS :<p>AMG 333 is TRPM8 antagonist with an IC50 of 13 nM,a Clinical Candidate for the Treatment of Migraine.</p>Formule :C20H12F5N3O4Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :453.32XEN907
CAS :XEN907 is a novel spiro oxindole NaV1.7 blocker. XEN907 also inhibits hNaV1.7 (IC50: 3 nM).Formule :C21H21NO4Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :351.4Esomeprazole magnesium salt
CAS :Esomeprazole magnesium, an oral proton pump inhibitor, curbs gastric acid by blocking H+, K+-ATPase; used in treating GERD.Formule :C17H21MgN3O3SCouleur et forme :SolidMasse moléculaire :371.74GNE-131
CAS :GNE-131 is a potent and specific inhibitor of human sodium channel NaV1.7 (IC50: 3 nM).Formule :C23H30N4O3SDegré de pureté :98.54% - 99.59%Couleur et forme :SolidMasse moléculaire :442.57Ref: TM-TQ0014
1mg111,00€5mg264,00€10mg376,00€25mg630,00€50mg880,00€100mg1.169,00€1mL*10mM (DMSO)283,00€Lansoprazole sodium
CAS :Lansoprazole sodium is a PPI used to treat acid reflux and peptic ulcers.Formule :C16H13F3N3NaO2SDegré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :391.34Rapastinel Trifluoroacetate
CAS :Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties.Formule :C20H32F3N5O8Degré de pureté :99.01% - 99.77%Couleur et forme :SolidMasse moléculaire :527.49Ref: TM-T5819
1mg39,00€5mg97,00€10mg160,00€25mg296,00€50mg416,00€100mg557,00€200mg743,00€1mL*10mM (DMSO)116,00€PF 05089771
CAS :PF 05089771 is a Selective inhibitor of Nav1.7 (IC50 = 11 nM) that interacts with the voltage-sensor domain of domain IV.Formule :C18H12Cl2FN5O3S2Degré de pureté :99.03% - 99.42%Couleur et forme :SolidMasse moléculaire :500.35(-)-Securinine
CAS :(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.Formule :C13H15NO2Degré de pureté :99.58% - 99.87%Couleur et forme :SolidMasse moléculaire :217.26Cinacalcet metabolite M4
CAS :Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.Formule :C10H12F3NDegré de pureté :97.13%Couleur et forme :SolidMasse moléculaire :203.2Ref: TM-T10814
5mg55,00€10mg74,00€25mg96,00€50mg137,00€100mg170,00€200mg244,00€500mg364,00€1mL*10mM (DMSO)51,00€Tegoprazan
CAS :Tegoprazan is an orally active, highly selective gastric H+/K+-ATPase inhibitor.Cost-effective and quality-assured.Formule :C20H19F2N3O3Degré de pureté :98.22%Couleur et forme :SolidMasse moléculaire :387.38Ref: TM-T17030
1mg52,00€5mg120,00€10mg180,00€25mg298,00€50mg393,00€100mg512,00€200mg727,00€1mL*10mM (DMSO)133,00€Alinidine hydrobromide
CAS :Alinidine hydrobromide, a specific bradycardic agent, diminishes the slope of the diastolic depolarization in sinoatrial tissue and Purkinje fibers [1].Formule :C12H14BrCl2N3Couleur et forme :SolidMasse moléculaire :351.07L-Allylglycine
CAS :L-Allylglycine is a potent inhibitor of the synthetic enzyme for GABA, glutamic acid decarboxylase.Formule :C5H9NO2Degré de pureté :≥98%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :115.13Acecainide hydrochloride
CAS :Acecainide hydrochloride (NAPA) is the major hepatic metabolite of procainamide.Cost-effective and quality-assured.Formule :C15H24ClN3O2Degré de pureté :98.023% - 99.81%Couleur et forme :SolidMasse moléculaire :313.835,7-Dichlorokynurenic acid
CAS :5,7-Dichlorokynurenic acid (5,7-dichlorokynurenic acid sodium) is an NMDA receptor antagonist.Formule :C10H5Cl2NO3Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :258.06TC-I2000
CAS :TC-I2000 is an TRPM8 channel blocker. Inhibits icilin-induced TRPM8 channel activation in rTRPM8-expressing CHO cells with IC50 of 53 nM.Formule :C23H18F4N2ODegré de pureté :99.778%Couleur et forme :SolidMasse moléculaire :414.4Ref: TM-T8449
5mg35,00€10mg50,00€25mg88,00€50mg119,00€100mg173,00€200mg259,00€1mL*10mM (DMSO)À demanderBI 01383298
CAS :BI 01383298 is a selective inhibitor of the sodium-citrate co-transporter (SLC13A5).Formule :C19H19Cl2FN2O3SDegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :445.34Levamlodipine hydrobromide
CAS :Levamlodipine hydrobromide is a medication used to lower blood pressure and prevent chest pain.Formule :C20H26BrClN2O5Couleur et forme :SolidMasse moléculaire :489.79CX614
