Transporteur membranaire/Canal ionique
Les inhibiteurs des transporteurs membranaires et des canaux ioniques sont des composés qui bloquent la fonction des protéines responsables du transport des ions, des nutriments et d'autres molécules à travers les membranes cellulaires. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie cellulaire, la transduction des signaux et la neurotransmission. Les inhibiteurs des transporteurs membranaires et des canaux ioniques sont également importants pour développer des traitements contre des troubles tels que l'épilepsie, les maladies cardiovasculaires et les syndromes métaboliques. Chez CymitQuimica, nous offrons une sélection diversifiée d'inhibiteurs de haute qualité des transporteurs membranaires et des canaux ioniques pour soutenir vos recherches en physiologie, neurosciences et pharmacologie.
Sous-catégories appartenant à la catégorie "Transporteur membranaire/Canal ionique"
- ABC(3 produits)
- ATPase(93 produits)
- Récepteur de l'adiponectine(5 produits)
- CFTR(64 produits)
- Récepteur CGRP(51 produits)
- Canal calcique(493 produits)
- Canal chlorure(49 produits)
- Récepteur GABA(336 produits)
- Transporteur de monoamine(23 produits)
- Transporteur de monocarboxylate(17 produits)
- NKCC(2 produits)
- NPC1L1(3 produits)
- Cotransporteur Na-K-Cl(8 produits)
- OAT(27 produits)
- OCT(7 produits)
- P-gp(53 produits)
- Canal potassique(276 produits)
- Pompe à protons(39 produits)
- SGLT(30 produits)
- Canal sodique(202 produits)
- Canal TRP/TRPV(92 produits)
Affichez 13 plus de sous-catégories
2270 produits trouvés pour "Transporteur membranaire/Canal ionique"
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GABAA receptor agent 1
CAS :<p>GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.</p>Formule :C13H8ClN3O2Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :273.675,5-Dimethyloxazolidine-2,4-dione
CAS :<p>5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.</p>Formule :C5H7NO3Degré de pureté :99.12%Couleur et forme :Drypowder PelletslargecrystalsMasse moléculaire :129.11Vinpocetine
CAS :<p>Vinpocetine (RGH-4405) is a selective inhibitor of cyclic GMP phosphodiesterase (PDE).</p>Formule :C22H26N2O2Degré de pureté :99.85% - 99.98%Couleur et forme :White Crystalline SolidMasse moléculaire :350.45FG 7142
CAS :<p>FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.</p>Formule :C13H11N3ODegré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :225.25Torsemide
CAS :<p>Torsemide (AC-4464), a sulfonylurea loop diuretic, has a long action duration, high plasma protein binding, and a long half-life.</p>Formule :C16H20N4O3SDegré de pureté :99.81%Couleur et forme :Crystalline SolidMasse moléculaire :348.42Nefiracetam
CAS :<p>Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.</p>Formule :C14H18N2O2Degré de pureté :97.37%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :246.3FFN 206 dihydrochloride
CAS :<p>FFN 206 dihydrochloride: fluorescent VMAT2 marker, detects subcellular sites, non-inhibitory to DAT.</p>Formule :C12H15ClN2O2Degré de pureté :98.96% - >99.99%Couleur et forme :SolidMasse moléculaire :254.71Piracetam
CAS :<p>Piracetam (UCB-6215), a cyclic derivative of the neurotransmitter gamma-aminobutyric acid (GABA), is used in therapy of the extensive cognitive disorders.</p>Formule :C6H10N2O2Degré de pureté :97.16%Couleur et forme :Crystals From Isopropanol SolidMasse moléculaire :142.16Afoxolaner
CAS :<p>Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs.</p>Formule :C26H17ClF9N3O3Degré de pureté :99.1% - 99.38%Couleur et forme :SolidMasse moléculaire :625.87Flufenamic acid
CAS :<p>Flufenamic acid (Arlef) is an anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties.</p>Formule :C14H10F3NO2Degré de pureté :98.68%Couleur et forme :White To Light Yellow Crystalline PowderMasse moléculaire :281.23Halothane
CAS :<p>Halothane (Anestan) 可以减弱内皮依赖性舒张作用。</p>Formule :C2HBrClF3Degré de pureté :98.50% - >99.99%Couleur et forme :Colorless Volatile Liquid Density 1 875 G / Cm3 Boiling Point 122 4°F (50 2°C) NoncombustibleMasse moléculaire :197.38Hydrochlorothiazide
CAS :<p>Hydrochlorothiazide (HCTZ) 是一种口服有效的噻嗪类的利尿药，可抑制转化 TGF-β/Smad 信号通路。它通过打开钙激活钾 (KCA) 通道发挥直接的血管松弛作用。它改善心脏功能，减少纤维化并具有降压作用。</p>Formule :C7H8ClN3O4S2Degré de pureté :99.43% - 99.50%Couleur et forme :Crystals Physical Description Crystals Or White Powder (Ntp 1992)Masse moléculaire :297.74L-Cycloserine
CAS :<p>L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.</p>Formule :C3H6N2O2Degré de pureté :99.45% - 99.92%Couleur et forme :Crystals White PowderMasse moléculaire :102.09Riparin III
CAS :<p>Riparin III is an alcamide isolated from Aniba riparia that has exhibited effects of antidepressant and anxiolytic activities in acute stress behavioral models.</p>Formule :C16H17NO4Degré de pureté :95.13%Couleur et forme :SolidMasse moléculaire :287.31BMS-394136
CAS :<p>BMS-394136 (BMS 394136) is a KV1.5 antagonist for the treatment of cardiovascular diseases such as arrhythmias and atrial fibrillation.</p>Formule :C24H21Cl2FN4ODegré de pureté :98.19% - 98.67%Couleur et forme :SolidMasse moléculaire :471.35Phenazopyridine hydrochloride
CAS :<p>Phenazopyridine HCl, an oral urinary analgesic, may cause nausea, anemia, and liver/kidney toxicity. Possibly carcinogenic.</p>Formule :C11H12ClN5Degré de pureté :99.27%Couleur et forme :Brownish-Yellow Crystals Aqueous Solutions Are Yellow To Brick-Red And Slightly Acidic; They May Be Stabilized By The AdditionMasse moléculaire :249.7RUVBL1/2 ATPase-IN-1
CAS :<p>RUVBL1/2 ATPase-IN-1 inhibits RUVBL1/2 ATPase (IC50: 6.0/7.7 μM); useful in cancer research.</p>Formule :C28H28F3N5ODegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :507.55Endovion
