Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.833 produits)
- Apoptose(6.315 produits)
- Cycle cellulaire/point de contrôle(4.875 produits)
- Chromatine/Épigénétique(2.613 produits)
- Signalisation du cytosquelette(1.567 produits)
- Altération de l'ADN/réparation de l'ADN(2.872 produits)
- Endocrinologie/Hormones(3.754 produits)
- Enzyme(3.672 produits)
- GPCR/G-Protéine(9.019 produits)
- Immunologie et Inflammation(3.904 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(415 produits)
- Signalisation MAPK(1.257 produits)
- Transporteur membranaire/Canal ionique(3.155 produits)
- Métabolisme(10.137 produits)
- Microbiologie/Virologie(7.620 produits)
- Neuroscience(10.446 produits)
- Autres inhibiteurs(35.847 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.429 produits)
- Protéases/Protéasome(1.691 produits)
- Cellules souche et Dérivés(732 produits)
- Tyrosine Kinase/Adaptateurs(1.982 produits)
- Ubiquitination(1.726 produits)
Affichez 16 plus de sous-catégories
66515 produits trouvés pour "Inhibiteurs"
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Ibandronate sodium monohydrate
CAS :Ibandronate sodium monohydrate (BM-210955) is a highly potent nitrogen-containing bisphosphonate used for the treatment of osteoporosis.Formule :C9H24NNaO8P2Degré de pureté :99.62%Couleur et forme :White Crystalline PowderMasse moléculaire :359.23Mesaconine
CAS :Mesaconine is an ingredient from Aconitum carmichaelii Debx..Formule :C24H39NO9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :485.57Apabetalone
CAS :Apabetalone (RVX000222) , an effective BET bromodomain inhibitor, has been investigated for the treatment of diabetes, atherosclerosis, and coronary arteryFormule :C20H22N2O5Degré de pureté :98.08% - ≥98%Couleur et forme :SolidMasse moléculaire :370.41-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID
CAS :1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.
Formule :C13H13NO5Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :263.25Trelagliptin succinate
CAS :Trelagliptin succinate (SYR-472 succinate) is a long-acting inhibitor of dipeptidyl peptidase-4 (DPP-4), being developed for the treatment of type 2 diabetes (Formule :C22H26FN5O6Degré de pureté :99.27% - 99.92%Couleur et forme :SolidMasse moléculaire :475.473-O-β-D-Glucopyranosylplatycodigenin
CAS :3-O-beta-D-Glucopyranosylplatycodigenin is isolated from the roots of Platycodon grandiflorum.Formule :C36H58O12Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :682.84Madecassoside
CAS :Madecassoside (Asiaticoside A) is a pentacyclic triterpene extracted from Centella asitica (L.) with anti-inflammatory, anti-oxidative and anti-aging activitiesFormule :C48H78O20Degré de pureté :99.46% - 99.85%Couleur et forme :White PowderMasse moléculaire :975.12Ref: TM-T2813
10mg49,00€25mg84,00€50mg120,00€100mg178,00€200mg289,00€500mg485,00€1mL*10mM (DMSO)49,00€TSPC
CAS :TSPC is an inhibitor for GA perception by in vitro and in planta evaluations.Formule :C9H5N3O2S2Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :251.28Methyl Aminolevulinate Hydrochloride
CAS :Methyl Aminolevulinate Hydrochloride (5-Aminolevulinic acid methyl ester) is used in photosentizer reagents for photodynamic therapy to treat conditions.Formule :C6H12ClNO3Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :181.62Levomefolate calcium
CAS :Levomefolate calcium is an artificial form of folate. It is a coenzymated form of folic acid and a more bioavailable alternative in dietary supplements.Formule :C20H23CaN7O6Degré de pureté :97.35%Couleur et forme :Off-White To Pale Yellow SolidMasse moléculaire :497.52Lilial
CAS :Lilial, also lysmeral or butylphenyl methylpropional, is a lily-scented perfume ingredient in cosmetics and laundry detergents.Formule :C14H20ODegré de pureté :97.28%Couleur et forme :LiquidMasse moléculaire :204.314-Ethylphenol
CAS :4-Ethylphenol is the volatile phenol associated with the aroma in wine.Formule :C8H10ODegré de pureté :97.76%Couleur et forme :Colorless Or White Needles; Tend To Yellow On Exposure To Light LiquidMasse moléculaire :122.16AT-9283 HCl
CAS :AT-9283, a multi-targeted kinase inhibitor, is used potentially for the treatment of multiple myeloma.Formule :C19H24ClN7O2Couleur et forme :SolidMasse moléculaire :417.895'-Guanylic acid disodium salt
CAS :5'-Guanylic acid disodium salt (GMP-5) belongs to the class of organic compounds known as purine ribonucleoside monophosphates.
