
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.849 produits)
- Apoptose(6.367 produits)
- Cycle cellulaire/point de contrôle(4.907 produits)
- Chromatine/Épigénétique(2.622 produits)
- Signalisation du cytosquelette(1.585 produits)
- Altération de l'ADN/réparation de l'ADN(2.873 produits)
- Endocrinologie/Hormones(3.758 produits)
- Enzyme(3.673 produits)
- GPCR/G-Protéine(9.049 produits)
- Immunologie et Inflammation(3.943 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(417 produits)
- Signalisation MAPK(1.259 produits)
- Transporteur membranaire/Canal ionique(3.164 produits)
- Métabolisme(10.149 produits)
- Microbiologie/Virologie(7.673 produits)
- Neuroscience(10.547 produits)
- Autres inhibiteurs(35.859 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.435 produits)
- Protéases/Protéasome(1.693 produits)
- Cellules souche et Dérivés(734 produits)
- Tyrosine Kinase/Adaptateurs(1.991 produits)
- Ubiquitination(1.743 produits)
Affichez 16 plus de sous-catégories
66517 produits trouvés pour "Inhibiteurs"
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TAPI-1 trifluoroacetate (163847-77-6(free base))
TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors.Formule :C28H38F3N5O7Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :613.62(R)-5-Oxopyrrolidine-2-carboxylic acid
CAS :(R)-5-Oxopyrrolidine-2-carboxylic acid (D-Pyroglutamic acid) is a cyclic derivative of glutamic acid, physiologically present in mammalian tissues.Formule :C5H7NO3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :129.11WHI-P180
CAS :WHI-P180 (Janex 3) is a potent EGFR and Cdk2 inhibitors with IC50 of 4.0 and 1.0 uM, respectively.Formule :C16H15N3O3Degré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :297.31KYP-2047
CAS :KYP-2047 is a very potent, selective Prolyl oligopeptidase (POP) inhibitor.Formule :C20H25N3O2Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :339.43Ref: TM-T8657
2mg43,00€5mg66,00€1mL*10mM (DMSO)75,00€10mg87,00€25mg161,00€50mg231,00€100mg349,00€200mg495,00€PFI-2 hydrochloride
CAS :PFI-2 hydrochloride ((R)-PFI-2 hydrochloride) is a potent, highly selective, and cell-active inhibitor of the methyltransferase activity of SETD7 (IC50: 2 nM),Formule :C23H26ClF4N3O3SDegré de pureté :99.31% - 99.91%Couleur et forme :SolidMasse moléculaire :535.98Ref: TM-T4583
1mg38,00€2mg49,00€5mg80,00€10mg111,00€1mL*10mM (DMSO)122,00€25mg200,00€50mg358,00€100mg523,00€500mg1.108,00€N-Formylcytisine
CAS :N-Formylcytisine ((-)-N-Formylcytisine) is a natural product isolated from the stem bark of Maackia amurensis.Formule :C12H14N2O2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :218.25LDN-192960
CAS :LDN-192960 is a potent inhibitor of Haspin and DYRK2 (IC50s: 10 nM and 48 nM).Formule :C18H20N2O2SDegré de pureté :99.01% - 99.51%Couleur et forme :SolidMasse moléculaire :328.43Ref: TM-TQ0111
1mg49,00€2mg64,00€5mg92,00€1mL*10mM (DMSO)104,00€10mg152,00€25mg295,00€50mg477,00€100mg763,00€200mg1.018,00€AZD8330
