Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.855 produits)
- Apoptose(6.375 produits)
- Cycle cellulaire/point de contrôle(4.911 produits)
- Chromatine/Épigénétique(2.633 produits)
- Signalisation du cytosquelette(1.588 produits)
- Altération de l'ADN/réparation de l'ADN(2.868 produits)
- Endocrinologie/Hormones(3.765 produits)
- Enzyme(3.673 produits)
- GPCR/G-Protéine(9.054 produits)
- Immunologie et Inflammation(3.954 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(417 produits)
- Signalisation MAPK(1.259 produits)
- Transporteur membranaire/Canal ionique(3.163 produits)
- Métabolisme(10.157 produits)
- Microbiologie/Virologie(7.674 produits)
- Neuroscience(10.550 produits)
- Autres inhibiteurs(35.862 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.438 produits)
- Protéases/Protéasome(1.692 produits)
- Cellules souche et Dérivés(733 produits)
- Tyrosine Kinase/Adaptateurs(1.992 produits)
- Ubiquitination(1.744 produits)
Affichez 16 plus de sous-catégories
66512 produits trouvés pour "Inhibiteurs"
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H4 Receptor antagonist 1
CAS :H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Formule :C16H17ClN4ODegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :316.79Rosamultin
CAS :Rosamultin has antioxidant, antiinflammatory/antinociceptive properties,and has anti-human immunodeficiency virus (HIV) activity.Formule :C36H58O10Degré de pureté :98% - 99.51%Couleur et forme :SolidMasse moléculaire :650.84LJH685
CAS :LJH685 is an effective pan-RSK inhibitor for RSK1/2/3 (IC50: 6/5/4 nM).Formule :C22H21F2N3ODegré de pureté :99.13% - 99.78%Couleur et forme :SolidMasse moléculaire :381.42Ref: TM-T6877
1mg37,00€1mL*10mM (DMSO)87,00€5mg88,00€10mg127,00€25mg240,00€50mg401,00€100mg603,00€200mg848,00€Methyl 3-phenylpropanoate
CAS :Methyl 3-phenylpropanoate (3-Phenylpropionic acid methyl ester) is a huamn endogenous metabolite.Formule :C10H12O2Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :164.2Euphorbia Factor L2
CAS :Euphorbia Factor L2 alleviates lipopolysaccharide-induced acute lung injury and inflammation through inhibits NF-κB activation.Formule :C38H42O9Degré de pureté :99.53% - 99.96%Couleur et forme :SolidMasse moléculaire :642.73NADPH tetracyclohexanamine
CAS :NADPH tetracyclohexanamine (NADPH (tetracyclohexanamine)) is a cofactor and biological reducing agent.
Formule :C45H82N11O17P3Degré de pureté :98.73% - 99.05%Couleur et forme :SolidMasse moléculaire :1142.12ML204
CAS :ML204 is a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels.Formule :C15H18N2Degré de pureté :98.1% - 99.72%Couleur et forme :SolidMasse moléculaire :226.32BMS-345541 hydrochloride
CAS :BMS-345541 hydrochloride is a selective IKK inhibitor (IKK2 and IKK1 with IC50 of 0.3 μM and 4 μM,respectively).Formule :C14H18ClN5Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :291.78Ref: TM-T8542
1mg38,00€2mg50,00€1mL*10mM (DMSO)52,00€5mg82,00€10mg119,00€25mg212,00€50mg356,00€100mg533,00€CP-724714
CAS :CP-724714 (CP724714) is an effective and selective HER2/ErbB2 inhibitor (IC50: 10 nM), >640-fold selectivity against EGFR, Abl, InsR, PDGFR, IRG-1R, Src, VEGFR2Formule :C27H27N5O3Degré de pureté :97.1% - 98.82%Couleur et forme :SolidMasse moléculaire :469.54Ref: TM-T4014
1mg42,00€2mg55,00€5mg90,00€1mL*10mM (DMSO)94,00€10mg148,00€25mg259,00€50mg429,00€100mg625,00€5-O-Demethylnobiletin
CAS :5-O-Demethylnobiletin is a natural anti-inflammatory that inhibits 5-LOX without altering COX-2 expression.