Formule :C10H14N5Na2O9PDegré de pureté :99.87% - >99.99%Couleur et forme :Odourless Colourless Or White Crystals Or White Crystalline PowderMasse moléculaire :425.20LY3405105
CAS :LY3405105 (1-Piperidinecarboxylic acid, 4-[[5-methyl-3-(1-methylethyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino]-, 1-[(2E)-4-(dimethylamino)-1-oxo-2-buten-1-yl]-3-Formule :C26H39N7O3Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :497.636-(4-Methoxyphenyl)-3-pyridazinamine
CAS :6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonistFormule :C11H11N3ODegré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :201.22Corynoxeine
CAS :Corynoxeine inhibits ERK1/2, curbs VSMC growth induced by PDGF-BB, and may prevent vascular diseases and restenosis post-angioplasty.Formule :C22H26N2O4Degré de pureté :98.61% - 99.94%Couleur et forme :SolidMasse moléculaire :382.45GS-441524
CAS :GS-441524 treatment of cats with naturally occurring feline infectious peritonitis.Formule :C12H13N5O4Degré de pureté :98.78% - 99.75%Couleur et forme :SolidMasse moléculaire :291.26(R)-MG-132
CAS :(R)-MG-132 (Z-Leu-D-leu-leu-al) is the enantiomer of MG-132. (R)-MG-132 stereoisomer is a more potent proteasome inhibitor than MG-132.Formule :C26H41N3O5Degré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :475.62Ref: TM-T12628
2mg38,00€5mg57,00€10mg79,00€25mg120,00€50mg177,00€100mg268,00€200mg398,00€1mL*10mM (DMSO)71,00€(2-Chloropyridin-4-yl)MethanaMine Hydrochloride
CAS :(2-Chloropyridin-4-yl)methanamine hydrochloride is a selective LOXL2 inhibitor(IC50 : 126 nM).Formule :C6H8Cl2N2Degré de pureté :97.23%Couleur et forme :SolidMasse moléculaire :179.05BPC 157 acetate(137525-51-0 free base)
BPC 157 acetate(137525-51-0 free base) is a 15-amino acid fragment of a gastric peptide (BPC) which has hepatoprotective effects.Formule :C64H102N16O24Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1479.61H3B-5942
CAS :H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).Formule :C31H34N4O2Degré de pureté :98.06% - ≥95%Couleur et forme :SolidMasse moléculaire :494.63Ref: TM-T5633
1mg51,00€5mg111,00€10mg167,00€25mg324,00€50mg462,00€100mg615,00€200mg830,00€1mL*10mM (DMSO)116,00€Tetradehydrothalictrifoline
CAS :Tetradehydrothalictrifoline is a nature product.