CAS :AZD8330 (ARRY-704) is a novel, selective, non-ATP competitive MEK 1/2 inhibitor with IC50 of 7 nM. Phase 1.Formule :C16H17FIN3O4Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :461.23Kudinoside D
CAS :Kudinoside D exerts anti-adipogenic effects through modulation of adipogenic transcription factors via AMPK signaling pathway.Formule :C47H72O17Degré de pureté :99.66% - 99.92%Couleur et forme :SolidMasse moléculaire :909.06Ref: TM-TN1836
1mg119,00€5mg269,00€1mL*10mM (DMSO)324,00€10mg374,00€25mg577,00€50mg783,00€100mg1.054,00€200mg1.423,00€3-Ethoxy-3-oxopropanoic acid
CAS :3-Ethoxy-3-oxopropanoic acid (Monoethyl malonic acid) belongs to the class of organic compounds known as dicarboxylic acids and derivatives.Formule :C5H8O4Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :132.11SDZ285428
CAS :SDZ285428 is a CYP24A1 inhibitor.Formule :C24H20ClN3ODegré de pureté :97.51%Couleur et forme :SolidMasse moléculaire :401.89Ref: TM-T4188
2mg37,00€5mg52,00€1mL*10mM (DMSO)58,00€10mg90,00€25mg170,00€50mg255,00€100mg375,00€200mg533,00€Irganox 1010
CAS :Irganox 1010 (Dovernox 10) is an agent of antioxidant.Formule :C73H108O12Degré de pureté :97.27% - 99.96%Couleur et forme :Pelletslargecrystals Othersolid Wetsolid PelletslargecrystalsMasse moléculaire :1177.63Hirsutine
CAS :Hirsutine induces apoptosis and is a potent Dengue virus inhibitor exhibiting low cytotoxicity.Hirsutine has anticancer, cardioprotective, anti-hypertensive andFormule :C22H28N2O3Degré de pureté :99.36% - 99.98%Couleur et forme :SolidMasse moléculaire :368.47Picropodophyllin
CAS :Picropodophyllin (PPP) is a selective IGF-1R inhibitor with IC50 of 1 nM, not affecting other growth factor receptors.Formule :C22H22O8Degré de pureté :98.38% - 99.83%Couleur et forme :SolidMasse moléculaire :414.41Ref: TM-T6943
5mg64,00€1mL*10mM (DMSO)69,00€10mg88,00€25mg170,00€50mg316,00€100mg535,00€500mg1.121,00€WNK463
CAS :WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).Formule :C21H24F3N7O2Degré de pureté :>99.99% - ≥95%Couleur et forme :SolidMasse moléculaire :463.46Dexmedetomidine
CAS :Dexmedetomidine: a central alpha-2 adrenergic agonist for general anesthesia.Formule :C13H16N2Degré de pureté :99% - >99.99%Couleur et forme :SolidMasse moléculaire :200.28(+)-Usnic acid
CAS :(+)-Usnic acid (D-Usnic Acid) is a naturally occurring dibenzofuran derivative found in several lichen species.Formule :C18H16O7Degré de pureté :98.22%Couleur et forme :SolidMasse moléculaire :344.322,2-Dihydroxyacetic acid
CAS :2,2-Dihydroxyacetic acid (Formylformic acid) is an organic compound that is both an aldehyde and a carboxylic acid, is associated with primary hyperoxaluria.Formule :C2H4O4Degré de pureté :99.25%Couleur et forme :White To Light Yellow Crystalline PowderMasse moléculaire :92.05Oxoadipic acid
CAS :Oxoadipic acid: metabolite from tryptophan and lysine, links TCA cycle to lysine synthesis, studied for mitochondrial transport.