Formule :C20H20O8Degré de pureté :99.83% - ≥95%Couleur et forme :SolidMasse moléculaire :388.37lavendustin C
CAS :lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.Formule :C14H13NO5Degré de pureté :98.06%Couleur et forme :Yellow To Tan PowderMasse moléculaire :275.26Ref: TM-T4185
1mg42,00€2mg55,00€1mL*10mM (DMSO)90,00€5mg93,00€10mg152,00€25mg330,00€50mg492,00€100mg707,00€(+)-Epicatechin
CAS :(+)-Epicatechin (Dexepicatechin) is a natural product and an antioxidant agent.Formule :C15H14O6Degré de pureté :98.92%Couleur et forme :SolidMasse moléculaire :290.276'-O-β-D-Glucosylgentiopicroside
CAS :1. 6'-O-beta-D-Glucosylgentiopicroside (6'-O-Glucosylgentiopicroside) may have antifungal activity.Formule :C22H30O14Degré de pureté :99.56% - 99.73%Couleur et forme :SolidMasse moléculaire :518.47Gymnemagenin
CAS :Gymnemagenin is a potent and selective antagonist for the β isoform of LXR, it has antihyperglycemic activity.Formule :C30H50O6Degré de pureté :99.29% - ≥95%Couleur et forme :SolidMasse moléculaire :506.71Nigakinone
CAS :Nigakinone, isolated from Kumu, is an alkaloid with the pharmacological activity.Formule :C15H10N2O3Degré de pureté :98.66% - 99.84%Couleur et forme :SolidMasse moléculaire :266.25Ref: TM-TQ0264
1mg62,00€1mL*10mM (DMSO)135,00€5mg144,00€10mg227,00€25mg375,00€50mg557,00€100mg797,00€L-Carnosine
CAS :L-Carnosine is an antioxidant found in muscles and brain, may slow aging-related biochemical changes.
Formule :C9H14N4O3Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :226.23BMS582949
CAS :BMS-582949 inhibits p38 MAPK with 13 nM IC50, blocking kinase activity and activation.Formule :C22H26N6O2Degré de pureté :98.11%Couleur et forme :SolidMasse moléculaire :406.48Ref: TM-T6789
1mg82,00€2mg114,00€5mg200,00€1mL*10mM (DMSO)200,00€10mg284,00€25mg477,00€50mg692,00€100mg973,00€BAY-474
CAS :BAY-474 is an inhibitor of tyrosine-protein kinase c-Met. It acts as an epigenetics probeFormule :C17H15N5Degré de pureté :98.98%Couleur et forme :SolidMasse moléculaire :289.33Ref: TM-T7900
1mg35,00€5mg71,00€1mL*10mM (DMSO)84,00€10mg112,00€25mg203,00€50mg294,00€100mg411,00€200mg553,00€Ixazomib
CAS :Ixazomib (MLN2238) is a boron-based peptide proteasome inhibitor targeting β5 site (IC50: 3.4 nM), also affecting β1 and β2 sites.Formule :C14H19BCl2N2O4Degré de pureté :98% - 99.77%Couleur et forme :SolidMasse moléculaire :361.03Velsecorat
CAS :Velsecorat (AZD7594) is an effective and selective nonsteroidal glucocorticoid receptor modulator (IC50: 0.9 nM).Formule :C32H32F2N4O6Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :606.62Ref: TM-TQ0225
1mg52,00€5mg114,00€1mL*10mM (DMSO)156,00€10mg158,00€25mg339,00€50mg505,00€100mg722,00€ICI 89406
CAS :ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.Formule :C19H22N4O3Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :354.4Lys-SMCC-DM1
