
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.754 produits)
- Apoptose(6.187 produits)
- Cycle cellulaire/point de contrôle(4.807 produits)
- Chromatine/Épigénétique(2.573 produits)
- Signalisation du cytosquelette(1.503 produits)
- Altération de l'ADN/réparation de l'ADN(2.893 produits)
- Endocrinologie/Hormones(3.702 produits)
- Enzyme(3.671 produits)
- GPCR/G-Protéine(8.964 produits)
- Immunologie et Inflammation(3.697 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.246 produits)
- Transporteur membranaire/Canal ionique(3.137 produits)
- Métabolisme(10.096 produits)
- Microbiologie/Virologie(7.552 produits)
- Neuroscience(10.303 produits)
- Autres inhibiteurs(35.769 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.402 produits)
- Protéases/Protéasome(1.670 produits)
- Cellules souche et Dérivés(742 produits)
- Tyrosine Kinase/Adaptateurs(1.921 produits)
- Ubiquitination(1.716 produits)
Affichez 16 plus de sous-catégories
66573 produits trouvés pour "Inhibiteurs"
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D-Lin-MC3-DMA
CAS :D-Lin-MC3-DMA, an ionizable cationic lipid, is a potent siRNA delivery vehicle.Formule :C43H79NO2Degré de pureté :95% - 99.86%Couleur et forme :LiquidMasse moléculaire :642.09Ref: TM-T5823
1mg38,00€5mg82,00€10mg109,00€25mg205,00€50mg314,00€100mg470,00€500mg1.054,00€1mL*10mM (DMSO)105,00€3'-Methoxyflavonol
CAS :3'-Methoxyflavonol is a potent, selective agonist of neuromedin U 2 receptor (NMU2R).Formule :C16H12O4Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :268.26Fluazinam
CAS :Fluazinam: a pyridinamine fungicide, broad-spectrum, strongly inhibits S. sclerotiorum mycelial growth.Formule :C13H4Cl2F6N4O4Degré de pureté :98% - 99.98%Couleur et forme :Light Yellow CrystalsMasse moléculaire :465.09Taminadenant
CAS :Taminadenant is an adenosine receptor antagonist.Formule :C10H8BrN7Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :306.12Ref: TM-T16980
2mg34,00€5mg49,00€10mg84,00€25mg114,00€50mg166,00€100mg236,00€200mg353,00€1mL*10mM (DMSO)54,00€D-α-Methylbenzyl isothiocyanate
CAS :D-alpha-Methylbenzyl isothiocyanate, an antioxidant and a chiral agent, induces phase II enzyme activity.Formule :C9H9NSDegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :163.24Benznidazol
CAS :Benznidazol (Benznidazole)e has an antiprotozoal activity by interfering with parasite protein biosynthesis, influencing cytokines production and stimulatingFormule :C12H12N4O3Degré de pureté :99.53% - >99.99%Couleur et forme :SolidMasse moléculaire :260.25BOT-64
CAS :BOT-64 is an IKK-2 inhibitor which targets the Ser177 and/or Ser181 residues in the kinase's activation loop domain.BOT-64 is a cell-permeable benzoxathioleFormule :C15H15NO2SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :273.35Ref: TM-T8705
1mg50,00€5mg110,00€10mg170,00€25mg323,00€50mg494,00€100mg665,00€200mg893,00€1mL*10mM (DMSO)102,00€JNJ-38158471
CAS :JNJ-38158471 (CS-2660), a highly selective, orally available, well tolerated VEGFR2 inhibitor, inhibits closely related tyrosine kinases such as Ret and Kit .Formule :C15H17ClN6O3Degré de pureté :97.08%Couleur et forme :SolidMasse moléculaire :364.79Ref: TM-T22349