Formule :C6H8O5Degré de pureté :96.61% - >99.99%Couleur et forme :SolidMasse moléculaire :160.12Nodakenin
CAS :Nodakenin ((+)-Marmesinin) is a compound with anti-allergic and anti-inflammatory activities.Formule :C20H24O9Degré de pureté :95.46% - 98.93%Couleur et forme :SolidMasse moléculaire :408.40Ref: TM-T3872
2mg34,00€1mL*10mM (DMSO)50,00€5mg52,00€10mg73,00€25mg105,00€50mg152,00€100mg215,00€200mg320,00€CNQX
CAS :CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively)Formule :C9H4N4O4Degré de pureté :99.70%Couleur et forme :Pale Yellow SolidMasse moléculaire :232.15Penicillin G potassium
CAS :Penicillin G potassium (Benzylpenicillin potassium) is the potassium salt form of penicillin G, a broad-spectrum penicillin antibiotic.Formule :C16H17KN2O4SDegré de pureté :98.55% - 99.84%Couleur et forme :LiquidMasse moléculaire :372.48PX-478
CAS :PX-478 is a HIF-1α inhibitor with selectivity, oral activity, and blood-brain barrier permeability.Formule :C13H20Cl4N2O3Degré de pureté :97% - 99.79%Couleur et forme :SolidMasse moléculaire :394.12Ref: TM-T6961
1mg39,00€5mg84,00€1mL*10mM (DMSO)84,00€10mg130,00€25mg193,00€50mg261,00€100mg411,00€200mg605,00€RO4987655
CAS :RO4987655 (RG7167) is an orally active and highly selective MEK inhibitor (IC50: 5.2 nM for MEK1/MEK2).Formule :C20H19F3IN3O5Degré de pureté :98.21%Couleur et forme :SolidMasse moléculaire :565.28Caftaric acid
CAS :Caftaric acid: a natural antioxidant, anti-inflammatory, antimutagenic, and Src kinase protein-protein interaction inhibitor.Formule :C13H12O9Degré de pureté :98.31% - 99.50%Couleur et forme :White PowderMasse moléculaire :312.23Ref: TM-T3S2390
1mg34,00€2mg46,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg92,00€25mg177,00€50mg295,00€100mg442,00€200mg620,00€Levamlodipine hydrobromide
CAS :Levamlodipine hydrobromide is a medication used to lower blood pressure and prevent chest pain.Formule :C20H26BrClN2O5Couleur et forme :SolidMasse moléculaire :489.79Gap 27
CAS :Gap 27 is a peptide(Ser-Arg-Pro-Thr-Glu-Lys-Thr-Ile-Phe-Ile-Ile) derived from connexin 43 that is a selective gap junction blocker.Formule :C60H101N15O17Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1304.531,4-D-Gulonolactone
CAS :1,4-D-Gulonolactone, precursor to vitamin C, is an enzyme substrate linked to oxidative stress and absent in scurvy-susceptible species.Formule :C6H10O6Degré de pureté :99.69%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :178.14d[Cha4]-AVP acetate(500170-27-4 free base)
'd[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'Formule :C52H75N13O13S2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :1154.37PF-07038124
CAS :PF-07038124 inhibits PDE4B2 (IC50=0.5 nM), IFNγ (IC50=1.06 nM), IL4 (IC50=4.1 nM), and IL-13 (IC50=125 nM).Formule :C18H22BNO4Couleur et forme :SolidMasse moléculaire :327.18Guanosine
CAS :Guanosine (DL-Guanosine) is a purine nucleoside formed from a beta-N9-glycosidic bond between guanine and a ribose ring and is essential for metabolism.Formule :C10H13N5O5Degré de pureté :97.36% - 99.95%Couleur et forme :SolidMasse moléculaire :283.24Harmol
CAS :Harmol (Methylpyridoindolol) is a β-carboline isolated from nature.Formule :C12H10N2ODegré de pureté :98.9% - 99.90%Couleur et forme :SolidMasse moléculaire :198.22Tacrine
