
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.781 produits)
- Apoptose(6.260 produits)
- Cycle cellulaire/point de contrôle(4.792 produits)
- Chromatine/Épigénétique(2.440 produits)
- Signalisation du cytosquelette(1.527 produits)
- Altération de l'ADN/réparation de l'ADN(2.968 produits)
- Endocrinologie/Hormones(3.706 produits)
- Enzyme(3.667 produits)
- GPCR/G-Protéine(9.005 produits)
- Immunologie et Inflammation(3.874 produits)
- Virus de la grippe(301 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.248 produits)
- Transporteur membranaire/Canal ionique(3.033 produits)
- Métabolisme(10.207 produits)
- Microbiologie/Virologie(7.591 produits)
- Neuroscience(10.382 produits)
- Autres inhibiteurs(36.042 produits)
- Oxydation-Réduction(42 produits)
- Signalisation PI3K/Akt/mTOR(1.444 produits)
- Protéases/Protéasome(1.724 produits)
- Cellules souche et Dérivés(825 produits)
- Tyrosine Kinase/Adaptateurs(2.035 produits)
- Ubiquitination(1.717 produits)
Affichez 16 plus de sous-catégories
66686 produits trouvés pour "Inhibiteurs"
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Epalrestat
CAS :Epalrestat (ONO2235), an aldose reductase inhibitor, helps manage diabetic neuropathy symptoms and slows disease progression.Formule :C15H13NO3S2Degré de pureté :99.2% - 99.54%Couleur et forme :Deep Red Acicular CrystalMasse moléculaire :319.4PIT
CAS :PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with an IC50 of 0.14 μM for human P2Y1.Formule :C20H16N2O5SDegré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :396.42Rolinsatamab
CAS :<p>Rolinsatamab: a humanized monoclonal antibody, blocks IL-4/IL-13, and modifies T cells, treating immune diseases.</p>Degré de pureté :> 95%Couleur et forme :LiquidMasse moléculaire :145.48 kDaPromestriene
CAS :Promestriene (3-propyl ethyl) (INN) is a synthetic estrogen and glucocorticoid used topically in a 1% cream formulation.Formule :C22H32O2Degré de pureté :99.35%Couleur et forme :White SolidMasse moléculaire :328.49Folic acid
CAS :<p>Folic acid (Vitamin B9) is a vitamin B9 that is essential for the synthesis of DNA/RNA and for the production new cells. Cost-effective and quality-assured.</p>Formule :C19H19N7O6Degré de pureté :99.19% - 99.27%Couleur et forme :Yellowish-Orange Crystals; Extremely Thin Platelets (Elongated @ 2 Ends) From Hot Water 482°FMasse moléculaire :441.40Dimethylsulfamoyl chloride
CAS :Dimethylsulfamoyl chloride (DMSC) is an organosulfur compoundused in organic synthesis and laboratory reagents.Formule :C2H6ClNO2SDegré de pureté :99.31%Couleur et forme :Less Liquid Colorless LiquidMasse moléculaire :143.59Nitazoxanide
CAS :Nitazoxanide (NSC-697855) is a synthetic benzamide antiprotozoal; it disrupts pyruvate electron transfer reactions.Formule :C12H9N3O5SDegré de pureté :99% - 99.93%Couleur et forme :SolidMasse moléculaire :307.28Chlorpheniramine maleate
CAS :Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.Formule :C20H23ClN2O4Degré de pureté :99.64% - 99.98%Couleur et forme :Odorless White Crystalline Solid Or White Powder With A Bitter TasteMasse moléculaire :390.87Samidorphan HCl
CAS :<p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>Formule :C21H27ClN2O4Degré de pureté :96.79% - 97.85%Couleur et forme :SoildMasse moléculaire :406.9Imiquimod
CAS :Imiquimod (R 837) is an immune response modifier that acts as a toll-like receptor 7 agonist.Formule :C14H16N4Degré de pureté :99.62% - >99.99%Couleur et forme :White To Off White Crystalline PowderMasse moléculaire :240.30Tidembersat
