
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.834 produits)
- Apoptose(6.315 produits)
- Cycle cellulaire/point de contrôle(4.878 produits)
- Chromatine/Épigénétique(2.613 produits)
- Signalisation du cytosquelette(1.568 produits)
- Altération de l'ADN/réparation de l'ADN(2.871 produits)
- Endocrinologie/Hormones(3.754 produits)
- Enzyme(3.672 produits)
- GPCR/G-Protéine(9.021 produits)
- Immunologie et Inflammation(3.904 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(415 produits)
- Signalisation MAPK(1.258 produits)
- Transporteur membranaire/Canal ionique(3.157 produits)
- Métabolisme(10.131 produits)
- Microbiologie/Virologie(7.620 produits)
- Neuroscience(10.484 produits)
- Autres inhibiteurs(35.844 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.429 produits)
- Protéases/Protéasome(1.689 produits)
- Cellules souche et Dérivés(731 produits)
- Tyrosine Kinase/Adaptateurs(1.982 produits)
- Ubiquitination(1.726 produits)
Affichez 16 plus de sous-catégories
66514 produits trouvés pour "Inhibiteurs"
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Ramosetron
CAS :Ramosetron 是一种血清素 5-HT3 受体拮抗剂,用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。Formule :C17H17N3ODegré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :279.34Echinatin
CAS :Echinatin (Retrochalcone) is a natural chalcone. Echinatin has hepatoprotective and anti-inflammatory effects. Cost effective and quality assured.Formule :C16H14O4Degré de pureté :97.13% - 99.61%Couleur et forme :SolidMasse moléculaire :270.28Ref: TM-T3926
1mg34,00€5mg66,00€1mL*10mM (DMSO)69,00€10mg105,00€25mg157,00€50mg225,00€100mg333,00€500mg797,00€KU-0060648
CAS :KU-0060648 is a dual inhibitor of DNA-PK and PI3Kα, PI3Kβ, PI3Kδ with IC50 of 8.6 nM and 4 nM, 0.5 nM, 0.1 nM respectively, less inhibition of PI3Kγ.Formule :C33H34N4O4SDegré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :582.71Oct3/4-inducer-1
CAS :Oct3/4-inducer-1 (2-(4-(4-methoxybenzyloxy)phenyl)acetonitrile) is an OCT3/4 inducer that promotes the expression and stabilization of OCT3/4.Formule :C15H12FNODegré de pureté :97.42% - ≥98%Couleur et forme :SolidMasse moléculaire :241.26Ref: TM-T3221
1mg34,00€5mg71,00€1mL*10mM (DMSO)77,00€10mg112,00€25mg200,00€50mg290,00€100mg404,00€200mg545,00€Disodium succinate
CAS :Disodium succinate is a sodium salt of succinate, key in metabolism and reactive oxygen species regulation.Formule :C4H4Na2O4Degré de pureté :97.162%Couleur et forme :White Solid Crystalline PowderMasse moléculaire :162.05MCU-i4
CAS :MCU-i4 is a novel negative modulator of the MCU, binding MICU1 and impairing muscle cell growth.Formule :C23H27N3O2Degré de pureté :99.45% - 99.98%Couleur et forme :SolidMasse moléculaire :377.48ML239
CAS :ML239 (CID-49843203) is a potent and selective inhibitor of breast cancer stem cells, with an IC50 of 1.16 μM.Formule :C13H10Cl3N3O2Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :346.6Nardosinone
CAS :Nardosinone inhibits H9c2 cell hypertrophy, protects neurons from OGD, and boosts neurite outgrowth by modifying key signaling pathways.Formule :C15H22O3Degré de pureté :98.82% - 99%Couleur et forme :SolidMasse moléculaire :250.33Leuphasyl TFA
CAS :Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.Formule :C31H40F3N5O9Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :683.67CPI-455 analogue
CAS :CPI-455 analogue (CPI-455 analogue) is an analogue of CPI-455 which is a KDM5 inhibitor.Formule :C16H14N4ODegré de pureté :98% - 98.13%Couleur et forme :SolidMasse moléculaire :278.31Lanreotide acetate