1mg38,00€5mg78,00€10mg103,00€25mg172,00€50mg250,00€100mg338,00€200mg464,00€1mL*10mM (DMSO)84,00€3-hydroxy-phthalicanhydrid
CAS :3-Hydroxyphthalic anhydride is used to synthesize 3-hydroxyphthalic anhydride modified human serum albumin.Formule :C8H4O4Degré de pureté :99.53%Couleur et forme :Beige PowderMasse moléculaire :164.12Tizoxanide
CAS :Tizoxanide (Desacetyl-nitazoxanide) is a metabolite of lamivudine.Formule :C10H7N3O4SDegré de pureté :98.89% - 99.28%Couleur et forme :SolidMasse moléculaire :265.25COG 133 Acetate
COG 133 Acetate, (C97H181N37O19) is a peptide with the sequence Ac-Leu-Arg-Val-Arg-Leu-Ala-Ser-His-Leu-Arg-Lys-Leu-Arg-Lys-Arg-Leu-Leu-amide.Formule :C99H185N37O21Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :2229.76Ref: TM-T21760L
1mg74,00€5mg202,00€10mg340,00€25mg472,00€50mg687,00€100mg938,00€1mL*10mM (DMSO)490,00€Raphin1
CAS :Raphin1 is an orally bioavailable, selective inhibitor of the regulatory phosphatase PPP1R15B (R15B).Formule :C8H8Cl2N4Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :231.08ML406
CAS :ML406 shows anti-tubercular activity via MtbbioA (DAPA synthase) enzyme inhibition(IC50 : 30 nM)Formule :C20H20N2O4Degré de pureté :98.69%Couleur et forme :SolidMasse moléculaire :352.38Pridopidine
CAS :Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.Formule :C15H23NO2SDegré de pureté :95.2% - 99.89%Couleur et forme :SolidMasse moléculaire :281.41SMCC
CAS :SMCC (N-Succinimidyl 4-(N-maleimidomethyl)cycl) is a heterobifunctional protein crosslinker.Formule :C16H18N2O6Degré de pureté :98.96% - 99.53%Couleur et forme :White Crystalline SolidMasse moléculaire :334.32M2N12
CAS :M2N12 selectively inhibits Cdc25C (IC50=0.09μM) and has anti-tumor properties, affecting Cdc25A and B as well.Formule :C20H16ClN5O2Degré de pureté :98.01%Couleur et forme :SolidMasse moléculaire :393.83Ref: TM-T11929
1mg84,00€5mg152,00€10mg236,00€25mg447,00€50mg670,00€100mg982,00€1mL*10mM (DMSO)167,00€Sarcosine
CAS :Sarcosine (Methylglycine) is a competitive inhibitor of the type I glycine transporter (GlyT1) and an N-methyl-D-aspartate receptor (NMDAR) co-agonist.Formule :C3H7NO2Degré de pureté :99.90%Couleur et forme :Deliquescent Water Soluble Physical Description Deliquescent Crystals Or Powder Has A Sweetish Taste (Ntp 1992)Masse moléculaire :89.092-Methylbutyraldehyde
CAS :2-Methylbutyraldehyde (2-Ethylpropanal) is a short-chain aldehyde compound and one of the burnt aroma substances in Atractylodes rhizome slices.Formule :C5H10ODegré de pureté :98.92%Couleur et forme :Colourless Clear LiquidMasse moléculaire :86.13Orthosphenic acid
CAS :Orthosphenic acid is a natural product isolated from M. triflora.Formule :C30H48O5Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :488.7Neuropeptide SF (human) acetate
Neuropeptide SF (human) aceate is a neuropeptide that augmented paraventricular CRH release and increased ACTH and corticosterone levels in the plasma.Formule :C67H98N18O17Degré de pureté :97.35%Couleur et forme :SolidMasse moléculaire :1427.61Flibanserin hydrochloride
