Transporteur membranaire/Canal ionique
Les inhibiteurs des transporteurs membranaires et des canaux ioniques sont des composés qui bloquent la fonction des protéines responsables du transport des ions, des nutriments et d'autres molécules à travers les membranes cellulaires. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie cellulaire, la transduction des signaux et la neurotransmission. Les inhibiteurs des transporteurs membranaires et des canaux ioniques sont également importants pour développer des traitements contre des troubles tels que l'épilepsie, les maladies cardiovasculaires et les syndromes métaboliques. Chez CymitQuimica, nous offrons une sélection diversifiée d'inhibiteurs de haute qualité des transporteurs membranaires et des canaux ioniques pour soutenir vos recherches en physiologie, neurosciences et pharmacologie.
Sous-catégories appartenant à la catégorie "Transporteur membranaire/Canal ionique"
- ABC(3 produits)
- ATPase(100 produits)
- Récepteur de l'adiponectine(5 produits)
- CFTR(66 produits)
- Récepteur CGRP(54 produits)
- Canal calcique(544 produits)
- Canal chlorure(53 produits)
- Récepteur GABA(369 produits)
- Transporteur de monoamine(30 produits)
- Transporteur de monocarboxylate(18 produits)
- NKCC(2 produits)
- NPC1L1(3 produits)
- Cotransporteur Na-K-Cl(10 produits)
- OAT(32 produits)
- OCT(7 produits)
- P-gp(55 produits)
- Canal potassique(283 produits)
- Pompe à protons(41 produits)
- SGLT(31 produits)
- Canal sodique(217 produits)
- Canal TRP/TRPV(96 produits)
Affichez 13 plus de sous-catégories
2575 produits trouvés pour "Transporteur membranaire/Canal ionique"
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(R)-BPO-27
CAS :(R)-BPO-27 is an orally active and potent ATP-competitive CFTR inhibitor (IC50: 4 nM) for the study of diarrhoea and polycystic kidney.Formule :C26H18BrN3O6Degré de pureté :99.1%Couleur et forme :SolidMasse moléculaire :548.34L-Palmitoylcarnitine
CAS :L-Palmitoylcarnitine (L-PC) inhibits Na/K ATPase activity and potentiates fibrinolytic enzymes and tPA to inhibit thrombosis.Formule :C23H45NO4Degré de pureté :97% - 99.81%Couleur et forme :SolidMasse moléculaire :399.61Clamikalant sodium
CAS :Clamikalant sodium (HMR 1098) is an ATP-dependent potassium channel (KATP) cardiac-selective blocker, used in the study of arrhythmias.Formule :C19H21ClN3NaO5S2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :493.96Ref: TM-T63330
1mg48,00€5mg90,00€10mg172,00€25mg346,00€50mg546,00€100mg855,00€200mg1.170,00€1mL*10mM (DMSO)99,00€β-Cyfluthrin
CAS :β-Cyfluthrin is a type II synthetic pyrethroid compound commonly utilized as an active ingredient in agricultural insecticide products.Formule :C22H18Cl2FNO3Couleur et forme :SolidMasse moléculaire :434.29MRS1845
CAS :MRS1845 is a selective inhibitor of store-operated calcium (SOC) channel (IC50 of 1.7 μM).Formule :C21H22N2O6Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :398.41Tetrabenazine-d6
CAS :Tetrabenazine D6 is the deuterium-labeled Tetrabenazine. Tetrabenazine is a VMAT-inhibitor used for the treatment of hyperkinetic movement disorder.Formule :C19H27NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :323.46PF-04856264
CAS :PF-04856264 is a Nav1.7 blocker.,modulates intracellular Ca 2+ signaling and chondrocyte secretome, raises the threshold of mechanical pain analgesic.Formule :C20H15N5O3S2Degré de pureté :97.43%Couleur et forme :SolidMasse moléculaire :437.5Ref: TM-T33943
1mg50,00€5mg105,00€10mg170,00€25mg340,00€50mg532,00€100mg893,00€1mL*10mM (DMSO)117,00€QO-58