CAS :Lanreotide acetate (BIM 23014 acetate) is a somatostatin analogue with antineoplastic activity, used for carcinoid syndromeFormule :C56H73N11O12S2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1156.39Cinchonain Ib
CAS :Cinchonain Ib is isolated from Eriobotrya japonica leaves.Formule :C24H20O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :452.41Wnt-C59
CAS :Wnt-C59 (C59)(C59) is a highly effective and specific Wnt signaling antagonis with PORCN enzymatic activity.Formule :C25H21N3ODegré de pureté :99.56% - 99.95%Couleur et forme :SolidMasse moléculaire :379.45Flavopiridol hydrochloride
CAS :Flavopiridol hydrochloride (MDL 107826A), an inhibitor of cyclin-dependent kinase, is a synthetic N-methylpiperidinyl chlorophenyl flavone compound.Formule :C21H21Cl2NO5Degré de pureté :98.87% - 99.88%Couleur et forme :SolidMasse moléculaire :438.3PRT4165
CAS :PRT4165 (NSC600157) is a potent PRC1-mediated H2A ubiquitylation inhibitor.Formule :C15H9NO2Degré de pureté :98.91% - 99.6%Couleur et forme :SolidMasse moléculaire :235.24Ref: TM-T3110
5mg43,00€10mg49,00€1mL*10mM (DMSO)50,00€25mg88,00€50mg112,00€100mg182,00€200mg254,00€500mg427,00€Talampanel
CAS :Talampanel (LY-300164), an oral selective AMPA receptor antagonist, exhibits anti-seizure and neuroprotective properties.Formule :C19H19N3O3Degré de pureté :98.3%Couleur et forme :SolidMasse moléculaire :337.37KML29
CAS :KML29 is highly selective and effective monoacylglycerol lipase (MAGL) inhibitor.Formule :C24H21F6NO7Degré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :549.42Ginsenoside Rb3
CAS :Ginsenoside Rb3 (Gypenoside IV) is a natural triterpenoid saponin, exhibiting inhibition effect on TNFα-induced NF-κB transcriptional activity.Formule :C53H90O22Degré de pureté :98% - 99.98%Couleur et forme :SolidMasse moléculaire :1079.27Ledipasvir hydrochloride
CAS :Ledipasvir hydrochloride, a hepatitis C NS5A inhibitor, has EC50 of 34 pM (1a) and 4 pM (1b), also inhibits SARS-CoV 3CL pro (IC50 1.62 µM).Formule :C49H55ClF2N8O6Couleur et forme :SolidMasse moléculaire :925.46Kanamycin sulfate
CAS :Kanamycin sulfate (Kanamycin monosulfate) is an aminoglycoside antibiotic. Kanamycin sulfate exhibits antimicrobial effect. Cost-effective and quality-assured.Formule :C18H38N4O15SDegré de pureté :99.63% - 99.96%Couleur et forme :Crystals From Methanol + Ethanol Off-White PowderMasse moléculaire :582.58Flumatinib mesylate
CAS :Flumatinib mesylate (HHGV678 mesylate) is a selective inhibitor of c-Abl, PDGFRβ and c-Kit, effectively overcomes drug resistance of certain KIT mutants.Formule :C30H33F3N8O4SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :658.69Ref: TM-T7861
1mg34,00€5mg84,00€10mg126,00€1mL*10mM (DMSO)132,00€25mg236,00€50mg371,00€100mg595,00€500mg1.234,00€Bay K 8644
CAS :Bay K 8644 (SQ 28,873) is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM.Formule :C16H15F3N2O4Degré de pureté :99.41%Couleur et forme :Yellow PowderMasse moléculaire :356.3Phe-Met-Arg-Phe, amide acetate
Phe-Met-Arg-Phe amide acetate (ED50=23 nM) triggers K+ current in caudodorsal neurons, co-localizes with neuropeptide Y in brain areas.Formule :C31H46N8O6SDegré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :658.82Clitorin
CAS :Clitorin has free radical scavenging property. It shows significant interactions with CD38, it may have anti-hyperglycemic potential.Formule :C33H40O19Degré de pureté :99.55% - 99.83%Couleur et forme :SolidMasse moléculaire :740.66Atorvastatin hemicalcium salt