CAS :Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.Formule :C20H22ClF3N4OCouleur et forme :SolidMasse moléculaire :426.87Aniline mustard
CAS :Aniline mustard (Mesylerythrol) is alkylating mustard with anti-neoplastic activity.Formule :C10H13Cl2NDegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :218.12Kv2-IN-A1
CAS :Kv2-IN-A1 is an inhibitor of Kv2.1 and Kv2.2.Formule :C20H17ClN4OSDegré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :396.89Mitiglinide
CAS :Mitiglinide (KAD-1229), an insulinotropic ATP-sensitive K+ channel antagonist, targets Kir6.2/SUR1; used in type 2 diabetes research.Formule :C19H25NO3Couleur et forme :SolidMasse moléculaire :315.412-Undecanol
CAS :2-Undecanol, a male pheromone from Lobiopa insularis, is also a floral volatile used by Hymenoptera species.Formule :C11H24ODegré de pureté :98%Couleur et forme :Clear Colorless LiquidMasse moléculaire :172.31Arabinose
CAS :Arabinose, a pentose sugar, is found in feces, cytoplasm, eukaryotes, sweet basil, and tamarind.Formule :C5H10O5Degré de pureté :98.71% - 99.93%Couleur et forme :Monoclinic Needles Or Prisms White Fine Crystalline PowderMasse moléculaire :150.13Talmapimod
CAS :Talmapimod (SCIO-469): Oral ATP-competitive p38α inhibitor, IC50 = 9 nM (p38α), 90 nM (p38β), >2000-fold selectivity over 20 kinases.Formule :C27H30ClFN4O3Degré de pureté :98% - 99.9%Couleur et forme :SolidMasse moléculaire :513Ref: TM-T12871
1mg50,00€2mg73,00€5mg109,00€10mg168,00€25mg358,00€50mg530,00€100mg758,00€1mL*10mM (DMSO)124,00€Mofezolac
CAS :Mofezolac (formerly known as Disopain or N-22) is a highly selective COX-1 (cyclooxygenase-1) inhibitor with COXs selectivity index > 6000Formule :C19H17NO5Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :339.34Fingolimod
CAS :Fingolimod (FTY-720A) is an antagonist of sphingosine 1-phosphate (S1P) (IC50 of 0.033 nM in K562 and NK cells).Formule :C19H33NO2Degré de pureté :99.53% - 99.6%Couleur et forme :SolidMasse moléculaire :307.47Ethyl potassium malonate
CAS :Ethyl potassium malonate, a competitive inhibitor of the enzyme succinate dehydrogenase, acts as a precursor to produce (trimethylsilyl)ethyl malonate, which isFormule :C5H7KO4Degré de pureté :99.71%Couleur et forme :White Crystals Or PowderMasse moléculaire :170.21Celosin H
CAS :Celosin H is a novel hepatoprotective triterpenoid saponin isolated from the methanol extract of Celosiae Semen.Formule :C47H72O20Degré de pureté :97.96% - 98.48%Couleur et forme :SolidMasse moléculaire :957.06GAL-021
CAS :GAL-021 an intravenous BKCa-channel blocker.Formule :C11H22N6ODegré de pureté :97.71% - 99.66%Couleur et forme :SolidMasse moléculaire :254.33Ref: TM-T3557
1mg34,00€5mg71,00€10mg98,00€25mg177,00€50mg268,00€100mg414,00€500mg888,00€1mL*10mM (DMSO)80,00€Anti-Inflammatory Peptide 1 Acetate
Anti-Inflammatory Peptide 1 Acetate (C45H82N12O14S2) inhibits PLA2 to reduce inflammation and pain.Formule :C47H86N12O16S2Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :1139.39Ref: TM-T21606L
2mg46,00€5mg64,00€10mg96,00€25mg138,00€50mg202,00€100mg301,00€200mg452,00€1mL*10mM (DMSO)150,00€Ethyl palmitate
