
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.849 produits)
- Apoptose(6.366 produits)
- Cycle cellulaire/point de contrôle(4.907 produits)
- Chromatine/Épigénétique(2.623 produits)
- Signalisation du cytosquelette(1.585 produits)
- Altération de l'ADN/réparation de l'ADN(2.872 produits)
- Endocrinologie/Hormones(3.759 produits)
- Enzyme(3.673 produits)
- GPCR/G-Protéine(9.051 produits)
- Immunologie et Inflammation(3.945 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(417 produits)
- Signalisation MAPK(1.259 produits)
- Transporteur membranaire/Canal ionique(3.162 produits)
- Métabolisme(10.149 produits)
- Microbiologie/Virologie(7.672 produits)
- Neuroscience(10.549 produits)
- Autres inhibiteurs(35.857 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.435 produits)
- Protéases/Protéasome(1.693 produits)
- Cellules souche et Dérivés(734 produits)
- Tyrosine Kinase/Adaptateurs(1.991 produits)
- Ubiquitination(1.743 produits)
Affichez 16 plus de sous-catégories
66517 produits trouvés pour "Inhibiteurs"
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Menadione bisulfite sodium
CAS :Menadione bisulfite sodium (Vitamin K3 sodium bisulfite) is used clinically to treat diseases caused by vitamin K deficiency and as a vitamin K supplement.Formule :C11H9NaO5SDegré de pureté :99.67%Couleur et forme :Crystalline PowderMasse moléculaire :276.24Pentagastrin
CAS :Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis ofFormule :C37H49N7O9SDegré de pureté :96.98% - 99.49%Couleur et forme :Fine Colorless Needle-Shaped Crystals From 2-Ethoxyethanol + Water SolidMasse moléculaire :767.893-Hydroxybenzaldehyde
CAS :3-Hydroxybenzaldehyde is a compound useful in organic synthesis.Formule :C7H6O2Degré de pureté :99.60%Couleur et forme :DrypowderMasse moléculaire :122.12Fasiglifam
CAS :Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.Formule :C29H32O7SDegré de pureté :99.82% - 99.9%Couleur et forme :SolidMasse moléculaire :524.63Ref: TM-T2351
1mg49,00€5mg90,00€1mL*10mM (DMSO)116,00€10mg141,00€25mg236,00€50mg356,00€100mg522,00€200mg713,00€7,3',4'-Tri-O-methylluteolin
CAS :7,3',4'-Tri-O-methylluteolin is anti-inflammatory, antibacterial, antifungal, and has moderate antitrypanosomal effects (MIC 19.0 ug/ml).
Formule :C18H16O6Degré de pureté :98.66% - 99.79%Couleur et forme :SolidMasse moléculaire :328.32KDU691
CAS :KDU691 is a PI4K inhibitor.Formule :C22H18ClN5O2Degré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :419.86Hydroxypropyl Cellulose
CAS :Hydroxypropyl cellulose (HPC), soluble in water and organics, serves as a food additive and DNA separation aid.Formule :C12H20N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :192.306Iso-H7 dihydrochloride
CAS :Iso-H7 dihydrochloride is a less potent inhibitor of phosphokinase C than H-7.Formule :C14H19Cl2N3O2SDegré de pureté :99.53%Couleur et forme :White Crystalline SolidMasse moléculaire :364.29Isosinensetin
CAS :1. Isosinensetin (6-Demethoxynobiletin) shows antioxidant and HIV-1 protease inhibiting activities.Formule :C20H20O7Degré de pureté :99.98% - ≥95%Couleur et forme :SolidMasse moléculaire :372.37Ref: TM-T2S0223