CAS :Atorvastatin hemicalcium salt (Atorvastatin Calcium) is an orally HMG-CoA reductase inhibitor that lowers cholesterol. Cost-effective and quality-assured.Formule :C33H34FN2O5CaDegré de pureté :99.27% - >99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :577.67Pritelivir
CAS :Pritelivir (BAY 57-1293) (BAY 57-1293) is a potent helicase-primase inhibitor with active against HSV-1 and HSV-2 (IC50: 20 nM).Formule :C18H18N4O3S2Degré de pureté :97.96% - 99.42%Couleur et forme :SolidMasse moléculaire :402.492-Pyridylethylamine dihydrochloride
CAS :2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Formule :C7H12Cl2N2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :195.09Ayanin
CAS :Ayanin: a vasorelaxant with potential in allergic asthma treatment; IL-4 inhibition IC50 of 2.2µM; non-selective PDE1-4 inhibitor for respiratory research.Formule :C18H16O7Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :344.32Thiazovivin
CAS :Thiazovivin, a ROCK inhibitor (IC50: 0.5 μM), increases the survival rate of hESC.Formule :C15H13N5OSDegré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :311.36Ref: TM-T2155
1mg34,00€2mg46,00€5mg64,00€1mL*10mM (DMSO)70,00€10mg98,00€25mg180,00€50mg304,00€100mg444,00€Pimozide
CAS :Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.Formule :C28H29F2N3ODegré de pureté :99.63% - >99.99%Couleur et forme :SolidMasse moléculaire :461.55A-740003
CAS :A-740003 is a potent P2X7 receptor blocker, inhibiting rat/human receptors (IC50: 18/40 nM), lessens pain in animals, and shrinks mouse neuroblastoma.Formule :C26H30N6O3Degré de pureté :96.53% - 99.68%Couleur et forme :SolidMasse moléculaire :474.55Sacubitril hemicalcium salt
CAS :Sacubitril hemicalcium salt (AHU377 calcium salt) is a potent NEP inhibitor with an IC50 of 5 nM.Formule :C48H56CaN2O10Degré de pureté :99.86% - 99.93%Couleur et forme :SolidMasse moléculaire :861.06Ref: TM-T4200
2mg39,00€5mg52,00€10mg64,00€1mL*10mM (DMSO)64,00€25mg94,00€50mg106,00€100mg155,00€200mg207,00€Sophoridine
CAS :Sophoridine, a natural Chinese anticancer drug, has a potent derivative 6b targeting DNA topoisomerase I in tumor cells, inducing apoptosis.Formule :C15H24N2ODegré de pureté :97.33% - 99.28%Couleur et forme :SolidMasse moléculaire :248.36Terephthalic acid
CAS :Terephthalic acid, an isomer of the three phthalic acids, serves as a precursor to the polyester PET, which is utilized in manufacturing plastic bottles andFormule :C8H6O4Degré de pureté :99.63%Couleur et forme :White When Purified To The Grade Required For Use As A Polyester Feedstock These May Alter Flow CharacteristicsMasse moléculaire :166.13Ac4GalNAz
CAS :Ac4GalNAz is an alkyl chain-based PROTAC linker that can be used in PROTAC synthesis.Formule :C16H22N4O10Degré de pureté :98.31% - 99.95%Couleur et forme :SolidMasse moléculaire :430.37Astragaloside A
CAS :Astragaloside A, saponin from Astragalus membranaceus, treats cardiovascular diseases.Formule :C41H68O14Degré de pureté :99.87% - 99.94%Couleur et forme :White PowderMasse moléculaire :784.97Ref: TM-T6395
1mg40,00€2mg50,00€5mg64,00€10mg93,00€1mL*10mM (DMSO)93,00€25mg159,00€50mg230,00€100mg350,00€200mg530,00€500mg853,00€ML346
CAS :ML346 is a novel activator of Hsp70.Formule :C14H12N2O4Degré de pureté :97.32% - 99.36%Couleur et forme :SolidMasse moléculaire :272.26Ref: TM-T3594
1mg38,00€2mg50,00€5mg80,00€1mL*10mM (DMSO)80,00€10mg109,00€25mg168,00€50mg259,00€100mg405,00€500mg888,00€Cromoglicic acid
CAS :Cromoglicic acid prevents the release of inflammatory chemicals such as histamine from mast cells.
