
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.519 produits)
- Apoptose(5.786 produits)
- Cycle cellulaire/point de contrôle(4.444 produits)
- Chromatine/Épigénétique(2.235 produits)
- Signalisation du cytosquelette(1.382 produits)
- Altération de l'ADN/réparation de l'ADN(2.823 produits)
- Endocrinologie/Hormones(3.499 produits)
- Enzyme(3.639 produits)
- GPCR/G-Protéine(8.314 produits)
- Immunologie et Inflammation(3.516 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(404 produits)
- Signalisation MAPK(1.199 produits)
- Transporteur membranaire/Canal ionique(2.786 produits)
- Métabolisme(9.417 produits)
- Microbiologie/Virologie(6.967 produits)
- Neuroscience(9.920 produits)
- Autres inhibiteurs(37.931 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.399 produits)
- Protéases/Protéasome(1.596 produits)
- Cellules souche et Dérivés(832 produits)
- Tyrosine Kinase/Adaptateurs(2.015 produits)
- Ubiquitination(1.646 produits)
Affichez 16 plus de sous-catégories
66627 produits trouvés pour "Inhibiteurs"
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GN44028
CAS :<p>GN44028 is a HIF-1 inhibitor with an IC50 of 14 nM, stopping HIF-1α activity but not mRNA or protein levels, or dimerization.</p>Formule :C18H15N3O2Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :305.33Roquinimex
CAS :<p>Roquinimex (FCF89) (Linomide) is a quinoline derivative immunostimulant which increases NK cell activity and macrophage cytotoxicity; inhibits angiogenesis and</p>Formule :C18H16N2O3Degré de pureté :97.69%Couleur et forme :SolidMasse moléculaire :308.33Adavosertib
CAS :<p>Adavosertib (MK-1775) is a small molecule inhibitor of the checkpoint kinase WEE1 (IC50: 5.2 nM). It hinders the G2 DNA damage checkpoint.</p>Formule :C27H32N8O2Degré de pureté :98.65% - 99.86%Couleur et forme :SolidMasse moléculaire :500.6Scutellarein
CAS :<p>Scutellarein (6-Hydroxyapigenin) reduces inflammatory responses by inhibiting Src kinase activity.</p>Formule :C15H10O6Degré de pureté :98.02% - 99.63%Couleur et forme :SolidMasse moléculaire :286.24OGT-IN-2
CAS :<p>OGT-IN-2: Potent OGT inhibitor, IC50: sOGT 30μM, ncOGT 53μM, for articular disease research.</p>Formule :C23H27ClN2O3SDegré de pureté :98.80%Couleur et forme :SolidMasse moléculaire :446.99Navoximod phosphate
CAS :<p>Navoximod phosphate is an indoleamine 2,3-dioxygenase (IDO) inhibitor, immunomodulator and antineoplastic.</p>Formule :C18H24FN2O6PCouleur et forme :SolidMasse moléculaire :414.37Mitiglinide calcium hydrate
CAS :<p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>Formule :C38H52CaN2O8Degré de pureté :98.97% - 99.96%Couleur et forme :White SolidMasse moléculaire :704.91Bisphenol A
CAS :<p>Bisphenol A: used in making polycarbonates/epoxy resins, has estrogen-like effects.</p>Formule :C15H16O2Degré de pureté :99.93%Couleur et forme :White Solid White Crystals Flakes PrillsMasse moléculaire :228.29Orientin
CAS :<p>1.</p>Formule :C21H20O11Degré de pureté :98.77% - 99.88%Couleur et forme :Yellow PowderMasse moléculaire :448.38α-calcium ketoglutarate monohydrate
CAS :<p>Alpha-calcium ketoglutarate monohydrate is the calcium salt form of Alpha-ketoglutarate, which is involved in the tricarboxylic acid cycle in organisms.</p>Formule :C5H6CaO6Degré de pureté :98.921%Couleur et forme :SolidMasse moléculaire :202.181-Methylguanidine hydrochloride