CAS :QO-58 is a novel Kv7 activator (opener) that activates neuronal Kv7/KCNQ/M channels, danti-nociceptive effects on inflammatory painFormule :C18H8Cl2F4N4ODegré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :443.18Flumazenil acid
CAS :Flumazenil is an antagonist of GABAA receptor. Flumazenil acid is a metabolite of Flumazenil.Formule :C13H10FN3O3Couleur et forme :SolidMasse moléculaire :275.24TGN-073
CAS :TGN-073 is an enhancer of aquaporin 4 (AQP4), a water channel in astrocytes. It shows an increase in lymphatic transport in the rat brain by up to 41%.Formule :C18H16N2O3SCouleur et forme :SolidMasse moléculaire :340.396Vigabatrin Hydrochloride
CAS :Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the GABA, irreversibly inhibiting the catabolism of GABA by GABA transaminase.Formule :C6H11NO2·HClDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :165.62Poneratoxin acetate
<p>Poneratoxin acetate is a neurotoxic peptide and modulator of NaV1.6/NaV1.7, lowering the activation threshold of voltage-gated sodium channels and causing pain.</p>Formule :C129H215N33O31S·xC2H4O2Couleur et forme :SolidMasse moléculaire :2756.35 (free base)VU041
CAS :VU041 inhibits mosquito Kir1 channels (IC50: An. gambiae 2.5μM, Ae. aegypti 1.7μM), less on mammalian Kir2.1 (12.7μM), and minimally on other Kir channels.Formule :C19H20F3N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :363.38(R)-Tegoprazan
CAS :(R)-Tegoprazan, a benzimidazole derivative, inhibits kidney H+/K+-ATPase (IC50: 98 nM). Potential in GI disease research.Formule :C20H19F2N3O3Couleur et forme :SolidMasse moléculaire :387.38(R)-Lercanidipine-d3 hydrochloride
CAS :(R)-lercanidipine D3 hydrochloride is a deuterium labeled (R)-Lercanidipine hydrochloride. (R)-Lercanidipine D3 (hydrochloride) is a calcium channel blocker.Formule :C36H42ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :651.21Tetramethrin
CAS :Tetramethrin is a type I pyrethroid insecticide that affects the inactivation process of sodium channels in insect neurons, prolonged sodium currents.Formule :C19H25NO4Degré de pureté :98.85%Couleur et forme :White Crystals Or PowderMasse moléculaire :331.41Dibucaine hydrochloride
CAS :Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.Formule :C20H30ClN3O2Degré de pureté :99.66%Couleur et forme :White PowderMasse moléculaire :379.92Jedi2
CAS :<p>Jedi2 is a Piezo1 activator rather than a specific Piezo2 activator. Jedi2 binds to the mouse Piezo1 proteins with a K d of 2770 μM [1].</p>Formule :C10H8O3SDegré de pureté :97.85%Couleur et forme :SolidMasse moléculaire :208.23Triamterene D5
CAS :Triamterene D5 is a deuterium-labeled Triamterene and can block epithelial Na+ channel (ENaC) in a voltage-dependent manner, used as a mild diuretic.Formule :C12H11N7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :258.29Pantoprazole sulfone
CAS :Pantoprazole sulfone, a metabolite from pantoprazole breakdown by CYP2C19 and CYP3A4, inhibits gastric H+/K+ ATPase.Formule :C16H15F2N3O5SCouleur et forme :SolidMasse moléculaire :399.37UBP608
CAS :UBP608 selectively inhibits NMDA GluN1/GluN2A receptors, 23x more than GluN1/GluN2D.Formule :C10H5BrO4Couleur et forme :SolidMasse moléculaire :269.05L-364,373
CAS :KV7.1 (KCNQ1) channel activatorFormule :C25H20FN3OCouleur et forme :SolidMasse moléculaire :397.44Lubiprostone hemiketal
CAS :Lubiprostone (hemiketal) (RU-0211 (hemiketal)), a selective activator of the chloride channel 2 (CLCN2), facilitates the treatment of chronic idiopathic constipation and opioid-induced constipation. It functions by enhancing CLCN2 channel activity, which boosts chloride ion secretion in the intestines, subsequently increasing fluid secretion and improving intestinal peristalsis. Additionally, Lubiprostone (hemiketal) may be utilized in research related to chronic constipation and cancer.Formule :C20H32F2O5Couleur et forme :SolidMasse moléculaire :390.46HSK16149