CAS :Ethyl palmate (palmitic acid ethyl ester) is a type of fatty acid ethyl ester (FAEE). Ethyl palmate can be used as a hair and skin conditioner.Formule :C18H36O2Degré de pureté :98.93% - 99.87%Couleur et forme :LiquidMasse moléculaire :284.48Amlodipine camsylate
CAS :Amlodipine camsylate is a medication used to lower blood pressure and prevent chest pain.Formule :C30H41ClN2O9SCouleur et forme :SolidMasse moléculaire :641.17Decursinol angelate
CAS :Decursinol angelate is anti-tumor, anti-inflammatory, anti-oxidant, hepatoprotective, and inhibits VEGF and cancer cell invasion.Formule :C19H20O5Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :328.36Berbamine dihydrochloride
CAS :Berbamine dihydrochloride (Berbamine), a natural compound derived from the Berberis amurensis plant, has been shown to exhibit antitumor activity in several Ys.Formule :C37H42Cl2N2O6Degré de pureté :95% - 99.99%Couleur et forme :SolidMasse moléculaire :681.65RIPGBM
CAS :RIPGBM is a selective inducer of apoptosis in glioblastoma multiforme cancer stem cells (EC50: ≤500 nM).Formule :C26H21FN2O3Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :428.45Ref: TM-T16754
2mg35,00€5mg54,00€10mg93,00€25mg177,00€50mg318,00€100mg530,00€200mg677,00€1mL*10mM (DMSO)60,00€Sanguinarine
CAS :Sanguinarine (Pseudochelerythrine) is a specific inhibitor of Rac1b with anti-microbial, anti-oxidant and anti-inflammatory properties.Formule :C20H14NO4Degré de pureté :99.04% - 99.76%Couleur et forme :SolidMasse moléculaire :332.331-Furfurylpyrrole
CAS :1-Furfurylpyrrole is a potential contributor of flavor and aroma to popcorn.Formule :C9H9NODegré de pureté :97.85%Couleur et forme :LiquidMasse moléculaire :147.17Abscisic Acid
CAS :Abscisic Acid (Dormin) is a plant hormone, which is involved in many plant developmental processes, modulates ion homeostasis and metabolism.Formule :C15H20O4Degré de pureté :99.52% - 99.73%Couleur et forme :White PowderMasse moléculaire :264.32HCH6-1
CAS :HCH6-1 is a competitive Formyl peptide receptor 1 (FPR1) antagonist.Formule :C28H27N3O4Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :469.53Ref: TM-T8313
1mg60,00€2mg87,00€5mg133,00€10mg203,00€25mg376,00€50mg563,00€100mg800,00€1mL*10mM (DMSO)147,00€Ginsenoside Rf
CAS :Ginsenoside Rf (Panaxoside Rf) is a trace component of ginseng root. Ginsenoside Rf inhibits N-type Ca2+ channel.Formule :C42H72O14Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :801.01Rhapontin
CAS :Rhapontin may reduce liver fat and better blood sugar/lipids, showing potential for treating type 2 diabetes.Formule :C21H24O9Degré de pureté :99% - 99.91%Couleur et forme :Light YellowMasse moléculaire :420.414-Methylumbelliferyl phosphate
CAS :4-Methylumbelliferyl phosphate (4-MUP) (4-MUP) is used as a fluorogenic substrate of alkaline phosphatases.Formule :C10H9O6PDegré de pureté :99.13% - 99.497%Couleur et forme :White Crystalline PowderMasse moléculaire :256.152-Hydroxy-4-methoxybenzaldehyde
CAS :2-Hydroxy-4-methoxybenzaldehyde (4-Methoxysalicylaldehyde) is an isomer of Vanillin, and a potent tyrosinase inhibitor, could be used to synthesis Urolithin M7.
