Transporteur membranaire/Canal ionique
Les inhibiteurs des transporteurs membranaires et des canaux ioniques sont des composés qui bloquent la fonction des protéines responsables du transport des ions, des nutriments et d'autres molécules à travers les membranes cellulaires. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie cellulaire, la transduction des signaux et la neurotransmission. Les inhibiteurs des transporteurs membranaires et des canaux ioniques sont également importants pour développer des traitements contre des troubles tels que l'épilepsie, les maladies cardiovasculaires et les syndromes métaboliques. Chez CymitQuimica, nous offrons une sélection diversifiée d'inhibiteurs de haute qualité des transporteurs membranaires et des canaux ioniques pour soutenir vos recherches en physiologie, neurosciences et pharmacologie.
Sous-catégories appartenant à la catégorie "Transporteur membranaire/Canal ionique"
- ABC(3 produits)
- ATPase(93 produits)
- Récepteur de l'adiponectine(5 produits)
- CFTR(64 produits)
- Récepteur CGRP(51 produits)
- Canal calcique(493 produits)
- Canal chlorure(49 produits)
- Récepteur GABA(336 produits)
- Transporteur de monoamine(23 produits)
- Transporteur de monocarboxylate(17 produits)
- NKCC(2 produits)
- NPC1L1(3 produits)
- Cotransporteur Na-K-Cl(8 produits)
- OAT(27 produits)
- OCT(7 produits)
- P-gp(53 produits)
- Canal potassique(276 produits)
- Pompe à protons(39 produits)
- SGLT(30 produits)
- Canal sodique(202 produits)
- Canal TRP/TRPV(92 produits)
Affichez 13 plus de sous-catégories
2270 produits trouvés pour "Transporteur membranaire/Canal ionique"
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Ataluren
CAS :<p>Ataluren (PTC124) is a novel, orally administered drug that targets nonsense mutations.</p>Formule :C15H9FN2O3Degré de pureté :99.16% - 99.84%Couleur et forme :SolidMasse moléculaire :284.24Raxatrigine hydrochloride
CAS :<p>Raxatrigine hydrochloride is a state-dependent sodium channel blocker and a Nav1.7 sodium channel inhibitor.</p>Formule :C18H20ClFN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :350.82Rostafuroxin
CAS :<p>Rostafuroxin (PST 2238) has been used in trials studying the treatment of Essential Hypertension.</p>Formule :C23H34O4Degré de pureté :99.08% - >99.99%Couleur et forme :SolidMasse moléculaire :374.51CX614
CAS :<p>CX614 is a positive allosteric modulator of the AMPA receptor concerning AMPA.</p>Formule :C13H13NO4Degré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :247.25Benzonatate
CAS :<p>Benzonatate is an antagonist of sodium channel protein.</p>Formule :C30H53NO11Degré de pureté :99.92%Couleur et forme :Colorless To Faintly Yellow Oil LiquidMasse moléculaire :603.74Miltirone
CAS :<p>Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.</p>Formule :C19H22O2Degré de pureté :99.22% - 99.66%Couleur et forme :SolidMasse moléculaire :282.38Aptiganel hydrochloride
CAS :<p>Aptiganel hydrochloride（Cerestat） is the salt form of Aptiganel.Aptiganel is a non-competitive NMDA antagonist with neuroprotective effects used in the treatment of stroke and focal cerebral ischemia.</p>Formule :C20H22ClN3Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :339.86KPT276
CAS :<p>KPT276 (KPT 276) is an orally bioavailable selective inhibitor of nuclear export (SINE) that irreversibly bind to CRM1 and block the function of CRM1.</p>Formule :C16H10F8N4ODegré de pureté :99.89% - >99.99%Couleur et forme :SolidMasse moléculaire :426.26Tariquidar dihydrochloride
CAS :<p>Tariquidar dihydrochloride, also known as XR9576 dihydrochloride, is a potent, specific P-glycoprotein (P-gp) inhibitor exhibiting high affinity (Kd = 5.1 nM).</p>Formule :C38H40Cl2N4O6Couleur et forme :SolidMasse moléculaire :719.65NBQX
CAS :<p>NBQX (FG9202) is a potent, selective and competitive AMPA receptor antagonist. Neuroprotective and anticonvulsant; active in vivo.</p>Formule :C12H8N4O6SDegré de pureté :97.66% - 99.42%Couleur et forme :SolidMasse moléculaire :336.28Etripamil
CAS :<p>Etripamil is a fast-acting intranasal L-type calcium-channel blocker for Paroxysmal Supraventricular Tachycardia.</p>Formule :C27H36N2O4Degré de pureté :99.47% - 99.83%Couleur et forme :SolidMasse moléculaire :452.59Kv2-IN-A1
CAS :<p>Kv2-IN-A1 is an inhibitor of Kv2.1 and Kv2.2.</p>Formule :C20H17ClN4OSDegré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :396.89Triclabendazole sulfoxide
CAS :<p>TCBZ-SO, a Triclabendazole metabolite, blocks ABCG2/BCRP and has anti-parasitic properties.</p>Formule :C14H9Cl3N2O2SDegré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :375.66CFTR(inh)-172
CAS :<p>CFTR(inh)-172 (CFTR Inhibitor-172) is a voltage-independent, selective CFTR inhibitor.</p>Formule :C18H10F3NO3S2Degré de pureté :98% - 99.72%Couleur et forme :SolidMasse moléculaire :409.4Lansoprazole sulfone
CAS :<p>Lansoprazole sulfone is a metabolite of the gastric pump inhibitor Lansoprazole.</p>Formule :C16H14F3N3O3SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :385.36Tiagabine
CAS :<p>Tiagabine (NO050328) is an Anti-epileptic Agent.</p>Formule :C20H25NO2S2Degré de pureté :99.25%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :375.55Ginsenoside Rc
CAS :<p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>Formule :C53H90O22Degré de pureté :98.83% - 99.56%Couleur et forme :White PowderMasse moléculaire :1079.27Tirofiban hydrochloride monohydrate
CAS :<p>Tirofiban（MK383） hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.</p>Formule :C22H39ClN2O6SDegré de pureté :98.81% - >99.99%Couleur et forme :White SolidMasse moléculaire :495.07Phe-Met-Arg-Phe, amide acetate