CAS :Tacrine (CS 12602) is an indirect cholinergic agonist and centrally acting anticholinesterase. It is approved for the treatment of Alzheimer's disease.Formule :C13H14N2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :198.26N-Formyl-Met-Ala-Ser TFA(17351-32-5 free base)
N-Formyl-Met-Ala-Ser (fMet-Ala-Ser) peptide targets neutrophil formyl peptide receptors.Formule :C14H22F3N3O8SDegré de pureté :98.21% - 99.79%Couleur et forme :SolidMasse moléculaire :449.4POL1-IN-1
CAS :POL1-IN-1 (Compound 3A) 是一种RNA 聚合酶 1 POL1抑制剂,IC50值低于 0.5 uM。 它能有效抑制A375恶性黑色素瘤细胞系中RNA 聚合酶I 的转录。
Formule :C21H20N6Degré de pureté :98% - 98.01%Couleur et forme :SolidMasse moléculaire :356.42N-Acetylputrescine hydrochloride
CAS :N-Acetylputrescine is a polyamine commonly occurring excreted in normal human urineFormule :C6H15ClN2ODegré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :166.657-Methoxyflavone
CAS :7-Methoxyflavone isolated from Zornia brasiliensis with antinociceptive effects.Formule :C16H12O3Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :252.26Cyclosporine
CAS :Cyclosporine is a calcineurin phosphatase pathway inhibitor, used as an immunosuppressant drug to prevent rejection in organ transplantation.Formule :C62H111N11O12Degré de pureté :99.68%Couleur et forme :White PowderMasse moléculaire :1202.61AG1024
CAS :AG1024 (Tyrphostin) suppresses IGF-1R autophosphorylation(IC50=7 μM), and is less potent for IR(IC50=57 μM).Formule :C14H13BrN2ODegré de pureté :98% - 99.37%Couleur et forme :SolidMasse moléculaire :305.1718α-Glycyrrhetinic acid
CAS :18α-Glycyrrhetinic acid (Enoxolone) is a pentacyclic triterpenoid derivative of the beta-amyrin type obtained from the hydrolysis of glycyrrhizic acid.Formule :C30H46O4Degré de pureté :98.54% - 99.68%Couleur et forme :SolidMasse moléculaire :470.68Ddr1-In-1
CAS :DDR1-IN-1 is an effective and specific DDR1 receptor tyrosine kinase inhibitor (IC50: 105 nM), about 3-fold selectivity over DDR2.Formule :C30H31F3N4O3Degré de pureté :99.83% - 99.93%Couleur et forme :SolidMasse moléculaire :552.59Ref: TM-T3337
1mg39,00€2mg50,00€5mg80,00€1mL*10mM (DMSO)95,00€10mg109,00€25mg167,00€50mg215,00€100mg334,00€200mg494,00€Pyridoxal 5'-phosphate monohydrate
CAS :Pyridoxal 5'-phosphate monohydrate is an active vitamin B6 metaboliteFormule :C8H12NO7PDegré de pureté :98.94% - 99.05%Couleur et forme :Slightly Yellow PowderMasse moléculaire :265.16Abafungin
CAS :Abafungin (Bay w 6341) is an antifungal agent with a broad-spectrum.Formule :C21H22N4OSDegré de pureté :98.11%Couleur et forme :SolidMasse moléculaire :378.49Chebulic acid
CAS :Chebulic acid, a phenolcarboxylic acid compound isolated from Terminalia chebula, has potent anti-oxidant activity,which breaks the cross-links of proteinsFormule :C14H12O11Degré de pureté :96% - 99.98%Couleur et forme :SolidMasse moléculaire :356.24SR8278
CAS :SR8278 is an REV-ERBα antagonist(EC50 = 0.47 μM), blocking activation of the receptor by the synthetic agonist GSK 4112Formule :C18H19NO3S2Degré de pureté :99.44% - 99.73%Couleur et forme :SolidMasse moléculaire :361.48Ref: TM-T7837