CAS :<p>Endovion (NS3728) is a pharmacological anion channel and an Anoctamin-1 (ANO 1) channel inhibitor. Endovion is also the specific VRAC/VSOAC blocker.</p>Formule :C16H9BrF6N6ODegré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :495.18NS8593 hydrochloride
CAS :<p>NS8593 hydrochloride (NS8593 HCl) is a potent and selective inhibitor of small conductance Ca2+-activated K+ channels (SK channels) .</p>Formule :C17H18ClN3Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :299.8Ropivacaine
CAS :<p>Ropivacaine (LEA-103 HCl) is a local anaesthetic drug belonging to the amino amide group.</p>Formule :C17H26N2ODegré de pureté :97.75% - >99.99%Couleur et forme :SolidMasse moléculaire :274.40Dyclonine hydrochloride
CAS :<p>Dyclonine hydrochloride (Dyclonine HCl) , an over the counter throat lozenge, is found in Sucretswith local anesthetic effect .</p>Formule :C18H27NO2·HClDegré de pureté :99.35%Couleur et forme :White Crystalline SolidMasse moléculaire :325.87(Z)-Capsaicin
CAS :<p>(Z)-Capsaicin (Zucapsaicin) is a medication used to treat osteoarthritis of the knee and Others neuropathic pain.(Z)-Capsaicin is a synthetic cis isomer of</p>Formule :C18H27NO3Degré de pureté :97.33% - 98.91%Couleur et forme :SolidMasse moléculaire :305.41Nicorandil
CAS :<p>Nicorandil (SG-75)(Ikorel) acts by relaxing the smooth muscle of the blood vessels, especially those of the venous system.</p>Formule :C8H9N3O4Degré de pureté :98.14% - >99.99%Couleur et forme :White Or Off-White PowderMasse moléculaire :211.17Alinidine
CAS :<p>Alinidine is an HCN channel blocker with antiarrhythmic effects and can be used for the study of angina pectoris.</p>Formule :C12H13Cl2N3Degré de pureté :98.91% - >99.99%Couleur et forme :SolidMasse moléculaire :270.16Tocainide hydrochloride
CAS :<p>Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) is a sodium channel blocker.</p>Formule :C11H17ClN2ODegré de pureté :97%Couleur et forme :SolidMasse moléculaire :228.72Flindokalner
CAS :<p>Flindokalner (BMS-204352) modulates potassium channels, enhances Kv7 subtypes and BKca, inhibits Kv7.1 (Ki=3.7μM), GABAA; has anxiolytic effects in vivo.</p>Formule :C16H10ClF4NO2Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :359.7URAT1 inhibitor 7
CAS :<p>URAT1 inhibitor 7, a uric acid transporter protein URAT1 inhibitor.URAT1 inhibitor 7 inhibits CYP2C9 and can be used in the study of hyperuricemia and gout.</p>Formule :C19H10ClFN4O3SDegré de pureté :97.65%Couleur et forme :SoildMasse moléculaire :428.82Glibenclamide
CAS :<p>Glibenclamide (Glyburide) is an antidiabetic sulfonylurea derivative with actions similar to those of chlorpropamide.</p>Formule :C23H28ClN3O5SDegré de pureté :99.05% - 99.75%Couleur et forme :SolidMasse moléculaire :494.00QX-314 chloride
CAS :<p>QX-314 chloride is a membrane-impermeable permanently charged blocker of sodium channel.</p>Formule :C16H27ClN2ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :298.85Gabapentin
CAS :<p>Gabapentin (Neurontin) is an Anti-epileptic Agent.</p>Formule :C9H17NO2Degré de pureté :99.55% - 99.91%Couleur et forme :White To Off-White Crystalline Solid; Crystals From Ethanol/Ether SolidMasse moléculaire :171.24NBQX disodium
CAS :<p>NBQX Disodium (FG9202 disodium) is a highly selective, competitive AMPA receptor antagonist with neuroprotective and anticonvulsant activity.</p>Formule :C12H6N4Na2O6SDegré de pureté :97.6% - 98.22%Couleur et forme :SolidMasse moléculaire :380.2415Clorsulon
CAS :<p>Clorsulon (L631529) is utilized for the treatment of Fasciola hepatica infections in calves and sheep.</p>Formule :C8H8Cl3N3O4S2Degré de pureté :99.66% - 99.87%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :380.66Miconazole
CAS :<p>Miconazole (R18134) is an imidazole antifungal agent that is used topically and by intravenous infusion.</p>Formule :C18H14Cl4N2ODegré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :416.13Omeprazole
CAS :<p>Omeprazole (Losec) is a proton pump inhibitor (PPI), Omeprazole(Losec) is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor.</p>Formule :C17H19N3O3SDegré de pureté :98.43% - 98.48%Couleur et forme :White SolidMasse moléculaire :345.42Pivagabine
CAS :<p>Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.</p>Formule :C9H17NO3Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :187.24Phenelzine sulfate
CAS :<p>Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.</p>Formule :C8H14N2O4SDegré de pureté :98.38% - 99.83%Couleur et forme :SolidMasse moléculaire :234.27Ropivacaine hydrochloride
CAS :<p>Ropivacaine hydrochloride (Ropivacaine monohydrochloride) is the hydrochloride salt of ropivacaine, a local anesthetic of the amide type with analgesic activity</p>Formule :C17H26N2O·HClDegré de pureté :99.85% - 99.95%Couleur et forme :SolidMasse moléculaire :310.86Oxybutynin
CAS :<p>Oxybutynin (Ditropan) is a synthetic anticholinergic agent that is used for treatment of urinary incontinence and overactive bladder syndrome.</p>Formule :C22H31NO3Degré de pureté :97.81% - 99.57%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :357.49N-Acetylprocainamide
CAS :<p>N-Acetylprocainamide (NAPA), the N-acetylated metabolite of Procainamide, is a Class III antiarrhythmic agent, while procainamide is a Class Ia antiarrhythmic</p>Formule :C15H23N3O2Degré de pureté :99.65% - 99.74%Couleur et forme :SolidMasse moléculaire :277.36VU591 hydrochloride
CAS :<p>VU591 hydrochloride is a selective Kir1.1 (ROMK) blocker with IC50 of 0.24 μM, not affecting Kir7.1, Kir2.1, Kir2.3, or Kir4.1, similar to VU 590.</p>Formule :C16H13ClN6O5Degré de pureté :98.93% - 99.22%Couleur et forme :SolidMasse moléculaire :404.76Emamectin Benzoate
CAS :<p>Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods</p>Formule :C56H81NO15Degré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :1008.256Acetohexamide