CAS :Lys-SMCC-DM1 (Lys-Nε-MCC-DM1) inhibits microtubule polymerization and is commonly used in breast cancer research. Cost-effective and quality-assured.Formule :C53H75ClN6O15SDegré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :1103.71Veratramine
CAS :Veratramine (NSC-23880)(NSC-17821; NSC-23880) is a potent signal transduction inhibitor for treating tumors.Formule :C27H39NO2Degré de pureté :99.7% - 99.75%Couleur et forme :SolidMasse moléculaire :409.60Carbidopa
CAS :Carbidopa (Lodosyn) is an aromatic-L-amino-acid decarboxylase inhibitor (IC50: 29±2 μM).Formule :C10H14N2O4Degré de pureté :98.01% - ≥98%Couleur et forme :SolidMasse moléculaire :226.23Hirsuteine
CAS :Hirsuteine: natural product; blocks nicotine effects on dopamine by hindering ion flow in receptor channels.Formule :C22H26N2O3Degré de pureté :99.36% - 99.83%Couleur et forme :SolidMasse moléculaire :366.45MHY1485
CAS :MHY1485 is an mTOR activator that is cell-permeable. MHY1485 inhibits autophagosome and lysosome fusion, thereby inhibiting autophagy. Cost-effective and quality-assured.Formule :C17H21N7O4Degré de pureté :97.74% - >99.99%Couleur et forme :SolidMasse moléculaire :387.39Motesanib
CAS :Motesanib (AMG 706) orally blocks VEGFR, PDGFR, Kit, Ret; curbing angiogenesis and cancer cell growth.Formule :C22H23N5ODegré de pureté :98% - 99.09%Couleur et forme :SolidMasse moléculaire :373.45Ref: TM-T2288
5mg34,00€1mL*10mM (DMSO)39,00€10mg49,00€25mg81,00€50mg114,00€100mg160,00€200mg230,00€500mg389,00€Pentagastrin
CAS :Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis ofFormule :C37H49N7O9SDegré de pureté :96.98% - 99.49%Couleur et forme :Fine Colorless Needle-Shaped Crystals From 2-Ethoxyethanol + Water SolidMasse moléculaire :767.89Punicalagin
CAS :Punicalagin, an ellagitannin in pomegranates, has antioxidant, anti-inflammatory, anticancer properties, and combats heart issues from high-fat diets.Formule :C48H28O30Degré de pureté :98% - 99.7%Couleur et forme :White Crystalline PowderMasse moléculaire :1084.723,4-Dicaffeoylquinic acid
CAS :3,4-Dicaffeoylquinic acid (Isochlorogenic acid B) has antioxidant activity.Formule :C25H24O12Degré de pureté :96.33% - 98.82%Couleur et forme :SolidMasse moléculaire :516.45Ref: TM-T6S1525
1mg40,00€5mg80,00€10mg101,00€1mL*10mM (DMSO)103,00€25mg167,00€50mg240,00€100mg355,00€500mg845,00€Tavapadon
CAS :Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.Formule :C19H16F3N3O3Degré de pureté :99.33% - 99.8%Couleur et forme :SolidMasse moléculaire :391.34Ref: TM-T16999
1mg77,00€5mg166,00€1mL*10mM (DMSO)178,00€10mg260,00€25mg475,00€50mg668,00€100mg888,00€Tectorigenin
CAS :Tectorigenin is an O-methylated isoflavone boosting osteoblasts and bone healing, yet inhibits osteoclasts and bone resorption.Formule :C16H12O6Degré de pureté :99.31% - 99.97%Couleur et forme :SolidMasse moléculaire :300.26Su1498
CAS :Su1498 (Tyrphostin SU 1498) is a selective inhibitor of the VEGF receptor 2, having negligible activity at several other serine/threonine and tyrosine kinases.