CAS :<p>MG derived from protein breakdown, may be toxic in renal failure but has anti-inflammatory properties, inhibiting iNOS and TNF- release.</p>Formule :C2H8ClN3Degré de pureté :98% - 99.02%Couleur et forme :CrystallineMasse moléculaire :109.56Phytic acid sodium salt
CAS :<p>Phytic acid sodium salt (Sodium phytate hydrate) functions as a [PO4]3- storage depot and a precursor for other inositol phosphates and pyrophosphates.</p>Formule :C6H18O24P6·xNaDegré de pureté :99.67%Couleur et forme :White Hygroscopic PowderMasse moléculaire :923.82Corn oil
CAS :<p>Corn oil is a kind of vegetable oil extracted from corn germ. Corn oil is mainly used as a carrier and solvent in scientific research. High-Quality, Low-Cost!</p>Degré de pureté :98%Couleur et forme :SolidHPI 1
CAS :<p>HPI 1 suppresses Hh pathway: IC50 = 1.5 μM (Shh, SAG), 4 μM (Gli2), 6 μM (Gli1) in Shh-LIGHT2 cells.</p>Formule :C27H29NO6Degré de pureté :97.6%Couleur et forme :SolidMasse moléculaire :463.52Gypsogenin
CAS :<p>Gypsogenin (639-14-5) is a naturally occurring biochemical that shows anti-ABL1 kinase and anti-chronic Myelogenous Leukemia activities.</p>Formule :C30H46O4Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :470.68Nimustine Hydrochloride
CAS :<p>Nimustine Hydrochloride (Nidran hydrochloride) has been used in trials studying the treatment of Glioblastoma.</p>Formule :C9H14Cl2N6O2Degré de pureté :98.80%Couleur et forme :SolidMasse moléculaire :309.15THPP-1
CAS :<p>THPP-1 is a potent and orally bioavailable inhibitor of PDE10A(Ki of 1 nM and 1.3 nM for human and rat PDE10A, respectively).</p>Formule :C23H21ClN6O3Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :464.9Trandolapril hydrochloride
CAS :<p>Trandolapril (RU44570) HCl, a non-mercapto prodrug for hypertension and heart issues, becomes active diacetyl form.</p>Formule :C24H35ClN2O5Couleur et forme :SolidMasse moléculaire :467.0Imperialine 3-β-D-glucoside
CAS :<p>Imperialine 3-β-D-glucoside (Sipeimine-3-beta-D-glucoside) is a natural product.</p>Formule :C33H53NO8Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :591.78[4-(4-phenylpiperazin-1-yl)oxan-4-yl]methanamine
CAS :<p>[4-(4-Phenylpiperazin-1-yl)oxan-4-yl]methanamine: A piperazine partial agonist for serotonin and dopamine, potential for treating depression/schizophrenia.</p>Formule :C16H25N3ODegré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :275.396"-O-Apiosyl-5-O-Methylvisammioside
CAS :<p>6”-O-Apiosyl-5-O-Methylvisammioside is one component of the traditional Chinese medicine Kang-Jing which has the functions of promoting blood circulation and</p>Formule :C27H36O14Degré de pureté :98% - 99.87%Couleur et forme :SolidMasse moléculaire :584.57BML-210
CAS :<p>BML-210 (CAY10433) is a new-type HDAC inhibitor.</p>Formule :C20H25N3O2Degré de pureté :96.37% - 98.12%Couleur et forme :SolidMasse moléculaire :339.43TAT-Gap19 acetate
<p>TAT-Gap19 acetate, a Cx43 HC inhibitor, crosses blood-brain barrier, reduces liver fibrosis in mice, and spares Cx43 GJCs.</p>Formule :C119H212N46O26Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :2703.25Vicriviroc
CAS :<p>Vicriviroc, also known as MK4176 is a CCR5 antagonist.</p>Formule :C28H38F3N5O2Couleur et forme :SolidMasse moléculaire :533.63Ipilimumab
CAS :<p>Ipilimumab (anti-CTLA-4) is an immunomodulatory monoclonal antibody directed against the cell surface antigen CTLA-4 and also a type of immune checkpoint</p>Degré de pureté :98.50% - 99.60%Couleur et forme :LiquidMasse moléculaire :148 kDa(+)-Isocorydine hydrochloride