Formule :C23H16O11Degré de pureté :99.55% - >99.99%Couleur et forme :Colorless Crystals From Ethanol + Ether Physical Description Solid (Ntp 1992)Masse moléculaire :468.371-(3-chloropyridin-2-yl)piperazine 2HCl
CAS :1-(3-Chloropyridin-2-yl)piperazine dihydrochloride is a versatile piperazine used in synthesis, coordination chemistry, and as a DPP4 inhibitor drug.Formule :C9H14Cl3N3Degré de pureté :97.2%Couleur et forme :SolidMasse moléculaire :270.587cis-4-Hydroxy-L-proline
CAS :cis-4-Hydroxy-L-proline hinders collagen synthesis, extracellular deposition, and fibroblast growth.Formule :C5H9NO3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :131.132-Hydroxy-4-methylbenzaldehyde
CAS :2-Hydroxy-4-methylbenzaldehyde is a human endogenous metabolite.Formule :C8H8O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :136.15CEF4 acetate
CEF4 acetate (CEF4 acetate (199727-68-9 free base)) is a polypeptide corresponding to amino acid sequence 342-351 of the influenza A virus nucleocapsid protein.Formule :C55H97N15O15Degré de pureté :95.27%Couleur et forme :SolidMasse moléculaire :1208.45Torin 2
CAS :Torin 2: mTOR inhibitor, IC50=0.25 nM, 800x more selective than PI3K, with EC50=28/35/118 nM for ATM/ATR/DNA-PK.Formule :C24H15F3N4ODegré de pureté :98.31% - 99.32%Couleur et forme :SolidMasse moléculaire :432.4SB-734117
CAS :SB-734117 inhibits productive replication of several HCMV strains.Formule :C14H16N6ODegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :284.32Ref: TM-T9580
1mg109,00€1mL*10mM (DMSO)224,00€5mg235,00€10mg349,00€25mg532,00€50mg745,00€100mg999,00€200mg1.333,00€Sapanisertib
CAS :Sapanisertib (INK 128) is an oral raptor-mTOR and rictor-mTOR inhibitor with potential cancer-fighting properties.Formule :C15H15N7ODegré de pureté :99.19% - >99.99%Couleur et forme :SolidMasse moléculaire :309.33Ref: TM-T1838
1mg40,00€2mg51,00€5mg85,00€1mL*10mM (DMSO)88,00€10mg96,00€25mg160,00€50mg235,00€100mg350,00€500mg838,00€DIM-C-pPhOCH3
CAS :DIM-C-pPhOCH3 (C-DIM5) is a Nerve Growth Factor-Induced Bα (NGFI-Bα, Nur77) agonistFormule :C24H20N2ODegré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :352.43JNK-IN-8
CAS :JNK-IN-8 (JNK Inhibitor XVI) is an irreversible JNK1/2/4 inhibitor (IC50: 4.7/18.7/1 nM).Formule :C29H29N7O2Degré de pureté :99.24% - >99.99%Couleur et forme :SolidMasse moléculaire :507.59Ref: TM-T2668
2mg44,00€5mg73,00€1mL*10mM (DMSO)82,00€10mg113,00€25mg197,00€50mg326,00€100mg482,00€200mg685,00€JHU37160
CAS :JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for hM4Di, and EC50 of 18.5 nM (hM3Dq), 0.2 nM (hM4Di) in HEK-293 cell assays.Formule :C19H20ClFN4Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :358.84Thiazole Orange
CAS :Thiazole Orange is a dye that can be used for reticulocyte analysis.Formule :C26H24N2O3S2Degré de pureté :99.29% - 99.93%Couleur et forme :SolidMasse moléculaire :476.61DSRM-3716
CAS :Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery ofFormule :C9H6INDegré de pureté :97.28% - 99.785%Couleur et forme :SolidMasse moléculaire :255.06Debrisoquin hydriodide