1mg63,00€5mg135,00€1mL*10mM (DMSO)165,00€10mg195,00€25mg326,00€50mg485,00€100mg700,00€Almotriptan Malate
CAS :Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.Formule :C17H25N3O2S·C4H6O5Degré de pureté :99.95%Couleur et forme :Pale Yellow SolidMasse moléculaire :469.55GSK-J4 Hydrochloride
CAS :GSK-J4 Hydrochloride (GSK J4 HCl) is a cell permeable, potent and selective histone demethylase(JMJD3 )inhibitor. It is an ethyl ester derivative of the GSK-J1.Formule :C24H28ClN5O2Degré de pureté :97.95% - 98.23%Couleur et forme :SolidMasse moléculaire :453.97Ref: TM-T4383
1mg38,00€2mg50,00€5mg84,00€10mg120,00€1mL*10mM (DMSO)132,00€25mg207,00€50mg344,00€100mg505,00€200mg707,00€Piboserod hydrochloride
CAS :Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.Formule :C22H32ClN3O2Couleur et forme :SolidMasse moléculaire :405.96Batatasin III
CAS :Batatasin III inhibits cancer migration and invasion by suppressing epithelial to mesenchymal transition and FAK-AKT signals and possesses anti-cancerFormule :C15H16O3Degré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :244.29Nitrocaramiphen hydrochloride
CAS :Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.Formule :C18H27ClN2O4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :370.87λ-Cyhalothrin
CAS :λ-Cyhalothrin (Icon) is a type II synthetic pyrethroid insecticide featuring a high-efficiency, broad-spectrum formula with an α-cyano group.Formule :C23H19ClF3NO3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :449.85D-Histidine
CAS :D-Histidine is an enantiomer of L-histidine. L-Histidine is an inhibitor of mitochondrial glutamine transport and also an essential amino acid for infants.
Formule :C6H9N3O2Degré de pureté :99.57%Couleur et forme :White Crystalline PowderMasse moléculaire :155.15OTX008
CAS :OTX008 (PTX008) is a selective galectin-1 inhibitor.Formule :C52H72N8O8Degré de pureté :96.38% - 99.84%Couleur et forme :SolidMasse moléculaire :937.18Ca-DTPA trisodium salt hydrate
CAS :Ca-DTPA trisodium hydrate: metal chelator, antidote for cadmium poisoning, non-toxic CMV replication inhibitor.Formule :C14H20CaN3NaO11Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :469.3935-FAM SE
CAS :5-FAM SE, a single-isomer green fluorophore, labels peptides, proteins, nucleotides.Formule :C25H15NO9Degré de pureté :96.19% - 99.93%Couleur et forme :Yellow To Orange SolidMasse moléculaire :473.39Bacopaside I
CAS :Bacopaside I, a saponin from Bacopa monniera, modulates Aquaporin-1, has neuroprotective, anti-Alzheimer's, antioxidative, and antidepressant effects.Formule :C46H74O20SDegré de pureté :98.66% - 99.51%Couleur et forme :SolidMasse moléculaire :979.13Ref: TM-TN1420
1mg67,00€5mg155,00€10mg255,00€1mL*10mM (DMSO)269,00€25mg409,00€50mg532,00€100mg745,00€Faropenem sodium
CAS :Faropenem sodium: Oral penem antibiotic for tuberculosis, pneumonia.Formule :C12H14NNaO5SDegré de pureté :99.41%Couleur et forme :Pale Yellow CrystalsMasse moléculaire :307.3PKC-iota inhibitor 1
CAS :PKC-iota inhibitor 1 is an inhibitor of protein kinase C-iota (PKC-ι ; IC50 : 0.34 μM)Formule :C21H22N6ODegré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :374.44Ref: TM-T8764