CAS :CX614 is a positive allosteric modulator of the AMPA receptor concerning AMPA.Formule :C13H13NO4Degré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :247.25Ref: TM-T19698
5mg52,00€10mg78,00€25mg119,00€50mg172,00€100mg259,00€200mg388,00€1mL*10mM (DMSO)55,00€ML277
CAS :ML277 (CID-53347902) was identified as a potent activator of KCNQ1 channels (EC(50)=260 nM).Formule :C23H25N3O4S2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :471.59Radiprodil
CAS :Radiprodil (RGH-896) is an oral NMDA NR2B antagonist for potential DPNP neuropathic pain treatment.Formule :C21H20FN3O4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :397.4Ref: TM-T5385
1mg48,00€2mg65,00€5mg96,00€10mg153,00€25mg240,00€50mg354,00€100mg532,00€1mL*10mM (DMSO)96,00€p-Hydroxybenzaldehyde
CAS :1.Formule :C7H6O2Degré de pureté :99.05% - 99.86%Couleur et forme :SolidMasse moléculaire :122.12PF-01247324
CAS :PF-01247324 is a selective and orally bioavailable Nav1.8 channel blocker (IC50: 196 nM).Formule :C13H10Cl3N3ODegré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :330.6Thiocolchicoside
CAS :<p>Thiocolchicoside, a muscle relaxant, has anti-inflammatory and analgesic properties; not for seizure-prone people.</p>Formule :C27H33NO10SDegré de pureté :99.11% - 99.39%Couleur et forme :SolidMasse moléculaire :563.62IDRA-21
CAS :IDRA-21 is a positive AMPA receptor modulator.Formule :C8H9ClN2O2SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :232.69Tenapanor
CAS :Tenapanor (RDX 5791), an NHE3 inhibitor, regulates sodium in the gut and kidney with a strong preclinical safety record and minimal side effects.Formule :C50H66Cl4N8O10S2Degré de pureté :99.49% - 99.85%Couleur et forme :SolidMasse moléculaire :1145.051-Aminocyclobutanecarboxylic acid
CAS :1-Aminocyclobutanecarboxylic acid (ACBC) is a NMDA receptor partial agonist. 1-Aminocyclobutanecarboxylic acid act at the glycine site, NR1[1].Formule :C5H9NO2Degré de pureté :99.94%Couleur et forme :White To Tan Powder Crystals Crystalline Powder And/Or With ChunksMasse moléculaire :115.13KCNQ2/3 activator-1
CAS :KCNQ2/3 activator-1 is a Kv7.2/Kv7.3 (KCNQ2/3) potassium channel activator.Formule :C23H29FN2ODegré de pureté :99.16% - 99.47%Couleur et forme :SolidMasse moléculaire :368.49Ref: TM-T9400
2mg40,00€5mg62,00€10mg94,00€25mg153,00€50mg235,00€100mg373,00€500mg938,00€1mL*10mM (DMSO)67,00€(2S)-6-Prenylnaringenin
CAS :(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Formule :C20H20O5Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :340.37Phenibut (hydrochloride)
CAS :Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Formule :C10H14ClNO2Degré de pureté :99.93%Couleur et forme :White Crystalline PowderMasse moléculaire :215.68VX-150
CAS :VX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).Formule :C21H17F4N2O7PDegré de pureté :97.58%Couleur et forme :SolidMasse moléculaire :516.34Ref: TM-T9683
1mg66,00€5mg144,00€10mg235,00€25mg472,00€50mg755,00€100mg1.206,00€1mL*10mM (DMSO)164,00€Nicainoprol
CAS :Nicainoprol (RU-42924) is a fast-sodium-channel blocking drug. Nicainoprol is a potent antiarrhythmic agent.Formule :C21H27N3O3Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :369.46Ref: TM-T4539
1mg140,00€5mg344,00€10mg512,00€25mg812,00€50mg1.093,00€100mg1.473,00€1mL*10mM (DMSO)350,00€Disopyramide phosphate
CAS :Disopyramide: Class 1a anti-arrhythmic, treats Ventricular Tachycardia, reduces heart muscle contractility.Formule :C21H32N3O5PCouleur et forme :SolidMasse moléculaire :437.47Tetrabenazine methanesulfonate
CAS :Tetrabenazine methanesulfonate: ex-antipsychotic/therapy for movement disorders, blocks neurotransmitter uptake, labels vesicle transport.Formule :C20H31NO6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.53(S)-(-)-5-Fluorowillardiine
CAS :(S)-(-)-5-Fluorowillardiine ((S)-5-Fluorowillardiine) is an AMPA receptor-specific agonistFormule :C7H8FN3O4Degré de pureté :99.69%Couleur et forme :Off-White SolidMasse moléculaire :217.15β-Pompilidotoxin Acetate