Formule :C8H8O3Degré de pureté :99.78%Couleur et forme :Colorless Needle-Like CrystalMasse moléculaire :152.15Ganoderic acid C1
CAS :Ganoderic acid C1: Anti-inflammatory, may treat asthma-related inflammation, anti-tumor, inhibits HIV-1 protease.Formule :C30H42O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :514.65Juglone
CAS :Juglone is a naphthoquinone from walnut and Juglandaceae, inhibits peptidyl-prolyl isomerases, RNA polymerases, and reduces rat kidney fibrosis.Formule :C10H6O3Degré de pureté :99.24%Couleur et forme :Red PowderMasse moléculaire :174.15Tianeptine
CAS :Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。Formule :C21H25ClN2O4SDegré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :436.95Benoxacor
CAS :Benoxacor (BRN-4190275) is an inert agricultural chemical. Benoxacor acts as an herbicide safener to protect crops from herbicide toxicity.Formule :C11H11Cl2NO2Degré de pureté :99.97%Couleur et forme :White SolidMasse moléculaire :260.12GluR6 antagonist-1
CAS :GluR6 antagonist-1 inhibits the pY binding site of tyrosine kinase p56lck SH2 domain.Formule :C15H11ClN2OSDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :302.78Arg-Gly-Asp TFA (99896-85-2(free base))
Arg-Gly-Asp TFA (RGD, 99896-85-2) is a tripeptide that promotes cell adhesion and integrin binding.Formule :C14H23F3N6O8Degré de pureté :99.2% - ≥98%Couleur et forme :SolidMasse moléculaire :460.36Fibrinogen-Binding Peptide fb-acetate
Fibrinogen-Binding Peptide mimics vitronectin site; blocks platelet adhesion to fibrinogen/vitronectin and aggregation.Formule :C31H51N7O10Degré de pureté :96.76%Couleur et forme :SolidMasse moléculaire :681.8(±)-Ibipinabant
CAS :(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Formule :C23H20Cl2N4O2SDegré de pureté :99.28% - 99.83%Couleur et forme :SolidMasse moléculaire :487.4Betazole dihydrochloride
CAS :Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.
Formule :C5H11Cl2N3Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :184.067T56-LIMKi
CAS :T56-LIMKi (T5601640) is a selective inhibitor of LIMK2.Formule :C19H14F3N3O3Degré de pureté :98.39% - 99.57%Couleur et forme :SolidMasse moléculaire :389.334-Oxofenretinide
CAS :4-Oxofenretinide (3-Keto fenretinide) , a recently identified fenretinide metabolite, induces marked G2-M cell cycle arrest and apoptosis.Formule :C26H31NO3Degré de pureté :96.89%Couleur et forme :SolidMasse moléculaire :405.53Ref: TM-T4189
1mg42,00€2mg52,00€5mg74,00€10mg107,00€25mg185,00€50mg278,00€100mg500,00€1mL*10mM (DMSO)90,00€Shanzhiside methyl ester
CAS :Shanzhiside methylester soothes neuropathic pain by triggering spinal GLP-1 receptors, boosting microglial β-endorphin through p38 MAPK.Formule :C17H26O11Degré de pureté :98.998% - 99.32%Couleur et forme :SolidMasse moléculaire :406.38Alectinib
CAS :Alectinib (RG-7853) is an ALK inhibitor that is selective, orally active, and ATP-competitive. Alectinib has antitumor activity. Cost-effective and quality-assured.Formule :C30H34N4O2Degré de pureté :98% - 99.38%Couleur et forme :SolidMasse moléculaire :482.62Ref: TM-T1936
2mg47,00€5mg69,00€10mg87,00€50mg105,00€100mg168,00€200mg259,00€500mg437,00€1mL*10mM (DMSO)73,00€Co 101244 hydrochloride
CAS :Co 101244 hydrochloride (4-Piperidinol, 1-[2-(4-hydroxyphenoxy)ethyl]-4-[(4-Methylphenyl)Methyl]-,hydrochloride) is an NR2B-containing NMDA receptor antagonist.Formule :C21H28ClNO3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :377.9Tomatine
