Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.764 produits)
- Apoptose(6.204 produits)
- Cycle cellulaire/point de contrôle(4.811 produits)
- Chromatine/Épigénétique(2.553 produits)
- Signalisation du cytosquelette(1.519 produits)
- Altération de l'ADN/réparation de l'ADN(2.906 produits)
- Endocrinologie/Hormones(3.703 produits)
- Enzyme(3.671 produits)
- GPCR/G-Protéine(8.966 produits)
- Immunologie et Inflammation(3.748 produits)
- Virus de la grippe(297 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.244 produits)
- Transporteur membranaire/Canal ionique(3.119 produits)
- Métabolisme(10.122 produits)
- Microbiologie/Virologie(7.569 produits)
- Neuroscience(10.314 produits)
- Autres inhibiteurs(35.802 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.411 produits)
- Protéases/Protéasome(1.681 produits)
- Cellules souche et Dérivés(752 produits)
- Tyrosine Kinase/Adaptateurs(1.947 produits)
- Ubiquitination(1.716 produits)
Affichez 16 plus de sous-catégories
66604 produits trouvés pour "Inhibiteurs"
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RSV-IN-7
CAS :RSV-IN-7 (example 253) is a RSV inhibitor ( EC 50 : < 0.4 μΜ) .Formule :C27H22F3N7O3Couleur et forme :SolidMasse moléculaire :549.50Antibacterial agent 69
Antibacterial agent 69 is a novel structural antimicrobial modulator that can be used against lethal multidrug-resistant bacterial infections (MIC: 2.978 μM).Formule :C24H19N3O4SCouleur et forme :SolidMasse moléculaire :445.49AMPK Activator SC4
CAS :SC4 is a potent, direct AMPK activator. SC4 preferentially activates α2 complexes and stimulates skeletal muscle glucose uptake.Formule :C26H18ClN3O4Couleur et forme :SolidMasse moléculaire :471.89DNA crosslinker 1 dihydrochloride
CAS :DNA Crosslinker 1 binds DNA minor groove with 1.1°C affinity increase; used in cancer research.Formule :C15H22Cl2N8OCouleur et forme :SolidMasse moléculaire :401.29Antitumor agent-51
Antitumor agent-51 targets osteosarcoma with 21.9 nM IC50, high selectivity, and low toxicity.Formule :C23H25N5O2SCouleur et forme :SolidMasse moléculaire :435.54EGFR/HER2-IN-8
EGFR/HER2-IN-8 inhibits EGFR, HER2, DHFR (IC50: 0.45, 0.244, 5.669 μM); useful in cancer research, safe and selective.Formule :C16H16N4O2SCouleur et forme :SolidMasse moléculaire :328.39DNA-PK-IN-6
CAS :DNA-PK-IN-6 inhibits DNA-PKcs, disrupting tumor DNA repair and triggering apoptosis; enhances radiotherapy and targets various tumors (WO2021197159A1).Formule :C19H21N7OCouleur et forme :SolidMasse moléculaire :363.42Dup-714
CAS :Dup-714 is a thrombin inhibitor.Formule :C21H33BN6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :460.33Elacestrant S enantiomer
Elacestrant S enantiomer is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.Formule :C30H38N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :458.63JNJ-1250132
CAS :JNJ-1250132 is a steroidal progesterone receptor modulator that inhibits binding of the receptor to DNA in vitro.Formule :C33H41NO4Couleur et forme :SolidMasse moléculaire :515.68(-)-Cevimeline hydrochloride hemihydrate
(-)-Cevimeline HCl hemihydrate, a muscarinic agonist, treats Sjogren's xerostomia. Quick absorption, species-dependent metabolism.Formule :C10H19ClNO1·5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :244.78LAS195319