Formule :C21H20NO4Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :350.39Methyl 3-phenylpropanoate
CAS :Methyl 3-phenylpropanoate (3-Phenylpropionic acid methyl ester) is a huamn endogenous metabolite.Formule :C10H12O2Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :164.2Sapanisertib
CAS :Sapanisertib (INK 128) is an oral raptor-mTOR and rictor-mTOR inhibitor with potential cancer-fighting properties.Formule :C15H15N7ODegré de pureté :99.19% - >99.99%Couleur et forme :SolidMasse moléculaire :309.33Ref: TM-T1838
1mg40,00€2mg51,00€5mg85,00€10mg96,00€25mg160,00€50mg235,00€100mg350,00€500mg838,00€1mL*10mM (DMSO)88,00€Trachelanthine
CAS :Trachelanthine is a natural product from Eupatorium fortunei.Formule :C15H27NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :301.38BDP-13176
CAS :BDP-13176 is a potent inhibitor of fascin 1(Kd of 90 nM and an IC50 of 240 nM). It has potential as an anti-metastatic agentFormule :C24H22Cl2N6O2Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :497.38MSX-127
CAS :MSX-127 elicites positive response in peptide CXCR4.Formule :C16H24N2O4Degré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :308.37(S)-Afatinib
CAS :(S)-Afatinib (BIBW2992) is an irreversible EGFR family inhibitor with IC50s of 0.5/0.4/10/14/1 nM for EGFRwt, L858R, L858R/T790M, HER2, and HER4, respectively.Formule :C24H25ClFN5O3Degré de pureté :99.22% - >99.99%Couleur et forme :Off-White SolidMasse moléculaire :485.9426RFa acetate
26RFa acetate is a hypothalamic neuropeptide with orexigenic activity in mammals[1].Formule :C129H201N37O38Degré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :2878.23,5,7,3′,4′-Pentamethoxyflavone
CAS :3,5,7,3′,4′-Pentamethoxyflavone (Quercetin 3,5,7,3,4-pentamethyl ether) is a natural product. It can induce adipogenesis on 3T3-L1 preadipocytes.Formule :C20H20O7Degré de pureté :98.87% - 99.73%Couleur et forme :SolidMasse moléculaire :372.372',7'-Dichlorofluorescein diacetate
CAS :2',7'-Dichlorofluorescein diacetate is a probe for tracking NO, ROS, and measuring oxidative stress.Formule :C24H14Cl2O7Degré de pureté :99.08% - 99.6%Couleur et forme :Off-White Crystal PowderMasse moléculaire :485.27Cichoric Acid
CAS :Cichoric Acid (Dicaffeoyltartaric acid) is a potent inhibitor of human immunodeficiency virus type-1 (HIV-1) integrase and the replication in tissues.Formule :C22H18O12Degré de pureté :97.87% - 98.77%Couleur et forme :SolidMasse moléculaire :474.37Eclitasertib
CAS :Eclitasertib is a potent inhibitor of receptor-interacting protein kinase 1 (RIPK1, IC50 of <1 µΜ).Formule :C19H18N6O3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :378.38Ref: TM-T9702
1mg101,00€2mg142,00€5mg215,00€10mg340,00€25mg618,00€50mg858,00€100mg1.224,00€1mL*10mM (DMSO)236,00€SYR127063
CAS :SYR127063 (BDBM-92454) (BDBM92454) is a potent and selective HER2 inhibitor, binds to HER2 in a reactive conformation.Formule :C23H20ClF3N4O3Degré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :492.88MLN8054 sodium
CAS :MLN8054 sodium is an Aurora A inhibitor.Formule :C25H14ClF2N4NaO2Couleur et forme :SolidMasse moléculaire :498.84Wogonoside
CAS :Wogonoside (Wogonin 7-O-glucuronide) acts as a positive allosteric modulator of the benzodiazepine site of the GABAA receptor.