<p>Phe-Met-Arg-Phe amide acetate (ED50=23 nM) triggers K+ current in caudodorsal neurons, co-localizes with neuropeptide Y in brain areas.</p>Formule :C31H46N8O6SDegré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :658.82Levosimendan
CAS :<p>Levosimendan (OR1259) is a calcium sensitizer for acute heart failure, enhancing cardiac contractility without raising calcium levels.</p>Formule :C14H12N6ODegré de pureté :99.37% - 99.91%Couleur et forme :Yellow Crystalline PowderMasse moléculaire :280.28Chloroprocaine
CAS :<p>Chloroprocaine: Na,K-ATPase inhibitor, IC50=13 mM, local anesthetic.</p>Formule :C13H19ClN2O2Couleur et forme :SolidMasse moléculaire :270.76AZD7325
CAS :<p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>Formule :C19H19FN4O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :354.38Ocinaplon
CAS :<p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>Formule :C17H11N5ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :301.3Esomeprazole
CAS :<p>Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.</p>Formule :C17H19N3O3SDegré de pureté :97.3%Couleur et forme :SolidMasse moléculaire :345.42Esomeprazole potassium salt
CAS :<p>Esomeprazole potassium, a potent oral proton pump inhibitor, curbs acid secretion in stomach cells, aiding GERD research.</p>Formule :C17H18KN3O3SCouleur et forme :SolidMasse moléculaire :383.51SAR7334 hydrochloride
CAS :<p>SAR7334 hydrochloride is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>Formule :C21H24Cl3N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.79Imidazenil
CAS :<p>Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.</p>Formule :C18H12BrFN4ODegré de pureté :98.4%Couleur et forme :SolidMasse moléculaire :399.22Pikamilone
CAS :<p>Pikamilone (Picamilon) is an intelligent medicine.</p>Formule :C10H12N2O3Degré de pureté :99.38%Couleur et forme :White Crystalline PowderMasse moléculaire :208.21Nisoxetine
CAS :<p>Nisoxetine is a selective NET (noradrenaline transporter) inhibitor (Kd=0.76 nM) capable of blocking voltage-gated sodium channels.</p>Formule :C17H21NO2Couleur et forme :SolidMasse moléculaire :271.35Pipequaline hydrochloride
CAS :<p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.</p>Formule :C22H25ClN2Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :352.9Flupirtine
CAS :<p>Flupirtine(D 9998) is a selective neuronal potassium channel opener as well as shows properties of NMDA receptor antagonist.</p>Formule :C15H17FN4O2Couleur et forme :SolidMasse moléculaire :304.32Icenticaftor
CAS :<p>Icenticaftor (QBW251) is an orally active potentiator of CFTR channel.</p>Formule :C12H13F6N3O3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :361.24KCNQ2/3 activator-1
CAS :<p>KCNQ2/3 activator-1 is a Kv7.2/Kv7.3 (KCNQ2/3) potassium channel activator.</p>Formule :C23H29FN2ODegré de pureté :99.16% - 99.47%Couleur et forme :SolidMasse moléculaire :368.49Rimtuzalcap
CAS :<p>Rimtuzalcap (CAD-1883), a selective modulator for SK channels, may treat movement disorders like SCA and ET.</p>Formule :C18H24F2N6ODegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :378.42Raxatrigine
CAS :<p>Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.</p>Formule :C18H19FN2O2Degré de pureté :98% - 99.43%Couleur et forme :SolidMasse moléculaire :314.35Nateglinide
CAS :<p>Nateglinide is an oral drug for type 2 diabetes, stimulating insulin release; may cause rare acute liver injury.</p>Formule :C19H27NO3Degré de pureté :99.93% - 99.94%Couleur et forme :White Crystalline PowderMasse moléculaire :317.42Gabazine free base
CAS :<p>Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.</p>Formule :C15H17N3O3Couleur et forme :SolidMasse moléculaire :287.31N-Me-aminopyrimidinone9
CAS :<p>N-Me-aminopyrimidinone9 is a sodium channel antagonist</p>Formule :C16H21N3OSDegré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :303.42GMQ hydrochloride
CAS :<p>GMQ hydrochloride, a potent ASIC modulator, activates ASIC3 at neutral pH and inhibits acid-induced peak current.</p>Formule :C10H12ClN5Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :237.692'-O-Methylisoliquiritigenin
CAS :<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Formule :C16H14O4Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :270.28Linerixibat
CAS :<p>Linerixibat (GSK2330672) is a highly effective, nonabsorbable ASBT inhibitor. Linerixibat can lower glucose in an animal model of type 2 diabetes.</p>Formule :C28H38N2O7SDegré de pureté :98.5% - 99.98%Couleur et forme :SolidMasse moléculaire :546.68Benzamil
CAS :<p>Benzamil blocks ENaC, inhibiting sodium transport (IC50=4 nM) and binds with Kd=5 nM to bovine kidney membranes.</p>Formule :C13H14ClN7ODegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :319.75ML329
CAS :<p>ML329 is a small molecule inhibitor of MITF, inhibiting TRPM-1 promoter activity.</p>Formule :C16H12N2O4SDegré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :328.34Acetoxyvalerensre
CAS :<p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>Formule :C17H24O4Degré de pureté :98.22%Couleur et forme :SolidMasse moléculaire :292.37DQP 1105
CAS :<p>DQP 1105 is a NMDA receptor antagonist.</p>Formule :C29H24BrN3O4Degré de pureté :98.6%Couleur et forme :SolidMasse moléculaire :558.42Piperazine
CAS :<p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>Formule :C4H10N2Couleur et forme :SolidMasse moléculaire :86.14UBP551
CAS :<p>UBP551 is a potent and selective NMDA receptors modulator.</p>Formule :C11H8O4Degré de pureté :98.69%Couleur et forme :SolidMasse moléculaire :204.18Omecamtiv mecarbil