CAS :<p>Acetohexamide (Acetohexamid) is an intermediate-acting, first-generation sulfonylurea with hypoglycemic activity.</p>Formule :C15H20N2O4SDegré de pureté :99.19% - 99.85%Couleur et forme :Crystals From 90% Aq EthanolMasse moléculaire :324.40Hydroxyhexamide
CAS :<p>Hydroxyhexamide ((±)-Hydroxyhexamid) is a pharmacologically active metabolite of Acetohexamide, used as a hypoglycemic agent.</p>Formule :C15H22N2O4SDegré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :326.41Gliclazide
CAS :<p>Gliclazide (SE1702), an oral antihyperglycemic agent, belongs to the sulfonylurea class of insulin secretagogues, which act by stimulating beta-cells of the</p>Formule :C15H21N3O3SDegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :323.41NS5806
CAS :<p>NS5806 activates K+ currents, slows KV4.2/4.3 decay with KChIP2, and boosts KV4.3/KChIP2 peaks (EC50=5.3μM).</p>Formule :C16H8Br2F6N6ODegré de pureté :97.95%Couleur et forme :SolidMasse moléculaire :574.07Meticrane
CAS :<p>Meticrane (Arresten) is a sulphonamide-derivative with thiazide-like diuretic activity.</p>Formule :C10H13NO4S2Degré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :275.34BIIB 722 Mesylate
CAS :<p>BIIB 722 Mesylate is a sodium-hydrogen exchange inhibitor with cardioprotective properties and can be used to study myocardial ischemia.</p>Formule :C19H23F3N6O5SDegré de pureté :99.57%Couleur et forme :SoildMasse moléculaire :504.483VU591
CAS :<p>VU591 is a selective extra-renal potassium channel inhibitor with an IC₅₀ of 0.24 μM.</p>Formule :C16H12N6O5Degré de pureté :99.29% - 99.53%Couleur et forme :SolidMasse moléculaire :368.3Nav1.8-IN-4
CAS :<p>Nav1.8-IN-4 is a potent Nav1.8 channel inhibitor with potential analgesic activity.Nav1.8-IN-4 can be used for pain and neurological related disorders.</p>Formule :C20H14F4N2O3Degré de pureté :99.83%Couleur et forme :SoildMasse moléculaire :406.33Tuvatexib
CAS :<p>Tuvatexib is a small molecule VDAC/HK2 dual modulator.</p>Formule :C21H23NO3Degré de pureté :97.29% - 99.80%Couleur et forme :SolidMasse moléculaire :337.41E 0747 FA
<p>E 0747 FA is an antiarrhythmic compound that inhibits the voltage of action potential Vmax in Purkinje fibers of porcine heart.E 0747 FA inhibits Na channels in cardiac cells.</p>Formule :C22H30ClN3O6Degré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :467.94Broflanilide
CAS :<p>Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 nM.</p>Formule :C25H14BrF11N2O2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :663.29Lansoprazole
CAS :<p>Lansoprazole (A-65006) is a 2, 2, 2-trifluoroethoxypyridyl derivative of timoprazole that is used in the therapy of STOMACH ULCERS and ZOLLINGER-ELLISON</p>Formule :C16H14F3N3O2SDegré de pureté :99.18% - 99.84%Couleur et forme :White Crystalline PowderMasse moléculaire :369.36NS1652
CAS :<p>NS1652 is an anion conductance inhibitor. NS1652 blocks chloride channel has an IC50 of 1.6 μM in human and mouse red blood cells.</p>Formule :C15H11F3N2O3Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :324.25VU6036720
<p>VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuit</p>Formule :C20H22ClFN4O2SDegré de pureté :98.1%Couleur et forme :SoildMasse moléculaire :436.93BI-749327
CAS :<p>BI-749327 is a high selectivity and orally bioavailable antagonist of TRPC6 (IC50s: 13 nM, 19 nM and 15 nM for mouse, human and guinea pig TRPC6).</p>Formule :C23H21F3N4O2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :442.43NS13001
CAS :<p>NS13001, an oral SK channel modulator, shows promise for SCA2 therapy; EC50: 1.8 µM (SK2), 0.14 µM (SK3).</p>Formule :C17H16ClN7Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :353.81Zamicastat
CAS :<p>Zamicastat (BIA 5-1058) inhibits DBH, P-gp (IC50=73.8μM), and BCRP (IC50=17.0μM).</p>Formule :C21H21F2N3OSDegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :401.47NMDA-IN-1
CAS :<p>NMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM).</p>Formule :C20H23ClFN3ODegré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :375.87Pramocaine hydrochloride
CAS :<p>Pramocaine hydrochloride (Pramoxine HCl), a topical anesthetic, is served as an antipruritic.</p>Formule :C17H27NO3·HClDegré de pureté :99.15% - 99.61%Couleur et forme :Crystals White Or Off White Crystalline PowderMasse moléculaire :329.86Cromolyn sodium
CAS :<p>Cromolyn sodium (FPL-670) is a chromone complex that acts by inhibiting the release of chemical mediators from sensitized mast cells.</p>Formule :C23H14Na2O11Degré de pureté :99.4% - 99.95%Couleur et forme :Colorless Crystals From Ethanol + Ether White Crystalline PowderMasse moléculaire :512.33VU0134992 hydrochloride
CAS :<p>VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).</p>Formule :C20H32BrClN2O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :447.841-EBIO
CAS :<p>1-EBIO (1-EBIO) is a calium channel agonist.</p>Formule :C9H10N2ODegré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :162.19FFN 511
CAS :<p>Fluorescent false neurotransmitter (FFN)</p>Formule :C17H20N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :284.35Clomethiazole
CAS :<p>Clomethiazole (Distraneurin) is an orally active GABAA agonist and it is an anticonvulsant agent. It has potential for treating convulsive status epilepticus.</p>Formule :C6H8ClNSDegré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :161.65TRPV4 agonist-1 free base
CAS :<p>TRPV4 agonist-1 free base (OUN67600) is an agonist of transient receptor potential vanilloid 4 (TRPV4;EC50 of 60 nM, in the hTRPV4 Ca2+ assay).</p>Formule :C25H22F2N4O2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :448.46Ethaverine hydrochloride
CAS :<p>Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.</p>Formule :C24H30ClNO4Degré de pureté :99.66% - 99.90%Couleur et forme :SolidMasse moléculaire :431.96T16Ainh-A01