CAS :Debrisoquin hydriodide is an organic antioxidant with potential for treating neurological issues like Parkinson's and depression.Formule :C10H14IN3Degré de pureté :99%Couleur et forme :SolidMasse moléculaire :303.14Resmetirom
CAS :Resmetirom (MGL-3196) is a THR-β agonist (EC50=0.21 μM), with high selectivity and oral activity. High-Quality, Low-Cost!Formule :C17H12Cl2N6O4Degré de pureté :99.05% - >99.99%Couleur et forme :SolidMasse moléculaire :435.22Ref: TM-T3595
1mg37,00€2mg49,00€1mL*10mM (DMSO)87,00€5mg93,00€10mg119,00€25mg202,00€50mg324,00€100mg482,00€500mg1.071,00€GSK2578215A
CAS :GSK2578215A is a potent and selective LRRK2 kinase inhibitor.Formule :C24H18FN3O2Degré de pureté :99.57% - 99.94%Couleur et forme :SolidMasse moléculaire :399.42Stigmasterol
CAS :Stigmasterol (Stigmasterin) is a phytosterol with a function in the maintenance of cell membranes. Stigmasterol lowers cholesterol levels. Cost-effective and quality-assured.Formule :C29H48ODegré de pureté :99.67% - 99.97%Couleur et forme :White SolidMasse moléculaire :412.69Otenabant
CAS :Otenabant (CP-945598) has been investigated for the treatment of Obesity.Formule :C25H25Cl2N7ODegré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :510.42Thonningianin A
CAS :Thonningianin A: an anti-cancer compound with antioxidant effects, GST inhibitor, and radical scavenger.Formule :C42H34O21Degré de pureté :98.37% - 99.94%Couleur et forme :SolidMasse moléculaire :874.71Ref: TM-T3S0218
1mg52,00€2mg67,00€5mg97,00€10mg160,00€1mL*10mM (DMSO)169,00€25mg263,00€50mg378,00€100mg568,00€Ginsenoside Rh1
CAS :Ginsenoside Rh1 (Sanchinoside B2) , one of the main constituents of Panax ginseng, exhibits anti-inflammatory effect.Formule :C36H62O9Degré de pureté :99% - 99.64%Couleur et forme :SolidMasse moléculaire :638.87HIV-1 Inhibitor 18A
CAS :HIV-1 Inhibitor 18A (HIV-1 Inhibitor-18A) specifically inhibits the entry of multiple HIV-1 isolates.Formule :C14H11N5O2SDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :313.33Ref: TM-T24141
1mg109,00€1mL*10mM (DMSO)207,00€5mg215,00€10mg296,00€25mg507,00€50mg712,00€100mg1.009,00€Riociguat
CAS :Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth muscle and is used to treat severe pulmonary arterialFormule :C20H19FN8O2Degré de pureté :99.28% - 99.95%Couleur et forme :SolidMasse moléculaire :422.42Proctolin
CAS :Proctolin is a bioactive neuropeptide that modulates interneuronal and neuromuscular synaptic transmission in a wide variety of arthropods.Formule :C30H48N8O8Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :648.75CTP disodium dihydrate
CAS :CTP disodium dihydrate is an agonist of P2X4 purinergic receptor
Formule :C9H18N3Na2O16P3Degré de pureté :98.51%Couleur et forme :White Crystalline PowderMasse moléculaire :563.15Lirinidine
CAS :(+)-Lirinidine shows antioxidative properties, inhibits melanoma and melanogenesis, and reduces collagen-related platelet aggregation.Formule :C18H19NO2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :281.35Neuropeptide S (Mouse) acetate
Neuropeptide S (Mouse) acetate is a bioactive peptide.Formule :C95H160N34O29Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :2242.5ARD-2128