CAS :Tomatine (lycopersicin) is an antiproliferatve agent of breast adenocarcinoma cells.Formule :C50H83NO21Degré de pureté :98.42% - 99.94%Couleur et forme :White To Light YellowMasse moléculaire :1034.19(±)-Praeruptorin A
CAS :(±)-Praeruptorin A could exhibit its anti-osteoclastogenic activity by inhibiting p38/Akt-c-Fos-NFATc1 signaling and PLCγ-independent Ca(2+) oscillation.Formule :C21H22O7Degré de pureté :98.9% - 99.73%Couleur et forme :SolidMasse moléculaire :386.40Alflutinib mesylate
CAS :Alflutinib mesylate (AST2818 mesylate) ,is an irreversible tyrosine kinase inhibitor that selectively inhibits EGFR mutations, especially T790M.Formule :C29H35F3N8O5SDegré de pureté :97.94% - 99.63%Couleur et forme :SolidMasse moléculaire :664.70Irisflorentin
CAS :Irisflorentin prevents cell death, boosts proteasomes via rpn-3, reduces egl-1, and lowers iNOS/NO in LPS-stimulated macrophages.Formule :C20H18O8Degré de pureté :98.6% - 99.81%Couleur et forme :SolidMasse moléculaire :386.35Licorice-saponin H2
CAS :Licorice-saponin H2 (Licoricesaponin H2) is a natural productFormule :C42H62O16Degré de pureté :99.58% - 99.76%Couleur et forme :SolidMasse moléculaire :822.93L-Argininamide dihydrochloride
CAS :L-Argininamide dihydrochloride aids research in DNA ligand binding studies and fluorescent aptasensor development.Formule :C6H17Cl2N5ODegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :246.14Piperaquine tetraphosphate tetrahydrate
CAS :Piperaquine tetraphosphate tetrahydrate is a potent anti-parasites agent.Formule :C29H32Cl2N6·4H3O4P·4H2ODegré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :999.6Ethoxyacetic acid
CAS :Ethoxyacetic acid is an endogenous metabolite of ethylene glycol monoethyl ether acetate.
Formule :C4H8O3Degré de pureté :≥98%Couleur et forme :Physical Description Liquid (Ntp 1992)Masse moléculaire :104.1Purine
CAS :Purine: an aromatic compound with fused pyrimidine & imidazole rings, turned into uric acid by enzymes; excessive uric acid can lead to gout.Formule :C5H4N4Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :120.11Fumaric acid
CAS :Fumaric acid reduces eotaxin-1 in TNF-α-activated fibroblasts via p38 MAPK/NF-κB. It's an oncometabolite found in high levels in tumors.Formule :C4H4O4Degré de pureté :98.77% - 98.80%Couleur et forme :Colorless Needles Monoclinic Prisms Or Leaflets From Water Solid CrystallineMasse moléculaire :116.07Fexofenadine
CAS :Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.Formule :C32H39NO4Degré de pureté :99.35%Couleur et forme :White To Off-White SolidMasse moléculaire :501.66L-Kynurenine
CAS :L-Kynurenine ((S)-Kynurenine)) is an endogenous agonist of aryl hydrocarbon receptor (AHR) ,inhibits allogeneic T cell proliferation. High-Quality, Low-Cost!Formule :C10H12N2O3Degré de pureté :98.44% - 99.91%Couleur et forme :Light Yellow CrystallineMasse moléculaire :208.21CID-1067700
CAS :CID-1067700 is one of the first identified competitive inhibitors of nucleotide binding by Ras-related GTPases(Rab7 with a Ki of 13 nM).Formule :C18H18N2O4S2Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :390.48Ref: TM-T7558
1mg34,00€2mg49,00€5mg71,00€10mg105,00€25mg178,00€50mg234,00€100mg303,00€1mL*10mM (DMSO)78,00€Tiagabine