1mg107,00€2mg152,00€5mg219,00€1mL*10mM (DMSO)226,00€10mg349,00€25mg583,00€50mg833,00€100mg1.134,00€500mg2.268,00€Ginsenoside Ra1
CAS :Ginsenoside Ra1 is a component from ginseng.Formule :C58H98O26Degré de pureté :97.44%Couleur et forme :SolidMasse moléculaire :1211.38Silychristin
CAS :Silychristin (Silicristin) is a plant growth regulator.Formule :C25H22O10Degré de pureté :99.53% - 99.74%Couleur et forme :SolidMasse moléculaire :482.44Epiberberine
CAS :1.Formule :C20H18NO4Degré de pureté :98.52% - 99.59%Couleur et forme :SolidMasse moléculaire :336.363-(2,4-Dihydroxyphenyl)propanoic acid
CAS :3-(2,4-Dihydroxyphenyl)propanoic acid (Hydroumbellic acid) is a metabolite that is produced by the metabolism of 3-(2, 4-dihydroxyphenyl)prop-2-enoic acid.Formule :C9H10O4Degré de pureté :98.12%Couleur et forme :SolidMasse moléculaire :182.17ENMD-2076
CAS :ENMD-2076, a multi-targeted kinase inhibitor, has specific activity against Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, FGFR2, Src, PDGFRα.Formule :C21H25N7Degré de pureté :97.63% - ≥95%Couleur et forme :SolidMasse moléculaire :375.47ML367
CAS :ML367 inhibits ATAD5 stabilization with low micromolar activity, serving as a probe molecule.Formule :C19H12F2N4Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :334.32Unifiram
CAS :Unifiram boosts cognition, enhances rat hippocampal signals (EC50=27 nM), and ups ACh in rat cortex.Formule :C13H15FN2O3SDegré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :298.332,2,2-Trichloroethanol
CAS :2,2,2-Trichloroethanol is an agonist of the nonclassical K2P channels TREK-1 and TRAAK.Formule :C2H3Cl3ODegré de pureté :99.74%Couleur et forme :LiquidMasse moléculaire :149.4urolithin M6
CAS :urolithin M6 (3,8,9,10-tetrahydroxy urolithin) (UM6) is an ellagitannin metabolite produced by gut microbiota, was identified as a putative galloflavin mimeticFormule :C13H8O6Degré de pureté :99.63%Couleur et forme :Light Beige To Dark Brown SolidMasse moléculaire :260.216-Epivoacarpine
CAS :16-Epivoacarpine is a natural product from Gelsemium elegans.
Formule :C21H24N2O4Degré de pureté :98.12% - 99.98%Couleur et forme :SolidMasse moléculaire :368.43γ-Linolenic acid
CAS :gamma-Linolenic acid (gamolenic acid), is an unsaturated fatty acid synthesized from linoleic acid (LA) by the enzyme delta-6-desaturase.Formule :C18H30O2Degré de pureté :95% - 98.5%Couleur et forme :SolidMasse moléculaire :278.43SB225002
CAS :SB225002 is a potent and selective CXCR2 antagonist inhibiting interleukin IL-8 binding to CXCR2.Formule :C13H10BrN3O4Degré de pureté :98.16% - 99.85%Couleur et forme :SolidMasse moléculaire :352.14Ref: TM-T1955
5mg48,00€1mL*10mM (DMSO)50,00€10mg63,00€25mg120,00€50mg213,00€100mg383,00€200mg585,00€500mg888,00€SD-169
CAS :SD-169 (SD 169) is a selective and ATP competitive the MAP kinases p38α and p38β inhibitor.Formule :C9H8N2ODegré de pureté :98.6%Couleur et forme :SolidMasse moléculaire :160.17Bavachinin
CAS :Bavachinin (Bavachinin A)(7-O-Methylbavachin) is a natural compound isolated from the Chinese herb Fructus Psoraleae with potent anti-angiogenic activity.Formule :C21H22O4Degré de pureté :98% - 99.67%Couleur et forme :SolidMasse moléculaire :338.40Neuraminidase-IN-1