1mg49,00€5mg97,00€1mL*10mM (DMSO)106,00€10mg160,00€25mg303,00€50mg437,00€100mg642,00€200mg914,00€Eflornithine hydrochloride hydrate
CAS :Eflornithine hydrochloride hydrate (DFMO hydrochloride hydrate) is an ornithine decarboxylase (ODC) inhibitor with antitumor activity. Cost-effective and quality-assured.Formule :C6H15ClF2N2O3Degré de pureté :99% - 99.88%Couleur et forme :White SolidMasse moléculaire :236.64S 14506 HCl
CAS :S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).Formule :C24H26FN3O2Couleur et forme :SolidMasse moléculaire :407.48L-745870 trihydrochloride
CAS :L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.Formule :C18H22Cl4N4Degré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :436.21Sipeimine
CAS :Sipeimine (Kashmirine) is an antiasthmatic M receptor antagonist, shifting the dose-response curve rightwards in Kaba-induced tracheal contractions.Formule :C27H43NO3Degré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :429.64IR-780 Iodide
CAS :IR-780 Iodide: a near-infrared dye for HIF-1α/glycolysis ABCB10-dependent human CSC characterization.Formule :C36H44ClIN2Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :667.12Sugammadex sodium
CAS :Sugammadex sodium (Org25969) , a synthetic derivative of γ-cyclodextrin, is a steroid-based neuromuscular blocker reversing agent.Formule :C72H104Na8O48S8Degré de pureté :99.43% - 99.8%Couleur et forme :SolidMasse moléculaire :2178.01APTS
CAS :Anionic dye 8-Aminopyrene-1,3,6-trisulfonic Acid (sodium salt), excites at 425 nm and emits at 503 nm, detects glucose and saccharides.Formule :C16H8NNa3O9S3Degré de pureté :97.17% - 99.79%Couleur et forme :Yellow SolidMasse moléculaire :523.4AZD 6482
CAS :AZD 6482 (KIN-193) is a potent and selective inhibitor of p110β and PI3Kβ with IC50 values of 0.69nM and 10nM.Cost-effective and quality-assured.Formule :C22H24N4O4Degré de pureté :99.87% - 99.95%Couleur et forme :SolidMasse moléculaire :408.45Nystatin
CAS :Nystatin (Fungicidin) is a topical and oral antifungal agent with activity against many species of yeast and candida albicans, which is used largely to treatFormule :C47H79NO19Degré de pureté :69.55% - 99.86%Couleur et forme :Yellow SuspensionMasse moléculaire :962.137L189
CAS :L189 is a human DNA ligase inhibitor, inhibits hLigI/III/IV (IC50: 5/9/5 μM).Formule :C11H10N4OSDegré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :246.29(S,R,S)-AHPC-Me
CAS :(S,R,S)-AHPC-Me is a VHL ligand for synthesizing the BET degrader ARV-771, which targets CRPC cells.Formule :C23H32N4O3SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :444.59Avanafil
CAS :Avanafil (TA1790) is a selective inhibitor of phosphodiesterase type 5 (PDE5) and is used as therapy of erectile dysfunction.Formule :C23H26ClN7O3Degré de pureté :99.03% - >99.99%Couleur et forme :White SolidMasse moléculaire :483.95KBU2046
CAS :KBU2046: oral anti-metastasis compound, enhances survival, targets chaperone complexes, not a typical HSP90 inhibitor.Formule :C15H11FO2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :242.24Ref: TM-T15646
2mg33,00€5mg50,00€1mL*10mM (DMSO)50,00€10mg71,00€25mg133,00€50mg200,00€100mg304,00€200mg425,00€AKT inhibitor VIII