CAS :<p>Omecamtiv mecarbil (CK-1827452) has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic</p>Formule :C20H24FN5O3Degré de pureté :98% - 99.23%Couleur et forme :SolidMasse moléculaire :401.43VU0134992
CAS :<p>VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μM</p>Formule :C20H31BrN2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :411.38Disopyramide phosphate
CAS :<p>Disopyramide: Class 1a anti-arrhythmic, treats Ventricular Tachycardia, reduces heart muscle contractility.</p>Formule :C21H32N3O5PCouleur et forme :SolidMasse moléculaire :437.47Acamprosate calcium
CAS :<p>Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.</p>Formule :C10H20CaN2O8S2Degré de pureté :98% - 99.93%Couleur et forme :White Odorless Or Nearly Odorless PowderMasse moléculaire :400.48GSK369796 Dihydrochloride
CAS :<p>GSK369796 Dihydrochloride (N-tert-butylisoquine),is an anti-malaria drug candidate.</p>Formule :C20H24Cl3N3ODegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :428.78Blebbistatin
CAS :<p>Blebbistatin ((±)-Blebbistatin) is a non-muscle myosin II (NMII)-selective and non-muscle myosin heavy chain 9 (MYH9)-specific inhibitor.Cost-effective and quality-assured.</p>Formule :C18H16N2O2Degré de pureté :99.88% - 99.97%Couleur et forme :Bright Yellow SolidMasse moléculaire :292.33TRPM8 antagonist WS-3
CAS :<p>TRPM8 antagonist WS-3 (Cyclohexanecarboxamide) is an agonist of TRPM8( EC50 : 3.7 μM).</p>Formule :C13H25NODegré de pureté :97.64%Couleur et forme :DrypowderMasse moléculaire :211.34VU6036720 hydrochloride
<p>VU6036720 hydrochloride inhibits Kir4.1/5.1. channels with 0.24 μM IC50; used in brain and kidney research.</p>Formule :C20H23Cl2FN4O2SCouleur et forme :SolidMasse moléculaire :473.39ML204
CAS :<p>ML204 is a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels.</p>Formule :C15H18N2Degré de pureté :98.1% - 99.72%Couleur et forme :SolidMasse moléculaire :226.32Afloqualone
CAS :<p>Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.</p>Formule :C16H14FN3ODegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :283.3α-Cyano-4-hydroxycinnamic acid
CAS :<p>α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) (α-CHCA) is an inhibitor of monocarboxylate transporter 1 (MCT1) that blocks pyruvate</p>Formule :C10H7NO3Degré de pureté :99.8% - 99.86%Couleur et forme :PowderMasse moléculaire :189.17BRITE-338733
CAS :<p>BRITE-338733 is a novel inhibitor of ATPase. BRITE 338733 inhibits the expression of RecA in bacteria (IC50=4.7 μM) for the bacterial infections treatment.</p>Formule :C27H35N3O2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :433.59Iptakalim Hydrochloride
CAS :<p>Iptakalim, a lipophilic para-amino compound, is a novel ATP-sensitive potassium channel (KATP) opener, as well as an α4β2-containing nicotinic acetylcholine</p>Formule :C9H22ClNDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :179.731IDRA-21
CAS :<p>IDRA-21 is a positive AMPA receptor modulator.</p>Formule :C8H9ClN2O2SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :232.69Temgicoluril
CAS :<p>Temgicoluril (mebikar) acts on GABA Receptor.</p>Formule :C8H14N4O2Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :198.22DL-Menthol
CAS :<p>DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.</p>Formule :C10H20ODegré de pureté :99.74%Couleur et forme :White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Masse moléculaire :156.27AMG 517
CAS :<p>AMG 517 is an effective and specific TRPV1 antagonist, antagonizes proton (IC50: 0.76 nM), capsaicin (IC50: 0.62 nM) and heat activation (IC50: 1.3 nM) of TRPV1</p>Formule :C20H13F3N4O2SDegré de pureté :99.77% - 99.85%Couleur et forme :SolidMasse moléculaire :430.4SN 2
CAS :<p>SN 2 is a novel and potent TRPML3 ion channel activator(EC50 = 1.13 μM). SN 2 also shares a similar antiviral effect against DENV2 and ZIKV.</p>Formule :C17H21NODegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :255.35CCTA-1523
CAS :<p>CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.</p>Formule :C16H15Cl2NO3Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :340.2YHO-13177
CAS :<p>YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells.</p>Formule :C20H22N2O3SDegré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :370.475,7-Dichlorokynurenic acid
CAS :<p>5,7-Dichlorokynurenic acid (5,7-dichlorokynurenic acid sodium) is an NMDA receptor antagonist.</p>Formule :C10H5Cl2NO3Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :258.06Songorine
CAS :<p>Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.</p>Formule :C22H31NO3Degré de pureté :98% - 99.92%Couleur et forme :SolidMasse moléculaire :357.49Vanilloid receptor antagonist 1
CAS :<p>Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.</p>Formule :C18H15N3O2Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :305.33Loreclezole
CAS :<p>Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.</p>Formule :C10H6Cl3N3Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :274.53KM 91104
CAS :<p>KM 91104 is a cell permeable inhibitor of V-ATPase. KM91104 specifically targets the interaction between V-ATPase subunit A3 and subunit B2.</p>Formule :C14H12N2O4Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :272.26Kavain
CAS :<p>Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation of</p>Formule :C14H14O3Degré de pureté :99.93% - ≥95%Couleur et forme :SolidMasse moléculaire :230.26AUT1
CAS :<p>AUT1 (AUT-1) is a novel specific modulator of Kv3 channels (EC50: 4.7 and 4.9 uM for Kv3.1b and Kv3.2a).</p>Formule :C18H19N3O4Degré de pureté :99.8% - 99.95%Couleur et forme :SolidMasse moléculaire :341.36Evifacotrep