CAS :Neuraminidase-IN-1 (Compound Y-1) is a novel neuraminidase inhibitor.Formule :C14H11N3O6Degré de pureté :97.75%Couleur et forme :SolidMasse moléculaire :317.25Ref: TM-T8555
2mg35,00€5mg55,00€1mL*10mM (DMSO)62,00€10mg92,00€25mg161,00€50mg244,00€100mg359,00€200mg505,00€Bilobetin
CAS :Bilobetin ameliorates insulin resistance by PKA-mediated phosphorylation of PPARα in rats fed a high-fat diet.Formule :C31H20O10Degré de pureté :97% - 99.69%Couleur et forme :SolidMasse moléculaire :552.48Ref: TM-T4S2128
1mg44,00€2mg66,00€5mg137,00€1mL*10mM (DMSO)177,00€10mg236,00€25mg403,00€50mg582,00€100mg800,00€BMY-25368
CAS :BMY-25368 is a long-acting antagonist of the H2-receptor.Formule :C19H25N3O3Couleur et forme :SolidMasse moléculaire :343.42Levobetaxolol hydrochloride
CAS :Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta blocker, used to lower the pressure in the eye in treating conditions such as glaucoma.Formule :C18H29NO3·HClDegré de pureté :98.80% - 99.69%Couleur et forme :SolidMasse moléculaire :343.89LEP(116-130)(mouse)
CAS :Leptin (116-130), mouse C64H109N19O24S, controls appetite and energy, sequence SCSLPQTSGLQKPES-NH2.Formule :C64H109N19O24SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1560.73Glycinamide Hydrochloride
CAS :Glycinamide Hydrochloride (2-Aminoacetamide hydrochloride) is a glycine pro-drug.Formule :C2H7ClN2ODegré de pureté :98% - 99.7%Couleur et forme :White To Off-White SolidMasse moléculaire :110.54Antibacterial agent 27
CAS :Antibacterial agent 27 has potent anti-Candida activity.Formule :C18H14N6Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :314.34Ref: TM-T9612
1mg42,00€1mL*10mM (DMSO)90,00€5mg92,00€10mg133,00€25mg241,00€50mg360,00€100mg537,00€200mg710,00€Cefoperazone
CAS :Cefoperazone (Medocef) inactivates PBPs, disrupting bacterial cell wall synthesis and division; inhibits rMrp2 [3H]E217βG uptake (IC50: 199 μM).Formule :C25H27N9O8S2Degré de pureté :98.99% - 99.76%Couleur et forme :SolidMasse moléculaire :645.67GSK2983559 active metabolite
CAS :GSK2983559 active metabolite (RIPK2-IN-1) is a potent, selective receptor-interacting protein-2 (RIP2) kinase inhibitor.Formule :C21H22N4O4S2Degré de pureté :97.07% - 99.57%Couleur et forme :SolidMasse moléculaire :458.55Physion 8-O-β-D-glucoside
CAS :Physion 8-O-β-D-glucoside is a tumor cell growth inhibitor.Formule :C22H22O10Degré de pureté :95.17% - 99.66%Couleur et forme :SolidMasse moléculaire :446.4Ganoderenic acid A
CAS :Ganoderenic acid A has a potent hepatoprotective, and cytotoxic effects, it shows inhibitory activity on human aldose reductase in vitro.Formule :C30H42O7Degré de pureté :97.27% - 98.50%Couleur et forme :SolidMasse moléculaire :514.653-phenoxy-8-azabicyclo[3.2.1]octane HCl
CAS :3-phenoxy-8-azabicyclo[3.2.1]octane hydrochloride: synthetic, D2 dopamine receptor agonist for dopamine signaling studies.Formule :C13H18ClNODegré de pureté :97.69%Couleur et forme :SolidMasse moléculaire :239.741Ref: TM-T50115
1mg38,00€1mL*10mM (DMSO)78,00€5mg82,00€10mg111,00€25mg182,00€50mg269,00€100mg389,00€200mg555,00€Mandelic acid