CAS :<p>T16Ainh-A01 is a potent TMEM16A chloride channel inhibitor with a 1 μM IC50, targeting CaCC.</p>Formule :C19H20N4O3S2Degré de pureté :97.18% - 98.15%Couleur et forme :SolidMasse moléculaire :416.52Vocacapsaicin hydrochloride
CAS :<p>Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and is used for pain relief.</p>Formule :C26H42ClN3O4Degré de pureté :99.66% - 99.80%Couleur et forme :SolidMasse moléculaire :496.08ATP synthase inhibitor 1
CAS :<p>ATP synthase inhibitor 1 is an inhibitor of the c subunit of the F1/FO-ATP synthase complex.</p>Formule :C17H18ClN3O3S2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :411.93GFB-8438
CAS :<p>GFB-8438 is a potent and subtype selective inhibitor of TRPC5(IC50s of 0.18 and 0.29 μM of hTRPC5 and hTRPC4, respectively).</p>Formule :C16H14ClF3N4O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :386.76Repaglinide
CAS :<p>Repaglinide, a benzoic acid derivative, stimulates insulin, treats type 2 diabetes, and may rarely cause acute liver injury.</p>Formule :C27H36N2O4Degré de pureté :99.73% - >99.99%Couleur et forme :White To Off-White SolidMasse moléculaire :452.59Domperidone EP Impurity A
CAS :<p>Domperidone EP Impurity A is used as pharmaceutical intermediates.</p>Formule :C12H14ClN3ODegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :251.71Sulfacarbamide
CAS :<p>Sulfacarbamide (Sulfanilylurea) is a blood sugar-lowering agent.</p>Formule :C7H9N3O3SDegré de pureté :95.6% - 99.72%Couleur et forme :SolidMasse moléculaire :215.23Econazole
CAS :<p>Econazole ((±)-Econazol) is an imidazole derivative that is commonly used as a topical antifungal agent.</p>Formule :C18H15Cl3N2ODegré de pureté :98.11% - 99.97%Couleur et forme :SolidMasse moléculaire :381.68Ornidazole (Levo-)
CAS :<p>Ornidazole (Levo-) (Levornidazole) is the levo-isomer of Ornidazole.</p>Formule :C7H10ClN3O3Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :219.63Tertiapin-Q
CAS :<p>Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner, inhibiting efflux to K(+).</p>Formule :C106H175N35O24S4Degré de pureté :98.06% - 98.09%Couleur et forme :SolidMasse moléculaire :2452CGP37157
CAS :<p>CGP37157 (7-Chloro-5-(2-chlorophenyl)-1,5-dihydro-4,1-benzothiazepine-2(3H)-one) is a Na+/Ca2+ exchanger inhibitor, inhibits Na+-induced Ca2+ release from</p>Formule :C15H11Cl2NOSDegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :324.22Manidipine dihydrochloride
CAS :<p>Manidipine dihydrochloride (Manidipine 2HCl) is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).</p>Formule :C35H40Cl2N4O6Degré de pureté :99.76% - 99.86%Couleur et forme :SolidMasse moléculaire :683.62D-AP5
CAS :<p>D-AP5 (D-APV) is a NMDA receptor antagonist.</p>Formule :C5H12NO5PDegré de pureté :98.77% - >99.99%Couleur et forme :White Fine Crystalline PowderMasse moléculaire :197.13Etifoxine hydrochloride
CAS :<p>Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug.</p>Formule :C17H18Cl2N2ODegré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :337.24CRAC intermediate 2
CAS :<p>CRAC intermediate 2 is a intermediate compound for CRAC inhibitor synthesis.</p>Formule :C11H7F6N3Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :295.18PF-04885614
CAS :<p>PF-04885614 is a potent inhibitor of NaV1.8, has potential for neurological and neurodevelopmental diseases treatment.</p>Formule :C13H14F3N3ODegré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :285.27Tolazamide
CAS :<p>Tolazamide (U-17835) is a sulphonylurea hypoglycemic agent with actions and uses similar to those of CHLORPROPAMIDE.</p>Formule :C14H21N3O3SDegré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :311.40Devapamil
CAS :<p>Devapamil (Devapamilo) is a phenylalkylamine that blocks L-type calcium currents from the inner side of membrane cells in a use-dependent manner.</p>Formule :C26H36N2O3Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :424.58Vigabatrin
CAS :<p>Vigabatrin (Sabril), an analogue of gamma-aminobutyric acid, is an irreversible inhibitor of 4-aminobutyrate Transaminase responsible for the catabolism of γ-</p>Formule :C6H11NO2Degré de pureté :99.47% - 99.88%Couleur et forme :SolidMasse moléculaire :129.16LAU159
CAS :<p>LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).</p>Formule :C17H12ClN3O2Degré de pureté :98.7% - 99.38%Couleur et forme :SolidMasse moléculaire :325.75Oxiracetam
CAS :<p>Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.</p>Formule :C6H10N2O3Degré de pureté :99.67%Couleur et forme :White Crystalline PowderMasse moléculaire :158.16Permethrin
CAS :<p>Permethrin (NRDC-143) is a pyrethroid insecticide commonly used in the treatment of LICE INFESTATIONS and SCABIES.</p>Formule :C21H20Cl2O3Degré de pureté :99.37% - 99.54%Couleur et forme :Colorless Crystals To A Viscous Liquid; Color White To Pale Yellow Permethrin Is A Pale Brown Liquid Relatively Water Insoluble Used As An InsecticideMasse moléculaire :391.29AR-C155858
CAS :<p>AR-C155858 is an inhibitor of monocarboxylate transporter MCT1 and MCT2 (Kis: 2.3 nM and 10 nM).</p>Formule :C21H27N5O5SDegré de pureté :98.96% - 99.42%Couleur et forme :SolidMasse moléculaire :461.53Oxybutynin chloride
CAS :<p>Oxybutynin chloride (Oxybutynin HCl) is an anticholinergic medication used to relieve urinary and bladder difficulties.</p>Formule :C22H32ClNO3Degré de pureté :99.27% - >99.99%Couleur et forme :White PowderMasse moléculaire :393.96BMS-191095
CAS :<p>BMS-191095 is mitochondrial ATP-sensitive potassium (mitoKATP) channel activator.</p>Formule :C22H21ClN4O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :408.88DCEBIO
CAS :<p>DCEBIO, a 1-EBIO derivative, enhances Cl- secretion via hIK1 K+ channel and apical conductance in T84 cells.</p>Formule :C9H8Cl2N2ODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :231.08Chlormezanone
CAS :<p>Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.</p>Formule :C11H12ClNO3SDegré de pureté :99.89% - >99.99%Couleur et forme :Crystals SolidMasse moléculaire :273.74Isoguvacine hydrochloride