CAS :<p>Evifacotrep: TRPC5 antagonist for neurological disease research (WO2020061162, compound 100).</p>Formule :C18H12ClF4N5O2Degré de pureté :98.6%Couleur et forme :SolidMasse moléculaire :441.77Guanidinoethyl sulfonate
CAS :<p>Guanidinoethyl sulfonate (Taurocyamine) is a competitive glycine receptor antagonist.</p>Formule :C3H9N3O3SDegré de pureté :99.43% - 99.47%Couleur et forme :SolidMasse moléculaire :167.19λ-Cyhalothrin
CAS :<p>λ-Cyhalothrin (Icon) is a type II synthetic pyrethroid insecticide featuring a high-efficiency, broad-spectrum formula with an α-cyano group.</p>Formule :C23H19ClF3NO3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :449.85AM92016
CAS :<p>AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.</p>Formule :C26H30Cl2N2O6SCouleur et forme :SolidMasse moléculaire :569.49RN-1734
CAS :<p>RN-1734 is selective TRPV4 channel antagonist(IC50 of 2.3 μM,5.9 μM,3.2 μM for hTRPV4, mTRPV4 and rTRPV4,respectively)</p>Formule :C14H22Cl2N2O2SDegré de pureté :99.1% - 99.3%Couleur et forme :SolidMasse moléculaire :353.31Esomeprazole magnesium salt
CAS :<p>Esomeprazole magnesium, an oral proton pump inhibitor, curbs gastric acid by blocking H+, K+-ATPase; used in treating GERD.</p>Formule :C17H21MgN3O3SCouleur et forme :SolidMasse moléculaire :371.74Cyclothiazide
CAS :<p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>Formule :C14H16ClN3O4S2Degré de pureté :98.23% - 99.49%Couleur et forme :Crystals From Dilute Alcohol SolidMasse moléculaire :389.88Eperisone hydrochloride
CAS :<p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>Formule :C17H26ClNODegré de pureté :99.80%Couleur et forme :White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter TasteMasse moléculaire :295.85SKA-31
CAS :<p>SKA-31 (Naphtho[1,2-d]thiazol-2-ylamine) is an activator of KCa3.1 and KCa2 channels (EC50s: 260, 2900, 2900 nM for KCa3.1, KCa2.1 and KCa2.2 respectively).</p>Formule :C11H8N2SDegré de pureté :99.38%Couleur et forme :SolidMasse moléculaire :200.26NBI-98782
CAS :<p>NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM)</p>Formule :C19H29NO3Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :319.44Ilaprazole sodium
CAS :<p>Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.</p>Formule :C19H17N4NaO2SDegré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :388.42Cis-ACBD
CAS :<p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>Formule :C6H9NO4Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :159.14Guan-fu base A hydrochloride(1394-48-5 free base)
CAS :<p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>Formule :C24H32NO6ClDegré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :465.97XEN907
CAS :<p>XEN907 is a novel spiro oxindole NaV1.7 blocker. XEN907 also inhibits hNaV1.7 (IC50: 3 nM).</p>Formule :C21H21NO4Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :351.4Quadrol
CAS :<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Formule :C14H32N2O4Degré de pureté :99.91% - 99.92%Couleur et forme :Viscous Liquid Liquid ViscousMasse moléculaire :292.41S107
CAS :<p>S107 stabilizes RyR2 by improving calstabin2 binding to mutant/PKA-phosphorylated channels.</p>Formule :C11H15NOSDegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :209.31RY785
CAS :<p>RY785 is a potent and selective inhibitor of voltage-gated potassium channel such as KV2.2 (IC50 = 50 nM). RY785 may be used in pain relief studies.</p>Formule :C21H20N4O2SDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :392.47Vanillyl butyl ether
CAS :<p>Vanillyl butyl ether (Butyl vanillyl ether) (VBE)is a capsaicin analogue,induce sensory irritation in humans,Vanillyl butyl ether is an alkoxy-substituted</p>Formule :C12H18O3Degré de pureté :99.57%Couleur et forme :Yellowish Liquid LiquidMasse moléculaire :210.27Rbin-1
CAS :<p>Rbin-1 (Ribozinoindole-1) is a potent,specific inhibitor of eukaryotic ribosome biogenesis.</p>Formule :C13H12N4SDegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :256.33Epaminurad
CAS :<p>Epaminurad (UR-1102) is an oral URAT1 inhibitor for gout research with a Ki of 0.057 μM, modestly affects OAT1/3.</p>Formule :C14H10Br2N2O3Couleur et forme :SolidMasse moléculaire :414.05Parimifasor
CAS :<p>Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.</p>Formule :C18H11Cl2F4N5ODegré de pureté :96.77% - 98.97%Couleur et forme :SolidMasse moléculaire :460.21DL-Willardiine
CAS :<p>DL-Willardiine (2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid) is an unnatural amino acid, a derivative of glutamate.</p>Formule :C7H9N3O4Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :199.16A2793
CAS :<p>A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.</p>Formule :C13H12ClNO3Degré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :265.69HC067047 Hydrochloride(883031-03-6 free base)
CAS :<p>HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.</p>Formule :C26H29ClF3N3O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :507.98Dotinurad
CAS :<p>Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).</p>Formule :C14H9Cl2NO4SDegré de pureté :97.43% - 98.04%Couleur et forme :SolidMasse moléculaire :358.2CTP disodium dihydrate
CAS :<p>CTP disodium dihydrate is an agonist of P2X4 purinergic receptor</p>Formule :C9H18N3Na2O16P3Degré de pureté :98.51%Couleur et forme :White Crystalline PowderMasse moléculaire :563.15PAP-1
CAS :<p>PAP-1 (5-(4-Phenoxybutoxy)psoralen) is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).</p>Formule :C21H18O5Degré de pureté :99.35% - 99.75%Couleur et forme :White SolidMasse moléculaire :350.36Levcromakalim
