Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.760 produits)
- Apoptose(6.191 produits)
- Cycle cellulaire/point de contrôle(4.809 produits)
- Chromatine/Épigénétique(2.579 produits)
- Signalisation du cytosquelette(1.502 produits)
- Altération de l'ADN/réparation de l'ADN(2.887 produits)
- Endocrinologie/Hormones(3.703 produits)
- Enzyme(3.671 produits)
- GPCR/G-Protéine(8.967 produits)
- Immunologie et Inflammation(3.704 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.248 produits)
- Transporteur membranaire/Canal ionique(3.137 produits)
- Métabolisme(10.092 produits)
- Microbiologie/Virologie(7.553 produits)
- Neuroscience(10.304 produits)
- Autres inhibiteurs(35.763 produits)
- Oxydation-Réduction(39 produits)
- Signalisation PI3K/Akt/mTOR(1.402 produits)
- Protéases/Protéasome(1.671 produits)
- Cellules souche et Dérivés(740 produits)
- Tyrosine Kinase/Adaptateurs(1.923 produits)
- Ubiquitination(1.717 produits)
Affichez 16 plus de sous-catégories
66570 produits trouvés pour "Inhibiteurs"
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Lobaric acid
CAS :Lobaric acid, from Stereocaulon lichen, has antioxidant and anticancer properties, inhibits PTP1B and 12(S)-LOX, and reduces TMV lesions in plants.Formule :C25H28O8Couleur et forme :SolidMasse moléculaire :456.48MSX-3 free acid
CAS :MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.Formule :C21H23N4O7PCouleur et forme :SolidMasse moléculaire :474.40FMK-MEA
CAS :FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor.Formule :C21H26FN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.46Nrf2 activator-6
CAS :Nrf2 activator-6, a tetrahydroisoquinoline, inhibits Kelch-Nrf2 at 5 nM IC50 (WO2021214470A1).Formule :C31H37ClFN5O5Couleur et forme :SolidMasse moléculaire :614.11Samuraciclib hydrochloride hydrate
Samuraciclib (CT7001) is a potent oral CDK7 inhibitor (IC50: 41 nM) with anti-breast cancer properties.Formule :C22H35ClN6O3Couleur et forme :SolidMasse moléculaire :521.7Ataprost
CAS :Ataprost (ONO 41483), an oral Carboprostacyclin analogue, is 2.6x more potent in inhibiting ADP-induced platelet aggregation and can relieve coronary spasm.Formule :C21H32O4Couleur et forme :SolidMasse moléculaire :348.48Hit 1
Hit 1 is an activator of insulin-degrading enzymes (IDE) (EC50: 5.5 μM) and reduces glucose-stimulated insulin secretion.Formule :C22H24N4O3S2Couleur et forme :SolidMasse moléculaire :456.58MB725
CAS :MB725 is a strong and selective inducer of viability reduction in several cancer cell lines containing the oncogenic p53-Y220C mutation.Formule :C18H21IN4O2SCouleur et forme :SolidMasse moléculaire :484.35PD-1/PD-L1-IN-13
PD-1/PD-L1-IN-13 is a potent immune checkpoint PD-1/PD-L1 inhibitor with an IC50 value of 10.2 nM for PD-1/PD- L1 interaction.PD-1/PD-L1-IN-13 promotes CD8+ T-Formule :C36H34ClF2N3O9Couleur et forme :SolidMasse moléculaire :726.12Tilpisertib fosmecarbil
CAS :Tilpisertib fosmecarbil is a potent inhibitor of serine/threonine kinases with anti-inflammatory properties.Formule :C35H36ClN8O7PCouleur et forme :SolidMasse moléculaire :747.14Terpendole E
CAS :Terpendole E is an atypical L5 site inhibitor.Formule :C28H39NO3Couleur et forme :SolidMasse moléculaire :437.61Heme Oxygenase-2-IN-1
Heme Oxygenase-2-IN-1 is a selective HO-2 inhibitor with IC50s: 14.9 μM (HO-1), 0.9 μM (HO-2).Formule :C19H17N3O2Couleur et forme :SolidMasse moléculaire :319.36Hoe 892