CAS :<p>Isoguvacine hydrochloride (1,2,3,6-tetrahydro-4-pyridinecarboxylic acid hydrochloride) is a GABA receptor agonist.</p>Formule :C6H10ClNO2Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :163.6Topiramate
CAS :<p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>Formule :C12H21NO8SDegré de pureté :99.79% - 99.92%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :339.36IA-Alkyne
CAS :<p>IA-Alkyne: TRPC agonist, cysteine-reactivity probe, potential in respiratory infection study.</p>Formule :C8H12INODegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :265.09Eact
CAS :<p>Eact is a potent TMEM16A activator that also triggers TRPV1, causing itch, pain, and heat sensitivity.</p>Formule :C22H24N2O5SDegré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :428.5Chlorpropamide
CAS :<p>Chlorpropamide (Diabinese) is a sulfonylurea hypoglycemic agent used in the treatment of non-insulin-dependent diabetes mellitus not responding to dietary</p>Formule :C10H13ClN2O3SDegré de pureté :98.90%Couleur et forme :Crystals From Dil Ethanol Physical Description White Crystalline Powder With A Slight Odor (Ntp 1992)Masse moléculaire :276.74Gut restricted-7
CAS :<p>Gut restricted-7 (GR-7) (GR-7) is a covalent and orally active pan-bile salt hydrolase (BSH) inhibitor.</p>Formule :C25H40FNaO6SDegré de pureté :98.81% - 99.27%Couleur et forme :SolidMasse moléculaire :510.64NaV1.7 inhibitor-1
CAS :<p>NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).</p>Formule :C23H30FNO4SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :435.55Omeprazole metabolite Omeprazole sulfone
CAS :<p>Omeprazole metabolite Omeprazole sulfone can inhibit proton pump.</p>Formule :C17H19N3O4SDegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :361.42Pentetrazol
CAS :<p>Pentylenetetrazol is a GABA(A) receptor antagonist, that displays activity as a central nervous system and respiratory stimulant.</p>Formule :C6H10N4Degré de pureté :99.7% - >99.99%Couleur et forme :Bitter Taste Aqueous Solutions Neutral To Litmus (Ntp 1992)Masse moléculaire :138.17Nikethamide
CAS :<p>Nikethamide is a stimulant which mainly influences the respiratory cycle. Widely known by its former sales name of Coramine, it was used in the mid-twentieth century as a medical countermeasure against tranquilizer overtreatments, before the advent of end</p>Formule :C10H14N2ODegré de pureté :99.42%Couleur et forme :Followed By A Faint Sensation Of The Warmth (Ntp 1992)Masse moléculaire :178.23Flumazenil
CAS :<p>Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervous</p>Formule :C15H14FN3O3Degré de pureté :99.72% - 99.98%Couleur et forme :Less Crystals Colourless CrystalsMasse moléculaire :303.29Eleclazine hydrochloride
CAS :<p>Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).</p>Formule :C21H17ClF3N3O3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :451.83Phenformin hydrochloride
CAS :<p>Phenformin hydrochloride (Phenformin HCl) is an agent belonging to the biguanide class of antidiabetics with antihyperglycemic activity.</p>Formule :C10H16ClN5Degré de pureté :97.11% - 99.80%Couleur et forme :Lactic AcidosisMasse moléculaire :241.72ML418
CAS :<p>ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.</p>Formule :C19H24ClN3O3Degré de pureté :99.3%Couleur et forme :SolidMasse moléculaire :377.874-Aminopyridine
CAS :<p>4-Aminopyridine (Dalfampridine) is a nonselective potassium (K+) channel blocker that binds to the cytoplasmic side of the cell membrane.</p>Formule :C5H6N2Degré de pureté :91.61%Couleur et forme :SolidMasse moléculaire :94.11NS19504
CAS :<p>NS19504 is an activator of Ca2+-activated K+ channel with EC50 of 11.0 µM.</p>Formule :C10H9BrN2SDegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :269.16CIQ
CAS :<p>CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. EC50 value: 2.7 μM for NR2C and 2.8 μM for NR2D.</p>Formule :C26H26ClNO5Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :467.94Omeprazole sulfide
CAS :<p>Omeprazole sulfide (Ufiprazole), a metabolite of Omeprazole, functions as a proton pump inhibitor.</p>Formule :C17H19N3O2SDegré de pureté :98.83%Couleur et forme :White To Slightly Collored Solid Solid CrystallineMasse moléculaire :329.42DSP-2230
CAS :<p>DSP-2230 is a selective blocker of Nav1.7/Nav1.8.</p>Formule :C20H20F3N5O2Degré de pureté :97.14%Couleur et forme :SolidMasse moléculaire :419.4ICA-27243
CAS :<p>ICA-27243: Potent KCNQ2/Q3 opener, oral, EC50 0.38 μM; less effective on KCNQ4, KCNQ3/Q5; antiepileptic.</p>Formule :C12H7ClF2N2ODegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :268.65Suloctidil
CAS :<p>Suloctidil is a peripheral vasodilator that was formerly used in the management of peripheral and cerebral vascular disorders.</p>Formule :C20H35NOSDegré de pureté :99.75% - >99.99%Couleur et forme :SolidMasse moléculaire :337.56Baclofen
CAS :<p>Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.</p>Formule :C10H12ClNO2Degré de pureté :98% - >99.99%Couleur et forme :1992)Masse moléculaire :213.66Linopirdine
CAS :<p>Linopirdine (DuP 996) is a TRPV1 agonist.</p>Formule :C26H21N3ODegré de pureté :99.45% - 99.78%Couleur et forme :SolidMasse moléculaire :391.46Azosemide
CAS :<p>Azosemide is a potent NKCC1 inhibitor (IC50s: 0.246 µM and 0.197 µM for hNKCC1A and NKCC1B).</p>Formule :C12H11ClN6O2S2Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :370.84Methocarbamol
CAS :<p>Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.</p>Formule :C11H15NO5Degré de pureté :99.96%Couleur et forme :Crystals From Benzene SolidMasse moléculaire :241.24Trichlormethiazide
CAS :<p>Trichlormethiazide (Naqua) is a short-acting, 3-dichloromethyl derivative of hydrochlorothiazide, belonging to the class of thiazide diuretics.</p>Formule :C8H8Cl3N3O4S2Degré de pureté :98.8% - 99.54%Couleur et forme :SolidMasse moléculaire :380.66Fluxametamide