CAS :HSK16149 is a novel ligand of voltage-gated calcium channel (VGCC) α 2 δ subunit with analgesic activity.Formule :C12H19NO2Couleur et forme :SolidMasse moléculaire :209.28SDZ 220-581 Ammonium salt
CAS :SDZ 220-581 Ammonium salt is a potent, orally active and competitive antagonist of NMDA receptor(pKi : 7.7).Formule :C16H20ClN2O5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.77N,N-Dimethylglycine hydrochloride
CAS :N,N-Dimethylglycine hydrochloride (N-Methylsarcosine hydrochloride) is a dietary supplement.Formule :C4H10ClNO2Degré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :139.58Lansoprazole-d4
CAS :Lansoprazole D4 (AG-1749 D4) is a deuterium labeled Lansoprazole. Lansoprazole is an inhibitor of proton pump which prevents the stomach from producing acid.Formule :C16H14F3N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :373.39Crinecerfont hydrochloride
CAS :SSR-125543, a potent CRF1 receptor non-peptide antagonist, effective in CAH research, taken orally.Formule :C27H29Cl2FN2OSCouleur et forme :SolidMasse moléculaire :519.5Fanapanel
CAS :Fanapanel (ZK200775) is a quinoxalinedione derivative and potent competitive antagonist of AMPAR for cerebrovascular-related studies.Formule :C14H15F3N3O6PCouleur et forme :SolidMasse moléculaire :409.25Pirmenol hydrochloride
CAS :Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μMFormule :C22H31ClN2OCouleur et forme :SolidMasse moléculaire :374.95Cabotegravir sodium
CAS :Cabotegravir sodium inhibits HIV integrase (IC50: 2.5 nM), metabolized by UGT1A1, with minimal ARV interaction.Formule :C19H16F2N3NaO5Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :427.34YM-244769
CAS :YM-244769 (3-Pyridinecarboxamide, N-[(3-aminophenyl)methyl]-6-[4-[(3-fluorophenyl)methoxy]phenoxy]-) is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3)Formule :C26H22FN3O3Degré de pureté :95.62%Couleur et forme :SolidMasse moléculaire :443.47(-)-α-Pinene
CAS :(-)-α-Pinene ((1S)-(-)-Alpha-Pinene) enhances the quantity of NREMS without affecting the intensity of NREMS by prolonging GABAergic synaptic transmission,Formule :C10H16Degré de pureté :98.02% - 98.60%Couleur et forme :Colourless LiquidMasse moléculaire :136.23GI-530159
CAS :TREK1/2 activator, selective over TRAAK/TASK3; hyperpolarizes neurons, depresses activity (EC50 = 0.76 μM).Formule :C27H20F6N2O2Couleur et forme :White CrystalsMasse moléculaire :518.4510,11-Dihydro-10-hydroxycarbamazepine-d4
CAS :10,11-Dihydro-10-hydroxycarbamazepine-d4 is a deuterated compound of 10,11-Dihydro-10-hydroxycarbamazepine.Formule :C15H10D4N2O2Masse moléculaire :258.31Torsemide (Standard)
CAS :Torsemide (Standard) is the standard substance of Torsemide, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Torsemide (AC-4464) is an anilinopyridine sulfonylurea belonging to the class of loop diuretics. Torsemide has a prolonged duration of action compared to other loop diuretics, is extensively protein bound in plasma and has a relatively long half-life.Formule :C16H20N4O3SMasse moléculaire :348.42Rosuvastatin Sodium
CAS :Rosuvastatin Sodium (ZD4522 Sodium) is a competitive HMG-CoA reductase (HMGCR) inhibitor (IC50=11 nM) with lipid-lowering and anti-atherosclerotic effects.Formule :C22H27FN3NaO6SCouleur et forme :SolidMasse moléculaire :503.521-N-Methyl-4-mercaptohistidine disulfide