β-Pompilidotoxin Acetate is a wasp venom peptide.Formule :C73H128N22O19Degré de pureté :98.64%Couleur et forme :SolidMasse moléculaire :1617.93Ref: TM-T21769L
2mg47,00€5mg66,00€10mg89,00€25mg154,00€50mg221,00€100mg314,00€200mg442,00€1mL*10mM (DMSO)136,00€Flupirtine
CAS :Flupirtine(D 9998) is a selective neuronal potassium channel opener as well as shows properties of NMDA receptor antagonist.Formule :C15H17FN4O2Couleur et forme :SolidMasse moléculaire :304.32Benzamil
CAS :Benzamil blocks ENaC, inhibiting sodium transport (IC50=4 nM) and binds with Kd=5 nM to bovine kidney membranes.Formule :C13H14ClN7ODegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :319.75Pilsicainide
CAS :Pilsicainide (SUN 1165 free acid) is a potent class Ic antiarrhythmic agent. Pilsicainide is a potent sodium channel blocker[1][2].Formule :C17H24N2OCouleur et forme :SolidMasse moléculaire :272.39BRITE-338733
CAS :BRITE-338733 is a novel inhibitor of ATPase. BRITE 338733 inhibits the expression of RecA in bacteria (IC50=4.7 μM) for the bacterial infections treatment.Formule :C27H35N3O2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :433.59Ref: TM-T22280
1mg46,00€2mg63,00€5mg97,00€10mg169,00€25mg329,00€50mg465,00€100mg655,00€200mg883,00€1mL*10mM (DMSO)105,00€α-Thujone
CAS :α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Formule :C10H16ODegré de pureté :97.02% - 98.41%Couleur et forme :Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Masse moléculaire :152.234-Acetamidobutanoic acid
CAS :4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.Formule :C6H11NO3Degré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :145.16rac-BHFF
CAS :rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.Formule :C17H21F3O3Degré de pureté :99.69% - >99.99%Couleur et forme :SolidMasse moléculaire :330.34Ref: TM-T4176
2mg43,00€5mg60,00€10mg96,00€25mg187,00€50mg311,00€100mg472,00€200mg657,00€1mL*10mM (DMSO)71,00€Benzocaine xHCl(94-09-7(free base))
Benzocaine shares a common receptor with all othe rLAs in the voltage-gated Na+ channel(IC50 of 0.8 mM tested with a potential of +30 mV).Formule :C9H11NO2·xHClDegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :N/APAP-1
CAS :PAP-1 (5-(4-Phenoxybutoxy)psoralen) is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).Formule :C21H18O5Degré de pureté :99.35% - 99.75%Couleur et forme :White SolidMasse moléculaire :350.36Ref: TM-TQ0179
2mg63,00€5mg88,00€10mg136,00€25mg291,00€50mg520,00€100mg550,00€200mg785,00€1mL*10mM (DMSO)90,00€Indecainide hydrochloride
CAS :Indecainide hydrochloride is a cardiac depressant.Formule :C20H25ClN2OCouleur et forme :SolidMasse moléculaire :344.88Elobixibat hydrate
CAS :Elobixibat hydrate, an IBAT inhibitor, IC50: 0.53 nM (human), 0.13 nM (mouse), 5.8 nM (canine); for CIC research.Formule :C36H47N3O8S2Couleur et forme :SolidMasse moléculaire :713.9RQ-00203078
CAS :RQ-00203078 is a highly selective, potent and orally available TRPM8 antagonist.Formule :C21H13ClF6N2O5SDegré de pureté :98% - 99.6%Couleur et forme :SolidMasse moléculaire :554.85A-967079
CAS :<p>A 967079 is a potent, selective, and bioavailable inhibitor of the TRPA1 channel, with IC50 values of 67 and 289 nM for the human and rat isoforms, respectively</p>Formule :C12H14FNODegré de pureté :98.34% - 99.75%Couleur et forme :SolidMasse moléculaire :207.24Cholesterol myristate
CAS :<p>Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.</p>Formule :C41H72O2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :597.01Zosuquidar
CAS :Zosuquidar (RS 33295-198) is a potent P-glycoprotein inhibitor with antitumor activity that inhibits tumor growth.Formule :C32H31F2N3O2Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :527.6Ref: TM-T6018L
1mg78,00€5mg160,00€10mg233,00€25mg378,00€50mg567,00€100mg825,00€200mg1.130,00€1mL*10mM (DMSO)180,00€Sodium ionophore III