CAS :<p>Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).</p>Formule :C20H16Cl2F3N3O3Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :474.26γ-Aminobutyric acid
CAS :<p>γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.</p>Formule :C4H9NO2Degré de pureté :99.95%Couleur et forme :White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderMasse moléculaire :103.12Cycloleucine
CAS :<p>Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.</p>Formule :C6H11NO2Degré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :129.16Linoleoyl glycine
CAS :<p>Linoleoyl glycine activates hKCNQ1/hKCNE1 channels, has analgesic properties, and is found in skin, spinal cord, and brain.</p>Formule :C20H35NO3Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :337.5Glipizide
CAS :<p>Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.</p>Formule :C21H27N5O4SDegré de pureté :99.67% - 99.75%Couleur et forme :SolidMasse moléculaire :445.54Diphenidol hydrochloride
CAS :<p>Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.</p>Formule :C21H28ClNODegré de pureté :99.15% - 99.33%Couleur et forme :Crystals Soluble In Methanol WaterMasse moléculaire :345.91Ciclopirox olamine
CAS :<p>Ciclopirox olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.</p>Formule :C14H24N2O3Degré de pureté :99.16% - >99.99%Couleur et forme :White To Yellow Solid Solid Particulate/PowderMasse moléculaire :268.35Dooku1
CAS :<p>Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.</p>Formule :C13H9Cl2N3OSDegré de pureté :98.87% - 99.74%Couleur et forme :SolidMasse moléculaire :326.2Caloxin 2A1 TFA
<p>Caloxin 2A1 TFA is a PM Ca2+ pump inhibitor that inhibits human red blood cell Ca2+-Mg2+-ATPase leakage.</p>Formule :C66H92F3N19O24Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :1592.55BMS-195270
CAS :<p>BMS-195270 is a bio-active chemical.</p>Formule :C15H9ClF3N3O2Degré de pureté :98.7%Couleur et forme :SolidMasse moléculaire :355.7Flavoxate hydrochloride
CAS :<p>Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.</p>Formule :C24H26ClNO4Degré de pureté :99.78%Couleur et forme :White SolidMasse moléculaire :427.92Tocainide
CAS :<p>Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus.</p>Formule :C11H16N2ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :192.26Celivarone
CAS :<p>Celivarone is a potassium channel blocker used in the study of arrhythmias, atrial flutter and atrial fibrillation.</p>Formule :C34H47NO4Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :533.74MRZ 2-514
CAS :<p>MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with Ki</p>Formule :C11H6BrN3O3Degré de pureté :98.459%Couleur et forme :SolidMasse moléculaire :308.09Prilocaine hydrochloride
CAS :<p>Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.</p>Formule :C13H21ClN2ODegré de pureté :99.97%Couleur et forme :Needles White Or Off White Crystalline PowderMasse moléculaire :256.77Z433927330
CAS :<p>Z433927330 is a potent and selective Aquaporin-7 (AQP7) inhibitor(IC50s of 0.2).</p>Formule :C20H20N4O3Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :364.4Bupivacaine hydrochloride
CAS :<p>Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.</p>Formule :C18H28N2O·HClDegré de pureté :99.9% - >99.99%Couleur et forme :SolidMasse moléculaire :324.89NEO 376
CAS :<p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>Formule :C20H24ClN3ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :357.88Bemegride
CAS :<p>Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.</p>Formule :C8H13NO2Degré de pureté :99.89%Couleur et forme :Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)Masse moléculaire :155.19IK1 inhibitor PA-6
CAS :<p>IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouse</p>Formule :C31H32N4O2Degré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :492.61Elexacaftor
CAS :<p>Elexacaftor (VX-445) is a cystic fibrosis transmembrane conductance regulator (CFTR) corrector.Cost-effective and quality-assured.</p>Formule :C26H34F3N7O4SDegré de pureté :98.87% - 99.87%Couleur et forme :SolidMasse moléculaire :597.65NS3623
CAS :<p>NS3623 is an activator of human ether-a-go-go-related gene potassium channels.</p>Formule :C15H10BrF3N6ODegré de pureté :97.06%Couleur et forme :SolidMasse moléculaire :427.18Lotilaner
CAS :<p>Lotilaner is a parasiticide.</p>Formule :C20H14Cl3F6N3O3SDegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :596.76EN6
CAS :<p>EN6, a small molecule, activates autophagy by modifying ATP6V1A, inhibiting mTORC1 and enhancing lysosomal function to clear TDP-43 aggregates.</p>Formule :C19H14F2N4O2Degré de pureté :95.74% - 97.04%Couleur et forme :SolidMasse moléculaire :368.34Mebeverine hydrochloride
CAS :<p>Mebeverine hydrochloride (Colofac Hydrochloride), a β-phenylethylamine derivative, is a potent α1 repector inhibitor, relaxing the muscles in and around the gut</p>Formule :C25H35NO5Degré de pureté :99.81% - 99.81%Couleur et forme :SolidMasse moléculaire :429.55Ethosuximide
CAS :<p>Ethosuximide (Zarontin) is an anticonvulsant, blocks the low voltage-activated T-type calcium channel used in the treatment of absence seizures unaccompanied by</p>Formule :C7H11NO2Degré de pureté :98.87% - 99.72%Couleur et forme :Crystals From Acetone And Ether SolidMasse moléculaire :141.17MK-7622
CAS :<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Formule :C25H25N3O2Degré de pureté :99.77% - 99.8%Couleur et forme :SolidMasse moléculaire :399.48DMT1 blocker 2
CAS :<p>Compound 12f, a DMT1 blocker, inhibits DMT1 with a 0.83 IC50, potentially blocking intestinal iron absorption.</p>Formule :C16H13N3ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :263.29AZD 7009