Formule :C22H20O11Degré de pureté :98.24% - >99.99%Couleur et forme :SolidMasse moléculaire :460.39Sinapine
CAS :Sinapine: an alkaloid with chemo-resistance, antioxidant, and radioprotective properties from cruciferous seeds.Formule :C16H24NO5Degré de pureté :98% - 99.68%Couleur et forme :White Or Light-Tan SolidMasse moléculaire :310.37Bromosporine
CAS :Bromosporine is a broad spectrum inhibitor for bromodomains for BRD2/4/9 and CECR2 (IC50: 0.41/0.29/0.122/0.017 μM), respectively.Formule :C17H20N6O4SDegré de pureté :99.65% - 99.79%Couleur et forme :SolidMasse moléculaire :404.44Ref: TM-T6255
1mg44,00€2mg57,00€5mg93,00€10mg133,00€25mg260,00€50mg416,00€100mg665,00€200mg888,00€1mL*10mM (DMSO)92,00€Amifostine trihydrate
CAS :Amifostine trihydrate (WR2721) is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.Formule :C5H15N2O3PS·3H2ODegré de pureté :99.71% - 99.80%Couleur et forme :SolidMasse moléculaire :268.27Fanotaprim
CAS :Fanotaprim is a dihydrofolate reductase (DHFR) inhibitor.Formule :C19H22N8ODegré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :378.43Ref: TM-T36692
1mg50,00€2mg71,00€5mg110,00€10mg170,00€25mg318,00€50mg442,00€100mg627,00€200mg845,00€1mL*10mM (DMSO)122,00€NSC 73150
CAS :6-Methyl-1H-pyrimidin-4-one (NSC 73150) shows antitumor effects, impeding growth in breast, lung, liver cancer, and inducing apoptosis.Formule :C12H12N4O2Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :244.25Ref: TM-T9398
1mg87,00€5mg192,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€200mg1.130,00€1mL*10mM (DMSO)170,00€AS8351
CAS :AS8351 inhibits histone demethylase, used with various compounds to turn human lung fibroblasts into cardiomyocytes.Formule :C17H13N3O2Degré de pureté :99.54% - 99.72%Couleur et forme :SolidMasse moléculaire :291.3Ref: TM-T4100
5mg48,00€10mg66,00€25mg110,00€50mg178,00€100mg333,00€200mg432,00€500mg707,00€1mL*10mM (DMSO)49,00€Articaine
CAS :Articaine (Hoe-045 free base), an amide anesthetic featuring an ester group, effectively relieves pain by reversibly binding to the α-subunit of the voltage-Formule :C13H20N2O3SCouleur et forme :SolidMasse moléculaire :284.37Quilseconazole
CAS :Quilseconazole is an effective, orally active fungal Cyp51 inhibitor. it also binds tightly to cryptococcal CYP51 but weakly inhibits humans CYP450 enzymes.Formule :C22H14F7N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :513.37Veratramine
CAS :Veratramine (NSC-23880)(NSC-17821; NSC-23880) is a potent signal transduction inhibitor for treating tumors.Formule :C27H39NO2Degré de pureté :99.7% - 99.75%Couleur et forme :SolidMasse moléculaire :409.60Brexpiprazole HCl
CAS :Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.Formule :C25H27N3O2S·xHClDegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :433.6Ref: TM-T8690
1mg124,00€5mg271,00€10mg408,00€25mg672,00€50mg945,00€100mg1.279,00€500mg2.547,00€1mL*10mM (DMSO)319,00€FRAX486 HCL(1232030-35-1 free base)
FRAX486 HCL is a potent p21-activated kinase (PAK) inhibitor with IC50 values of 14, 33, 39 and 575 nM for PAK1, PAK2, PAK3 and PAK4 respectively.Formule :C25H24Cl3FN6ODegré de pureté :98.85% - 99.82%Couleur et forme :SolidMasse moléculaire :549.86Chlorotoluron
CAS :Chlorotoluron (Dicuran), a phenylurea herbicide, targets broad-leaved weeds in winter cereals.Formule :C10H13ClN2ODegré de pureté :99.61%Couleur et forme :Colorless Crystals Colourless Crystals Or White PowderMasse moléculaire :212.68Cdk5 Substrate acetate