CAS :Hoe 892 is a stable thia-thimo-analogue of prostacyclin and acts as a platelet aggregation inhibitor.Formule :C20H33NO4SCouleur et forme :SolidMasse moléculaire :383.55NLRP3-IN-7
NLRP3-IN-7 (Compound 36) is a selective inhibitor of the NLRP3 inflammasome and is able to assemble the NLRP3 inflammasome.Formule :C18H15ClN2O4S3Couleur et forme :SolidMasse moléculaire :454.97TH-6
TH-6, a potent HDAC inhibitor (IC50: HDAC1-0.115, 2-0.135, 3-0.242, 6-0.138, 8-2.120 μM), blocks cell migration, invasion, and has anti-tumor properties.Formule :C22H24FN3O5Couleur et forme :SolidMasse moléculaire :429.44CDK-IN-9
CDK-IN-9: A potent CDK inhibitor, gels to enhance CDK12/DDB1 binding, targets CDK2/E (IC50: 4 nM), induces apoptosis via dephosphorylation.Formule :C21H24N8SCouleur et forme :SolidMasse moléculaire :420.53H 218-54
CAS :H 218-54 is a renin inhibitor.Formule :C37H56N2O5SCouleur et forme :SolidMasse moléculaire :640.92L-365260 hemihydrate
L-365260 hemihydrate: selective oral CCK-B/gastrin blocker, Ki=1.9/2.0 nM, competes with guinea pig receptors.Formule :C24H24N4O3Couleur et forme :SolidMasse moléculaire :407.47LY2934747
CAS :LY2934747 is a novel, potent, and systemically bioavailable mGlu2/3 receptor agonist, exhibiting both antipsychotic and analgesic properties in vivo.Formule :C10H13NO4Couleur et forme :SolidMasse moléculaire :211.21RORγt/DHODH-IN-3
RORγt/DHODH-IN-3 (compound (S)-14d) is a potent, orally active dual inhibitor of RORγt (IC50: 0.098 μM) and DHODH (IC50: 0.432 μM).RORγt/DHODH-IN-1 hasFormule :C24H26ClF6N3O3SCouleur et forme :SolidMasse moléculaire :585.99Carbonic anhydrase inhibitor 4
CA inhibitor 4, photoprobe; targets hCA I-XIV; Ki: 640-1166 nM.Formule :C21H18N2O4SCouleur et forme :SolidMasse moléculaire :394.44HER2-IN-12
HER2-IN-12 is an HER2 inhibitor with an IC50 value of 121 nM and can be used to study cancers such as breast cancer.Formule :C17H18BrN5O2SCouleur et forme :SolidMasse moléculaire :436.33Brostallicin HCl
CAS :Brostallicin, a synthetic MGB, inhibits DNA replication in cancer cells, inducing cell death, effective against MMR-defective tumors.Formule :C30H36BrClN12O5Couleur et forme :SolidMasse moléculaire :760.04Gemilukast
CAS :Gemilukast (ONO-6950) is a cysteinyl leukotriene 1 and 2 receptor inhibitor that inhibits bronchoconstriction and is used in the treatment of asthma.Formule :C36H37F2NO5Degré de pureté :98.27% - 99.5%Couleur et forme :SolidMasse moléculaire :601.68Ref: TM-T11388
1mg115,00€5mg274,00€10mg472,00€25mg914,00€50mg1.415,00€100mg2.517,00€1mL*10mM (DMSO)363,00€Gabaculine HCl
CAS :Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.Formule :C7H10ClNO2Couleur et forme :SolidMasse moléculaire :175.61Topo I-IN-1
Topo I-IN-1 (14d) is a powerful Topo I inhibitor with antitumor effects and DNA intercalation, inducing apoptosis.Formule :C20H14BrN3O2Couleur et forme :SolidMasse moléculaire :408.25Elocalcitol
CAS :Elocalcitol is a calcitriol analog for inhibition of prostate cell growth.Formule :C29H43FO2Couleur et forme :SolidMasse moléculaire :442.65PKCiota-IN-1
CAS :PKCiota-IN-1: Strong PKC-ι inhibitor (IC50=2.7 nM); also blocks PKC-α/ε (IC50s=45/450 nM).Formule :C25H22FN5OCouleur et forme :SolidMasse moléculaire :427.47Aplysin
CAS :Aplysin suppresses breast cancer cells and protects liver cells by blocking PI3K/AKT/FOXO3a and preventing oxidative damage.Formule :C15H19BrOCouleur et forme :SolidMasse moléculaire :295.21FXIa-IN-10