CAS :1-N-Methyl-4-mercaptohistidine disulfide is a Duchenne chloroplast coupling factor 1 redox modulator that inhibits light-triggered CF1 ATPase activity.Formule :C14H20N6O4S2Degré de pureté :97.67% - ≥98%Couleur et forme :SoildMasse moléculaire :400.48Muzolimine
CAS :Muzolimine: a long-acting, high-capacity diuretic for kidney failure/hypertension; withdrawn due to serious neurological side effects.Formule :C11H11Cl2N3OCouleur et forme :SolidMasse moléculaire :272.13Benzocaine hydrochloride
CAS :Benzocaine hydrochloride (Ethyl 4-aminobenzoate hydrochloride) is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers andFormule :C9H11NO2·HClDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :201.65Afoxolaner (Standard)
CAS :Afoxolaner (Standard) is the standard substance of Afoxolaner, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs. Afoxolaner acts on the insect GABA and glutamate receptors, inhibiting GABA & glutamate-regulated uptake of chloride ions, resulting in excess neuronal stimulation and death of the arthropod.Formule :C26H17ClF9N3O3Masse moléculaire :625.87Norverapamil-d7 HCl
CAS :Norverapamil-d7 HCl (D591-d7 HCl) is a 2H-labeled Norverapamil HCl, a calcium channel blocker and P-gp inhibitor, also a coronary vasodilator.Formule :C26H37ClN2O4Couleur et forme :SolidMasse moléculaire :484.08SKA-121
CAS :SKA-121 is a selective KCa3.1 activator (EC50s: 109 nM and 4.4 μM for KCa3.1 and KCa2.3, respectively).Formule :C12H10N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :198.22Esomeprazole sodium-d6
CAS :Esomeprazole sodium-d6 is a deuterated compound of Esomeprazole sodium.Formule :C17H12D6N3NaO3SMasse moléculaire :373.44Naspm
CAS :Naspm is a synthetic analogue of Joro spider toxin and is a antagonist iscalcium permeable AMPA (CP-AMPA) receptors.Formule :C22H34N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :370.53Pantoprazole Sulfide
CAS :Pantoprazole sulfide, a metabolite of pantoprazole, is formed by CYP2C19 and CYP3A4 enzymes.Formule :C16H15F2N3O3SCouleur et forme :SolidMasse moléculaire :367.37Primidone (Standard)
CAS :Primidone (Standard) is the standard substance of Primidone, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Primidone (NCI-C56360) is a potent anticonvulsant agent. It is a neuronal voltage-gated sodium channel blocker and has value in the study of epilepsy, essential tremor, and psychiatric disorders.Formule :C12H14N2O2Couleur et forme :Crystals (Ntp 1992)Masse moléculaire :218.25YM-244769 dihydrochloride
CAS :YM-244769 dihydrochloride is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3) with an IC50 of 18 nM.Formule :C26H24Cl2FN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :516.39Luciferase, firefly
CAS :Luciferase, firefly is a reporter gene in cellular imaging studies to quantify target gene expression levels and measure intracellular ATP content,Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :N/AUnifiram
CAS :Unifiram boosts cognition, enhances rat hippocampal signals (EC50=27 nM), and ups ACh in rat cortex.Formule :C13H15FN2O3SDegré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :298.33Kavain
CAS :Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation ofFormule :C14H14O3Degré de pureté :99.93% - ≥95%Couleur et forme :SolidMasse moléculaire :230.26Lomerizine
CAS :<p>Lomerizine, a blocker of diphenylmethylpiperazine Ca2+ channel, is used to prevent migraines.</p>Formule :C27H30F2N2O3Couleur et forme :SolidMasse moléculaire :468.54DL-AP5
CAS :DL-AP5 is the racemic form of a selective N-methyl-D-aspartate (NMDA) receptor antagonist with anticonvulsant effects.Formule :C5H12NO5PDegré de pureté :99.33%Couleur et forme :White Fine Crystalline PowderMasse moléculaire :197.13Levamlodipine hydrobromide