Cdk5, a serine/threonine kinase active in neurons, phosphorylates proteins like histone H1; its synthetic substrate has a Km of 5 µM.Formule :C55H103N15O14Degré de pureté :96.21%Couleur et forme :SolidMasse moléculaire :1198.5Spinosad
CAS :Spinosad: natural insecticide from S. spinosa, mix of spinosyn A & D, targets insect nAChRs.Formule :C41H65NO10Degré de pureté :99.06% - >99.99%Couleur et forme :Solid PowderMasse moléculaire :731.96Glypromate acetate(32302-76-4 free base)
Glypromate acetate is a neuroprotective agent, is a weak NMDA receptor agonist.Formule :C14H23N3O8Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :361.35Ref: TM-T7778L
2mg37,00€5mg52,00€10mg74,00€25mg119,00€50mg160,00€100mg225,00€200mg314,00€1mL*10mM (DMSO)57,00€Ζ-Stat
CAS :ζ-Stat (NSC37044), a specific and atypical inhibitor of PKC-ζ with an IC50 of 5 μM, demonstrates the ability to inhibit proliferation and induce apoptosis inFormule :C10H8O10S3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :384.36Hexa-D-arginine
CAS :Hexa-D-arginine is an inhibitor of furin,blocks the activation of Pseudomonas aeruginosa exotoxin A in vivo.Formule :C36H75N25O6Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :954.14MS-049 oxalate salt
CAS :MS-049 oxalate salt is a potent and selective inhibitor of protein arginine methyltransferases (PRMTs) PRMT 4 and PRMT6.Formule :C17H26N2O5Couleur et forme :SolidMasse moléculaire :338.4NSC 405020
CAS :NSC 405020 is a noncatalytic inhibitor of MT1-MMP.Formule :C12H15Cl2NODegré de pureté :96.93% - 99.07%Couleur et forme :SolidMasse moléculaire :260.16PF-06454589
CAS :PF-06454589 is a potent inhibitor of LRRK2.Formule :C14H16N6ODegré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :284.32Ref: TM-T7729
2mg34,00€5mg52,00€10mg75,00€25mg128,00€50mg187,00€100mg290,00€200mg419,00€1mL*10mM (DMSO)52,00€Capmatinib 2HCl.H2O
CAS :Capmatinib 2HCl.H2O (NVP-INC280 2HCl.H2O) is an orally bioavailable inhibitor of the proto-oncogene c-Met (HGFR)with potential antineoplastic activity.Formule :C23H21Cl2FN6O2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :503.36Ref: TM-T8825
2mg34,00€5mg48,00€10mg63,00€25mg84,00€50mg92,00€100mg126,00€500mg250,00€1mL*10mM (DMSO)50,00€ARS-1620
CAS :ARS-1620 is a covalent inhibitor of K-RASG12C.Formule :C21H17ClF2N4O2Degré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :430.84Protein kinase inhibitors 1 hydrochlorid
Protein kinase inhibitors 1 hydrochlorid (Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base))) is a novel inhibitor of HIPK2 with an IC50 of 74Formule :C18H18ClN5O3SDegré de pureté :98.00% - 98.78%Couleur et forme :SolidMasse moléculaire :419.88TW-37
CAS :TW-37 is an nonpeptide inhibitor to recombinant Bcl-2, Bcl-xL and Mcl-1 (Ki: 0.29/1.11/0.26 μM).Formule :C33H35NO6SDegré de pureté :97.06% - ≥95%Couleur et forme :SolidMasse moléculaire :573.7Ref: TM-T6281
1mg38,00€2mg50,00€5mg65,00€10mg107,00€25mg202,00€50mg334,00€100mg495,00€1mL*10mM (DMSO)90,00€3,5,6,7,8,3',4'-Heptemthoxyflavone
CAS :3,5,6,7,8,3',4'-Heptemthoxyflavone has neuroprotective, chemopreventive, anti-allergic, anti-inflammatory, immunomodulatory, and photoprotective effects.Formule :C22H24O9Degré de pureté :99.38% - 99.93%Couleur et forme :SolidMasse moléculaire :432.42Ref: TM-TN1088