CAS :Tidembersat is a small molecule compound used to treat and/or prevent degenerative diseases such as Huntington's chorea, schizophrenia, neurological.Formule :C20H19F2NO4Degré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :375.37p-MPPI hydrochloride
CAS :p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.Formule :C25H28ClIN4O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :578.87Ref: TM-T16421
2mg40,00€5mg59,00€10mg93,00€25mg145,00€50mg235,00€100mg371,00€200mg550,00€1mL*10mM (DMSO)89,00€AZD-8529 mesylate
CAS :AZD-8529 mesylate is a highly selective, and orally bioavailable positive allosteric modulator of mGluR2 (EC50: 285 nM).Formule :C25H28F3N5O6SDegré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :583.58Ref: TM-T10432L
1mg57,00€5mg120,00€10mg188,00€25mg432,00€50mg747,00€100mg1.093,00€200mg1.454,00€1mL*10mM (DMSO)156,00€Ethyleneurea
CAS :Ethyleneurea (Imidazolidinone) is used as a formaldehyde scavenger and intermediate.Formule :C3H6N2ODegré de pureté :98.47%Couleur et forme :White To Pale-Yellow White To Pale-Yellow Powder Or CrystalsMasse moléculaire :86.09Atovaquone
CAS :Atovaquone (Atavaquone) is a hydroxynaphthoquinone that has antimicrobial activity and is being used in antimalarial protocols.Formule :C22H19ClO3Degré de pureté :98% - 99.85%Couleur et forme :Yellow To Orange Crystalline SolidMasse moléculaire :366.84Vitamin D2
CAS :Ergocaliferol (Vitamin D2), derived from ergosterol by UV, inhibits bladder tumor promotion and leukemia, and blocks DNA Polymerase.Formule :C28H44ODegré de pureté :98.73% - 99.89%Couleur et forme :Prisms From Acetone 1998)Masse moléculaire :396.65Ciliobrevin D
CAS :Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor.Formule :C17H8Cl3N3O2Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :392.62Ref: TM-T14965
1mg64,00€2mg92,00€5mg140,00€10mg215,00€25mg424,00€50mg625,00€100mg873,00€1mL*10mM (DMSO)157,00€STAT3-IN-1
CAS :STAT3-IN-1 selective and orally active inhibitor of STAT3(in HT29 and MDA-MB 231 cells, with IC50 values of 1.82 μM and 2.14 μM , respectively), induces tumorFormule :C28H29NO6Degré de pureté :95.89% - 95.89%Couleur et forme :SolidMasse moléculaire :475.53Ref: TM-T13009
1mg60,00€2mg88,00€5mg131,00€10mg192,00€25mg349,00€50mg523,00€100mg753,00€500mg1.549,00€1mL*10mM (DMSO)137,00€Diclofenac sodium
CAS :<p>Diclofenac sodium (GP 45840) is a non-steroidal anti-inflammatory agent (NSAID) with antipyretic and analgesic actions.</p>Formule :C14H10Cl2NNaO2Degré de pureté :98.21% - 99.73%Couleur et forme :White Or Off-White PowderMasse moléculaire :318.13Homosalate
CAS :Homosalate is an organic UV filter, an ester of salicylic acid and 3,3,5-trimethylcyclohexanol.Formule :C16H22O3Degré de pureté :99.48%Couleur et forme :Physical Description Viscous Or Light Yellow To Slightly Tan Liquid Or Oil (Ntp 1992)Masse moléculaire :262.34Diminazene Aceturate
CAS :Diminazene is a trypanocidal agent.Formule :C22H29N9O6Degré de pureté :96.86% - 99.58%Couleur et forme :SolidMasse moléculaire :515.52Adenosine 5'-monophosphate monohydrate
CAS :<p>Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.</p>Formule :C10H14N5O7P·H2ODegré de pureté :97.68% - 98.49%Couleur et forme :White PowderMasse moléculaire :365.24ZX-29
CAS :ZX-29: Strong ALK inhibitor; IC50 - ALK 2.1 nM, L1196M 1.3 nM, G1202R 3.9 nM; triggers autophagy; anti-cancer.Formule :C23H28ClN7O3SDegré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :518.03Ref: TM-T13416
1mg92,00€5mg230,00€10mg364,00€25mg620,00€50mg848,00€100mg1.121,00€200mg1.510,00€1mL*10mM (DMSO)264,00€Dofequidar fumarate