CAS :<p>(+)-Isocorydine hydrochloride (Isocorydine HCl) is a eukaryote protein kinases Inhibitor.</p>Formule :C20H24ClNO4Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :377.873-hydroxycephem
CAS :<p>3-hydroxycephem is a useful organic compound for research related to life sciences. The catalog number is T4581 and the CAS number is 54639-48-4.</p>Formule :C28H24N2O5SDegré de pureté :98.74%Couleur et forme :White Or Off-White Crysalline PowderMasse moléculaire :500.572'-O-Methylisoliquiritigenin
CAS :<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Formule :C16H14O4Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :270.28Sultopride hydrochloride
CAS :<p>Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.</p>Formule :C17H27ClN2O4SDegré de pureté :≥95%Couleur et forme :White Or Yellowish PowderMasse moléculaire :390.93Avotaciclib trihydrochloride
CAS :<p>Avotaciclib trihydrochloride (BEY1107) is an oral CDK1 inhibitor targeting advanced pancreatic cancer.</p>Formule :C13H14Cl3N7ODegré de pureté :99%Couleur et forme :SolidMasse moléculaire :390.65LY 303511 hydrochloride
CAS :<p>LY 303511 hydrochloride is a potent mTOR inhibitor</p>Formule :C19H19ClN2O2Degré de pureté :98.47%Couleur et forme :SolidMasse moléculaire :342.82GSK621
CAS :<p>GSK621 is a specific and potent AMPK activator.</p>Formule :C26H20ClN3O5Degré de pureté :97.02% - 97.05%Couleur et forme :SolidMasse moléculaire :489.91Dehydrocostuslactone
CAS :<p>Dehydrocostuslactone, from Aucklandia, offers anti-inflammatory, anticancer, and more health benefits.</p>Formule :C15H18O2Degré de pureté :99.46% - 99.8%Couleur et forme :White PowderMasse moléculaire :230.3S 3304
CAS :<p>S 3304 is a novel matrix metalloproteinases inhibitor which is specific for MMP-2 and MMP-9.</p>Formule :C24H20N2O4S2Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :464.562-((9R,10S,11R,15S)-12,14-dioxo-9,10-dih
CAS :<p>Compound 8 can bind to GID1, By the results of the in vitro binding assays, chemical 8 showed greater effects than did 67D in an in vivo experimental system.</p>Formule :C24H23NO4Degré de pureté :97.82%Couleur et forme :SolidMasse moléculaire :389.44Isavuconazole
CAS :<p>Isavuconazole (RO-0094815) is an azole antifungal with MICs 0.002-0.5 mg/liter against C. albicans to C. glabrata.</p>Formule :C22H17F2N5OSDegré de pureté :99.74% - >99.99%Couleur et forme :SolidMasse moléculaire :437.47HZ-1157
CAS :<p>HZ-1157 (DHFR-inhibitor) is a hepatitis C virus (HCV) inhibitor with inhibitory activities toward HCV NS3/4A protease.</p>Formule :C12H16N4ODegré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :232.28GW4869
CAS :<p>GW4869 (GW69A) is a selective and non-competitive inhibitor of neutral sphingomyelinase N-SMase (IC50=1 μM).</p>Formule :C30H30Cl2N6O2Degré de pureté :98.12% - 98.47%Couleur et forme :SolidMasse moléculaire :577.5glatiramer Acetate
CAS :<p>GA: synthetic copolymer for RRMS and CIS treatment.</p>Formule :C25H45N5O13Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :623.65Metoclopramide
CAS :<p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>Formule :C14H22ClN3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :299.8010074-A4
CAS :<p>10074-A4 is a c-Myc binding compound that associates with c-Myc370–409 and behaves like a “ligand cloud” around a “protein cloud”, with distinct features from</p>Formule :C18H14Cl2N2O3SDegré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :409.29FMOC-3VVD-OH