FXIa-IN-10 is a potent, orally bioavailable inhibitor of Activator XI (FXIa) (Ki: 0.17 nM).Formule :C23H18Cl2F3N9O2Couleur et forme :SolidMasse moléculaire :580.35GRP78-IN-1
GRP78-IN-1 binds to GRP78 protein, inhibits cell growth, and triggers apoptosis in breast cancer; has -8.07 kcal/mol binding energy.Formule :C21H23FO3Couleur et forme :SolidMasse moléculaire :342.4Massarilactone H
CAS :Massarilactone H, a polyketide, is a neuraminidase inhibitor, with an IC 50 of 8.18 µM .Formule :C11H12O5Couleur et forme :SolidMasse moléculaire :224.21OP-5244 sodium
OP-5244 sodium: potent oral CD73 inhibitor (IC50: 0.25 nM), potential in cancer research by hindering adenosine, reversing immunosuppression.Formule :C19H28ClN5NaO9PCouleur et forme :SolidMasse moléculaire :559.87Anticancer agent 65
CAS :Anticancer agent 65: Effective on A549 cells, IC50 1.07 μM, halts S phase, triggers apoptosis, elevates p53/p21, causes ROS and MMP collapse.Formule :C36H63NO5Couleur et forme :SolidMasse moléculaire :589.89CDK/HDAC-IN-1
CDK/HDAC-IN-1 inhibits CDK2/4/6 & HDAC6 with IC50s: 60.9, 276, 27.2, and 128.6 nM respectively.Formule :C20H18N4O4Couleur et forme :SolidMasse moléculaire :378.38Gimatecan
CAS :Gimatecan (STI481) is a potent topoisomerase I inhibitor. Gimatecan is an orally bioavailable camptothecin analogue with antitumor activity.Formule :C25H25N3O5Degré de pureté :98.47%Couleur et forme :SolidMasse moléculaire :447.48GR 122222X
CAS :GR 122222X is an inhibitor of topoisomerase II.Formule :C26H35N5O11SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :625.65Tofogliflozin
CAS :Tofogliflozin specifically inhibits SGLT2; IC50s are 2.9 nM (human), 14.9 nM (rat), 6.4 nM (mouse).Formule :C22H26O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.44LRRK2-IN-5
LRRK2-IN-5 is an oral, BBB-penetrating selective inhibitor for LRRK2 with IC50s: 1.2μM (GS) and 16μM (WT); halts LRRK2 autophosphorylation.Formule :C24H26F2N4O2SCouleur et forme :SolidMasse moléculaire :472.55BMS-986034
CAS :BMS-986034 is a GPR119 agonist.Formule :C24H24Cl2N6O4Couleur et forme :SolidMasse moléculaire :531.39MraY-IN-1
MraY-IN-1 inhibits MraY (IC50: 140μM), fights E. coli K12, B. subtilis W23, P. fluorescens (MIC50: 7-46μg/ml), for antimicrobial research.Formule :C35H46N3O5Couleur et forme :SolidMasse moléculaire :588.76Saphenamycin
CAS :Saphenamycin is an antibiotic from a strain of Streptomyces.Formule :C23H18N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :402.40ER272
CAS :ER272 is a natural PKC activator, inducing hippocampal neurogenesis.Formule :C24H34O6Couleur et forme :SolidMasse moléculaire :418.52Pociredir
CAS :Pociredir (FTX-6058), a potent EED inhibitor (KD=0.163 nM), may help in SCD research.Formule :C22H18FN5O2Couleur et forme :SolidMasse moléculaire :403.41MRS2279 diammonium
CAS :MRS2279 diammonium, a P2Y1 antagonist with K i 2.5 nM, IC 50 51.6 nM, blocks ADP-induced platelet aggregation, pK b 8.05.Formule :C13H24ClN7O8P2Couleur et forme :SolidMasse moléculaire :503.77IACS-8779 disodium
CAS :IACS-8779 disodium: potent STING agonist, strong systemic anti-tumor effects, effective in melanoma model.Formule :C21H23N9Na2O10P2S2Couleur et forme :SolidMasse moléculaire :733.52EGFR-IN-18
EGFR-IN-18 strongly inhibits L858R/T790M/C797S mutant EGFR (4.9 nM) and also targets wild-type EGFR (47 nM).Formule :C33H28N6O3SCouleur et forme :SolidMasse moléculaire :588.68(2S,4S)-Sacubitril