CAS :ARD-2128: potent oral PROTAC that degrades AR, curbing prostate cancer growth with no toxicity.Formule :C45H50ClN7O6Degré de pureté :98.8%Couleur et forme :SolidMasse moléculaire :820.37NSC 405020
CAS :NSC 405020 is a noncatalytic inhibitor of MT1-MMP.Formule :C12H15Cl2NODegré de pureté :96.93% - 99.07%Couleur et forme :SolidMasse moléculaire :260.16Ralfinamide
CAS :Ralfinamide (Priralfinamide) is an orally available Na-channel blocker for the treatment of neuropathic pain and other pain conditions.Formule :C17H19FN2O2Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :302.34HeE1-2Tyr
CAS :HeE1-2Tyr, a pyridobenzothiazole, inhibits flavivirus RdRp including West Nile, Dengue, SARS-CoV-2 (IC50: 27.6 µM).Formule :C33H30N2O6SDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :582.67Tris(benzyltriazolylmethyl)amine
CAS :Tris(benzyltriazolylmethyl)amine (TBTA) is a tertiary amine. It complexes with, and stabilizes, copper(I) to accelerate azide-alkyne cycloadditions.Formule :C30H30N10Degré de pureté :99.58% - 99.82%Couleur et forme :SolidMasse moléculaire :530.63Hederacoside D
CAS :Hederacoside D is a bioactive saponins from Hedera helix.Formule :C53H86O22Degré de pureté :94.94% - 99.80%Couleur et forme :SolidMasse moléculaire :1075.24Vinorelbine ditartrate
CAS :Vinorelbine ditartrate (KW-2307) is a natural alkaloid and an anti-mitotic agent. Vinorelbine ditartrate has anti-tumor activity. Cost-effective and quality-assured.Formule :C45H54N4O8·2C4H6O6Degré de pureté :98% - 99.93%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :1079.11HEX3 acetate(688805-40-5 free base)
HEX3 acetate is a fragment of the adenoviral hexon. Hexon is the major capsid protein of adenovirion and is comprised of three identical polypeptide chains.Formule :C49H82N12O16Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :1095.26Quilseconazole
CAS :Quilseconazole is an effective, orally active fungal Cyp51 inhibitor. it also binds tightly to cryptococcal CYP51 but weakly inhibits humans CYP450 enzymes.Formule :C22H14F7N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :513.37Bromosporine
CAS :Bromosporine is a broad spectrum inhibitor for bromodomains for BRD2/4/9 and CECR2 (IC50: 0.41/0.29/0.122/0.017 μM), respectively.Formule :C17H20N6O4SDegré de pureté :99.65% - 99.79%Couleur et forme :SolidMasse moléculaire :404.44Ref: TM-T6255
1mg44,00€2mg57,00€1mL*10mM (DMSO)92,00€5mg93,00€10mg133,00€25mg260,00€50mg416,00€100mg665,00€200mg888,00€BDP-13176
CAS :BDP-13176 is a potent inhibitor of fascin 1(Kd of 90 nM and an IC50 of 240 nM). It has potential as an anti-metastatic agentFormule :C24H22Cl2N6O2Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :497.38IDO5L
CAS :IDO5L (INCB024360 analogue) is an effective IDO1 inhibitor(IC50=10 nM).Formule :C9H7ClFN5O2Degré de pureté :99.49% - 99.75%Couleur et forme :SolidMasse moléculaire :271.64Ref: TM-T2647
1mL*10mM (DMSO)35,00€10mg50,00€25mg86,00€50mg124,00€100mg187,00€200mg321,00€500mg505,00€Ellagic Acid Dihydrate