CAS :<p>FMOC-3VVD-OH is an active chemical.</p>Formule :C36H51N3O7Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :637.81GSK-5959
CAS :<p>GSK-5959 is a selective BRPF1 inhibitor with IC50 ~80 nM, 100-fold more specific than 35 other bromodomains.</p>Formule :C22H26N4O3Degré de pureté :98.35% - 98.65%Couleur et forme :SolidMasse moléculaire :394.474-Carboxyquinoline
CAS :<p>4-Carboxyquinoline (4-Quinolinecarboxylic acid) showed anti-tumor activity against L1210 leukemia and B16 melanoma.</p>Formule :C10H7NO2Degré de pureté :99.46% - 99.69%Couleur et forme :White To Light Yellow Crystal PowderMasse moléculaire :173.17Trientine-2HCl
CAS :<p>Trientine-2HCl treats Wilson's disease by chelating copper; also stabilizes epoxy resins and aids in isoelectric focusing.</p>Formule :C6H20Cl2N4Degré de pureté :≥98%Couleur et forme :White Crystalline PowderMasse moléculaire :219.15Cryptotanshinone
CAS :<p>Cryptotanshinone: STAT3 inhibitor, IC50 4.6 μM; blocks STAT3 Tyr705 phosphorylation, minor effect on Ser727, no impact on STAT1/5.</p>Formule :C19H20O3Degré de pureté :97.94% - ≥95%Couleur et forme :Orange Needle CrystalMasse moléculaire :296.36Thioredoxin reductase peptide acetate
<p>Thioredoxin reductase peptide acetate, residues 53-67, aids TrxR research, similar to glutathione reductase but has a unique C-terminal selenylsulfide.</p>Formule :C68H110N18O20S2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :1563.84TBA-354
CAS :<p>TBA-354 is anti-tuberculous and active against Mycobacterium tuberculosis strain H37Rv.</p>Formule :C19H15F3N4O5Degré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :436.34VEGFR-2-IN-5
CAS :<p>VEGFR-2-IN-5 (UNC0064-12), multikinase inhibitor and has a -NH2 terminal linker for further synthesis.</p>Formule :C19H24N8Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :364.45Tat-NR2B9c acetate
<p>Tat-NR2B9c acetate inhibits PSD-95, NMDAR & nNOS interactions; EC50: 6.7 nM (PSD-95d2), 670 nM (d1); IC50: 0.5 μM (NR2A), 8 μM (NR2B); neuroprotective.</p>Formule :C107H192N42O32Degré de pureté :98.46%Couleur et forme :SolidMasse moléculaire :2578.93CRBN modulator-1
CAS :<p>CRBN modulator-1 (WUN29654) is a Thalidomide analog and CRBN modulator,has an IC50 of 3.5 μM and a Ki of 0.98 μM.</p>Formule :C17H12N2O5Degré de pureté :99.24% - 99.36%Couleur et forme :SolidMasse moléculaire :324.29SB-3CT
CAS :<p>SB-3CT is a potent and specific gelatinase inhibitor for MMP-2(Ki=13.9 nM) and MMP-9(Ki=600 nM).</p>Formule :C15H14O3S2Degré de pureté :98% - 99.38%Couleur et forme :SolidMasse moléculaire :306.4Enavogliflozin
CAS :<p>Enavogliflozin (DWP-16001) is an orally available small molecule and sodium glucose transporter 2 inhibitor.</p>Formule :C24H27ClO6Degré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :446.92AGK2
CAS :<p>AGK2(IC50=3.5 μM) is an effective, and specific SIRT2 inhibitor.</p>Formule :C23H13Cl2N3O2Degré de pureté :98.68% - 99.17%Couleur et forme :SolidMasse moléculaire :434.27(±)-Methyl Jasmonate
CAS :<p>Methyl 2-(3-oxo-2-(pent-2-en-1-yl)cyclopentyl)acetate ((±)-Jasmonic Acid methyl ester)induces the synthesis of proteinase inhibitors in plant leaves.</p>Formule :C13H20O3Degré de pureté :98.95% - 99.39%Couleur et forme :Colorless Liquid Clear To Pale Yellow LiquidMasse moléculaire :224.3MK-0557
CAS :<p>MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).</p>Formule :C22H19FN4O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :406.41SKF89976A hydrochloride