CAS :(2S,4S)-Sacubitril (Sacubitril Impurity C) is a stereoisomer derived from Sacubitril which is a potent NEP inhibitor.Formule :C24H29NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :411.49AZD 2066 hydrate
AZD 2066 hydrate is a selective, orally active, and brain-penetrant antagonist of mGluR5. It exhibits antinociceptive effects [1].Formule :C19H18ClN5O3Couleur et forme :SolidMasse moléculaire :386.33Sequoiaflavone
CAS :Sequoiaflavone is a biflavone isolated from Ginkgo biloba.Formule :C31H20O10Couleur et forme :SolidMasse moléculaire :552.48Antibiotic LL Z1640-2
CAS :Antibiotic LL Z1640-2 is an inhibitor against the TAK1 activity.Formule :C19H22O7Couleur et forme :SolidMasse moléculaire :362.38Aurora/LIM kinase-IN-1
Aurora/LIM kinase-IN-1 (Compound F114) is a dual inhibitor targeting aurora and lim kinases, potentially useful in GBM cancer treatment efforts.Formule :C16H20N6OCouleur et forme :SolidMasse moléculaire :312.37EP-7041 HCl
CAS :EP-7041 is a novel, potent, and selective Factor XIa inhibitor.Formule :C19H27ClN4O4Couleur et forme :SolidMasse moléculaire :410.89GPBAR1-IN-3
CAS :GPBAR1-IN-3 (Compound 14) is both a selective agonist for GPBAR1, with an EC50 value of 0.17 μM, and an antagonist for CysLT1R [1].Formule :C21H23NO2Couleur et forme :SolidMasse moléculaire :321.41MDK-3298
CAS :MDK-3298 is a reversible covalent inhibitor of Mcl-1, a target of protein-protein interaction (PPI).Formule :C35H32BN3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :617.46Zalunfiban dihydrochloride
Zalunfiban (RUC-4) is a potent αIIbβ3 platelet antagonist, IC50 45 nM, used in myocardial infarction research.Formule :C16H20Cl2N8O2SCouleur et forme :SolidMasse moléculaire :459.35Avorelin acetate
CAS :Avorelin acetate is a luteinizing hormone releasing hormone (LH-RH) agonist.Formule :C67H89N17O14Couleur et forme :SolidMasse moléculaire :1356.55MS117
MS117 is a first-in-class and cell-active irreversible covalent inhibitor of protein arginine methyltransferase 6 (PRMT6) (IC50 = 18 nM) [1].Formule :C17H22N4OCouleur et forme :SolidMasse moléculaire :298.38Leukotriene F4
CAS :LTF4, made in vitro from LTE4 with enzymes, contracts vascular muscle weakly; potency is LTD4 > LTC4 > LTE4 >> LTF4.Formule :C28H44N2O8SCouleur et forme :SolidMasse moléculaire :568.72(R)-BAY-899
(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.Formule :C25H19F2N5O2Couleur et forme :SolidMasse moléculaire :459.45PI3Kα-IN-8
PI3Kα-IN-8 is a selective inhibitor of PI3Kα (IC50: 0.012 μM).Formule :C26H27BrN4O2Couleur et forme :SolidMasse moléculaire :507.42MEIS-IN-1
CAS :MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.Formule :C24H21F3N2O4Couleur et forme :SolidMasse moléculaire :458.43P7170
CAS :P7170 is an anti-cancer agent active as an mTORC1/C2 and activin receptor-like kinase 1 (ALK1) inhibitor.Formule :C21H16F3N9Couleur et forme :SolidMasse moléculaire :451.42Nedocromil sodium
CAS :Nedocromil sodium is a pharmacologic stabilizer of mast cells, has been shown to normalize cytokine levels and attenuate cardiac remodeling.Formule :C19H17NNaO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.335Numidargistat
CAS :CB-1158 is a potent and orally bioavailable inhibitor of arginase (IC50s: 86 and 296 nM for recombinant human arginase 1 and 2).Formule :C11H22BN3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :287.12NK1 receptor antagonist 2