CAS :Levamlodipine hydrobromide is a medication used to lower blood pressure and prevent chest pain.Formule :C20H26BrClN2O5Couleur et forme :SolidMasse moléculaire :489.791-Aminocyclobutanecarboxylic acid
CAS :1-Aminocyclobutanecarboxylic acid (ACBC) is a NMDA receptor partial agonist. 1-Aminocyclobutanecarboxylic acid act at the glycine site, NR1[1].Formule :C5H9NO2Degré de pureté :99.94%Couleur et forme :White To Tan Powder Crystals Crystalline Powder And/Or With ChunksMasse moléculaire :115.13BPU-11
CAS :BPU-11 (Biphenyl Urea 11) is an HCN4 CLP ligand that acts by modulating channel function and completely abolishing the cAMP-induced shift in V1/2.Formule :C32H31N5ODegré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :501.62YHO-13177
CAS :YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells.Formule :C20H22N2O3SDegré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :370.47MDK-4025
CAS :MDK-4025 is an inhibitor of the high voltage-activated (HVA) Ca2+ current in pyramidal neurons.Formule :C19H15ClODegré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :294.77Radiprodil
CAS :Radiprodil (RGH-896) is an oral NMDA NR2B antagonist for potential DPNP neuropathic pain treatment.Formule :C21H20FN3O4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :397.4Ref: TM-T5385
1mg48,00€2mg65,00€5mg96,00€10mg153,00€25mg240,00€50mg354,00€100mg532,00€1mL*10mM (DMSO)96,00€HC-030031
CAS :HC-030031 (TOSLAB 829227) is a potent TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2 and 5.3 μM, respectively.Formule :C18H21N5O3Degré de pureté :99.69% - ≥95%Couleur et forme :SolidMasse moléculaire :355.39Evifacotrep
CAS :Evifacotrep: TRPC5 antagonist for neurological disease research (WO2020061162, compound 100).Formule :C18H12ClF4N5O2Degré de pureté :98.6%Couleur et forme :SolidMasse moléculaire :441.77Ref: TM-T40042
1mg92,00€5mg178,00€10mg286,00€25mg440,00€50mg655,00€100mg973,00€200mg1.468,00€1mL*10mM (DMSO)152,00€Ginkgolide A
CAS :Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.Formule :C20H24O9Degré de pureté :98.76% - 99.81%Couleur et forme :White PowderMasse moléculaire :408.40CCTA-1523
CAS :CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.Formule :C16H15Cl2NO3Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :340.2Ref: TM-T9587
1mg87,00€5mg192,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€200mg1.130,00€1mL*10mM (DMSO)192,00€DL-Menthol
CAS :DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.Formule :C10H20ODegré de pureté :99.74%Couleur et forme :White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Masse moléculaire :156.27VU0134992
CAS :VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μMFormule :C20H31BrN2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :411.38Ref: TM-T8372
1mg71,00€5mg131,00€10mg190,00€25mg323,00€50mg459,00€100mg632,00€200mg852,00€1mL*10mM (DMSO)156,00€Phenibut (hydrochloride)
CAS :Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Formule :C10H14ClNO2Degré de pureté :99.93%Couleur et forme :White Crystalline PowderMasse moléculaire :215.68(S)-ATPO
CAS :<p>(S)-ATPO is Competitive antagonist at GluR1-4 (AMPA-preferring) receptors.</p>Formule :C11H19N2O7PDegré de pureté :98.37% - 99.41%Couleur et forme :SolidMasse moléculaire :322.25Omecamtiv mecarbil
CAS :<p>Omecamtiv mecarbil (CK-1827452) has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic</p>Formule :C20H24FN5O3Degré de pureté :98% - 99.23%Couleur et forme :SolidMasse moléculaire :401.43Procyclidine hydrochloride