CAS :<p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>Formule :C22H26ClNO2Degré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :371.9Pomalidomide-C2-COOH
<p>Pomalidomide-C2-COOH: a synthetic E3 ligase linker for PROTAC, with CRBN-based Pomalidomide.</p>Formule :C16H15N3O6Degré de pureté :97.65%Couleur et forme :SolidMasse moléculaire :345.31Dexelvucitabine
CAS :<p>Dexelvucitabine (RVT), a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.</p>Formule :C9H10FN3O3Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :227.19Hemin
CAS :<p>Hemin (Hemin chloride) is a chlorinated iron-containing porphyrin, a heme oxygenase (HO)-1 inducer.</p>Formule :C34H32ClFeN4O4Degré de pureté :97.169% - 99.59%Couleur et forme :Dark Purple Crystalline PowderMasse moléculaire :651.94Boc-GABA-OH
CAS :<p>Boc-GABA-OH serves as a PROTAC linker essential for synthesizing UNC6852, an EED-targeted PROTAC[1].</p>Formule :C9H17NO4Degré de pureté :99%Couleur et forme :White Crystalline PowderMasse moléculaire :203.24Daclatasvir dihydrochloride
CAS :<p>Daclatasvir dihydrochloride is an oral antiviral that treats chronic hepatitis C by inhibiting HCV's NS5A; rare liver enzyme elevation, seldom causes jaundice.</p>Formule :C40H52Cl2N8O6Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :811.8BIBR 1532
CAS :<p>BIBR 1532 is an effective, specific and non-competitive telomerase inhibitor (IC50: 100 nM, in a cell-free assay).</p>Formule :C21H17NO3Degré de pureté :98.49% - 98.90%Couleur et forme :SolidMasse moléculaire :331.36AMD 3465 hexahydrobromide
CAS :<p>AMD 3465 hexahydrobromide (GENZ-644494 (hexahydrobromide)) is a CXCR4 receptor antagonist with potential anticancer and anti-HIV activity.</p>Formule :C24H44Br6N6Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :896.07Sudan IV
CAS :<p>Sudan IV (Solvent Red 24) is a lysochrome (fat-soluble dye) diazo dye used for the staining of triglycerides,lipids and lipoproteins on frozen paraffin sections</p>Formule :C24H20N4OCouleur et forme :Dark Red Solid PowderMasse moléculaire :380.44GSK2656157
CAS :<p>GSK2656157 is a highly specific and ATP-competitive PERK inhibitor (IC50: 0.9 nM) in a cell-free assay.</p>Formule :C23H21FN6ODegré de pureté :98.59% - >99.99%Couleur et forme :SolidMasse moléculaire :416.45Tussilagone
CAS :<p>Tussilagone has anti-cancer, anti-oxidant, anti-inflammatory effects and modulates dendritic cells, potentially treating colon cancer and neuro-inflammation.</p>Formule :C23H34O5Degré de pureté :98.17% - 99.63%Couleur et forme :SolidMasse moléculaire :390.51Dicyclanil
CAS :<p>Dicyclanil, a regulator of insect growth, is a veterinary medicine for the protection against early-season myiasis.</p>Formule :C8H10N6Degré de pureté :≥95%Couleur et forme :White Microcrystalline PowderMasse moléculaire :190.21Secoisolariciresinol
CAS :<p>Secoisolariciresinol is an enterolignan precursor, it has antioxidant, and estrogen-like activities, it can significantly suppress triglyceride (TG)</p>Formule :C20H26O6Degré de pureté :99.34% - 99.51%Couleur et forme :White PowderMasse moléculaire :362.42ω-Pentadecalactone
CAS :<p>ω-Pentadecalactone (Exaltolide) is the fragrance structural group macrocyclic lactone and lactide derivatives used as a fragrance ingredient.</p>Formule :C15H28O2Degré de pureté :98%Couleur et forme :Liquid OthersolidMasse moléculaire :240.38Feruloylputrescine
CAS :<p>Feruloylputrescine is a natural product.</p>Formule :C14H20N2O3Degré de pureté :97.7% - 99.71%Couleur et forme :SolidMasse moléculaire :264.32Esculentoside A