CAS :NK1 Receptor Antagonist 2, a compound targeting the NK1 receptor, holds potential for tinnitus and hearing loss research.Formule :C31H35F7N4O2Couleur et forme :SolidMasse moléculaire :628.62AMG-548 hydrochloride
AMG-548 hydrochloride: orally active, p38α inhibitor (Ki=0.5 nM), 1000x less for p38γ/δ, also blocks TNFα (IC50=3 nM) & inhibits casein kinase 1 δ/ε.Formule :C29H28ClN5OCouleur et forme :SolidMasse moléculaire :498.02Intoplicine
CAS :Intoplicine is an inhibitor of DNA topoisomerase I and II.Formule :C21H24N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :348.44RORγt inverse agonist 29
RORγt inverse agonist 29 is a potent, selective, orally active RORγt inverse agonist with an IC50 value of 21 nM.Formule :C25H24N2O5SCouleur et forme :SolidMasse moléculaire :464.53QPX7728 methoxy acetoxy methy ester
CAS :QPX7728 methoxy acetoxy methy ester is an inhibitor of boronic acid β-lactamase.Formule :C14H14BFO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.07LRRK2-IN-3
CAS :LRRK2-IN-3: potent, selective oral LRRK2 blocker, BBB-penetrant, IC50 of 0.6 nM in hPBMCs, for Parkinson's research.Formule :C25H29ClF2N6O2Couleur et forme :SolidMasse moléculaire :518.99Canosimibe
CAS :Canosimibe is a cholesterol absorption inhibitorFormule :C44H60FN3O10Couleur et forme :SolidMasse moléculaire :809.96T-3861174
CAS :T-3861174 is a prolyl tRNA synthetase (PRS) inhibitor, exhibiting significant in vitro anti-tumor activity with GCN2-ATF4 pathway activation.Formule :C26H25FN6O2Couleur et forme :SolidMasse moléculaire :472.51Anti-inflammatory agent 18
Anti-inflammatory agent 18: NO activity blocker (IC50: 15.94 μM), hampers HMGB1-induced inflammation, potential for COVID-19, sepsis study.Formule :C30H50O6Couleur et forme :SolidMasse moléculaire :506.71Cav 3.2 inhibitor 3
Cav 3.2 inhibitor 3 is a potent inhibitor of the Cav3.2 T-type Ca2+channel (IC50: 0.1534 μM) and has a low binding affinity for D2 receptors.Formule :C32H37N3O2Couleur et forme :SolidMasse moléculaire :495.66FTO-IN-1 TFA
FTO-IN-1 TFA: FTO enzyme inhibitor, anti-obesity, IC50 < 1μM, potential cancer research tool.Formule :C20H17Cl2F3N4O4Couleur et forme :SolidMasse moléculaire :505.27DS01080522
DS01080522: PRKACA inhibitor, IC50: kinase 0.8 nM, CREB 66 nM; potential for cancer research.Formule :C23H20Cl2N4O3Couleur et forme :SolidMasse moléculaire :471.34HG-12-6
CAS :HG-12-6 is a type II IRAK4 inhibitor, targeting its inactive form with an IC50 of 165 nM, and is used in autoimmunity and inflammation.Formule :C29H27F3N6O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :580.62GSK789
CAS :GSK789 is a selective inhibitor of the first bromodomains (BD1) of the bromo and extra terminal domain (BET) proteins.Formule :C26H33N5O3Couleur et forme :SolidMasse moléculaire :463.57UCN-01
CAS :inhibitor of Akt, protein kinase C, PDK1 and cyclin-dependent kinasesFormule :C28H26N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.53Top/HDAC-IN-1
Top/HDAC-IN-1: Dual Top/HDAC inhibitor, potent against HDAC1-3,6,8 and HCT116 cells; blocks G2 phase, induces apoptosis.Formule :C29H27N5O4Couleur et forme :SolidMasse moléculaire :509.56PSB 36
CAS :A1 adenosine receptor antagonistFormule :C21H30N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.49Myxothiazol
CAS :Myxothiazol blocks mitochondrial complex III and triggers SESN2, a gene important for stress response.Formule :C25H33N3O3S2Couleur et forme :SolidMasse moléculaire :487.68Factor B-IN-3