CAS :Tiagabine (NO050328) is an Anti-epileptic Agent.Formule :C20H25NO2S2Degré de pureté :99.25% - 99.67%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :375.55Hemiphloin
CAS :Hemiphloin: natural flavonoid with anti-inflammatory properties, potential skin disease therapy.Formule :C21H22O10Degré de pureté :99.26% - 99.95%Couleur et forme :SolidMasse moléculaire :434.39AZ505
CAS :AZ505 is an effective and specific SMYD2 inhibitor (IC50: 0.12 μM).Formule :C29H38Cl2N4O4Degré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :577.54Ref: TM-TQ0100
1mg60,00€5mg130,00€10mg178,00€25mg295,00€50mg462,00€100mg623,00€1mL*10mM (DMSO)165,00€Crizotinib
CAS :Crizotinib (PF-02341066) is an ATP-competitive small-molecule tyrosine kinases inhibitor of c-MET (IC50: 8 nM) and ALK (IC50: 20 nM) receptor.Formule :C21H22Cl2FN5ODegré de pureté :99% - 99.87%Couleur et forme :SolidMasse moléculaire :450.34Ref: TM-T1661
2mgÀ demander5mg33,00€10mg49,00€25mg55,00€50mg64,00€100mg88,00€500mg147,00€1mL*10mM (DMSO)50,00€Cuminaldehyde
CAS :Cuminaldehyde: a natural anti-fibrillation aldehyde with anticancer properties and a pleasant aroma.Formule :C10H12ODegré de pureté :98%Couleur et forme :Colourless LiquidMasse moléculaire :148.2JNJ-31020028
CAS :JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, human; pIC50=8.22, rat).Formule :C34H36FN5O2Degré de pureté :95.92% - 99.65%Couleur et forme :SolidMasse moléculaire :565.68Orobol
CAS :Orobol (3’,4’,5,7-tetrahydroxy-isoflavon) is an inhibitor of tyrosine-specific protein kinase and phosphatidylinositol turnover.Formule :C15H10O6Degré de pureté :98% - 98%Couleur et forme :SolidMasse moléculaire :286.24Huperzine B
CAS :1.
Formule :C16H20N2ODegré de pureté :99.83% - ≥95%Couleur et forme :SolidMasse moléculaire :256.34GW604714X
CAS :GW604714X (2,4-Thiazolidinedione, 5-[[5-[6-(4-acetyl-1-piperazinyl)-3-nitro-2-pyridinyl]-2-fluorophenyl]methylene]-) were found to be potent inhibitors ofFormule :C21H18FN5O5SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :471.46TTA-A2
CAS :TTA-A2: T-type calcium channel blocker; anticonvulsant targeting Cav3.1, Cav3.2; IC50 of 89/92 nM; potential for treating neurological conditions.Formule :C20H21F3N2O2Degré de pureté :99.5% - 99.9%Couleur et forme :SolidMasse moléculaire :378.39Ref: TM-T8944
1mg99,00€5mg241,00€10mg385,00€25mg707,00€50mg1.009,00€100mg1.333,00€1mL*10mM (DMSO)265,00€Rebastinib
CAS :DCC-2036 (Rebastinib (DCC-2036)) is a conformational control Bcr-Abl inhibitor for Abl1(WT, IC50: 0.8 nM) and Abl1(T315I, IC50: 4 nM), also inhibits LYN, SRC,
Formule :C30H28FN7O3Degré de pureté :99.53% - 99.79%Couleur et forme :SolidMasse moléculaire :553.59MI-136
CAS :MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.Formule :C23H21F3N6SDegré de pureté :98.63% - 99.12%Couleur et forme :SolidMasse moléculaire :470.51Ref: TM-T6889
1mg44,00€5mg93,00€10mg140,00€25mg264,00€50mg447,00€100mg692,00€200mg964,00€1mL*10mM (DMSO)92,00€Vonoprazan
CAS :Vonoprazan (TAK-438 (free base)) is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduodenal ulcer andFormule :C17H16FN3O2SDegré de pureté :99.87% - 99.92%Couleur et forme :SolidMasse moléculaire :345.393-Methoxyphenylethylamine
CAS :3-Methoxyphenylethylamine 是一种生物活性化学品。Formule :C9H13NODegré de pureté :97.07%Couleur et forme :Less Liquid Colorless LiquidMasse moléculaire :151.21Glycylsarcosine