CAS :AKT inhibitor VIII (AKTi-1/2) is a highly specific Akt1/2 inhibitor (IC50: 58/210 nM). The selectivity for Akt1 is higher about 36-fold than Akt3.Formule :C34H29N7ODegré de pureté :98.31% - 98.65%Couleur et forme :Pale Yellow SolidMasse moléculaire :551.64AC1NS4RE
CAS :It is a tyrosine kinase inhibitor.Formule :C15H13ClN2ODegré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :272.73Dovitinib lactate hydrate
CAS :Dovitinib lactate hydrate (TKI258) is the Lactate of Dovitinib, which is a multitargeted RTK inhibitor, mostly for class III (FLT3/c-Kit).Formule :C24H27FN6O4Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :482.51Rottlerin
CAS :Rottlerin (NSC-56346), a Mallotus Philippinensis extract, inhibits PKC (3-100 μM IC50); triggers apoptosis by activating caspase 3.Formule :C30H28O8Degré de pureté :97.41% - 99.44%Couleur et forme :Orange To Brown PowderMasse moléculaire :516.54Oclacitinib
CAS :Oclacitinib (PF-03394197)(PF03394197) is a potent and selective JAKs inhibitor with IC50 of 10-99 nM; not inhibit a panel of 38 non-JAK kinases (IC50 's > 1000Formule :C15H23N5O2SDegré de pureté :98% - 98.45%Couleur et forme :White To Off-White SolidMasse moléculaire :337.44Agarotetrol
CAS :Agarotetrol is a flavonoid derivative isolated from agarwood.Formule :C17H18O6Degré de pureté :99.29% - 99.96%Couleur et forme :SolidMasse moléculaire :318.32Tetrindole mesylate
CAS :Tetrindole mesylate is a MAO-A inhibitor.Formule :C21H30N2O3SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :390.54Leucomethylene blue mesylate
CAS :Leucomethylene blue mesylate (TRx0237 mesylate) is a second-generation tau protein aggregation inhibitor for the treatment of AD and frontotemporal dementia.Formule :C16H19N3S·2CH4O3SDegré de pureté :97.47% - 99.99%Couleur et forme :SolidMasse moléculaire :477.62Ref: TM-T7003
2mg37,00€5mg52,00€1mL*10mM (DMSO)52,00€10mg71,00€25mg114,00€50mg182,00€100mg314,00€200mg474,00€ML-SI3
CAS :CCG-143140 is a GLP-1 receptor inverse agonists.Formule :C23H31N3O3SDegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :429.581,2-Dipalmitoyl-sn-glycerol
CAS :1,2-Dipalmitoyl-sn-glycerol ((S)-1,2-Dipalmitin) is an analog of the PKC-activating second messenger diacylglycerol (DAG). It weakly activates PKC.Formule :C35H68O5Degré de pureté :97.84% - 99.78%Couleur et forme :SolidMasse moléculaire :568.91Choline Fenofibrate
CAS :Choline Fenofibrate (Trilipix) is a choline formulation of fenofibrate, a synthetic phenoxy-isobutyric acid derivate and prodrug with antihyperlipidemic
Formule :C22H28ClNO5Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :421.91AQW-051 fumarate
CAS :AQW-051 fumarate is an α7 nicotinic ACh receptor partial agonist that may act as a cognitive-enhancing agent.Formule :C23H26N2O5Couleur et forme :SolidMasse moléculaire :410.475-Phenylvaleric Acid
CAS :5-Phenylvaleric Acid (Benzenepentanoic acid) is a pentanoic acid of bacterial origin, occasionally found in human biofluids.Formule :C11H14O2Degré de pureté :97.159%Couleur et forme :SolidMasse moléculaire :178.23Nevirapine hemihydrate
CAS :Nevirapine hemihydrate is a non-nucleoside reverse transcriptase inhibitor (NNRTI) studied for potential treatment of HIV-1 infection and AIDS.Formule :C30H30N8O3Couleur et forme :SolidMasse moléculaire :550.62Dihydrotanshinone I