CAS :LAS195319 is a potent and selective inhaled PI3Kδ Inhibitor (IC50 = 0.5 nM) for the Treatment of Respiratory Diseases.Formule :C29H26N10O3SCouleur et forme :SolidMasse moléculaire :594.65LY 292728
CAS :LY 292728 is a highly potent antagonist of leukotriene B4 receptor.Formule :C34H29FO9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :600.59THR-β agonist 5
CAS :THR-β agonist 5 (compound 54) is a potent THR-β agonist, with an EC 50 of <50 nM [1].Formule :C22H23N5O2Couleur et forme :SolidMasse moléculaire :389.45L-threo-Sphingosine C-18
CAS :L-threo-Sphingosine C-18 is a protein kinase C inhibitor.Formule :C18H37NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :299.49AChE-IN-10
AChE-IN-10 (24r) inhibits AChE (IC50=2.4 nM), reducing amyloid buildup, tau phosphorylation, and promotes neuron health.Formule :C23H27F2NO4SCouleur et forme :SolidMasse moléculaire :451.53KH-259
KH-259: potent, selective CNS-penetrant HDAC6 inhibitor with 0.26 μM IC50; shows antidepressant effects in mice.Formule :C20H25N3O2Couleur et forme :SolidMasse moléculaire :339.43Anticancer agent 64
CAS :Anticancer agent 64 (5m) induces apoptosis, has IC50 2.4μM in CCRF-CEM, activates caspases, cleaves PARP, affects mitochondria.Formule :C31H46N2O2SCouleur et forme :SolidMasse moléculaire :510.77β-Secretase Inhibitor III
β-Secretase Inhibitor III is a highly selective inhibitor of BACE1 with a Ki value of 0.13 nM.Formule :C20H20F2N4O3SCouleur et forme :SolidMasse moléculaire :434.46ATR-IN-19
CAS :ATR-IN-19 (Compound 15 R-configure) is an ATR inhibitor [1].Formule :C18H19N7OSCouleur et forme :SolidMasse moléculaire :381.45IRAK4-IN-11
IRAK4-IN-11 (compound 6) is a potent inhibitor of IRAK4 with an IC 50 of 0.008 μM. IRAK4-IN-11 exhibits cell pIRAK4 potencies with an IC 50 of 0.19 μM [1].Formule :C16H19N7OCouleur et forme :SolidMasse moléculaire :325.37EGFR/HER2-IN-5
EGFR/HER2-IN-5: Irreversible, oral dual EGFR inhibitor, IC50 0.6 nM, targets L858R/T790M mutations, anti-tumor in vivo for lung cancer study.Couleur et forme :SolidIsobetanin
CAS :Isobetanin is a betacyanin that has been shown to enhance vitexin-2-O-xyloside mediated inhibition of proliferation of T24 bladder cancer cells.
Formule :C24H26N2O13Couleur et forme :SolidMasse moléculaire :550.47(Rac)-Nebivolol
CAS :(Rac)-Nebivolol, a racemic β1-adrenergic blocker (IC50=0.8 nM), has vasodilatory properties and mitigates ethanol-induced cardiac harm.Formule :C22H25F2NO4Couleur et forme :SolidMasse moléculaire :405.43PD-1/PD-L1-IN-16
PD-1/PD-L1-IN-16 is a potent inhibitor of PD-1/PD-L1 (IC50: 53.2 nM) and has shown research potential for tumour immunotherapy.Formule :C34H30N4O4Couleur et forme :SolidMasse moléculaire :558.632R,4S-Sacubitril
CAS :2R,4S-Sacubitril (Sacubitril Enantiomer) is the impurity of Sacubitril which is a neprilysin inhibitor.Formule :C24H28NO51CaDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :430.49AM9405
AM9405: peripheral CB1/5-HT3 agonist, suppresses gut motility, relieves GI disorder symptoms in mice.Formule :C24H33BrN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.44Tofacitinib Prodrug-1