Formule :C25H30N2O2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :390.52Oxytetracycline Dihydrate
CAS :Oxytetracycline Dihydrate (Terramycin Dihydrate) is a prescription antibiotic, interfering with the ability of bacteria to produce essential proteins.Formule :C22H24N2O9·2H2ODegré de pureté :99.80%Couleur et forme :CrystallineMasse moléculaire :496.461-Naphthol
CAS :1-Naphthol (Furro ER) is an excited state proton transfer (ESPT) fluorescent molecular probe for sensing thermotropic microenvironmental changes of pluronicFormule :C10H8ODegré de pureté :98.8%Couleur et forme :Yellow Monoclinic Needles From Water Liquid PelletslargecrystalsMasse moléculaire :144.17Deoxyshikonin
CAS :1.Formule :C16H16O4Degré de pureté :99.36% - ≥95%Couleur et forme :SolidMasse moléculaire :272.32-(1,8-naphthyridin-2-yl)phenol
CAS :2-NP is a STAT1 enhancer.Formule :C14H10N2ODegré de pureté :99.33% - 99.82%Couleur et forme :SolidMasse moléculaire :222.24Ref: TM-T2168
5mg57,00€1mL*10mM (DMSO)63,00€10mg90,00€25mg177,00€50mg281,00€100mg444,00€200mg647,00€500mg982,00€Camelliaside B
CAS :Camelliaside B possesses deglycosylation activity.Formule :C32H38O19Degré de pureté :95.92% - 99.92%Couleur et forme :SolidMasse moléculaire :726.63LY3177833
CAS :LY3177833 is an Cdc7 kinase inhibitor (IC50 : 3.3 nM)Formule :C16H12FN5ODegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :309.3Ref: TM-T7810
1mg38,00€5mg80,00€1mL*10mM (DMSO)87,00€10mg109,00€25mg212,00€50mg318,00€100mg477,00€200mg677,00€Pre-084
CAS :Pre-084 is a high affinity, selective σ1 agonist.Formule :C19H28ClNO3Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :353.88Demethylsuberosin
CAS :7-Demethylsuberosin (7-demethylsuberosin) is a coumarin compound isolated from Angelica gigas Nakai,and has anti-inflammatory activity,and exhibited inhibitoryFormule :C14H14O3Degré de pureté :98.17% - 98.36%Couleur et forme :SolidMasse moléculaire :230.26SB 204990
CAS :SB 204990 is a lactone prodrug of SB-201076, a potent and specific ATP citrate lyase inhibitor.Cost-effective and quality-assured.Formule :C18H22Cl2O5Degré de pureté :96.32% - 99.6%Couleur et forme :SolidMasse moléculaire :389.27KUN56321
CAS :KUN56321, a luminescent compound, enhances efficiency and lowers drive voltage in organic light-emitting devices.Formule :C23H15BrN2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :399.28Methuosis inducer 1
CAS :Methuosis inducer 1 is a potent methuosis inducer, with nticancer activity.Formule :C27H20F3N5ODegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :487.48Ref: TM-T7262
1mg84,00€5mg177,00€1mL*10mM (DMSO)188,00€10mg268,00€25mg482,00€50mg708,00€100mg1.044,00€TFAP
CAS :TFAP (N-(5-Aminopyridin-2-yl)-4-(trifluoromethyl)benzamide) is a selective cyclooxygenase-1 (COX-1) inhibitorFormule :C13H10F3N3ODegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :281.23Oprozomib
CAS :Oprozomib inhibits 20S proteasome β5/LMP7, is orally available, and may have cancer-fighting properties. IC50: β5 - 36 nM; LMP7 - 82 nM.Formule :C25H32N4O7SDegré de pureté :98% - 99.87%Couleur et forme :SolidMasse moléculaire :532.61LYN-1604 dihydrochloride
CAS :LYN-1604 is a novel ULK1 activator.It inducing cell death involved in ATF3, RAD21, and caspase3, accompanied by autophagy and apoptosis.Formule :C33H45Cl4N3O2Degré de pureté :98.95% - 99.92%Couleur et forme :SolidMasse moléculaire :657.54Ref: TM-T8808L