CAS :<p>Levcromakalim (BRL 38227) is an activator of the ATP-sensitive K+ channel.</p>Formule :C16H18N2O3Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :286.33ML213
CAS :<p>ML213 (CID-3111211) is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM,</p>Formule :C17H23NODegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :257.37YHO-13351
CAS :<p>YHO-13351 is an ABCG2 inhibitor that induces sensitization of cancer stem cells/initiating-like side population cells to irinotecan.</p>Formule :C27H37N3O7S2Degré de pureté :97.88%Couleur et forme :SolidMasse moléculaire :579.73DL-AP5
CAS :<p>DL-AP5 is the racemic form of a selective N-methyl-D-aspartate (NMDA) receptor antagonist with anticonvulsant effects.</p>Formule :C5H12NO5PDegré de pureté :99.33%Couleur et forme :White Fine Crystalline PowderMasse moléculaire :197.13Pico145
CAS :<p>Pico145 (HC-608) is a remarkable inhibitor of TRPC1/4/5 channels.</p>Formule :C23H20ClF3N4O5Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :524.88rac-BHFF
CAS :<p>rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.</p>Formule :C17H21F3O3Degré de pureté :99.69% - >99.99%Couleur et forme :SolidMasse moléculaire :330.34Lomerizine
CAS :<p>Lomerizine, a blocker of diphenylmethylpiperazine Ca2+ channel, is used to prevent migraines.</p>Formule :C27H30F2N2O3Couleur et forme :SolidMasse moléculaire :468.54Flupirtine maleate
CAS :<p>Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.</p>Formule :C15H17FN4O2·C4H4O4Degré de pureté :99.5% - 99.9%Couleur et forme :Off-White Crystalline PowderMasse moléculaire :420.39Selinexor (KPT-330)
CAS :<p>Selinexor (KPT-330) is an orally available, small molecule inhibitor of CRM1 (exportin 1 or XPO1), with potential antineoplastic activity.</p>Formule :C17H11F6N7ODegré de pureté :98% - 99.97%Couleur et forme :SolidMasse moléculaire :443.31TRPM4-IN-1
CAS :<p>TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.</p>Formule :C15H11Cl2NO4Degré de pureté :97.22%Couleur et forme :SolidMasse moléculaire :340.16(S)-(-)-5-Fluorowillardiine hydrochloride
CAS :<p>(S)-(-)-5-Fluorowillardiine hydrochloride is a potent and specific agonist of AMPAR.</p>Formule :C7H9ClFN3O4Couleur et forme :SolidMasse moléculaire :253.62Unifiram
CAS :<p>Unifiram boosts cognition, enhances rat hippocampal signals (EC50=27 nM), and ups ACh in rat cortex.</p>Formule :C13H15FN2O3SDegré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :298.33Tricaine methanesulfonate
CAS :<p>Tricaine methanesulfonate (TMS/MS-222) is an anesthetic used in hatcheries and studies to immobilize fish for marking, transport, and invasive procedures.</p>Formule :C10H15NO5SDegré de pureté :99.259% - 99.86%Couleur et forme :White PowderMasse moléculaire :261.30Methyl homoveratrate
CAS :<p>Methyl homoveratrate, a McN5691 (RWJ-26240) metabolite detected in vivo in plasma, urine, and fecal extracts, functions as a voltage-sensitive calcium channel</p>Formule :C11H14O4Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :210.23SSD114 HCl
CAS :<p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>Formule :C18H21ClF3N3ODegré de pureté :99.03% - 99.95%Couleur et forme :SolidMasse moléculaire :387.83BzATP triethylammonium salt
CAS :<p>BzATP triethylammonium salt is a P2X7 receptor agonist.</p>Formule :C30H39N6O15P3Degré de pureté :95% - 99.57%Couleur et forme :SolidMasse moléculaire :816.59MK6-83
CAS :<p>MK6-83 is the transient receptor potential channel ML3 agonist.</p>Formule :C16H20N2O2S2Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :336.479-Phenanthrol
CAS :<p>9-Phenanthrol is inhibitor of the transient receptor potential melastatin 4 (TRPM) channel, a Ca2+ -activated non-selective cation channel.</p>Formule :C14H10ODegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :194.23Amifampridine phosphate
CAS :<p>Amifampridine treats rare muscle diseases like LEMS and congenital myasthenias, targeting specific enzyme defects.</p>Formule :C5H10N3O4PCouleur et forme :SolidMasse moléculaire :207.12O4I1
CAS :<p>O4I1 is an effective Oct3/4 inducer.</p>Formule :C16H15NO2Degré de pureté :96.25% - 99.47%Couleur et forme :SolidMasse moléculaire :253.3Sepimostat dimethanesulfonate
CAS :<p>Sepimostat dimethanesulfonate (FUT-187) is a neuroprotective NR2B receptor antagonist with an inhibition Ki of 27.7 μM.</p>Formule :C23H27N5O8S2Couleur et forme :SolidMasse moléculaire :565.62Quinine hydrobromide
CAS :<p>Quinidine: oral, selective P450db inhibitor, K+ channel blocker (IC50=19.9μM), antiarrhythmic, used in malaria research.</p>Formule :C20H25BrN2O2Couleur et forme :SolidMasse moléculaire :405.336ICA-121431
CAS :<p>ICA-121431: a potent Nav1.7 inhibitor (IC50=19 nM for rat), minimal effect on human Nav1.5/Nav1.7.</p>Formule :C23H19N3O3S2Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :449.55Vonoprazan
CAS :<p>Vonoprazan (TAK-438 (free base)) is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduodenal ulcer and</p>Formule :C17H16FN3O2SDegré de pureté :99.87% - 99.92%Couleur et forme :SolidMasse moléculaire :345.39Eniporide hydrochloride
CAS :<p>Eniporide hydrochloride (EMD-96785 hydrochloride) serves as a robust inhibitor of the sodium/hydrogen (Na+/H+) exchange process.</p>Formule :C14H17ClN4O3SCouleur et forme :SolidMasse moléculaire :356.83Selamectin
CAS :<p>Selamectin (UK-124114) is a macrocyclic lactone derivative of ivermectin, an anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening in</p>Formule :C43H63NO11Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :769.96Esomeprazole hemistrontium