1mg93,00€5mg200,00€10mg295,00€25mg497,00€50mg710,00€100mg964,00€1mL*10mM (DMSO)227,00€Zimlovisertib
CAS :Zimlovisertib (PF-06650833) is an effective, selective and orally active inhibitor of interleukin-1 receptor-associated kinase 4 (IRAK4).Formule :C18H20FN3O4Degré de pureté :98.21%Couleur et forme :SolidMasse moléculaire :361.37TASIN-1
CAS :TASIN-1 is a small molecule inhibitor of mutant adenomatous polyposis coli (APC).Formule :C18H28N2O3SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :352.49Ref: TM-T22632
1mg37,00€5mg79,00€10mg124,00€25mg255,00€50mg409,00€100mg605,00€500mg1.288,00€1mL*10mM (DMSO)87,00€GSK-J4
CAS :GSK-J4 (GSK J4 HCl) is a cell permeable prodrug of GSK-J1, a dual inhibitor of the H3K27me3/me2 demethylases JMJD3/KDM6B and UTX/KDM6A. Cost effective and quality assured.Formule :C24H27N5O2Degré de pureté :98.24% - 99.98%Couleur et forme :SolidMasse moléculaire :417.5Ref: TM-T3100
2mg52,00€5mg86,00€10mg122,00€25mg215,00€50mg345,00€100mg523,00€200mg663,00€1mL*10mM (DMSO)134,00€Robustine
CAS :Robustine is a natural product, exhibits inhibitory potency against human phosphodiesterase 5 (hPDE5A) in vitro.Formule :C12H9NO3Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :215.2IRAK-1-4 Inhibitor I
CAS :IRAK-1-4 Inhibitor I is a dual inhibitor of IRAK4 and IRAK1.Formule :C20H21N5O4Degré de pureté :98% - 99.89%Couleur et forme :SolidMasse moléculaire :395.41Ref: TM-T2457
1mg42,00€5mg74,00€10mg104,00€25mg212,00€50mg356,00€100mg512,00€500mg1.071,00€1mL*10mM (DMSO)74,00€Sitravatinib
CAS :Sitravatinib (MGCD516) (MGCD516) is an inhibitor targeting multiple RTKs involved in driving sarcoma cell growth, including c-Met, c-Kit, PDGFRα/β, PDGFR, andFormule :C33H29F2N5O4SDegré de pureté :98.9% - 99.85%Couleur et forme :SolidMasse moléculaire :629.68Ref: TM-T4349
5mg49,00€10mg74,00€25mg130,00€50mg200,00€100mg319,00€200mg507,00€500mg800,00€1mL*10mM (DMSO)69,00€Miquelianin
CAS :Miquelianin (Quercetin 3-glucuronide) is a potent stilbene oxidase inhibitor, it has antioxidant, anti-atherogenic, and anti-inflammatory activities.Formule :C21H18O13Degré de pureté :98.83% - 99.52%Couleur et forme :SolidMasse moléculaire :478.36L-Leucyl-L-Leucine methyl ester hydrochloride
CAS :L-Leucyl-L-Leucine methyl ester hydrochloride (Leu-Leu-ome hydrochloride) is a dipeptide condensation product of L-leucine methyl ester. Cost-effective and quality-assured.Formule :C13H27ClN2O3Degré de pureté :98.41% - 99.63%Couleur et forme :SolidMasse moléculaire :294.81rosmarinate acid
CAS :Rosmarinate acid(Rosemary acid) inhibits MAO-A, MAO-B and COMT enzymes with IC50s of 50.1, 184.6 and 26.7 μM, respectivelyFormule :C18H16O8Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :360.31Ref: TM-TN7057
5mg55,00€10mg82,00€25mg126,00€50mg182,00€100mg273,00€200mg409,00€1mL*10mM (DMSO)74,00€VK-II-36
CAS :VK-II-36, a carvedilol analog, suppresses sarcoplasmic reticulum (SR) Ca(2+) release but does not block the β-receptor.Formule :C26H26N2O5Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :446.49PDE4-IN-20
CAS :EAPT, a selective PDE4 inhibitor, controls cAMP levels and has potential for treating inflammatory diseases.Formule :C13H12F3N3O2Degré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :299.25β-catenin-IN-2
CAS :β-catenin-IN-2 is a potent inhibitor of β-catenin that can be used in colorectal cancer research.Formule :C15H14FN3Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :255.29Ref: TM-T9696