Tofacitinib Prodrug-1: an oral prodrug reducing Tofacitinib's side effects, treats ulcerative colitis in mice effectively with low toxicity.Formule :C36H39ClN10O7Couleur et forme :SolidMasse moléculaire :759.21FXIa-6f
CAS :FXIa-6f is a high affinity, orally bioavailable macrocyclic FXIa inhibitor with antithrombotic activity in preclinical speciesFormule :C31H29ClF2N4O4Couleur et forme :SolidMasse moléculaire :595.04MSX-3 free acid
CAS :MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.Formule :C21H23N4O7PCouleur et forme :SolidMasse moléculaire :474.40Dihydrokainic acid
CAS :EAAT2(GLT1)-selective non-transportable inhibitor of L-glutamate and L-aspartate uptakeFormule :C10H17NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :215.25HPK1-IN-3
HPK1-IN-3: Selective HPK1 inhibitor, ATP-competitive, IC50=0.25nM; boosts IL-2 in PBMCs, EC50=108nM.Formule :C23H22F4N6O2Couleur et forme :SolidMasse moléculaire :490.45CVS-1578
CAS :CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.Formule :C20H30N6O5SCouleur et forme :SolidMasse moléculaire :466.55Oxeclosporin
CAS :Oxeclosporin is a hydroxyethyl derivative of serine(8)-cyclosporine; inhibits proliferation and functions of lymphocytes.Formule :C64H115N11O14Couleur et forme :SolidMasse moléculaire :1262.66RAD51-IN-8
RAD51-IN-8 inhibits RAD51-BRCA2 interaction and H4A4 with EC50 of 19 μM; a micromolar PPI inhibitor.Formule :C16H14Cl2FN3O2Couleur et forme :SolidMasse moléculaire :370.21MAP3K14-IN-173
CAS :MAP3K14-IN-173 is a potent MAP3K14 kinase inhibitor.Formule :C29H31N7O2Couleur et forme :SolidMasse moléculaire :509.60DC4SMe
CAS :DC4SMe, a prodrug for targeted tumor therapy and ADC synthesis, has IC50s: 1.9 nM (Ramos), 2.9 nM (Namalwa), 1.8 nM (HL60/s).Formule :C35H31ClN5O7PS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :764.21L 671776
CAS :L 671776 is an inositol monophosphatase inhibitor.Formule :C23H32O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :388.5BI-2540
CAS :BI-2540 is a HIV non-nucleoside reverse transcriptase ( NNRT ) inhibitor .Formule :C24H15ClF5NO5Couleur et forme :SolidMasse moléculaire :527.83MALT1-IN-5
CAS :MALT1-IN-5 is a potent inhibitor of the MALT1 protease and can be used in cancer research.Formule :C17H17ClF2N6O3Couleur et forme :SolidMasse moléculaire :426.80Beloxepin
CAS :Beloxepin is an oral dual selective inhibitor of serotonin and norepinephrine uptake.Formule :C19H21NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :295.38Agosterol A
CAS :Agosterol A is isolated from marine sponge Spongia.Formule :C33H52O8Couleur et forme :SolidMasse moléculaire :576.76SM-433 hydrochloride
SM-433 hydrochloride, a Smac mimetic & IAP inhibitor, binds XIAP BIR3; potent IC50 <1 μM. (Patent WO2008128171A2)Formule :C32H44ClN5O4Couleur et forme :SolidMasse moléculaire :598.18AChE/BuChE-IN-3
CAS :AChE/BuChE-IN-3 inhibits AChE (IC50: 0.65 μM), BuChE (IC50: 5.77 μM), crosses BBB, and hinders Aβ1-42 aggregation for Alzheimer's research.Formule :C30H30F3N3O6Couleur et forme :SolidMasse moléculaire :585.57D-Cl-amidine hydrochloride
D-Cl-amidine hydrochloride is a potent and highly selective inhibitor of PAD1. It exhibits excellent tolerance and does not induce significant toxicity [1].Formule :C14H20Cl2N4O2Couleur et forme :SolidMasse moléculaire :347.24DHU-Se1