CAS :Ellagic Acid Dihydrate inhibit the CYP1A1-dependent activation of benzo[a]pyrene.Formule :C14H10O10Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :338.22Alizarin Cyanine Green F
CAS :Alizarin Cyanine Green F (NSC-41838) is an agent of green dye.Formule :C28H20N2Na2O8S2Degré de pureté :98%Couleur et forme :Dark Blue-Green Powder SolidMasse moléculaire :622.58Arctigenin
CAS :(-)-Arctigenin ((-)-Arctigenin) is found in burdock.Formule :C21H24O6Degré de pureté :98% - 99.51%Couleur et forme :SolidMasse moléculaire :372.41Pirozadil
CAS :Pirozadil shows hypolipidemic activity.Formule :C27H29NO10Degré de pureté :97.54% - 98.31%Couleur et forme :SolidMasse moléculaire :527.52Octreotide Acetate
CAS :Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.Formule :C51H70N10O12S2Degré de pureté :99.03% - 99.87%Couleur et forme :Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised SolidMasse moléculaire :1079.30ON123300
CAS :ON123300 is a potent and multi-targeted kinase inhibitor for CDK4/Ark5/PDGFRβ/FGFR1/RET/Fyn (IC50: 3.9/5/26/26/9.2/11 nM).Formule :C24H27N7ODegré de pureté :99.53% - 99.7%Couleur et forme :SolidMasse moléculaire :429.52SRI 31215 TFA
CAS :SRI 31215 TFA acts as a triplex inhibitor of matriptase, hepsin and HGFA and mimics the activity of HAI-1/2, endogenous inhibitors of HGF activation.Formule :C27H34F3N5O3Degré de pureté :98.25% - 99.97%Couleur et forme :SolidMasse moléculaire :533.6Ref: TM-T5478
1mg40,00€5mg92,00€1mL*10mM (DMSO)96,00€10mg128,00€25mg248,00€50mg370,00€100mg527,00€200mg713,00€Jujuboside A
CAS :Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Formule :C58H94O26Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :1207.35cangrelor tetrasodium
CAS :Cangrelor tetrasodium is a reversible and selective antagonist of platelet P2Y12, with prompt and potent antiplatelet effects.
Formule :C17H21Cl2F3N5Na4O12P3S2Degré de pureté :98.51% - 98.6%Couleur et forme :SolidMasse moléculaire :864.29dGTP
CAS :dGTP (2'-Deoxyguanosine-5'-triphosphate) is one of the guanosine nucleotides which is highly susceptible to oxidative damage to 8-O-GDP, 8-O-dGTP, 8-O-GTP, andFormule :C10H16N5O13P3Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :507.184-Methylsalicylic acid
CAS :4-Methylsalicylic acid is used to inhibit the medium chain acyl-CoA synthetase.Formule :C8H8O3Degré de pureté :99.64%Couleur et forme :Solid Solid CrystallineMasse moléculaire :152.15Osimertinib
CAS :Osimertinib (AZD-9291) is a small molecule tyrosine kinase receptor inhibitor and antineoplastic agent that is used in the therapy of selected forms of NSCLC.Formule :C28H33N7O2Degré de pureté :99.32% - >99.99%Couleur et forme :SolidMasse moléculaire :499.61Ref: TM-T2490
2mg34,00€5mg52,00€1mL*10mM (DMSO)52,00€10mg55,00€25mg67,00€50mg80,00€100mg94,00€500mg114,00€1g138,00€2g197,00€5g329,00€Methyl purple
CAS :Methyl purple is an introduced quinone-imide redox dye that has been shown to be an exceptionally sensitive monitor of photosystem I activity in chloroplasts.Formule :C24H32ClN3Degré de pureté :≥98%Couleur et forme :Dark Green PowderMasse moléculaire :397.99Syrosingopine