CAS :Mandelic acid is a metabolite of adrenaline and found in skincare, used as an analytical reagent, dye precursor, and linked to phenylketonuria.Formule :C8H8O3Degré de pureté :99.45% - 99.95%Couleur et forme :White Solid SolidMasse moléculaire :152.154-[(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]benzoic acid
CAS :4-[(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]benzoic acid: potent, selective antitumor agent; low water solubility; potentially toxic at high doses.Formule :C11H7NO4SDegré de pureté :98.4%Couleur et forme :SolidMasse moléculaire :249.24Aminoadipic acid
CAS :Aminoadipic acid, a lysine metabolism intermediate, inhibits kynurenic acid production and antagonizes NMDA receptor activity.Formule :C6H11NO4Degré de pureté :99.7% - 99.84%Couleur et forme :SolidMasse moléculaire :161.16T.cruzi Inhibitor hydrochloride
T.cruzi Inhibitor is a Trypanosoma cruzi inhibitor.Formule :C22H26ClF3N2ODegré de pureté :97.98% - 99.43%Couleur et forme :SolidMasse moléculaire :426.91Euphorbiasteroid
CAS :Euphorbiasteroid (Euphobiasteroid) (25-50 μM) decreased differentiation of 3T3-L1 cells via reduction of intracellular triglyceride (TG) accumulation.Formule :C32H40O8Degré de pureté :98% - 99.96%Couleur et forme :SolidMasse moléculaire :552.66Ref: TM-T3220
2mg37,00€5mg52,00€10mg71,00€1mL*10mM (DMSO)80,00€25mg114,00€50mg167,00€100mg240,00€200mg355,00€Chemerin-9 (149-157) acetate
Chemerin-9 (149-157) acetate, a nonapeptide C-terminal fragment of chemerin, retains full protein's activity as chemerinR agonist.Formule :C56H70N10O15Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :1123.23Fmoc-Gly-Ser(psi(Me,Me)pro)-OH acetate
Fmoc-Gly-Ser(psi(Me,Me)pro)-OH acetate is a dipeptide.Formule :C25H28N2O8Degré de pureté :94.78%Couleur et forme :SolidMasse moléculaire :484.5VEGFR2-IN-2
CAS :VEGFR2-IN-2 has anti-inflammatory and analgesic activities.Formule :C15H11BrN2ODegré de pureté :99.504%Couleur et forme :SolidMasse moléculaire :315.16Ref: TM-T9724
1mg35,00€5mg73,00€1mL*10mM (DMSO)93,00€10mg105,00€25mg195,00€50mg311,00€100mg445,00€200mg617,00€FIN56
CAS :FIN56 is a specific inducer of ferroptosis.Formule :C25H31N3O5S2Degré de pureté :99.72% - 99.78%Couleur et forme :SolidMasse moléculaire :517.66Ref: TM-T4066
2mg42,00€5mg63,00€1mL*10mM (DMSO)72,00€10mg89,00€25mg192,00€50mg341,00€100mg535,00€200mg748,00€Autocamtide-2-related inhibitory peptide, myristoylated acetate(201422-04-0 free base)
Myristoylated autocamtide-2-related inhibitory peptide acetate is a cell-permeable CaM kinase II inhibitor.Formule :C80H146N22O22Degré de pureté :97.03%Couleur et forme :SolidMasse moléculaire :1768.15Taurolithocholic acid sodium salt
CAS :Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, butFormule :C26H44NNaO5SDegré de pureté :99.79% - 99.93%Couleur et forme :SolidMasse moléculaire :505.69PJ34 hydrochloride
CAS :PJ34 hydrochloride (PJ34 HCl) is a potent specific inhibitor of PARPl/2.Formule :C17H18ClN3O2Degré de pureté :98.87% - ≥95%Couleur et forme :SolidMasse moléculaire :331.8ML348
CAS :ML348 (GNF-Pf-1127) is a selective and reversible lysophospholipase 1 (LYPLA1) inhibitor (IC50 = 210 nM).Formule :C18H17ClF3N3O3Degré de pureté :99% - 99.88%Couleur et forme :SolidMasse moléculaire :415.79Ref: TM-T3439