DHU-Se1: potent anti-inflammatory, releases reactive selenium from macrophages, inhibits iNOS/TNF-α, blocks M0 to M1 polarization.Formule :C23H23N3OSSeCouleur et forme :SolidMasse moléculaire :468.47STA 2
CAS :STA 2 is an analogue of TXA2, a thromboxane receptor in the colonic epithelium.Formule :C21H34O3SCouleur et forme :SolidMasse moléculaire :366.56LAF-153
CAS :LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.Formule :C18H32N2O7Couleur et forme :SolidMasse moléculaire :388.46ATX inhibitor 22
ATX inhibitor 22 is a novel inhibitor of ATX (autotaxin) (IC50: 218.9 μM) that lacks inhibitory activity against LPAR1.Formule :C19H17Cl3F2N2O4SCouleur et forme :SolidMasse moléculaire :513.77SI-109
CAS :SI-109 is a potent inhibitor of STAT3 SH2 domain (Ki=9 nM),and with antitumor activity.Formule :C40H44F2N7O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :835.79GYKI-53784
CAS :GYKI-53784 (LY 303070) is an effective selective AMPA receptor antagonist.Formule :C19H20N4O3Couleur et forme :SolidMasse moléculaire :352.39Antibacterial agent 78
Antibacterial agent 78 (compound 30) is an antibacterial agent with improved cytotoxicity profile[1].Formule :C16H23N3S2Couleur et forme :SolidMasse moléculaire :321.5HDAC-IN-9
HDAC-IN-9, a dual tubulin/HDAC inhibitor, impedes A549 cell invasion/migration and shows strong anti-tumor/angiogenic effects.Formule :C33H38N2O4Couleur et forme :SolidMasse moléculaire :526.67Unoprostone
CAS :Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.Formule :C22H38O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :382.53SphK1-IN-1
SphK1-IN-1: SphK1 ATPase inhibitor, IC50=2.48 μM, potential for cancer research.Formule :C22H22N6O2Couleur et forme :SolidMasse moléculaire :402.45LSD1/2-IN-3
LSD1/2-IN-3 selectively inhibits LSD1 (Ki 11 nM) over LSD2 (Ki 7 μM), and hinders tumor stem cell proliferation.Formule :C9H8BrF2NCouleur et forme :SolidMasse moléculaire :248.07Antimalarial agent 2
Antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects.Formule :C27H25N3O5Couleur et forme :SolidMasse moléculaire :471.5DHFR-IN-4
CAS :DHFR-IN-4 is a potent dihydrofolate reductase (DHFR) inhibitor with anti-tumour activity, inhibits EGFR and HER2 and can be used to study pancreatic cancer.Formule :C18H21N5O2SDegré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :371.46OP-2507
CAS :OP-2507, a prostacyclin agonist, is used potentially for the treatment of hepatic insufficiency and hypertension.Formule :C25H41NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :419.6LY3130481
CAS :LY3130481: TARP γ-8 dependent AMPA receptor blocker; selectively targets AMPA/TARP γ-8 with 65 nM IC50.Formule :C19H18N4O3SCouleur et forme :SolidMasse moléculaire :382.44TBK1/IKKε-IN-1
CAS :TBK1/IKKε-IN-1 is a dual inhibitor of TBK1 and IKKε (IC50s of <100 nM).Formule :C28H26N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :498.53LEO 134310
CAS :LEO 134310: Selective, non-steroidal GR agonist with 14 nM EC50, for topical skin disease treatment.Formule :C34H40N2O8Couleur et forme :SolidMasse moléculaire :604.69GSK 932121
CAS :GSK 932121: potent antimalarial, targets P. falciparum by inhibiting cytochrome bc1 in the electron transport chain.Formule :C20H15ClF3NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.79GNE-2256