CAS :<p>Esomeprazole hemistrontium, potent oral proton pump inhibitor, reduces gastric acid by blocking H+, K+-ATPase.</p>Formule :C34H36N6O6S2SrCouleur et forme :SolidMasse moléculaire :776.44Ononetin
CAS :<p>Ononetin (2',4'-Dihydroxy-2-(4-methoxyphenyl)acetophenone) is a TRPM3 channel blocker(IC50: 0.3 μM).</p>Formule :C15H14O4Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :258.27NPPB
CAS :<p>NPPB is a chloride channel blocker with IC50 of 80 nM .</p>Formule :C16H16N2O4Degré de pureté :99.95%Couleur et forme :Light Yellow To Yellow SolidMasse moléculaire :300.31Flecainide acetate
CAS :<p>Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).</p>Formule :C19H24F6N2O5Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :474.39Ivacaftor
CAS :<p>Ivacaftor (VX-770) (VX-770) is a potentiator of CFTR targeting G551D-CFTR (EC50: 100 nM) and F508del-CFTR (EC50: 25 nM) in Fisher rat thyroid cells,</p>Formule :C24H28N2O3Degré de pureté :99% - 99.98%Couleur et forme :SolidMasse moléculaire :392.494-Acetamidobutanoic acid
CAS :<p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>Formule :C6H11NO3Degré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :145.16Azumolene sodium anhydrous
CAS :<p>Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.</p>Formule :C13H8BrN4NaO3Couleur et forme :SolidMasse moléculaire :371.13Myomodulin acetate(110570-93-9 free base)
<p>Myomodulin acetate is present in two identified aplysia neurons that contain myomodulin A the ARC motor neuron B16 and the abdominal neuron L10.</p>Formule :C38H71N11O10S2Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :906.17NS6180
CAS :<p>NS6180 is a potent and selective KCa3.1 channel inhibitor(IC50= 9 nM). It prevents T-cell activation and inflammation.</p>Formule :C16H12F3NOSDegré de pureté :99.83% - ≥95%Couleur et forme :SolidMasse moléculaire :323.33Azimilide Dihydrochloride
CAS :<p>Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the IKs and IKr with antiarrhythmic activity.</p>Formule :C23H30Cl3N5O3Degré de pureté :97.59% - ≥95%Couleur et forme :SolidMasse moléculaire :530.88RQ-00203078
CAS :<p>RQ-00203078 is a highly selective, potent and orally available TRPM8 antagonist.</p>Formule :C21H13ClF6N2O5SDegré de pureté :98% - 99.6%Couleur et forme :SolidMasse moléculaire :554.85Jujuboside A
CAS :<p>Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.</p>Formule :C58H94O26Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :1207.35Amlodipine mesylate
CAS :<p>Amlodipine mesylate, an oral dihydropyridine Ca2+ blocker, treats angina, hypertension, and may be used in cancer research.</p>Formule :C21H29ClN2O8SCouleur et forme :SolidMasse moléculaire :504.98DS-1971a
CAS :<p>DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.</p>Formule :C20H21ClFN5O3SDegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :465.93Flecainide hydrochloride
CAS :<p>Flecainide is a medication used to prevent and treat abnormally fast heart rates. This includes ventricular and supraventricular tachycardias.</p>Formule :C17H21ClF6N2O3Degré de pureté :97.79%Couleur et forme :SolidMasse moléculaire :450.81Rufinamide
CAS :<p>Rufinamide (E 2080), a triazole derivative, is used as voltage-gated sodium channel blocker for the treatment of seizure disorders.</p>Formule :C10H8F2N4ODegré de pureté :99.77% - >99.99%Couleur et forme :White PowderMasse moléculaire :238.19Ibutilide Fumarate
CAS :<p>Ibutilide Fumarate is a class III antiarrhythmic, prolonging action potentials by enhancing sodium influx, and can extend QT interval.</p>Formule :(C20H36N2O3S)2·C4H4O4Degré de pureté :99.68% - 99.74%Couleur et forme :SolidMasse moléculaire :885.23TRAM-34
CAS :<p>TRAM-34 (Triarylmethane-34), an effective and specific inhibitor of the intermediate-conductance Ca2+-activated K+ channel, does not block cytochrome P450.</p>Formule :C22H17ClN2Degré de pureté :99.01% - 99.91%Couleur et forme :SolidMasse moléculaire :344.84Ko 143
CAS :<p>Ko 143 is a selective inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2; BCRP).</p>Formule :C26H35N3O5Degré de pureté :99.01% - 99.89%Couleur et forme :SolidMasse moléculaire :469.57Chloroprocaine hydrochloride
CAS :<p>Chloroprocaine hydrochloride (Chloroprocaine HCl) is a local anesthetic during surgical procedures.</p>Formule :C13H20Cl2N2O2Degré de pureté :99.65%Couleur et forme :White Crystalline PowderMasse moléculaire :307.22BAY-8002
CAS :<p>BAY-8002 is a potent dual MCT1/2 inhibitor (IC50 values are 3, 8, and 12 nM at rat (C6), human (DLD-1) and mouse (4T1) MCT1 respectively).</p>Formule :C20H14ClNO5SDegré de pureté :98.7% - 99.13%Couleur et forme :SolidMasse moléculaire :415.85Ropivacaine hydrochloride monohydrate
CAS :<p>Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.</p>Formule :C17H29ClN2O2Degré de pureté :99.94% - 99.95%Couleur et forme :White SolidMasse moléculaire :328.88Tetraethylammonium chloride
CAS :<p>Tetraethylammonium chloride is a quaternary ammonium compound.</p>Formule :C8H20ClNDegré de pureté :≥95%Couleur et forme :White Solid Solid Particulate/PowderMasse moléculaire :165.7Ro 25-6981 Maleate
CAS :<p>Ro 25-6981 Maleate is an NMDA receptor antagonist used in the study of neurological disorders such as Parkinson's and epilepsy.</p>Formule :C26H33NO6Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :455.54JNJ-28583113
CAS :<p>JNJ-28583113 is a TRPM2 antagonist, inducing phosphorylation of GSK3α and β subunits, protecting cells from oxidative stress-induced cell death.</p>Formule :C19H21F3N2O2Degré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :366.38SRI-41315