CAS :Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.Formule :C19H30ClNODegré de pureté :99.24% - 99.88%Couleur et forme :Crystals From Petroleum Ether White PowderMasse moléculaire :323.9Pikamilone
CAS :Pikamilone (Picamilon) is an intelligent medicine.Formule :C10H12N2O3Degré de pureté :99.38%Couleur et forme :White Crystalline PowderMasse moléculaire :208.21γ-Acetylenic GABA
CAS :γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.Formule :C6H9NO2Couleur et forme :SolidMasse moléculaire :127.143Esomeprazole potassium salt
CAS :Esomeprazole potassium, a potent oral proton pump inhibitor, curbs acid secretion in stomach cells, aiding GERD research.Formule :C17H18KN3O3SCouleur et forme :SolidMasse moléculaire :383.51(S)-(-)-5-Fluorowillardiine
CAS :(S)-(-)-5-Fluorowillardiine ((S)-5-Fluorowillardiine) is an AMPA receptor-specific agonistFormule :C7H8FN3O4Degré de pureté :99.69%Couleur et forme :Off-White SolidMasse moléculaire :217.15β-Pompilidotoxin Acetate
β-Pompilidotoxin Acetate is a wasp venom peptide.Formule :C73H128N22O19Degré de pureté :98.64%Couleur et forme :SolidMasse moléculaire :1617.93Ref: TM-T21769L
2mg47,00€5mg66,00€10mg89,00€25mg154,00€50mg221,00€100mg314,00€200mg442,00€1mL*10mM (DMSO)136,00€Myomodulin acetate(110570-93-9 free base)
Myomodulin acetate is present in two identified aplysia neurons that contain myomodulin A the ARC motor neuron B16 and the abdominal neuron L10.Formule :C38H71N11O10S2Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :906.17Levamlodipine hydrochloride
CAS :Levamlodipine hydrochloride is a medication used to lower blood pressure and prevent chest pain.Formule :C20H26Cl2N2O5Couleur et forme :SolidMasse moléculaire :445.34Ivacaftor
CAS :Ivacaftor (VX-770) (VX-770) is a potentiator of CFTR targeting G551D-CFTR (EC50: 100 nM) and F508del-CFTR (EC50: 25 nM) in Fisher rat thyroid cells,Formule :C24H28N2O3Degré de pureté :99% - 99.98%Couleur et forme :SolidMasse moléculaire :392.49Ref: TM-T2588
1mg38,00€2mgÀ demander5mg81,00€10mg127,00€25mg205,00€50mg304,00€100mg439,00€200mgÀ demander1mL*10mM (DMSO)88,00€TRPM8 antagonist WS-3
CAS :TRPM8 antagonist WS-3 (Cyclohexanecarboxamide) is an agonist of TRPM8( EC50 : 3.7 μM).Formule :C13H25NODegré de pureté :97.64%Couleur et forme :DrypowderMasse moléculaire :211.34NBQX
CAS :NBQX (FG9202) is a potent, selective and competitive AMPA receptor antagonist. Neuroprotective and anticonvulsant; active in vivo.Formule :C12H8N4O6SDegré de pureté :97.66% - 99.93%Couleur et forme :SolidMasse moléculaire :336.28Ref: TM-T4113
1mg40,00€2mg52,00€5mg88,00€10mg120,00€25mg235,00€50mg354,00€100mg525,00€200mg757,00€1mL*10mM (DMSO)96,00€NPPB
CAS :NPPB is a chloride channel blocker with IC50 of 80 nM .Formule :C16H16N2O4Degré de pureté :99.95%Couleur et forme :Light Yellow To Yellow SolidMasse moléculaire :300.31Ononetin
CAS :Ononetin (2',4'-Dihydroxy-2-(4-methoxyphenyl)acetophenone) is a TRPM3 channel blocker(IC50: 0.3 μM).Formule :C15H14O4Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :258.27Vonoprazan
CAS :Vonoprazan (TAK-438 (free base)) is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduodenal ulcer andFormule :C17H16FN3O2SDegré de pureté :99.87% - 99.92%Couleur et forme :SolidMasse moléculaire :345.39ICA-121431
CAS :ICA-121431: a potent Nav1.7 inhibitor (IC50=19 nM for rat), minimal effect on human Nav1.5/Nav1.7.Formule :C23H19N3O3S2Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :449.55Sepimostat dimethanesulfonate
CAS :Sepimostat dimethanesulfonate (FUT-187) is a neuroprotective NR2B receptor antagonist with an inhibition Ki of 27.7 μM.Formule :C23H27N5O8S2Couleur et forme :SolidMasse moléculaire :565.62Indecainide hydrochloride