CAS :Dihydrotanshinone I (DHTS) is a natural compound extracted from Salvia miltiorrhiza Bunge used for treating of cardiovascular diseases.Formule :C18H14O3Degré de pureté :97.4% - 99.59%Couleur et forme :SolidMasse moléculaire :278.30Nordihydroguaiaretic acid
CAS :Nordihydroguaiaretic acid (NDGA) is a natural lipoxygenase (5-LOX) inhibitor. Nordihydroguaiaretic acid has antioxidant effect. Cost-effective and quality-assured.Formule :C18H22O4Degré de pureté :97.82% - 99.91%Couleur et forme :SolidMasse moléculaire :302.36ARV-825
CAS :ARV-825: PROTAC recruits BRD4 to cereblon for rapid BRD4 degradation in all tested BL cells.Formule :C46H47ClN8O9SDegré de pureté :97.15% - 98%Couleur et forme :SolidMasse moléculaire :923.43NVP-BHG712
CAS :NVP-BHG712 is a specific EphB4 inhibitor with ED50 of 25 nM that discriminates between VEGFR and EphB4 inhibition; also shows activity against c-Raf, c-Src andFormule :C26H20F3N7ODegré de pureté :97.32% - 98.63%Couleur et forme :SolidMasse moléculaire :503.48Ref: TM-T6348
1mg34,00€5mg74,00€1mL*10mM (DMSO)84,00€10mg105,00€25mg200,00€50mg371,00€100mg557,00€200mg790,00€Calcitonin eel acetate
Calcitonin eel acetate (Calcitonin eel acetate (57014-02-5 Free base)) is the regulation of calcium homeostasis thyroid hormone peptide.Formule :C148H245N43O49S2Degré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :3474.96Benzamidine hydrochloride
CAS :Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin.Formule :C7H9ClN2Degré de pureté :99.25% - 99.97%Couleur et forme :White To Off-White PowderMasse moléculaire :156.61Lerisetron
CAS :Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Formule :C18H20N4Degré de pureté :99.15% - 99.82%Couleur et forme :SolidMasse moléculaire :292.38Esonarimod
CAS :Esonarimod (KE-298) is an antirheumatic drug.Formule :C14H16O4SDegré de pureté :97.44%Couleur et forme :SolidMasse moléculaire :280.344-Phenoxybenzylamine
CAS :4-Phenoxybenzylamine inhibits the function of the NS3 protein by stabilizing an inactive conformation with an IC50 of about 500 μM against HCV NS3/4a .Formule :C13H13NODegré de pureté :97.26%Couleur et forme :SolidMasse moléculaire :199.25WHI-P258
CAS :WHI-P258, a weak JAK3 inhibitor, is used as a negative control in drug development.Formule :C16H15N3O2Degré de pureté :99.66% - 99.92%Couleur et forme :SolidMasse moléculaire :281.31Lophanthoidin B
CAS :Lophanthoidin B is a natural product isolated from the herbs of Rabdosia lophanthoides.Formule :C24H32O8Degré de pureté :98.00% - 98.00%Couleur et forme :SolidMasse moléculaire :448.51Tanshinone I
CAS :Tanshinone I (Tanshinone A), an active principle isolated from the herbal medicine Salvia miltiorrhiza, displays cytotoxicity against tumor cells.Formule :C18H12O3Degré de pureté :98.31% - 98.70%Couleur et forme :SolidMasse moléculaire :276.29NSC 404988
CAS :NSC 404988 is a benzamide bioactive used for drug synthesis, metabolite analysis, and studying drug metabolism.Formule :C11H14ClNODegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :211.69Alytesin acetate
Alytesin acetate is an amphibian bombesin-like peptide.