1mg35,00€5mg78,00€1mL*10mM (DMSO)101,00€10mg117,00€25mg212,00€50mg316,00€100mg447,00€200mg628,00€N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.Formule :C30H39N5O8Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :597.66Lefamulin
CAS :Lefamulin (BC-3781) is a semi-synthetic compound that inhibits the synthesis of bacterial protein, which is required for bacteria to grow.Formule :C28H45NO5SDegré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :507.73Ref: TM-T7588
1mg70,00€5mg150,00€1mL*10mM (DMSO)167,00€10mg215,00€25mg358,00€50mg517,00€100mg707,00€200mg973,00€Vesnarinone
CAS :Vesnarinone (Arkin) (INN) is a mixed phosphodiesterase 3 inhibitor and ion-channel modifier that has modest, dose-dependent, positive inotropic activity, butFormule :C22H25N3O4Degré de pureté :96.69% - 98.13%Couleur et forme :SolidMasse moléculaire :395.45Ref: TM-T3465
2mg34,00€1mL*5mM (DMSO)47,00€5mg50,00€10mg75,00€25mg111,00€50mg*5mM (DMSO)198,00€100mg296,00€200mg427,00€GDC-0152
CAS :GDC-0152 is a potent inhibitor of IAPs.Formule :C25H34N6O3SDegré de pureté :97.18% - 99.32%Couleur et forme :SolidMasse moléculaire :498.64Theaflavin 3,3′-digallate
CAS :Theaflavin 3,3'-digallate, a major polyphenol found in black tea, is an inducer of oxidative stress which has anti-inflammatory and cancerFormule :C43H32O20Degré de pureté :98.71% - 99.86%Couleur et forme :SolidMasse moléculaire :868.70Ref: TM-T5429
1mg87,00€5mg169,00€10mg268,00€1mL*10mM (DMSO)268,00€25mg462,00€50mg647,00€100mg873,00€200mg1.153,00€3,4-Dimethoxyphenol
CAS :3,4-Dimethoxyphenol (4-Hydroxyveratrole) is an active biochemical.Formule :C8H10O3Degré de pureté :98.57%Couleur et forme :Red Crystal PowderMasse moléculaire :154.161-Ethyl-6-aminouracil
CAS :1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have highFormule :C6H9N3O2Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :155.15p-Fluoro-L-phenylalanine
CAS :p-Fluoro-L-phenylalanine: TH substrate, studies enzyme regulation, binds E. coli L-leucine receptor, KD 0.26μM.Formule :C9H10FNO2Degré de pureté :99.63%Couleur et forme :White To Off-White PowderMasse moléculaire :183.182-Methylpentanedioic acid
CAS :2-Methylpentanedioic acid, a succinic acid metabolite, occurs naturally in human urine.Formule :C6H10O4Degré de pureté :98% - 99.13%Couleur et forme :White Solid CrystallineMasse moléculaire :146.14Ruxolitinib
CAS :Ruxolitinib (INCB018424) is a JAK1/2 inhibitor (IC50=3.3/2.8 nM) that is potent and selective.Formule :C17H18N6Degré de pureté :99.4% - >99.99%Couleur et forme :SolidMasse moléculaire :306.36Ref: TM-T1829
5mg55,00€1mL*10mM (DMSO)62,00€10mg71,00€25mg96,00€50mg110,00€100mg146,00€200mg231,00€500mg393,00€MHP
CAS :MHP (Methyl caprooyl tyrosinate) is an activator of sphingosine kinase (SPHK1), and significantly stimulates CAMP mRNA and protein production in KC.Formule :C16H23NO4Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :293.36Ref: TM-T4658
1mg34,00€2mg46,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg101,00€25mg207,00€50mg334,00€100mg537,00€200mg762,00€JNJ16259685