1mg90,00€5mg215,00€10mg340,00€25mg575,00€50mg822,00€100mg1.108,00€500mg2.242,00€1mL*10mM (DMSO)250,00€NT157
CAS :NT157, a small tyrphostin, inhibits IRS, IGF-1R, and STAT3 in TME, reducing cancer cell survival.Formule :C16H14BrNO5SDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :412.26DOPEXAMINE
CAS :Dopexamine is a dopaminergic agonistFormule :C22H32N2O2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :356.5Ref: TM-T8653
1mg131,00€2mg188,00€5mg284,00€10mg430,00€25mg710,00€50mg998,00€100mg1.349,00€1mL*10mM (DMSO)306,00€Bayogenin
CAS :Bayogenin is an alfalfa saponin, Bayogenin shows moderate potency of glycogen phosphorylase inhibition.Formule :C30H48O5Degré de pureté :99.69% - 99.76%Couleur et forme :SolidMasse moléculaire :488.70Diprotin A
CAS :Diprotin A (Ile-Pro-Ile) (Ile-Pro-Ile) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.Formule :C17H31N3O4Degré de pureté :99.29%Couleur et forme :White PowderMasse moléculaire :341.45HEX3 acetate(688805-40-5 free base)
HEX3 acetate is a fragment of the adenoviral hexon. Hexon is the major capsid protein of adenovirion and is comprised of three identical polypeptide chains.Formule :C49H82N12O16Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :1095.26Asiatic acid
CAS :Asiatic acid (Dammarolic acid) is the aglycone of asiaticoside used in wound healing with antioxidant, anti-inflammatory, and neuroprotective properties.Formule :C30H48O5Degré de pureté :98.01% - 99.52%Couleur et forme :Solid PowderMasse moléculaire :488.70Imeglimin hydrochloride
CAS :Imeglimin hydrochloride (EMD 387008 hydrochloride） is an oral hypoglycemic agent. Imeglimin improves insulin sensitivity.Cost-effective and quality-assured.Formule :C6H14ClN5Degré de pureté :99.25% - 99.94%Couleur et forme :SolidMasse moléculaire :191.66Ref: TM-T7486
1mg39,00€2mg50,00€5mg82,00€10mg117,00€25mg207,00€50mg344,00€100mg520,00€200mg730,00€1mL*10mM (DMSO)195,00€AMG-208
CAS :AMG-208 is a highly selective c-Met inhibitor with IC50 of 9 nM. Phase 1.Formule :C22H17N5O2Degré de pureté :98.56%Couleur et forme :SolidMasse moléculaire :383.4MG-132
CAS :MG-132 (Z-Leu-Leu-Leu-al) is a 26S proteasome inhibitor, cell-permeable and reversible,an autophagy activator, induces apoptosis. High-Quality, Low-Cost!Formule :C26H41N3O5Degré de pureté :95% - 99.99%Couleur et forme :White To Off-White PowderMasse moléculaire :475.62Ref: TM-T2154
10mg46,00€25mg84,00€50mg137,00€100mg205,00€200mg356,00€500mg447,00€1mL*10mM (DMSO)44,00€Wnt-C59
CAS :Wnt-C59 (C59)(C59) is a highly effective and specific Wnt signaling antagonis with PORCN enzymatic activity.Formule :C25H21N3ODegré de pureté :99.56% - 99.95%Couleur et forme :SolidMasse moléculaire :379.45Rec 15/2615 (hydrochloride)
CAS :Rec 15/2615 is an α1B-AR antagonist (Ki = 0.45 nM), more selective over α1A/D/L-ARs, lowers rabbit aorta contractions, and reduces dog blood pressure.Formule :C26H35Cl2N5O5Couleur et forme :SolidMasse moléculaire :568.49I-49 free base
I-49 free base (Pyrido[4,3-d]pyrimidin-7(6H)-one, 2-methyl-4-[[(1R)-1-[2-methyl-3-(trifluoromethyl)phenyl]ethyl]amino]-6-(tetrahydro-2H-pyran-4-yl)-) is a novelFormule :C23H26ClF3N4O2Degré de pureté :99.64% - 99.88%Couleur et forme :SolidMasse moléculaire :482.92Duloxetine