CAS :<p>Esculentoside A dampens inflammation in ALI, modulates T cells, and could treat autoimmune diseases and BXSB mice by adjusting cytokines and renal cells.</p>Formule :C42H66O16Degré de pureté :98% - 99.85%Couleur et forme :SolidMasse moléculaire :826.96Chrysosplenol D
CAS :<p>Chrysosplenol D, an efflux pump inhibitor that can potentiate the activity of commercially important antibiotics and antimalarials.</p>Formule :C18H16O8Degré de pureté :97.87% - 99.98%Couleur et forme :SolidMasse moléculaire :360.31Murrayone
CAS :<p>Murrayone from M. paniculata, a bioactive coumarin, prevents cancer metastasis and reduces ADP-induced platelet aggregation.</p>Formule :C15H14O4Degré de pureté :98.01% - 98.79%Couleur et forme :SolidMasse moléculaire :258.27[Sar9,Met(O2)11]-Substance P
CAS :<p>[Sar9,Met(O2)11]-Substance P (NA) is an agonist of NK1 receptor.</p>Formule :C64H100N18O15SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1393.66D-Mannose
CAS :<p>D-Mannose (D-(+)-Mannose) is a carbohydrate. D-Mannose plays an important role in human metabolism, especially in the glycosylation of specific proteins.</p>Formule :C6H12O6Degré de pureté :99.21% - 99.68%Couleur et forme :Colorless Crystals Or White Granular Powder With Water (Uscg 1999)Masse moléculaire :180.16Bis(maltolato)oxovanadium(IV)
CAS :<p>BMOV: oral pan-PTP inhibitor, mimics insulin, anti-diabetic, improves heart function in diabetes, IC50s: 126-201 nM.</p>Formule :C12H10O7VDegré de pureté :99.65% - 99.918%Couleur et forme :SolidMasse moléculaire :317.15WEE1-IN-3
CAS :<p>WEE1-IN-3 (JUN76288) is a potent Wee1 kinase inhibitor with an IC50 of <10 nM. It treatment of cancer and other proliferative diseases.</p>Formule :C28H31N7O2Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :497.59Telaprevir
CAS :<p>Telaprevir (Incivek) (VX-950) is an effective inhibitor of HCV NS3-4A serine protease (IC50: 0.35 μM).</p>Formule :C36H53N7O6Degré de pureté :96.9% - 98.89%Couleur et forme :SolidMasse moléculaire :679.85ELR510444
CAS :<p>ELR510444 (LR510444) is a novel microtubule disruptor; inhibits MDA-MB-231 cell proliferation with IC50 of 30.9 nM.</p>Formule :C19H16N2O2S2Degré de pureté :97.67% - 98.69%Couleur et forme :SolidMasse moléculaire :368.47Tetrahydropalmatine hydrochloride
CAS :<p>Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.</p>Formule :C21H26ClNO4Degré de pureté :98% - 99.59%Couleur et forme :SolidMasse moléculaire :391.888LY3200882
CAS :<p>LY3200882 is a highly selective inhibitor of TGF-β receptor type 1 (TGFβRI).</p>Formule :C24H29N5O3Degré de pureté :99.46% - 99.63%Couleur et forme :SolidMasse moléculaire :435.52GLPG2938
CAS :<p>GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent and</p>Formule :C20H19F6N7O2Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :503.4Columbianadin
CAS :<p>Columbianadin (Zosimin), one of the main bioactive constituents of the roots of Angelica pubescens Maxim.</p>Formule :C19H20O5Degré de pureté :98.44% - 99.48%Couleur et forme :SolidMasse moléculaire :328.36Geniposide
CAS :<p>Geniposide is an iridoid glycoside with a variety of biological activities including neuroprotective, anti-diabetic, antiproliferative, and antioxidative</p>Formule :C17H24O10Degré de pureté :99.17% - 99.54%Couleur et forme :SolidMasse moléculaire :388.37Diclofenac deanol