CAS :JNJ16259685 (TN.T 16259685) is a selective mGluR1 antagonist, and inhibits the synaptic activation of mGluR1 in a concentration-dependent manner with IC50 of 19Formule :C20H23NO3Degré de pureté :98.31%Couleur et forme :SolidMasse moléculaire :325.4Ref: TM-T5512
1mg46,00€2mg62,00€5mg95,00€1mL*10mM (DMSO)95,00€10mg133,00€25mg278,00€50mg424,00€100mg620,00€PKG inhibitor peptide TFA (82801-73-8 free base)
PKG inhibitor peptide TFA (82801-73-8 free base) is an inhibitor of ATP-competitive cGMP-dependent protein kinase (PKG).Formule :C40H75F3N18O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1057.13Carboxyatractyloside
CAS :Carboxyatractyloside (Carboxyatractyloside tripotassium salt) is a natural product.Formule :C31H46O18S2Degré de pureté :99.56% - 99.83%Couleur et forme :White PowderMasse moléculaire :770.82Acenaphthylene
CAS :Acenaphthylene is environmental polycyclic aromatic hydrocarbon (PAH)pollutantsFormule :C12H8Degré de pureté :99.73%Couleur et forme :Yellow Needles Fungicides And In The Manufacture Of PlasticsMasse moléculaire :152.19BDC2.5 mimotope 1040-31 acetate
BDC2.5 mimotope 1040-31 acetate, an agonistic peptide, targets BDC2.5 T cells effectively, known as p31.Formule :C65H101N17O16SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :1408.69PKD-IN-1
CAS :CRT0066101 is an inhibitor of PKD.Formule :C18H19ClN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :342.82RFRP-1 (human) acetate(311309-25-8 free base)
RFRP-1 (human) acetate: potent NPFF2/1 agonist, alters rat/rabbit cardiac functions, and regulates rat prolactin.Formule :C69H105N19O16SDegré de pureté :96.84%Couleur et forme :SolidMasse moléculaire :1488.77Dovitinib
CAS :Dovitinib is an orally active, multi-targeted tyrosine kinase (RTK) inhibitor with anti-tumor effects.Cost-effective and quality-assured.
Formule :C21H21FN6ODegré de pureté :99.35% - 99.92%Couleur et forme :SolidMasse moléculaire :392.43Levolansoprazole
CAS :Levolansoprazole ((S)-Lansoprazole), a proton pump inhibitor, irreversibly inhibits H+/K+-stimulated ATPase pumps in parietal cells (IC50: 5.2 μM).Formule :C16H14F3N3O2SDegré de pureté :98.629%Couleur et forme :SolidMasse moléculaire :369.36Ref: TM-T20714
1mg105,00€5mg234,00€1mL*10mM (DMSO)241,00€10mg326,00€25mg495,00€50mg655,00€100mg879,00€200mg1.161,00€BAR 501 impurity
CAS :BAR 501 impurity 在 BAR501 制剂中发现的一种杂质，可作为 G 蛋白偶联胆汁酸激活受体 (GP-BAR1) 的激动剂。 BAR501 杂质 (10 µM) 在 GP-BAR1 报告基因检测中诱导荧光素酶活性增加 150%。Formule :C26H46O3Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :406.64Presatovir
CAS :Presatovir (GS-5806) (GS-5806) is a novel, orally bioavailable RSV fusion inhibitor (mean EC50: 0.43 nM).Formule :C24H30ClN7O3SDegré de pureté :99.14% - 99.92%Couleur et forme :SolidMasse moléculaire :532.06D-JNKI-1 acetate
D-JNKI-1 acetate (AM-111 acetate) is a highly potent and cell-permeable peptide inhibitor of JNK.Formule :C166H290N66O42Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :3882.5Ref: TM-T10937L
1mg156,00€5mg296,00€10mg442,00€25mg707,00€50mg1.009,00€1mL*10mM (DMSO)1.089,00€100mg1.333,00€D-Tagatose
CAS :D-Tagatose, a rare hexoketose and isomer of d-galactose, is naturally found in Sterculia setigera gum and various dairy products.Formule :C6H12O6Degré de pureté :99.78% - 99.96%Couleur et forme :White Crystalline PowderMasse moléculaire :180.16PHYTOL