CAS :GNE-2256, also known as molecule 19, is an orally active compound that inhibits Interleukin 1 receptor-associated kinase 4 (IRAK4) with a K i of 1.4 nM and hasFormule :C24H27FN6O4Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :482.51Antileishmanial agent-6
Antileishmanial agent-6: potent against Leishmania donovani, IC50 0.54μM; cytotoxic IC50 10.2μM.Formule :C24H26O8Couleur et forme :SolidMasse moléculaire :442.46MK-7445
CAS :MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase.Formule :C21H13Cl2N7OCouleur et forme :SolidMasse moléculaire :450.28Dopamine D3 receptor antagonist-2
Dopamine D3 receptor antagonist-2 is a dopamine D3 receptor selective (Ki=2.16 nM) or multi-targeting dual ligand that shows potential effects in CNS disorders.Formule :C23H27Cl2N3O3Couleur et forme :SolidMasse moléculaire :464.38BAY-091
CAS :BAY-091 is a novel potent and highly selective PIP4K2A kinase inhibitor.Formule :C26H21FN4O2Degré de pureté :97.66% - 99.23%Couleur et forme :SoildMasse moléculaire :440.47Ref: TM-T60147
1mg82,00€5mg177,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€500mgÀ demander1mL*10mM (DMSO)188,00€Antibacterial agent 90
Antibacterial agent 90 (6n), a pleuromutilin derivative, targets Gram-positive pathogens and Mycoplasma pneumoniae.Formule :C30H42N2O6Couleur et forme :SolidMasse moléculaire :526.66CXCR7 modulator 2
CAS :CXCR7 modulator 2 is a 7-type C-X-C chemokine receptor (CXCR7) modulator with a Ki of 13 nM.Formule :C29H42N6O3Couleur et forme :SolidMasse moléculaire :522.68Sargachromanol E
CAS :Sargachromanol E is a compound isolated from the marine brown alga, Sargassum horneri. It has been studied for its inhibitory effect on skin ageing.Formule :C27H40O4Couleur et forme :SolidMasse moléculaire :428.6Lentiginosine
CAS :Lentiginosine is a selective amyloglucosidase inhibitor.Formule :C8H15NO2Couleur et forme :SolidMasse moléculaire :157.21WM382
CAS :WM382, a potent dual PMIX/X inhibitor, has IC50s of 1.4 nM/0.03 nM and effective against various malaria stages.Formule :C29H36N4O4Couleur et forme :SolidMasse moléculaire :504.62ETP-47037
CAS :ETP-47037: strong PI3Kα inhibitor (IC50: 0.99 nM), also targets PI3Kβ, δ, γ; may protect telomeres.Formule :C20H27N9O3SCouleur et forme :SolidMasse moléculaire :473.555-HT6R/MAO-B modulator 1
5-HT6R/MAO-B modulator 1 blocks 5-HT6R and permanently inhibits MAO-B, protects glial cells, and reverses memory loss.Formule :C33H38N4O3SCouleur et forme :SolidMasse moléculaire :570.74MMAF sodium
CAS :MMAF sodium, a potent tubulin inhibitor in ADCs like Vorsetuzumab mafodotin and SGN-CD19A, acts as an antitumor agent.Formule :C39H64N5NaO8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :753.94LY 178210
CAS :LY 178210 is a 5-hydroxytryptamine receptor agonist.Formule :C18H25N3OCouleur et forme :SolidMasse moléculaire :299.41K027
K027 is a potent organophosphate (OP) inhibitor of acetylcholinesterase (AChE) reactivation. k027 can be used to study Alzheimer's disease.Formule :C15H18Br2N4O2Couleur et forme :SolidMasse moléculaire :446.1412(S)-HETE
CAS :Enpatoran hydrochloride (M5049 hydrochloride) is a TLR7/8 inhibitor with antiviral activity that is used in the study of autoimmune diseases.
Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.47AMG-315
CAS :AMG-315: Chiral AEA analogue, potent CB1 agonist (Ki 7.8 nM, EC50 0.6 nM), stable against hydrolyzing/oxidative enzymes.Formule :C24H41NO2Couleur et forme :SolidMasse moléculaire :375.59KCL-440
CAS :RS 57639 is a bioactive chemical.Formule :C18H18N2O2Couleur et forme :SolidMasse moléculaire :294.35Tubulin inhibitor 17
Compound 3b inhibits tubulin polymerization, IC50 12.38 µM, with anticancer properties and promotes cell apoptosis.Formule :C17H16N2OCouleur et forme :SolidMasse moléculaire :264.32MRTX849 acid
CAS :MRTX849 acid, used to make PROTAC LC-2, effectively degrades KRAS G12C at 0.25-0.76 μM DC50.Formule :C34H37ClFN7O4Couleur et forme :SolidMasse moléculaire :662.16S39625
CAS :S39625 is a stable, potent topoisomerase I inhibitor with anticancer properties, resistant to efflux transporters, inducing gamma-H2AX at nanomolar levels.Formule :C25H22N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :430.4511-trans Leukotriene E4
CAS :Slow isomerization of the C-11 double bond of LTE4 leads to the formation of 11-trans LTE4. 11-trans LTE4 is equipotent to LTE4 in contracting guinea pig ileum.Formule :C23H37NO5SCouleur et forme :SolidMasse moléculaire :439.61U92016A hydrochloride
CAS :U92016A hydrochloride: potent, orally active 5-HT1A agonist, metabolically stable, high intrinsic activity, Ki=0.2 nM.Formule :C19H26ClN3Couleur et forme :SolidMasse moléculaire :331.89TAP311
TAP311 is an inhibitor of cholesteryl ester transfer protein (CETP)(IC50 of 62 nM).Formule :C34H40F6N6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :710.71YKL-1-116
CAS :YKL-1-116 is an effective, selective, and covalent CDK7 inhibitor.Formule :C34H38N8O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :606.72NLRP3-IN-4
NLRP3-IN-4 is an effective, oral NLRP3 inflammasome inhibitor with potent anti-inflammatory effects on colitis.Formule :C22H22N2O5Couleur et forme :SolidMasse moléculaire :394.42HBV-IN-11
CAS :HBV-IN-11 is a potent inhibitor of HBsAg secretion (EC50: 0.46 μM).Formule :C21H24ClNO6Couleur et forme :SolidMasse moléculaire :421.87Domitroban
CAS :Domitroban, also known as S-145, is a thromboxane (Tx) A2-receptor antagonist with partial agonistic activity in vascular smooth muscle.Formule :C20H27NO4SCouleur et forme :SolidMasse moléculaire :377.5c-Met-IN-2
CAS :c-Met-IN-2 is a selective and orally available c-Met inhibitor (IC50: 0.6 nM) with antitumor activity.Formule :C24H21FN10ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :484.49Rodatristat ethyl
CAS :Rodatristat ethyl is an oral TPH1 inhibitor reducing 5-HT levels & lowering PAH at low doses.Formule :C29H31ClF3N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :590.04ATR-IN-7
CAS :ATR-IN-7 is a potent inhibitor of ATR.Formule :C21H22FN7OCouleur et forme :SolidMasse moléculaire :407.44Org-6906
CAS :DCB-3503, a tylophorine analog, may treat cancer and suppress immunity by blocking protein synthesis and modulating HSC70's ATPase activity.Formule :C13H16ClNDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :221.73Chitin synthase inhibitor 5
Calpain Inhibitor-2, lipophilic, inhibits calpain; shows anti-proliferative effects on melanoma, PC-3 cells; blocks 80% DU-145 cell invasion.Formule :C23H22BrN3O5Couleur et forme :SolidMasse moléculaire :500.34Tenellin
CAS :Tenellin is a fungal metabolite that inhibits Mg2+-, Ca2+-, and Na+/K+-ATPase activities in erythrocytes. Tenellin is cytotoxic to Sf9 and Sf21 insect cells.Formule :C21H23NO5Couleur et forme :SolidMasse moléculaire :369.41PLAP-IN-1
CAS :PLAP-IN-1: Potent, selective inhibitor of PLAP, IC50 of 32 nM; doesn't notably inhibit TNAP.Formule :C25H21Cl2N3O5Couleur et forme :SoildMasse moléculaire :514.36Tonapofylline
CAS :Tonapofylline, orally active, selectively blocks A1 adenosine receptor (Ki: 7.4 nM), used in heart failure research.Formule :C22H32N4O4Degré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :416.51Antitumor agent-54
Compound C11 inhibits 14-3-3η protein (KD: 35 μM), targets liver cancer cells, blocks G1-S phase, and induces apoptosis.Formule :C29H32N2O3Couleur et forme :SolidMasse moléculaire :456.58