2mg44,00€5mg65,00€10mg92,00€25mg215,00€50mg334,00€100mg537,00€200mg750,00€500mg1.134,00€Periplogenin
CAS :1.Formule :C23H34O5Degré de pureté :98.41% - 99.91%Couleur et forme :SolidMasse moléculaire :390.51FAUC-365
CAS :FAUC-365 is a D3 dopamine receptor agonist.Formule :C23H25Cl2N3OSDegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :462.44Ref: TM-T21667
1mg50,00€5mg105,00€1mL*10mM (DMSO)116,00€10mg160,00€25mg305,00€50mg485,00€100mg700,00€500mg1.459,00€Tectoridin
CAS :Tectoridin activates estrogen/thyroid receptors; has anti-inflammatory, antioxidant, hypoglycemic effects; inhibits rat aldose reductase (IC: 1.4-15.5 μM).Formule :C22H22O11Degré de pureté :99.02% - 99.48%Couleur et forme :SolidMasse moléculaire :462.40Salcaprozate sodium
CAS :Salcaprozate sodium (SNAC) enhances oral delivery of heparin and insulin by boosting lipophilic transcellular absorption.Formule :C15H20NNaO4Degré de pureté :99.08% - 99.75%Couleur et forme :SolidMasse moléculaire :301.32Skimmin
CAS :Skimmin reduces inflammation, enhances kidney function, and inhibits IgG and glomerular damage in rat kidney disease.Formule :C15H16O8Degré de pureté :97.55% - 99.77%Couleur et forme :SolidMasse moléculaire :324.282-Undecanol
CAS :2-Undecanol, a male pheromone from Lobiopa insularis, is also a floral volatile used by Hymenoptera species.Formule :C11H24ODegré de pureté :98%Couleur et forme :Clear Colorless LiquidMasse moléculaire :172.315-Methylcytidine
CAS :5-Methylcytidine is a modified nucleoside derived from 5-methylcytosine and is a minor constituent of RNA as well as DNA for certain organisms.Formule :C10H15N3O5Degré de pureté :99.02% - 99.88%Couleur et forme :SolidMasse moléculaire :257.24ML281
CAS :ML281 is a potent and selective STK33 inhibitor with IC50 of 14 nM.Formule :C22H19N3O2SDegré de pureté :99.12% - 99.87%Couleur et forme :SolidMasse moléculaire :389.47Ref: TM-T3423
1mg34,00€5mg75,00€1mL*10mM (DMSO)84,00€10mg92,00€25mg178,00€50mg295,00€100mg474,00€500mg1.035,00€1-Furfurylpyrrole
CAS :1-Furfurylpyrrole is a potential contributor of flavor and aroma to popcorn.Formule :C9H9NODegré de pureté :97.85%Couleur et forme :LiquidMasse moléculaire :147.17Rhapontin
CAS :Rhapontin may reduce liver fat and better blood sugar/lipids, showing potential for treating type 2 diabetes.Formule :C21H24O9Degré de pureté :99% - 99.91%Couleur et forme :Light YellowMasse moléculaire :420.41GNE-7915 tosylate
CAS :GNE-7915 tosylate is a potent, selective, and brain-penetrant LRRK2 inhibitor, boasting an IC50 value of 9 nM.Formule :C26H29F4N5O6SCouleur et forme :SolidMasse moléculaire :615.6Ac9-25 acetate
Ac9-25 acetate is an annexin AI peptide and activates the neutrophil reduced nicotinamide adenine dinucleotide phosphate oxidase through FPR but not throughFormule :C101H147N23O35Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :2243.38Rosarin
CAS :Rosarin reduces inflammation and protects nerves by inhibiting iNOS, IL-1β, TNF-α in mouse kidneys and brain.Formule :C20H28O10Degré de pureté :99.14% - 99.95%Couleur et forme :Brown Fine Powder With Characteristic OdorMasse moléculaire :428.43Ref: TM-T3887
100mgÀ demander1mg55,00€5mg109,00€1mL*10mM (DMSO)131,00€10mg170,00€25mg304,00€50mg442,00€N-(4-methoxyphenyl)prop-2-enamide