CAS :Phytol is a diterpene alcohol with antinociceptive, antioxidant, anti-inflammatory, and antiallergic properties, activating PPARα.Formule :C20H40ODegré de pureté :97.71% - 99.62%Couleur et forme :LiquidMasse moléculaire :296.53Seletalisib
CAS :Seletalisib (UCB5857) (UCB5857) is a potent and specific PI3Kδ inhibitor (IC50: 12 nM).Formule :C23H14ClF3N6ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :482.85Ref: TM-TQ0044
1mg54,00€2mg77,00€5mg114,00€1mL*10mM (DMSO)119,00€10mg178,00€25mg313,00€50mg447,00€100mg625,00€Tiaprofenic acid
CAS :Tiaprofenic acid (Acido tiaprofenico) is a non-steroidal anti-inflammatory drug used to treat pain, especially arthritic pain.Formule :C14H12O3SDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :260.31PF-3758309
CAS :PF-3758309 (PF-03758309) (IC50=1.3 nM), a pyrrolopyrazole inhibitor of PAK4, has effective ATP-competition.Formule :C25H30N8OSDegré de pureté :97.70%Couleur et forme :SolidMasse moléculaire :490.62Norfluoxetine Hydrochloride
CAS :Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.Formule :C16H17ClF3NODegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :331.76TAK-632
CAS :TAK-632 is a potent pan-Raf inhibitor.Formule :C27H18F4N4O3SDegré de pureté :98% - 99.5%Couleur et forme :SolidMasse moléculaire :554.52Bradykinin
CAS :Bradykinin is an inflammatory mediator.Formule :C50H73N15O11Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :1060.21Tectorigenin 7-O-Xylosyl Glucoside
CAS :Tectorigenin 7-O-Xylosyl Glucoside (Tectorigenin 7-O-xylosylglucoside) is a natural productFormule :C27H30O15Degré de pureté :99.65% - 99.97%Couleur et forme :SolidMasse moléculaire :594.52Refametinib
CAS :Refametinib (RDEA119) (RDEA119, Bay 86-9766) is an effective, ATP non-competitive and specific inhibitor of MEK1/2 (IC50: 19/47 nM).Formule :C19H20F3IN2O5SDegré de pureté :99.85% - >99.99%Couleur et forme :SolidMasse moléculaire :572.34Ref: TM-T6636
2mg43,00€5mg63,00€1mL*10mM (DMSO)79,00€10mg93,00€25mg147,00€50mg222,00€100mg326,00€200mg485,00€Apilimod
CAS :Apilimod (STA 5326) inhibits the production of IL-12 and IL-23 and reduces dendritic cell infiltration in psoriasis.Formule :C23H26N6O2Degré de pureté :99.38% - 99.89%Couleur et forme :SolidMasse moléculaire :418.492-Benzylsuccinic acid
CAS :2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite.Formule :C11H12O4Degré de pureté :99.01% - ≥95%Couleur et forme :SolidMasse moléculaire :208.21BAI1
CAS :BAI1 (Bax channel blocker) is a potent inhibitor of Bax-mediated mitochondrial cytochrome C release (IC50: 0.52 μM).Formule :C19H21Br2N3ODegré de pureté :99.96% - ＞99.99%Couleur et forme :SolidMasse moléculaire :467.2Amino-PEG7-acid
CAS :Amino-PEG7-acid is a PEG-based PROTAC linker that can be used in PROTAC synthesis.Formule :C17H35NO9Degré de pureté :98.28%Couleur et forme :SolidMasse moléculaire :397.46MERS-CoV-IN-1
CAS :MERS-CoV-IN-1: potent inhibitor for coronavirus, aids in preventing MERS/SARS.Formule :C19H17NO2Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :291.34PFI-90
CAS :PFI-90, a selective histone demethylase (KDM3B) inhibitor, targets PAX3-FOXO1 action and demonstrates potential antitumor activity.Formule :C11H10N4ODegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :214.22Deoxycytidine triphosphate