CAS :Duloxetine is an inhibitor of serotonin-norepinephrine reuptake(Ki of 4.6 nM),with treatment of major depressive disorder and generalized anxiety disorder.Formule :C18H19NOSDegré de pureté :99.71% - 99.89%Couleur et forme :SolidMasse moléculaire :297.41Dynasore
CAS :Dynasore, a cell-permeable dynamin inhibitor, blocks GTPase of dynamin 1/2 and Drp1 (IC50: 15 μM) without affecting other small GTPases.Formule :C18H14N2O4Degré de pureté :95.85% - 99.22%Couleur et forme :SolidMasse moléculaire :322.31Ref: TM-T1848
5mg49,00€10mg79,00€25mg140,00€50mg259,00€100mg374,00€200mg560,00€500mg883,00€1mL*10mM (DMSO)87,00€6-fluoro-3-(4-1,2,5,6-tetrahydropyridyl)indole
CAS :6-Fluoro-3-(4-tetrahydropyridyl)indole: a potential anticancer indole derivative and drug lead.Formule :C13H13FN2Degré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :216.25Kartogenin
CAS :Kartogenin (KGN) is an activator of the smad4/smad5 pathway, and promotes the selective differentiation of multipotent mesenchymal stem cells into chondrocytes.Formule :C20H15NO3Degré de pureté :96.25% - 97.79%Couleur et forme :SolidMasse moléculaire :317.34ICCB280
CAS :ICCB280 was capable of inducing differentiation and apoptosis of ATRA-resistant patient blasts strongly signify that the activity of this compound can overcome
Formule :C23H18N2O4Degré de pureté :98.04%Couleur et forme :SolidMasse moléculaire :386.4Dihydrorhodamine 123
CAS :Dihydrorhodamine 123 (DHR 123) is a fluorescent probe (λex=488 nm, λem=525 nm). oxidized in the presence of reactive oxygen species. High-Quality, Low-Cost!Formule :C21H18N2O3Degré de pureté :97.75% - 99.53%Couleur et forme :SolidMasse moléculaire :346.38Platycodin D
CAS :Platycodin D may stimulate TNF-α synthesis or inhibit degradation of TNF-α mRNA.Formule :C57H92O28Degré de pureté :99.2% - 99.65%Couleur et forme :SolidMasse moléculaire :1225.32LOX-IN-3 dihydrochloride monohydrate
CAS :LOX-IN-3 dihydrochloride monohydrate is an oral lysyl oxidase inhibitor for research in fibrosis, cancer, and angiogenesis.Formule :C13H17Cl2FN2O3SCouleur et forme :SolidMasse moléculaire :371.25Benzopinacole
CAS :Benzopinacole is an anti-amoeba drug that can be used as an intermediate to synthesize a variety of compounds.Formule :C26H22O2Degré de pureté :99.47%Couleur et forme :White Crystalline PowderMasse moléculaire :366.45H-Val-Pro-Pro-OH
CAS :H-Val-Pro-Pro-OH is an inhibitor of Angiotensin I converting enzyme (ACE)( IC50 : 9 μM).Formule :C15H25N3O4Degré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :311.38Bifendate
CAS :Bifendate (Bifendatatum) is commonly used to treat the transaminase elevation that caused by viral hepatitis and drug-induced liver injury.
Formule :C20H18O10Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :418.35Norisoboldine
CAS :Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.Formule :C18H19NO4Degré de pureté :98.12% - 99.7%Couleur et forme :SolidMasse moléculaire :313.35NH2-C6-NH-Boc
CAS :NH2-C6-NH-Boc is a PROTAC linker. NH2-C6-NH-Boc can be used in the synthesis the Mcl-1 inhibitor based on PROTAC.Formule :C11H24N2O2Degré de pureté :99.97%Couleur et forme :Clear Light Yellow Viscous LiquidMasse moléculaire :216.32Enzastaurin
CAS :Enzastaurin (LY317615) (LY317615) is an effective PKCβ selective inhibitor (IC50: 6 nM), 6- to 20-fold selectivity against PKCα/γ/ε.Formule :C32H29N5O2Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :515.6
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