CAS :Factor B-IN-3 is a potent inhibitor of complement factor B. Factor B-IN-3 can be used to study inflammatory and immune-related diseases.Formule :C24H29N3O4Couleur et forme :SolidMasse moléculaire :423.5KRAS G12D inhibitor 3
CAS :KRAS G12D Inhibitor 3, a compound targeting the KRAS G12D mutation, demonstrates potent antitumor efficacy with an inhibitory concentration (IC50) of less thanFormule :C34H31ClF3N5O2Couleur et forme :SolidMasse moléculaire :634.09Soyacerebroside II
CAS :Soyacerebroside II is a Ca2+ ionophore; both I and II inhibit IL-18 in PBMCs and modulate immune responses.Formule :C40H75NO9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :714.02Gepotidacin hydrochloride
CAS :Gepotidacin (GSK-2140944) is a potent DNA topoisomerase inhibitor, a novel antibacterial efficacious against various anaerobes.Formule :C24H29ClN6O3Couleur et forme :SolidMasse moléculaire :484.98Taranabant
CAS :Taranabant: potent CB1 receptor inverse agonist; inhibits agonists with 0.13 nM Ki in vitro.Formule :C27H25ClF3N3O2Degré de pureté :99.06% - 99.06%Couleur et forme :SolidMasse moléculaire :515.96Antileishmanial agent-5
Antileishmanial agent-4, a ribonucleoside analogue, targets L.infantum and T.cruzi with EC50s of 0.68 μM and 0.83 μM.Formule :C17H17ClN4O4Couleur et forme :SolidMasse moléculaire :376.79FAAH/MAGL-IN-1
FAAH/MAGL-IN-1 (SIH 3) inhibits FAAH & MAGL with IC50 of 31 & 29 nM, useful in neuropathic pain research.Formule :C15H9Cl2N3O3Couleur et forme :SolidMasse moléculaire :350.16BMS 310705
CAS :BMS 310705, an Epothilone B analog, targets ovarian/renal/bladder/lung cancer, inducing apoptosis via mitochondria.Formule :C27H42N2O6SCouleur et forme :SolidMasse moléculaire :522.70CCR4 antagonist 2
CAS :CCR4 antagonist 2 (Compound 31) is a novel potent, orally bioavailable small molecule antagonists of CC chemokine receptor 4 (CCR4) that inhibits TregFormule :C26H28Cl2N6ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :511.45GSK8814
CAS :GSK8814 is a selective and ATAD2/2B bromodomain chemical probe and inhibitor (binding constant pKd=8.1 and a pKi=8.9 in BROMOscan).Formule :C28H35F2N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.61PF 03709270
CAS :PF 03709270 is an oral prodrug of sulopenem with broad-spectrum antibacterial effects on gram-positive and gram-negative bacteria.Formule :C19H27NO7S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.61ONO-DI-004
CAS :ONO-DI-004 is a selective EP1 Prostanoid receptor agonist.Formule :C24H38O6Couleur et forme :SolidMasse moléculaire :422.55CYP2C19-IN-1
CYP2C19-IN-1: potent CYP2C19 inhibitor, non-genotoxic, non-hepatotoxic, blocks RdRP (Ki: 6.16 μM), useful for ZIKV research.Formule :C26H26N2O6SCouleur et forme :SolidMasse moléculaire :494.56Anti-MRSA agent 2
CAS :Anti-MRSA agent 2 inhibits MRSA at 0.098 μg/ml, with low toxicity and disrupts bacterial membranes and DNA.Formule :C18H10Br2N2OCouleur et forme :SolidMasse moléculaire :430.09Antibiotic MA 144M2
CAS :Antibiotic MA 144M2, an anthracycline glycoside, targets gram-positive bacteria and tumors, derived from Streptomyces and aclacinomycin A conversion.Formule :C42H55NO16Couleur et forme :SolidMasse moléculaire :829.88AP5
CAS :AP5: GPR40 agonist, positive allosteric modulator; rat hIP1 EC50: 0.49 nM.Formule :C28H28FNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.52