CAS :dCTP is a nucleotide used in DNA synthesis, PCR, cDNA creation, and sequencing.Formule :C9H16N3O13P3Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :467.16glycohyodeoxycholic acid
CAS :glycohyodeoxycholic acid is a major metabolite of the secondary bile acid hyodeoxycholic acid in humans.Formule :C26H43NO5Degré de pureté :99.33% - 99.81%Couleur et forme :SolidMasse moléculaire :449.62Nafamostat mesylate
CAS :Nafamostat mesylate (FUT-175), a synthetic serine protease inhibitor, has been used for the treatment of allergic disorders such as asthma, allergic rhinitisFormule :C19H17N5O2·2CH4O3SDegré de pureté :97.36% - 99.76%Couleur et forme :Tan To Pale Orange SolidMasse moléculaire :539.582-Chloroadenosine
CAS :2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectivelyFormule :C10H12ClN5O4Degré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :301.69H-L-Lys(Poc)-OH HCl
CAS :N-ε-propargyloxycarbonyl-L-lysine hydrochloride (N6-((Prop-2-yn-1-yloxy)carbonyl)-L-lysine hydrochloride) is a modified amino acid for cancer therapyFormule :C10H17ClN2O4Degré de pureté :99.79% - 99.93%Couleur et forme :SolidMasse moléculaire :264.71Alofanib
CAS :Alofanib (RPT835) selectively inhibits FGFR2 in KATO III cells with IC50 <10 nM; doesn’t affect FGFR1/3 or FGF2-FGFR2 binding.Formule :C19H15N3O6SDegré de pureté :99.53% - 99.81%Couleur et forme :SolidMasse moléculaire :413.4Efaproxiral Sodium
CAS :Efaproxiral Sodium (RSR13 sodium), a synthetic allosteric modifier of hemoglobin, is utilized for brain metastases originating from breast cancer.Formule :C20H23NO4·NaDegré de pureté :97.92%Couleur et forme :SolidMasse moléculaire :363.38Cerlapirdine
CAS :Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.Formule :C22H23N3O3SDegré de pureté :98.77%Couleur et forme :SolidMasse moléculaire :409.5Ref: TM-T30798
1mg81,00€5mg170,00€1mL*10mM (DMSO)198,00€10mg274,00€25mg543,00€50mg780,00€100mg1.074,00€MOSLOFLAVONE
CAS :MOSLOFLAVONE showed promising anti-inflammatory activity via inhibition of TNF-α and IL-1β with IC50 values of 0.71 μM and 7.8 μM, respectively.Formule :C17H14O5Degré de pureté :98.42% - ≥95%Couleur et forme :SolidMasse moléculaire :298.293-TERT-BUTYL-4-HYDROXYANISOLE
CAS :3-tert-Butyl-p-hydroxyanisole is an antioxidant which is produced via water chlorination.Formule :C11H16O2Degré de pureté :99.65%Couleur et forme :White Solid WaxyMasse moléculaire :180.24Taladegib
CAS :Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.Formule :C26H24F4N6ODegré de pureté :98.75% - >99.99%Couleur et forme :SolidMasse moléculaire :512.5Diphenyleneiodonium chloride
CAS :Diphenyleneiodonium chloride (DPI) inhibits iNOS & eNOS (IC50: 50 nM & 0.3 μM) and has wide-ranging bactericidal properties.Formule :C12H8ClIDegré de pureté :99.71% - 99.86%Couleur et forme :SolidMasse moléculaire :314.55Pimelic acid
CAS :Pimelic acid aids lysine synthesis, is one methylene longer than adipic acid, and is made from cyclohexanone or salicylic acid.Formule :C7H12O4Degré de pureté :99.85%Couleur et forme :OthersolidMasse moléculaire :160.17Methyl p-tert-butylphenylacetate
CAS :Methyl p-tert-butylphenylacetate is a flavouring ingredient.Formule :C13H18O2Degré de pureté :99.96%Couleur et forme :Less Oily Liquid; Sweet Somewhat Woody-Camphoraceous Odour Colourless Oily Liquid; Sweet Somewhat Woody-Camphoraceous OdourMasse moléculaire :206.28