Formule :C70H110N22O19SDegré de pureté :95.79%Couleur et forme :SolidMasse moléculaire :1595.82Ref: TM-TP2219L
1mg245,00€2mg366,00€5mg550,00€10mg787,00€25mg1.198,00€50mg1.596,00€100mg2.175,00€500mg4.351,00€Nitecapone
CAS :Nitecapone is a reversible inhibitor of S-COMT (IC50 values of 300 nM in rat liver)Formule :C12H11NO6Degré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :265.222,3-dihydro-1H-indene-5-sulfonamide
CAS :2,3-dihydro-1H-indene-5-sulfonamide is Carbonic anhydrase 12 (human) inhibitor.Formule :C9H11NO2SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :197.25Ref: TM-T8611
1mg58,00€1mL*10mM (DMSO)99,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€Nitrofen
CAS :Nitrofen is a selective contact herbicide. Nitrofen is a protoporphyrinogen oxidase and retinal dehydrogenase inhibitor.Formule :C12H7Cl2NO3Degré de pureté :99.92%Couleur et forme :Less Crystals Or Black Solid Used As A Pre- Or Post-Emergence HerbicideMasse moléculaire :284.09Sinigrin
CAS :Sinigrin, a glucosinolate used to test and identify myrosinase enzymes, serves as a reference for isolating glucosinolates.Formule :C10H16KNO9S2Degré de pureté :99.93%Couleur et forme :White To Beige Crystalline PowderMasse moléculaire :397.45(-)-(S)-Equol
CAS :(-)-(S)-Equol (4',7-Dihydroxyisoflavan) is an orally bioavailable, non-steroidal estrogen naturally produced by the metabolism of the isoflavonoid daidzein.Formule :C15H14O3Degré de pureté :99.13% - 99.52%Couleur et forme :SolidMasse moléculaire :242.27(Arg)9 TFA (143413-47-2 free base)
CAS :(Arg)9 TFA (Peptide R9 TFA) is a cell-penetrating peptide. (Arg)9 TFA exhibits neuroprotective activity with an IC50 of 0.78 μM in the glutamic acid model.Formule :C56H111F3N36O12Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1537.71Acetyl hexapeptide 38 Acetate
Acetyl hexapeptide-38 Acetate, a breast volume enhancer, boosts fat synthesis in targeted areas.Formule :C32H59N9O12Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :761.85Rapastinel Trifluoroacetate
CAS :Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties.Formule :C20H32F3N5O8Degré de pureté :99.01% - 99.77%Couleur et forme :SolidMasse moléculaire :527.49Ref: TM-T5819
1mg39,00€5mg97,00€1mL*10mM (DMSO)116,00€10mg160,00€25mg296,00€50mg416,00€100mg557,00€200mg743,00€Cridanimod
CAS :Cridanimod (10-carboxymethyl-9-acridanone, CMA) is a potent STING agonist that directly binds to STING and triggers a strong antiviral response through the TBK1Formule :C15H11NO3Degré de pureté :99.91% - 99.96%Couleur et forme :SolidMasse moléculaire :253.25Alprenolol tartrate
CAS :Alprenolol tartrate is a 5-HT1A antagonist.Formule :C19H29NO8Couleur et forme :SolidMasse moléculaire :399.446-OAU
CAS :6-OAU is a GPR84 agonist, activates it in HEK293 cells with a 105 nM EC50.Formule :C12H21N3O2Degré de pureté :98.14% - 99.01%Couleur et forme :SolidMasse moléculaire :239.31Ref: TM-T2036
1mg152,00€2mg203,00€1mL*10mM (DMSO)285,00€5mg313,00€10mg447,00€25mg713,00€50mg1.018,00€100mg1.369,00€8-Chloroadenosine
CAS :8-Chloroadenosine (NSC-354258) is a 5' AMP-activated protein kinase agonist potentially for the treatment of chronic lymphocytic leukemia.Formule :C10H12ClN5O4Degré de pureté :98.75% - 99.84%Couleur et forme :SolidMasse moléculaire :301.69Ref: TM-T19661
1mg34,00€5mg114,00€1mL*10mM (DMSO)158,00€10mg178,00€25mg314,00€50mg467,00€100mg665,00€500mg1.333,00€(R)-GNE-140
CAS :(R)-GNE-140 (GNE-140) is an effective LDHA/LDHB inhibitor (IC50s: 3/5 nM) and is 18-fold more potent than S enantiomer.Formule :C25H23ClN2O3S2Degré de pureté :98.25% - 98.91%Couleur et forme :SolidMasse moléculaire :499.04Lansoprazole sodium
CAS :Lansoprazole sodium is a PPI used to treat acid reflux and peptic ulcers.Formule :C16H13F3N3NaO2SDegré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :391.34