CAS :Glycylsarcosine (GLYCYL-SARCOSINE) is a dipeptide obtained by formal condensation of the carboxy group of glycine with the amino group of sarcosineFormule :C5H10N2O3Degré de pureté :98.47%Couleur et forme :SolidMasse moléculaire :146.14Esomeprazole Sodium
CAS :Esomeprazole Sodium ((S)-Omeprazole sodium) is the S-isomer of omeprazole with selective and irreversible proton pump inhibitor activity.Formule :C17H18N3O3S·NaDegré de pureté :98.17% - >99.99%Couleur et forme :SolidMasse moléculaire :367.4Gossypol
CAS :Gossypol (BL 193) Acetate is a polyphenolic aldehyde that permeates cells and acts as an inhibitor for several dehydrogenase enzymes.Formule :C30H30O8Degré de pureté :98.52% - 99.89%Couleur et forme :SolidMasse moléculaire :518.55GSK-2881078
CAS :GSK-2881078 is a selective androgen receptor modulato (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting.Formule :C14H13F3N2O2SDegré de pureté :98.16% - 98.81%Couleur et forme :SolidMasse moléculaire :330.33Cichoric Acid
CAS :Cichoric Acid (Dicaffeoyltartaric acid) is a potent inhibitor of human immunodeficiency virus type-1 (HIV-1) integrase and the replication in tissues.Formule :C22H18O12Degré de pureté :97.87% - 98.77%Couleur et forme :SolidMasse moléculaire :474.37Pomalidomide-C7-NH2 hydrochloride
CAS :Pomalidomide-C7-NH2 HCl, a synthetic E3 ligase ligand-linker for PROTAC, with CRBN ligand.Formule :C20H26N4O4Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :386.44Glycyl-glutamine
CAS :Glycyl-glutamine (Glycyl-L-glutamine monohydrate) is an inhibitory neuropeptide derived from beta-endorphin.Formule :C7H13N3O4Degré de pureté :99.51%Couleur et forme :White Solid CrystallineMasse moléculaire :203.2Timosaponin B III
CAS :Timosaponin B III (Anemarsaponin BIII) is a bioactive steroidal saponin isolated from Anemarrhena asphodeloides Bge.Formule :C45H74O18Degré de pureté :98% - 99.75%Couleur et forme :SolidMasse moléculaire :903.06FR 180204
CAS :FR 180204 is a potent and selective ATP-competitive inhibitor of ERK1 and ERK2.Formule :C18H13N7Degré de pureté :98% - 99.74%Couleur et forme :SolidMasse moléculaire :327.34Ref: TM-T1956
1mg43,00€2mg55,00€5mg86,00€10mg138,00€25mg221,00€50mg331,00€100mg497,00€1mL*10mM (DMSO)94,00€PKR-IN-C16
CAS :PKR-IN-C16: inhibits PKR autophosphorylation and translation blockade; binds ATP site; IC50 of 186-210 nM; protects cells from ER stress damage.Formule :C13H8N4OSDegré de pureté :97.8%Couleur et forme :SolidMasse moléculaire :268.29Ref: TM-T16550
1mg40,00€2mg52,00€5mg84,00€10mg130,00€25mg260,00€50mg409,00€100mg605,00€1mL*10mM (DMSO)105,00€Abl Cytosolic Substrate acetate
Abl Cytosolic Substrate acetate is a substrate for Abelson tyrosine kinase (Abl ).Formule :C66H105N15O18Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1396.65MC-Gly-Gly-Phe
CAS :MC-Gly-Gly-Phe is a cleavable linker. MC-Gly-Gly-Phe can be used for antibody-drug conjugates (ADC).Formule :C23H28N4O7Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :472.49CBL0137 hydrochloride
CAS :CBL0137 hydrochloride (Curaxin-137 hydrochloride) is an inhibitor of the histone chaperone FACT, which also activates p53 and inhibits NF-κB.Cost-effective and quality-assured.Formule :C21H25ClN2O2Degré de pureté :99.35% - 99.86%Couleur et forme :SolidMasse moléculaire :372.88