CAS :<p>AZD 7009 is a novel antiarrhythmic compound that inhibits the sodium current of hNav1.5 in CHO K1 cells with an IC50 of 11 uM.</p>Formule :C23H34N4O5Degré de pureté :98.42% - 98.51%Couleur et forme :SoildMasse moléculaire :446.54Moxidectin
CAS :<p>Moxidectin (CL301423) is an anthelmintic for heartworm/intestinal worms in dogs, cats, horses, cattle, and sheep; oral/topical/injectable.</p>Formule :C37H53NO8Degré de pureté :97.38%Couleur et forme :Appearance White Or Pale Yellow Amorphous PowderMasse moléculaire :639.82Phenibut
CAS :<p>Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).</p>Formule :C10H13NO2Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :179.22γ-DGG acetate(6729-55-1 free base)
CAS :<p>gamma-DGG acetate(6729-55-1 free base) (γ-D-Glutamylglycine) is a competitive blocker of AMPA receptor.</p>Formule :C9H16N2O7Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :264.23GET73
CAS :<p>GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5.</p>Formule :C13H16F3NO2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :275.27Etimizol
CAS :<p>Etimizol improves memory by aiding the consolidation stage, effective against amnesia from hypoxia or brain injury.</p>Formule :C9H14N4O2Degré de pureté :99%Couleur et forme :SolidMasse moléculaire :210.23Oxybuprocaine hydrochloride
CAS :<p>Oxybuprocaine hydrochloride (Oxybuprocaine HCl), a local anesthetic, is used especially in otolaryngology and ophthalmology.</p>Formule :C17H29ClN2O3Degré de pureté :>99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :344.88DCPIB
CAS :<p>DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μM</p>Formule :C22H28Cl2O4Degré de pureté :99.79% - 99.87%Couleur et forme :SolidMasse moléculaire :427.36Doxapram hydrochloride hydrate
CAS :<p>Doxapram hydrochloride hydrate (Doxapram HCl) inhibits TASK-1, TASK-3, TASK-1/TASK-3 heterodimeric channel function with EC50 of 0.41, 37, 9 μM, respectively.</p>Formule :C24H33ClN2O3C24H30N2O2·ClH·H2ODegré de pureté :99.64% - >99.99%Couleur et forme :SolidMasse moléculaire :432.99Glimepiride
CAS :<p>Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.</p>Formule :C24H34N4O5SDegré de pureté :97.84% - 98.87%Couleur et forme :White Cyrstalline SolidMasse moléculaire :490.62Disopyramide
CAS :<p>Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.</p>Formule :C21H29N3ODegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :339.473,4,5-Trimethoxycinnamic acid
CAS :<p>3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at the</p>Formule :C12H14O5Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :238.24Butamben
CAS :<p>Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.</p>Formule :C11H15NO2Degré de pureté :99.43%Couleur et forme :Crystals From Alc Physical Description Yellow Powder Insoluble In Water (Ntp 1992)Masse moléculaire :193.24Penicillin G sodium salt
CAS :<p>Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of its sodium or potassium salts in the treatment of a</p>Formule :C16H17N2NaO4SDegré de pureté :98.11%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :356.37Leptomycin A
CAS :<p>Leptomycin A from Streptomyces inhibits CRM1, reducing HIV-1 replication, less potent than Leptomycin B, blocks protein nuclear export.</p>Formule :C32H46O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :526.7EVT-401
<p>EVT-401 (P2X7 receptor antagonist-1), a purinergic P2X7 receptor antagonist, demonstrates efficacy in combating neuroinflammation [1].</p>Formule :C22H20F4N2O3Couleur et forme :SolidMasse moléculaire :436.4Cavα2δ-IN-1
CAS :<p>Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a Ki</p>Formule :C18H27N5OCouleur et forme :SolidMasse moléculaire :329.448Nitrazolam
CAS :<p>Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.</p>Formule :C17H13N5O2Couleur et forme :SolidMasse moléculaire :319.32Elgodipine
CAS :<p>Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.</p>Formule :C29H33FN2O6Degré de pureté :98.95% - 99.50%Couleur et forme :SolidMasse moléculaire :524.58GS-9191 PM
<p>GS-9191 PM: novel antitumorviral bis-amide prodrug, inhibits MDR1/BCRP, has antiproliferative activity.</p>Formule :C11H16N6ODegré de pureté :99.79%Couleur et forme :SoildMasse moléculaire :248.28TRPA1 Antagonist 3
CAS :<p>TRPA1 Antagonist 3 is a compound with photoswitchable properties that acts as an agonist on the TRPA1 channel, providing the ability for optical control.</p>Formule :C11H8ClN3Couleur et forme :SolidMasse moléculaire :217.66(1S,3R)-3-Aminocyclopentane carboxylic acid
CAS :<p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>Formule :C6H11NO2Couleur et forme :SolidMasse moléculaire :129.16GsMTx4
CAS :<p>GsMTx-4, mechanosensitive and stretch-activated ion channel inhibitor (CAS 1209500-46-8).</p>Formule :C185H273N49O45S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4095.84BeKm-1
CAS :<p>Potent, selective hERG (KV11.1) blocker; doesn't affect 14 other K+ channels; extends QTc in rabbit heart dose-dependently.</p>Formule :C174H261N51O52S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4091.65GeX-2
CAS :<p>GeX-2 is a truncated analogue of αO-conotoxin. It has the ability to activate GABAB receptors and inhibit α9α10nAChR as well as CaV2.2 channels. Additionally, GeX-2 is effective in alleviating pain in a rat model of chronic constriction injury.</p>Formule :C103H169N43O27Couleur et forme :SolidMasse moléculaire :2441.72α,β-Methylene-ATP dilithium
CAS :<p>α,β-Methylene ATP dilithium, a phosphonic analog of ATP, serves as a ligand for P2X3 and P2X7 receptors.</p>Formule :C11H16Li2N5O12P3Couleur et forme :SolidMasse moléculaire :517.07GpTx-1 TFA
<p>GpTx-1 TFA is a polypeptide NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It exhibits potent inhibitory activity on the NaV1.7 channel with an IC50 value of 10 nM, demonstrating excellent selectivity over NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM) with >20-fold and >950-fold selectivity, respectively.</p>Couleur et forme :Odour SolidWAY-326766