CAS :<p>SRI-41315 is an eRF1 degrader that acts as a molecular glue at the ribosomal decoding center.SRI-41315 induces extended pauses at the termination codon.</p>Formule :C22H19N3O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :357.41Riluzole
CAS :<p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>Formule :C8H5F3N2OSDegré de pureté :99.71% - 99.88%Couleur et forme :PowderMasse moléculaire :234.2Doxapram
CAS :<p>Doxapram (Dopram) is a respiratory stimulant that inhibits TASK-1, TASK-3, and TASK-1/TASK-3 heterodimer channels.</p>Formule :C24H30N2O2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :378.51Darigabat
CAS :<p>Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.</p>Formule :C22H21FN4O3SDegré de pureté :98.42% - 99.29%Couleur et forme :SolidMasse moléculaire :440.49Methionine
CAS :<p>Methionine (D-Methionine) (MRX-1024; D-Methionine) is an effective chemoprotective agent which can also inhibit the neuronal activity through GABAA receptor</p>Formule :C5H11NO2SDegré de pureté :99.13% - 99.62%Couleur et forme :SolidMasse moléculaire :149.21BL-1249
CAS :<p>BL-1249 is a selective and potent non-steroidal potassium channel activator with anti-inflammatory activity that activates K2P2.1 (TREK-1) and K2P10.1 (TREK-2).</p>Formule :C17H17N5Degré de pureté :98% - 98.25%Couleur et forme :SolidMasse moléculaire :291.35VU590
CAS :<p>VU590 is an inhibitor of extrarenal medullary potassium ROMK.VU590 inhibits Kir7.1 and modulates uterine myometrial contractility and melanocortin signalling.</p>Formule :C24H32N4O7Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :488.53Bupivacaine
CAS :<p>Bupivacaine (AH-250) is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels</p>Formule :C18H28N2ODegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :288.43Dimiracetam
CAS :<p>Dimiracetam, a NMDA-receptor antagonist, is used potentially for the treatment of neuropathic pain.</p>Formule :C6H8N2O2Degré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :140.14ZT-1a
CAS :<p>ZT-1a is a SPAK inhibitor.ZT-1a inhibits SPAK.ZT-1a can be used for the prevention and treatment of neurodegenerative and neurocognitive disorders.</p>Formule :C22H15Cl3N2O2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :445.73Safinamide
CAS :<p>Safinamide: reversible MAO-B inhibitor, enhances dopamine, blocks glutamate release, sodium, calcium channels; may treat Parkinson's, RLS, epilepsy.</p>Formule :C17H19FN2O2Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :302.34Apinocaltamide
CAS :<p>Apinocaltamide (ACT-709478) is an orally available and selective T-type calcium channel blocker that cross BBB for Cav3.1, Cav3.2, and Cav3.3,epilepsy.</p>Formule :C22H18F3N5ODegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :425.41Lanicemine dihydrochloride
CAS :<p>Lanicemine dihydrochloride (AZD-6765 dihydrochloride) is an NMDA channel blocker with antidepressant activity and can be used to study neurological diseases.</p>Formule :C13H16Cl2N2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :271.19HUP30
CAS :<p>HUP30 is a potent vasodilating agent. HUP30 can stimulate soluble guanylyl cyclase, activate K+ channels, and block extracellular Ca2+ influx.</p>Formule :C14H15N3O3SDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :305.35N-Methyl-L-leucin
CAS :<p>N-Methyl-L-leucine ((S)-4-Methyl-2-(methylamino)pentanoic acid) is a novel calcium channel antagonist used in pain research.</p>Formule :C7H15NO2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :145.2CX717
CAS :<p>CX 717 is a positive allosteric modulator of AMPA receptor which has an antidepressant-like effect.</p>Formule :C11H11N3O3Degré de pureté :99.81%Couleur et forme :SoildMasse moléculaire :233.23Mtb ATP synthase-IN-1
CAS :<p>Mtb ATP synthase-IN-1 is a potent, low-toxicity M. tuberculosis inhibitor with good oral bioavailability and metabolic stability.</p>Formule :C17H13N3O4Degré de pureté :98.28%Couleur et forme :SolidMasse moléculaire :323.30VB124
CAS :<p>VB124 is an orally active, potent and selective MCT4 inhibitor. VB124 blocked lactate importand expor in MDA-MB-231 cells.Cost-effective and quality-assured.</p>Formule :C23H23ClN2O4Degré de pureté :99.21% - 99.57%Couleur et forme :SoildMasse moléculaire :426.89PF 03716556
CAS :<p>PF 03716556 (PF-3716556) , an effective and specific P-CAB (potassium-competitive acid blocker), is utilized for the treatment of gastroesophageal reflux</p>Formule :C22H26N4O3Degré de pureté :99.79% - 99.85%Couleur et forme :SolidMasse moléculaire :394.47Propoxycaine hydrochloride
CAS :<p>Propoxycaine hydrochloride is an ester local anesthetic that inhibits voltage-gated sodium channels, modulates nerve impulses, and induces loss of sensation.</p>Formule :C16H27ClN2O3Degré de pureté :97.25%Couleur et forme :SolidMasse moléculaire :330.85Bupivacaine-d9
CAS :<p>Bupivacaine-d9 is a deuterated compound of Bupivacaine. Bupivacaine has a CAS number of 38396-39-3. Bupivacaine is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels with the IC50 of 69.5 μM. Bupivacaine can be used for the research of chronic pain.</p>Formule :C18H19D9N2OCouleur et forme :SolidMasse moléculaire :297.48SAR7334
CAS :<p>SAR7334 (TRCP6-IN-1) is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>Formule :C21H22ClN3ODegré de pureté :99.62% - 99.71%Couleur et forme :SolidMasse moléculaire :367.87Eleclazine