CAS :<p>Dofequidar fumarate (MS-209)(MS-209 fumarate), a quinoline-based compound administered orally, is known for counteracting multidrug resistance (MDR) through the</p>Formule :C34H35N3O7Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :597.66Ref: TM-T11071
1mg39,00€2mg50,00€5mg85,00€10mg125,00€25mg245,00€50mg472,00€100mg687,00€500mg1.444,00€CXCR7 antagonist-1
CAS :CXCR7 antagonist-1 is a specific antagonist of the binding of the SDF-1 chemokine or I-TAC to the chemokine receptor CXCR7.Formule :C21H19FN6ODegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :390.41Zidebactam
CAS :Zidebactam (WCK-5107) is an effective β-lactamase inhibitor. Zidebactam also is a penicillin-binding protein2 inhibitor (IC50: 0.26 μg/mL).Formule :C13H21N5O7SDegré de pureté :96.85% - 99.69%Couleur et forme :SolidMasse moléculaire :391.4AZ7550 hydrochloride
CAS :AZ7550 hydrochloride (AZ7550 hydrochloride ), an active metabolite of AZD9291, inhibits the activity of IGF1R (IC50: 1.6 μM).Formule :C27H32ClN7O2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :522.04Caulophyllogenin
CAS :Caulophyllogenin, from Kalopanax pictus, is a PPARγ agonist with anti-inflammatory properties, targeting diabetes and obesity.Formule :C30H48O5Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :488.7CCX140
CAS :CCX140 (CCX140-B) (CCX140-B) is an antagonist of CCR2.Formule :C20H13ClF3N5O3SDegré de pureté :99.66% - 99.95%Couleur et forme :SolidMasse moléculaire :495.86MS31 trihydrochloride (2366264-12-0 free base)
MS31 trihydrochloride (2366264-12-0 free base) is a potent, highly affinity and selective fragment-like methyllysine reader protein spindlin 1 (SPIN1) inhibitorFormule :C20H30Cl3N3O2Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :450.83Ref: TM-T12111L
1mg195,00€5mg390,00€10mg572,00€25mg914,00€50mg1.216,00€100mg1.673,00€1mL*10mM (DMSO)399,00€Onvatilimab
CAS :<p>Onvatilimab (JNJ-61610588) is a human IgG1 κ monoclonal antibody with antitumor effects for advanced head and neck cancers.</p>Degré de pureté :98.11% (SEC-HPLC) - > 95%Couleur et forme :LiquidMasse moléculaire :144.52 kDaPenicillamine
CAS :Penicillamine (Artamine), possessing antineoplastic properties, induces apoptosis by a p53-mediated mechanism and inhibits angiogenesis by chelating with copperFormule :C5H11NO2SDegré de pureté :99.69% - 99.8%Couleur et forme :Fine White Or Practically White Crystalline Powder SolidMasse moléculaire :149.214-Nonylphenol polyethoxylate
CAS :4-Nonylphenol polyethoxylate (Nonoxinol-9) is a typical surfactant used as a vaginal spermicide. Spermicides are locally acting non-hormonal contraceptives.Formule :(C2H4O)nC15H24ODegré de pureté :98%Couleur et forme :Compounds With N20 Are Pale-Yellow To Off-White Pastes Or Waxes Liquid LiquidMasse moléculaire :514.69AZD7624
CAS :AZD7624 is an p38 inhibitor. It has potent anti-inflammatory activity.Formule :C27H30FN5O3Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :491.56Ref: TM-T14381
1mg73,00€5mg160,00€10mg250,00€25mg455,00€50mg682,00€100mg1.017,00€1mL*10mM (DMSO)170,00€Captopril
CAS :Captopril (SA333) is a potent and specific inhibitor of peptidyl-dipeptidase A.Formule :C9H15NO3SDegré de pureté :98.34% - 99.85%Couleur et forme :White To Off-White Crystalline Powder SolidMasse moléculaire :217.29DNA2 inhibitor C5
CAS :DNA2 inhibitor C5 is a specific cancer sensitizer with an IC50 of 20 μM, targeting multiple DNA2 activities.Formule :C10H6N2O5Degré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :234.16Ref: TM-T15146