CAS :Sodium ionophore III (ETH2120) is a Na+ ionophore suitable for the test of sodium activity in plasma, serum, and blood.Formule :C34H52N2O4Degré de pureté :99.51% - 99.78%Couleur et forme :SolidMasse moléculaire :552.79AZD-9056 free base
CAS :AZD9056 is a potent, selective, orally bioavailable P2X7 receptor antagonist.Formule :C24H35ClN2O2Couleur et forme :SolidMasse moléculaire :419DQP 1105
CAS :<p>DQP 1105 is a NMDA receptor antagonist.</p>Formule :C29H24BrN3O4Degré de pureté :98.6%Couleur et forme :SolidMasse moléculaire :558.42Tiludronate
CAS :Tiludronate, an oral bisphosphonate, treats metabolic bone disorders and inhibits osteoclasts.Formule :C7H9ClO6P2SCouleur et forme :SolidMasse moléculaire :318.61Drotaverine hydrochloride
CAS :Drotaverine hydrochloride is a type 4 cyclic nucleotide phosphodiesterase (PDE4) inhibitor，and is an antispasmodic drug, used to enhance cervical dilationFormule :C24H32ClNO4Degré de pureté :99.81%Couleur et forme :Pale-Yellow Crystalline SolidMasse moléculaire :433.968Piperazine
CAS :Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.Formule :C4H10N2Couleur et forme :SolidMasse moléculaire :86.14Felbamate
CAS :Felbamate (W-554) is an Anti-epileptic Agent.Formule :C11H14N2O4Degré de pureté :99% - >99.99%Couleur et forme :White Powder SolidMasse moléculaire :238.24TCN 201
CAS :TCN 201 is a selective antagonist of NMDA receptors containing the NR2A subunit.Formule :C21H17ClFN3O4SDegré de pureté :98.5%Couleur et forme :SolidMasse moléculaire :461.89Songorine
CAS :Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.Formule :C22H31NO3Degré de pureté :98% - 99.92%Couleur et forme :SolidMasse moléculaire :357.49MDK-4025
CAS :MDK-4025 is an inhibitor of the high voltage-activated (HVA) Ca2+ current in pyramidal neurons.Formule :C19H15ClODegré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :294.77Pyr10
CAS :Pyr10, a pyrazole derivative, selectively inhibits TRPC3, not STIM1/Orai1, with IC50 of 0.72 μM in TRPC3-HEK293, and 13.08 μM in BRL-2H3 cells.Formule :C18H13F6N3O2SDegré de pureté :99.69% - 99.7%Couleur et forme :SolidMasse moléculaire :449.37Methyl homoveratrate
CAS :Methyl homoveratrate, a McN5691 (RWJ-26240) metabolite detected in vivo in plasma, urine, and fecal extracts, functions as a voltage-sensitive calcium channelFormule :C11H14O4Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :210.23Fipronil
CAS :Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.Formule :C12H4Cl2F6N4OSDegré de pureté :97.21%Couleur et forme :Solid PowderMasse moléculaire :437.15Tricaine methanesulfonate
CAS :Tricaine methanesulfonate (TMS/MS-222) is an anesthetic used in hatcheries and studies to immobilize fish for marking, transport, and invasive procedures.Formule :C10H15NO5SDegré de pureté :99.259% - 99.86%Couleur et forme :White PowderMasse moléculaire :261.30Amifampridine phosphate
CAS :Amifampridine treats rare muscle diseases like LEMS and congenital myasthenias, targeting specific enzyme defects.Formule :C5H10N3O4PCouleur et forme :SolidMasse moléculaire :207.12GMQ hydrochloride
CAS :<p>GMQ hydrochloride, a potent ASIC modulator, activates ASIC3 at neutral pH and inhibits acid-induced peak current.</p>Formule :C10H12ClN5Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :237.69Iptakalim Hydrochloride
CAS :Iptakalim, a lipophilic para-amino compound, is a novel ATP-sensitive potassium channel (KATP) opener, as well as an α4β2-containing nicotinic acetylcholineFormule :C9H22ClNDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :179.731GSK369796 Dihydrochloride
CAS :GSK369796 Dihydrochloride (N-tert-butylisoquine),is an anti-malaria drug candidate.Formule :C20H24Cl3N3ODegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :428.78Ref: TM-T7195
1mg79,00€2mg101,00€5mg149,00€10mg195,00€25mg373,00€50mg562,00€100mg802,00€1mL*10mM (DMSO)145,00€9-Phenanthrol
CAS :<p>9-Phenanthrol is inhibitor of the transient receptor potential melastatin 4 (TRPM) channel, a Ca2+ -activated non-selective cation channel.</p>Formule :C14H10ODegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :194.23