CAS :Indecainide hydrochloride is a cardiac depressant.Formule :C20H25ClN2OCouleur et forme :SolidMasse moléculaire :344.88Selinexor (KPT-330)
CAS :Selinexor (KPT-330) is an orally available, small molecule inhibitor of CRM1 (exportin 1 or XPO1), with potential antineoplastic activity.Formule :C17H11F6N7ODegré de pureté :98% - 99.97%Couleur et forme :SolidMasse moléculaire :443.316-Methylflavone
CAS :6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Formule :C16H12O2Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :236.27Homo-VK-II-36
CAS :Homo-VK-II-36 (Homo-V-II-36) is a carvedilol analogue that acts by inhibiting store- overload-induced calcium release through the RyR2 channel.Formule :C27H28N2O5Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :460.52Flupirtine maleate
CAS :Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.Formule :C15H17FN4O2·C4H4O4Degré de pureté :99.5% - 99.9%Couleur et forme :Off-White Crystalline PowderMasse moléculaire :420.39Vanilloid receptor antagonist 1
CAS :Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.Formule :C18H15N3O2Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :305.33Ref: TM-T9247
1mg99,00€5mg235,00€10mg354,00€25mg602,00€50mg847,00€100mg1.206,00€1mL*10mM (DMSO)47,00€7-Chlorokynurenic acid sodium salt
CAS :7-CKA sodium salt: NMDA receptor antagonist, glycine B site (IC50: 0.56 μM), blocks glutamate reuptake (Ki: 0.59 μM).Formule :C10H6ClNNaO3Couleur et forme :SolidMasse moléculaire :246.6Optovin
CAS :Optovin is a TRPA1 activator, which is reversibly photoactivated.Formule :C15H13N3OS2Degré de pureté :99.47% - 99.67%Couleur et forme :SolidMasse moléculaire :315.41Ref: TM-T6617
2mg39,00€5mg57,00€10mg93,00€25mg160,00€50mg250,00€100mg406,00€200mg592,00€1mL*10mM (DMSO)64,00€Linerixibat
CAS :Linerixibat (GSK2330672) is a highly effective, nonabsorbable ASBT inhibitor. Linerixibat can lower glucose in an animal model of type 2 diabetes.Formule :C28H38N2O7SDegré de pureté :98.5% - 99.98%Couleur et forme :SolidMasse moléculaire :546.68Azumolene sodium anhydrous
CAS :Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.Formule :C13H8BrN4NaO3Couleur et forme :SolidMasse moléculaire :371.13Zosuquidar
CAS :Zosuquidar (RS 33295-198) is a potent P-glycoprotein inhibitor with antitumor activity that inhibits tumor growth.Formule :C32H31F2N3O2Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :527.6Ref: TM-T6018L
1mg73,00€5mg152,00€10mg220,00€25mg358,00€50mg537,00€100mg782,00€200mg1.071,00€1mL*10mM (DMSO)170,00€α-Cyano-4-hydroxycinnamic acid
CAS :α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) (α-CHCA) is an inhibitor of monocarboxylate transporter 1 (MCT1) that blocks pyruvateFormule :C10H7NO3Degré de pureté :99.8% - 99.86%Couleur et forme :PowderMasse moléculaire :189.17AZD-9056 free base
CAS :AZD9056 is a potent, selective, orally bioavailable P2X7 receptor antagonist.Formule :C24H35ClN2O2Couleur et forme :SolidMasse moléculaire :419A-803467
CAS :A-803467 is a selective NaV1.8 channel blocker.Formule :C19H16ClNO4Degré de pureté :96.94% - 98%Couleur et forme :SolidMasse moléculaire :357.79Glibenclamide potassium
CAS :Glibenclamide potassium, a more soluble form of Glibenclamide, exists as anhydrous and hydrate salts.Formule :C23H27ClKN3O5SCouleur et forme :SolidMasse moléculaire :532.09Efonidipine hydrochloride
CAS :Efonidipine HCl (NZ-105) blocks T-type/L-type calcium channels; used in hypertension treatment.Formule :C34H39ClN3O7PCouleur et forme :SolidMasse moléculaire :668.12