1mg60,00€2mg85,00€5mg119,00€10mg188,00€25mg432,00€50mg638,00€100mg908,00€500mg1.825,00€1mL*10mM (DMSO)118,00€Bronopol
CAS :Bronopol (BNPD): Low-toxicity antimicrobial, highly effective against Gram-negative bacteria.Formule :C3H6BrNO4Degré de pureté :98.96% - 99.85%Couleur et forme :White Crystalline PowderMasse moléculaire :199.992-Chlorophenothiazine
CAS :2-Chlorophenothiazine is used as the intermediate of Chlorpromazine hydrochloride.Formule :C12H8ClNSDegré de pureté :98.18%Couleur et forme :Gray PowderMasse moléculaire :233.72Bufexamac
CAS :Bufexamac (Bufexamic acid) is a COX inhibitor for IFN-α release with anti-inflammatory, analgesic, and antipyretic action.Formule :C12H17NO3Degré de pureté :99.73%Couleur et forme :Acicular CrystalMasse moléculaire :223.27Amatuximab
CAS :Amatuximab is a chimeric humanized IgG1/k antibody targeting MSLN with antitumor effects for solid tumors.Degré de pureté :SDS-PAGE:95.2%;SEC-HPLC:98.4%Couleur et forme :LiquidMasse moléculaire :144.31 kDaBRD4 Inhibitor-10
CAS :<p>BRD4 Inhibitor-10 is an inhibitor of BRD4-BD1 (IC50: 8 nM).</p>Formule :C25H27N5O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :429.51Aminoguanidine hydrochloride
CAS :Aminoguanidine hydrochloride (Hydrazinecarboximidamide) is a diamine oxidase and NO synthase inhibitor, used in the treatment of diabetic nephropathy.Formule :CH6N4·HClDegré de pureté :99.80%Couleur et forme :White To Off-White SolidMasse moléculaire :110.55Hydroxy-PEG4-(CH2)2-Boc
CAS :Hydroxy-PEG4-(CH2)2-Boc, an uncleavable ADC linker from patent WO2004008101A2, is used in ADC synthesis.Formule :C15H30O7Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :322.39ATN-224
CAS :ATN-224, oral SOD1 inhibitor, hinders endothelial cell activity; dose-dependent with 17.5 nM IC50.Formule :C10H28MoN2O2S4Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :432.564-Hydroxynonenal
CAS :4-Hydroxynonenal (4-HNE) (4-HNE) is an oxidative/nitrosative stress biomarker. It is a substrate and an inhibitor of acetaldehyde dehydrogenase 2 (ALDH2).Formule :C9H16O2Degré de pureté :95.12% - 98%Couleur et forme :Clear Colorless LiquidMasse moléculaire :156.22Viridicatol
CAS :Viridicatol, with potent antibacterial activity against Staphylococcus aureus(MIC: 15.6 μg/mL), is isolated from the fermentation of an endophytic fungusFormule :C15H11NO3Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :253.25Ref: TM-T13305
1mg85,00€5mg170,00€10mg274,00€25mg467,00€50mg655,00€100mg929,00€500mg1.853,00€1mL*10mM (DMSO)207,00€Clorgyline hydrochloride
CAS :<p>Clorgyline hydrochloride (Clorgiline hydrochloride), a white powder, is served as monoamine oxidase inhibitor.</p>Formule :C13H15Cl2NO·HClDegré de pureté :99.8% - 99.82%Couleur et forme :SolidMasse moléculaire :308.63Niclosamide olamine
CAS :<p>Niclosamide olamine (Niclosamide Ethanolamine salt) is an Repellent, Insect Attractant and Chemosterilant.</p>Formule :C15H15Cl2N3O5Degré de pureté :99.89%Couleur et forme :Bright Yellow Crystalline Physical Description Yellow Solid Insoluble In Water (Ntp 1992)Masse moléculaire :388.20D-Mannitol
CAS :D-Mannitol (Mannitol) is a diuretic and renal diagnostic aid related to sorbitol.Formule :C6H14O6Degré de pureté :99.66% - 99.68%Couleur et forme :Orthorhombic Needles From Alc (Ntp 1992)Masse moléculaire :182.17Cyclandelate
CAS :Cyclandelate (BS 572), a direct-acting smooth muscle relaxant, is used to dilate blood vessels.Formule :C17H24O3Degré de pureté :97.01% - 97.03%Couleur et forme :Crystals SolidMasse moléculaire :276.37