CAS :<p>Diclofenac deanol: a phenylacetic acid NSAID with anti-inflammatory, analgesic, and antipyretic effects; favors COX-2 inhibition.</p>Formule :C18H22Cl2N2O3Couleur et forme :SolidMasse moléculaire :385.29DG172 dihydrochloride
CAS :<p>DG172 dihydrochloride (DG-172 dihydrochloride) is an antagonist of PPARβ/δ(IC50 : 27 nM).</p>Formule :C20H22BrCl2N3Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :455.2Levobupivacaine hydrochloride
CAS :<p>Levobupivacaine hydrochloride ((S)-(-)-Bupivacaine monohydrochloride) is a reversible neuronal sodium channel inhibitor, used as a long-acting local anesthetic.</p>Formule :C18H28N2O·HClDegré de pureté :99.74%Couleur et forme :White Crystalline PowderMasse moléculaire :324.89XMD8-87
CAS :<p>XMD8-87 (ACK1-B19), a TNK2 inhibitor, strongly blocks TNK2 phosphorylation and mutations in tumors.</p>Formule :C24H27N7O2Degré de pureté :98.05% - 99.89%Couleur et forme :SolidMasse moléculaire :445.52Ionox 330
CAS :<p>Ionox 330 (Ahydol) is an alkylphenol compound used as an antioxidant.</p>Formule :C54H78O3Degré de pureté :99.95%Couleur et forme :White Solid PowderMasse moléculaire :775.203-hydroxy-phthalicanhydrid
CAS :<p>3-Hydroxyphthalic anhydride is used to synthesize 3-hydroxyphthalic anhydride modified human serum albumin.</p>Formule :C8H4O4Degré de pureté :99.53%Couleur et forme :Beige PowderMasse moléculaire :164.12WH-4-023
CAS :<p>WH-4-023 (Dual LCK/SRC inhibitor) is a potent and orally active Lck/Src inhibitor. It also potently inhibits SIK.</p>Formule :C32H36N6O4Degré de pureté :98% - 99.75%Couleur et forme :SolidMasse moléculaire :568.674,4'-DIMETHOXYBENZIL
CAS :<p>4,4'-Dimethoxybenzil (p-Anisil) is a human intestinal carboxyl esterase (hiCE) inhibitor( Ki : 70 nM).</p>Formule :C16H14O4Degré de pureté :99.04%Couleur et forme :Yellow Fine Crystalline PowderMasse moléculaire :270.28Pinealon Acetate
<p>Pinealon Acetategland has antioxidant activity and can directly interact with the cell genome.</p>Formule :C17H30N6O10Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :478.45Cynaroside
CAS :<p>Cynaroside (Luteolin 7-O-Glucoside) is a flavone, a flavonoid-like chemical compound. It has an anti-oxidant effect, inhibiting lipid and protein oxidation.</p>Formule :C21H20O11Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :448.38GSK2636771
CAS :<p>GSK2636771, an effective, specific, orally bioavailable, PI3Kβ inhibitor, has been used in cancer, lymphoma, solid neoplasm, recurrent solid neoplasm, and</p>Formule :C22H22F3N3O3Degré de pureté :98.58% - ≥95%Couleur et forme :SolidMasse moléculaire :433.42L-Propargylglycine
CAS :<p>L-Propargylglycine ((S)-Propargylglycine) is an inhibitor of the enzyme.</p>Formule :C5H7NO2Degré de pureté :99.63% - 99.83%Couleur et forme :White Crystalline PowderMasse moléculaire :113.11Platycodin D2
CAS :<p>Platycodin D2 enhances immune response to Hep B in mice with minimal hemolysis, acting as a safe Th1/Th2 adjuvant.</p>Formule :C63H102O33Degré de pureté :97.24%Couleur et forme :SolidMasse moléculaire :1387.46Broparestrol (E)-
CAS :<p>Broparestrol (E)- has antifertility activity and is a potent inhibitor of rodent mammary tumorigenesis.</p>Formule :C22H19BrDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :363.29Oxfenicine
CAS :<p>Oxfenicine, a 4-Hydroxy-L-phenylglycine, inhibits CPT-1, boosts glucose tolerance & insulin sensitivity in obese, insulin-resistant mice.</p>Formule :C8H9NO3Degré de pureté :99.22%Couleur et forme :White SolidMasse moléculaire :167.16