CAS :N-(4-methoxyphenyl)prop-2-enamide (N-(4-Methoxyphenyl)acrylamide) is an acrylamide analog used as a molecular structural unit.Formule :C10H11NO2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :177.2Ref: TM-T50041
1mg34,00€1mL*10mM (DMSO)54,00€5mg62,00€10mg93,00€25mg141,00€50mg207,00€100mg309,00€200mg439,00€HSDVHK-NH2 acetate
P11 acetate is an integrin αvβ3-vitronectin interaction antagonist(IC50 = 2.74 nM).Formule :C32H52N12O11Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :780.39WNK-IN-11
CAS :WNK-IN-11 (Allosteric WNK Kinase Inhibitor) is an allosteric With-No-Lysine (WNK) kinase inhibitor,WNK1(IC50 : 4 nM)Formule :C21H21Cl2N5OSDegré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :462.4Ref: TM-T5456
1mg87,00€5mg172,00€1mL*10mM (DMSO)188,00€10mg280,00€25mg474,00€50mg683,00€100mg964,00€500mg1.918,00€Pheanthine
CAS :Pheanthine is an extract of the fruit of Gyrocarpus jacquinii and shows induction of C/EBPα activity.Formule :C38H42N2O6Degré de pureté :98.71%Couleur et forme :SolidMasse moléculaire :622.75U-104
CAS :U-104 (NSC-213841) is an effective carbonic anhydrase (CA) inhibitor for CA IX( Ki=45.1 nM) and CA XII(Ki=4.5 nM).Formule :C13H12FN3O3SDegré de pureté :98.76% - 99.88%Couleur et forme :SolidMasse moléculaire :309.32Ref: TM-T2017
5mg34,00€10mg50,00€1mL*10mM (DMSO)55,00€25mg93,00€50mg135,00€100mg236,00€200mg379,00€500mg617,00€FRAX486 HCL(1232030-35-1 free base)
FRAX486 HCL is a potent p21-activated kinase (PAK) inhibitor with IC50 values of 14, 33, 39 and 575 nM for PAK1, PAK2, PAK3 and PAK4 respectively.Formule :C25H24Cl3FN6ODegré de pureté :98.85% - 99.82%Couleur et forme :SolidMasse moléculaire :549.86C15AlkOPP
CAS :C15AlkOPP is an FPP analogue, bearing an alkyne group to allow for post-prenylation protein labeling.Formule :C18H30O8P2Couleur et forme :SolidMasse moléculaire :436.37Sapropterin dihydrochloride
CAS :Sapropterin dihydrochloride (6R-BH4 dihydrochloride) is phenylalanine hydroxylase agonist that is approved for the treatment of BH4 responsive PKU.Formule :C9H17Cl2N5O3Degré de pureté :98% - 99.88%Couleur et forme :White Crystalline SolidMasse moléculaire :314.17TP0463518
CAS :TP-0463518 is a highly potent HIF prolyl hydroxylase (PHD) inhibitor (IC50s: 13 nM and 18 nM for human and rat PHD2, respectively).Formule :C20H18ClN3O6Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :431.83TW-37
CAS :TW-37 is an nonpeptide inhibitor to recombinant Bcl-2, Bcl-xL and Mcl-1 (Ki: 0.29/1.11/0.26 μM).Formule :C33H35NO6SDegré de pureté :97.06% - ≥95%Couleur et forme :SolidMasse moléculaire :573.7Ref: TM-T6281
1mg38,00€2mg50,00€5mg65,00€1mL*10mM (DMSO)90,00€10mg107,00€25mg202,00€50mg334,00€100mg495,00€G15
CAS :G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)Formule :C19H16BrNO2Degré de pureté :98.46% - 98.59%Couleur et forme :SolidMasse moléculaire :370.24Pseudolaric acid B β-D-glucoside
CAS :Pseudolaric acid B β-D-glucoside (Pseudolaric acid B-glucopyranoside) is a natural product from Pseudolarix amabilis.Formule :C29H38O13Degré de pureté :98.55% - ≥95%Couleur et forme :SolidMasse moléculaire :594.60dasiglucagon acetate