CAS :Syrosingopine is a dual inhibitor of MCT1 and MCT4, 60 times more potent against MCT4, preventing lactate and H+ efflux.Cost-effective and quality-assured.Formule :C35H42N2O11Degré de pureté :99.25% - 99.78%Couleur et forme :SolidMasse moléculaire :666.71Ref: TM-TN2252
1mg63,00€5mg135,00€1mL*10mM (DMSO)192,00€10mg200,00€25mg343,00€50mg515,00€100mg710,00€N2,N2-Dimethylguanosine
CAS :Urinary N2,N2-Dimethylguanosine levels higher in colorectal cancer than in villous adenoma or healthy adults.Formule :C12H17N5O5Degré de pureté :98.01%Couleur et forme :White SolidMasse moléculaire :311.29Triheptanoin
CAS :Triheptanoin (IND 106011) is a fatty acid metabolic modulator. It potentially for the treatment of fatty acid oxidation disorders and GLUT1.Formule :C24H44O6Degré de pureté :99.51%Couleur et forme :Colourless LiquidMasse moléculaire :428.6Thymine
CAS :Thymine: Derived from DNA hydrolysis or methylcyanoacetylurea, found in DNA (not RNA), binds adenine, used in biochemical research.Formule :C5H6N2O2Degré de pureté :99.77% - 99.97%Couleur et forme :SolidMasse moléculaire :126.11Stearic acid
CAS :Stearic acid reduces tumor load, cuts visceral fat, gels foods/pharma, boosts insulin signaling, and ups milk yield without weight impact.Formule :C18H36O2Degré de pureté :99.40% - 99.81%Couleur et forme :White Solid LeafletsMasse moléculaire :284.48WZ-3146
CAS :WZ3146: EGFR(L858R/E746_A750) inhibitor, IC50=2 nM, selective, doesn't block ERBB2(T798I).Formule :C24H25ClN6O2Degré de pureté :97.15%Couleur et forme :SolidMasse moléculaire :464.95Ref: TM-T6733
1mg50,00€2mg71,00€5mg92,00€1mL*10mM (DMSO)101,00€10mg170,00€25mg301,00€50mg484,00€100mg692,00€Verbenalin
CAS :Verbenalin (Verbenaloside) induces angiogenesis via a programmed PI3K/Akt/eNOS/VEGF signaling axis.Formule :C17H24O10Degré de pureté :98.81% - 99.88%Couleur et forme :Off-White PowderMasse moléculaire :388.37LOX-IN-3 dihydrochloride
CAS :LOX-IN-3 dihydrochloride is an inhibitor of lysyl oxidase (LOX).Formule :C13H15Cl2FN2O2SDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :353.24Ref: TM-T39986
1mg54,00€5mg114,00€1mL*10mM (DMSO)120,00€10mg178,00€25mg334,00€50mg557,00€100mg888,00€200mg1.251,00€Decursinol angelate
CAS :Decursinol angelate is anti-tumor, anti-inflammatory, anti-oxidant, hepatoprotective, and inhibits VEGF and cancer cell invasion.Formule :C19H20O5Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :328.36GW604714X
CAS :GW604714X (2,4-Thiazolidinedione, 5-[[5-[6-(4-acetyl-1-piperazinyl)-3-nitro-2-pyridinyl]-2-fluorophenyl]methylene]-) were found to be potent inhibitors ofFormule :C21H18FN5O5SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :471.46Rabeprazole Sulfide
CAS :Rabeprazole Sulfide (Rabeprazole Related Compound E) is an antiulcer drug in the class of proton pump inhibitors.Formule :C18H21N3O2SDegré de pureté :99.34% - 99.78%Couleur et forme :Off-White Crystalline PowderMasse moléculaire :343.44FMOC-L-1,2,3,4-TETRAHYDRONORHARMAN-3-CAR
CAS :Fmoc-Tpi-OH, a THN derivative, is used in synthesizing pharmaceuticals and agrochemicals.Formule :C27H22N2O4Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :438.47