CAS :<p>WAY-326766 increases ion transport through mutant CFTR and can be used to alter the lifespan of eukaryotes.WAY-326766 can be used to treat cystic fibrosis (CF).</p>Formule :C21H23N3O5Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :397.42AChE/Aβ-IN-1
<p>AChE/Aβ-IN-1 (compound 32) is a potent, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 86 nM and an NMDA receptor antagonist targeting the</p>Formule :C20H25BrN4Couleur et forme :SolidMasse moléculaire :401.34Anisatin
<p>Anisatin is a useful organic compound for research related to life sciences and the catalog number is T124719.</p>Formule :C15H20O8Couleur et forme :SolidMasse moléculaire :328.317Trans (2,3)-Dihydrotetrabenazine
CAS :<p>Trans (2,3)-Dihydrotetrabenazine is a Tetrabenazine metabolite, shows inhibition activity on vesicular monoamine transporter (VMAT2).</p>Formule :C19H29NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :319.44LRRK2-IN-15
<p>LRRK2-IN-15 is an inhibitor of LRRK2. It exhibits an IC50 value of 5 nM in PBMC cells and 1.5 μM for BCRP. This compound is utilized in the research of Parkinson's disease.</p>Couleur et forme :Odour SolidTP-050
CAS :<p>TP-050: potent, selective NMDAR agonist, EC50 0.51 µM (GluN2A), 9.6 µM (GluN2D), BBB permeable, boosts hippocampal LTP.</p>Formule :C16H15ClF2N6OCouleur et forme :SolidMasse moléculaire :380.78Albanin A
<p>Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.</p>Formule :C20H18O6Couleur et forme :SolidMasse moléculaire :354.358Jingzhaotoxin-XII TFA
<p>Jingzhaotoxin-XII (JzTx-XII) TFA is a specific inhibitor of the Kv4.1 channel, exhibiting an IC50 of 0.363 μM. It interacts with the channel by altering gating behavior.</p>Couleur et forme :Odour Solid3-Aminopropylphosphinic acid
CAS :<p>3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).</p>Formule :C3H10NO2PCouleur et forme :SolidMasse moléculaire :123.092Huwentoxin I
CAS :<p>Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.</p>Formule :C161H246N48O44S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3750.36LY-466195
CAS :<p>LY-466195 is a competitive antagonist of GLUK5 receptor.</p>Formule :C16H24F2N2O4Couleur et forme :SolidMasse moléculaire :346.37Hyp9
CAS :<p>Hyp9, a specific agonist for the transient receptor potential canonical 6 (TRPC6) channel, is utilized in spinal cord injury (SCI) research [1].</p>Formule :C18H26O5Couleur et forme :SolidMasse moléculaire :322.40AChE/Aβ-IN-2
<p>AChE/Aβ-IN-2 (compound 33) is a powerful, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 135 nM.</p>Formule :C20H25ClN4Couleur et forme :SolidMasse moléculaire :356.89Chlorotoxin TFA
<p>Chlorotoxin TFA, a scorpion venom peptide, blocks chloride channels and has anti-cancer properties.</p>Formule :C160H250F3N53O49S11Couleur et forme :SolidMasse moléculaire :4109.74JAMI1001A
CAS :<p>JAMI1001A enhances AMPA receptor signaling, slows deactivation/desensitization for flip/flop isoforms.</p>Formule :C16H17F3N4O3SCouleur et forme :SolidMasse moléculaire :402.39SLC26A3-IN-2
CAS :<p>Vilobelimab (CaCP-29) is a human-mouse chimeric IgG antibody targeting human complement component 5a, a C5a inhibitor that inhibits neutrophil activation.</p>Formule :C19H13ClN2O2SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :368.84Homocarnosine
CAS :<p>Homocarnosine is an endogenous dipeptide in cerebral regions and cerebrospinal fluid.</p>Formule :C10H16N4O3Couleur et forme :SolidMasse moléculaire :240.26Idactamab
CAS :<p>Idactamab (INT-001) is a monoclonal antibody to the human amino acid transport protein ASCT2.</p>Degré de pureté :> 95%Couleur et forme :LiquidMasse moléculaire :146.2 kDaAnticonvulsant agent 9
<p>Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.</p>Formule :C22H24N4O2Couleur et forme :SolidMasse moléculaire :376.45Crofelemer
CAS :<p>Crofelemer (Provir) is an orally active antidiarrheal agent. It targets the cystic fibrosis transmembrane conductance regulator (CFTR) and calcium-activated chloride channels (CACC), which are responsible for chloride and fluid secretion in the gastrointestinal tract. Crofelemer is applicable for research in diarrhea-related conditions.</p>Couleur et forme :Solid2,4,6-Tri-tert-butylphenol
CAS :<p>2,4,6-Tri-tert-butylphenol inhibits the Ca2+ ATPase activity of human red blood cell membranes and can be used in related research in the field of life sciences.</p>Formule :C18H30ODegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :262.43Bendroflumethiazide
CAS :<p>Bendroflumethiazide (Naturetin) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE. It has been used in the treatment of familial hyperkalemia, hypertension, edema, and urinary tract disorders. (From Martindale, The Extra Pharmacopoeia, 30th ed, p810)</p>Formule :C15H14F3N3O4S2Degré de pureté :98% - >99.99%Couleur et forme :Crystals From Dioxane SolidMasse moléculaire :421.41Levamlodipine besylate Hemipentahydrate
CAS :<p>Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.</p>Formule :C20H25ClN2O5·C6H6O3SH2OCouleur et forme :SolidMasse moléculaire :1224.18Analgesic/antidepressant agent-1
<p>Analgesic/antidepressant agent-1 (Compound k1) is an orally active N-acetylamino chloro ketone derivative capable of crossing the blood-brain barrier. It exhibits high affinity for NMDA receptors and demonstrates analgesic, anti-inflammatory, and antidepressant properties, with low psychotomimetic activity.</p>Formule :C22H25ClN2O2Couleur et forme :SolidMasse moléculaire :384.9Resolvin D2 methyl ester
CAS :<p>RvD2 is an anti-inflammatory lipid made from docosahexaenoic acid by 15- and 5-lipoxygenase. Its methyl ester may serve as a prodrug.</p>Formule :C23H34O5Couleur et forme :SolidMasse moléculaire :390.52