Dasiglucagon acetate: new, stable glucagon for hypoglycemia with better absorption and longer half-life.Formule :C154H226N38O52Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :3441.67Nexturastat A
CAS :Nexturastat A is an effective and specific HDAC6 inhibitor (IC50: 5 nM). Its selectivity is >190-fold than other HDACs.Formule :C19H23N3O3Degré de pureté :99.40% - 99.57%Couleur et forme :SolidMasse moléculaire :341.4Paris saponin VII
CAS :Paris saponin VII (Dioscini) shows inhibitory effects on cell proliferation.Formule :C51H82O21Degré de pureté :99.51% - 99.63%Couleur et forme :SolidMasse moléculaire :1031.18LY2874455
CAS :LY2874455 has been used in trials studying the treatment of Advanced Cancer.Formule :C21H19Cl2N5O2Degré de pureté :97.22% - 99.46%Couleur et forme :SolidMasse moléculaire :444.31Ref: TM-T2361
1mg47,00€5mg92,00€1mL*10mM (DMSO)101,00€10mg145,00€25mg281,00€50mg447,00€100mg670,00€200mg888,00€Osimertinib mesylate
CAS :Osimertinib mesylate (AZD-9291 mesylate) is an EGFR third-generation inhibitor. Osimertinib mesylate has antitumor activity. Cost-effective and quality-assured.
Formule :C29H37N7O5SDegré de pureté :99.46% - >99.99%Couleur et forme :SolidMasse moléculaire :595.71(S)-CPI203
CAS :CPI-203 is an effective BET bromodomain inhibitor (IC50: 37 nM for BRD4).Formule :C19H18ClN5OSDegré de pureté :99.01% - 99.92%Couleur et forme :SolidMasse moléculaire :399.9Ref: TM-T6026
2mg34,00€5mg55,00€1mL*10mM (DMSO)58,00€10mg89,00€25mg170,00€50mg269,00€100mg424,00€200mg593,00€CGS 21680 Hydrochloride
CAS :CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.Formule :C23H29N7O6·HClDegré de pureté :96.74% - 99.53%Couleur et forme :SolidMasse moléculaire :535.98Ref: TM-T6441
1mg38,00€2mg50,00€5mg81,00€1mL*10mM (DMSO)95,00€10mg109,00€25mg215,00€50mg389,00€100mg575,00€Diquafosol tetrasodium
CAS :Diquafosol Tetrasodium is a P2Y2 receptor agonist that stimulates the secretion of mucins from ocular tissues Diquafosol tetrasodium (INS365) improves tear filmFormule :C18H22N4Na4O23P4Degré de pureté :98.25% - 99.97%Couleur et forme :SolidMasse moléculaire :878.23Galanin Receptor Ligand M35 TFA
Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).Formule :C109H154N27F3O28Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :2347.62JNJ-63576253
CAS :JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).Formule :C23H22ClF3N6O2SDegré de pureté :98.71%Couleur et forme :SolidMasse moléculaire :538.97AP1189 acetate
CAS :AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.Formule :C16H18N6O4Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :358.35SR 57227 hydrochloride
CAS :SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.Formule :C10H14ClN3·HClDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :248.15trans-Cinnamaldehyde
CAS :Trans-Cinnamaldehyde (Phenylacrolein) exhibits anti-inflammatory activities and antidepressant-like effects in stressed mid-aged rats as a COX-2 inhibitor.Formule :C9H8ODegré de pureté :98.07%Masse moléculaire :132.16ICI 63197
CAS :ICI 63197 (2-Amino-6-methyl-4-propyl-[1,2,4]triazolo[1,5-a]pyrimidin-5(4H)-one) is a PDE4 inhibitor.Formule :C9H13N5ODegré de pureté :99.70%Couleur et forme :White SolidMasse moléculaire :207.23