CAS :<p>Eleclazine (GS-6615) is a novel and selective voltage-gated sodium channel inhibitor with antiarrhythmic properties that reduces peak sodium current (INaP).</p>Formule :C21H16F3N3O3Degré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :415.37MCT-IN-1
CAS :<p>MCT-IN-1 (compound 2) acts as a potent inhibitor of the monocarboxylate transporter (MCT), demonstrating IC50 values of 9 nM for MCT1 and 14 nM for MCT4.</p>Formule :C19H26N2O3Couleur et forme :SolidMasse moléculaire :330.42Eperisone
CAS :<p>Eperisone: a muscle relaxant for stiffness and pain, relaxes muscles, improves circulation, and mitigates pain by inhibiting reflexes and vasodilation.</p>Formule :C17H25NOCouleur et forme :SolidMasse moléculaire :259.39Flavoxate
CAS :<p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>Formule :C24H25NO4Couleur et forme :SolidMasse moléculaire :391.46VGSC blocker-1
CAS :<p>VGSC blocker-1 inhibits 34.9% INa in nNav1.5 at 1 μM, reduces MDA-MB-231 invasion by 0.3%, non-toxic.</p>Formule :C24H32F2N2Couleur et forme :SolidMasse moléculaire :386.52FSC231
CAS :<p>FSC231 is a PICK1 inhibitor with analgesic activity, activating GSK-3β and ERK1/2.</p>Formule :C13H10Cl2N2O3Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :313.14Amlodipine besilate impurity G
CAS :<p>Amlodipine besilate impurity G is a Calcium Channel antagonist with potential application in the study of neurological diseases and is an impurity in the</p>Formule :C17H18ClNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :335.78Cinepazide
CAS :<p>Cinepazide: a vasodilator targeting adenosine A2 receptors, treats various vascular diseases.</p>Formule :C22H31N3O5Couleur et forme :White PowderMasse moléculaire :417.5Amlodipine hydrochloride
CAS :<p>Amlodipine hydrochloride is a salt of Amlodipine --- a medication used to lower blood pressure and prevent chest pain.</p>Formule :C20H26Cl2N2O5Couleur et forme :SolidMasse moléculaire :445.34PBFI-AM
CAS :<p>PBFI-AM is a useful tool to determine intracellular K + content [1] .</p>Formule :C58H62N2O24Couleur et forme :SolidMasse moléculaire :1171.11Methocarbamol D5
CAS :<p>Methocarbamol is a central muscle relaxant. Methocarbamol D5 is deuterium labeled Methocarbamol.</p>Formule :C11H15NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :246.27Topiramate D12
CAS :<p>Topiramate D12 is a deuterium labeled Topiramate. Topiramate is an agent of broad-spectrum antiepileptic. Topiramate is an antagonist of GluR5 receptor.</p>Formule :C12H21NO8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :351.44Propafenone D7 hydrochloride
CAS :<p>Propafenone D7 hydrochloride is the deuterium labeled Propafenone, and is a classic anti-arrhythmic medication.</p>Formule :C21H28ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :384.95Repaglinide D5
CAS :<p>Repaglinide D5 is deuterium labeled Repaglinide. Repaglinide is an insulin secretagogue for treatment type-2 diabetes mellitus.</p>Formule :C27H36N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :457.62Nifedipine-d6
CAS :<p>Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel.</p>Formule :C17H18N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.37BAY-390
CAS :<p>BAY-390, a selective TRPA1 inhibitor, crosses species, penetrates brains, with IC50s: 16-82 nM. Used in inflammation research.</p>Formule :C13H15F4NOCouleur et forme :SolidMasse moléculaire :277.26Dofetilide D4
CAS :<p>Dofetilide D4 (UK 68789 D4), a deuterium-labeled version of Dofetilide, is categorized as a Class III antiarrhythmic medication.</p>Formule :C19H27N3O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :445.59Bumetanide-d5
CAS :<p>Bumetanide D5 is a deuterium-labeled Bumetanide. Bumetanide is a Na+-K+-Cl- (NKCC1) inhibitor (IC50s: 0.68 and 4.0 μM for hNKCC1A and hNKCC2A).</p>Formule :C17H20N2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :369.45FFN 511 hydrochloride
CAS :<p>FFN 511 hydrochloride is a fluorescent pseudo-neurotransmitter (FFNs) targeting VMA T2 that can be used to label baraminergic nerve endings.</p>Formule :C17H21ClN2O2Degré de pureté :99.83%Couleur et forme :SoildMasse moléculaire :320.81ORM-10103
CAS :<p>ORM-10103 is a novel potent and selective inhibitor of the Na+/Ca2+ exchanger (NCX).ORM-10103 inhibited NCX currents with estimated IC50 values of 55 and 67 nM</p>Formule :C20H16N2O4Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :348.35MNI-caged-NMDA
CAS :<p>NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group</p>Formule :C14H17N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :323.30Tetradifon
CAS :<p>Tetradifon is a broad-spectrum organochlorine acaricide that inhibits mitochondrial OSCP, blocking energy production (IC50=4.5-27nmoL/mg) with oligomycin-like effects.</p>Formule :C12H6Cl4O2SDegré de pureté :99.84%Couleur et forme :Yellowish Odorless OilMasse moléculaire :356.05A-317491 sodium salt hydrate
<p>A-317491 sodium salt hydrate is a non-nucleotide P2X3 and P2X2/3 receptor antagonist, which inhibits calcium flux mediated by the receptors.</p>Formule :C33H29NNaO9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :606.57Diphenidol
CAS :<p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>Formule :C21H27NOCouleur et forme :Needles From Petroleum Ether SolidMasse moléculaire :309.45DL-AP7
CAS :<p>DL-AP7: competitive NMDA antagonist, anticonvulsant, inhibits NMDA convulsions, impairs mice learning.</p>Formule :C7H16NO5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :225.18LY 303511
CAS :<p>LY303511, an inactive analogue of LY294002, is a mTOR inhibitor and no inhibition for PI3-K.</p>Formule :C19H18N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :306.36
