Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.795 produits)
- Apoptose(6.256 produits)
- Cycle cellulaire/point de contrôle(4.836 produits)
- Chromatine/Épigénétique(2.591 produits)
- Signalisation du cytosquelette(1.534 produits)
- Altération de l'ADN/réparation de l'ADN(2.880 produits)
- Endocrinologie/Hormones(3.748 produits)
- Enzyme(3.670 produits)
- GPCR/G-Protéine(8.981 produits)
- Immunologie et Inflammation(3.789 produits)
- Virus de la grippe(299 produits)
- Signalisation JAK/STAT(415 produits)
- Signalisation MAPK(1.250 produits)
- Transporteur membranaire/Canal ionique(3.148 produits)
- Métabolisme(10.143 produits)
- Microbiologie/Virologie(7.591 produits)
- Neuroscience(10.343 produits)
- Autres inhibiteurs(35.823 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.420 produits)
- Protéases/Protéasome(1.680 produits)
- Cellules souche et Dérivés(748 produits)
- Tyrosine Kinase/Adaptateurs(1.958 produits)
- Ubiquitination(1.720 produits)
Affichez 16 plus de sous-catégories
66564 produits trouvés pour "Inhibiteurs"
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Edoxaban Tosylate Monohydrate
CAS :Edoxaban(DU-176) is an oral factor Xa (FXa) inhibitor in clinical development for stroke prevention.Formule :C31H40ClN7O8S2Degré de pureté :99.86% - 99.91%Couleur et forme :SolidMasse moléculaire :738.27Tucidinostat
CAS :Tucidinostat is an oral HDAC1/2/3/10 inhibitor (IC50: 67-160 nM), weaker on HDAC8/11, inactive on HDAC4/5/6/7/9.Formule :C22H19FN4O2Degré de pureté :97.01% - 99.95%Couleur et forme :SolidMasse moléculaire :390.41Ref: TM-T4481
5mg60,00€10mg95,00€25mg159,00€50mg250,00€100mg399,00€200mg558,00€500mg832,00€1mL*10mM (DMSO)60,00€PD153035
CAS :PD153035 (NSC-669364) hydrochloride is an effective and selective inhibitor of EGFR (Ki/IC50: 5.2/29 pM, in cell-free assays); little inhibitory against FGFR,Formule :C16H14BrN3O2Degré de pureté :98.47% - 99.29%Couleur et forme :SolidMasse moléculaire :360.21Hypotaurine
CAS :Hypotaurine (2-Aminoethanesulfinic acid), functioning as an intermediate in the biosynthesis of taurine from cysteine within astrocytes, acts as an endogenousFormule :C2H7NO2SDegré de pureté :98% - ≥98%Couleur et forme :WhiteMasse moléculaire :109.15MG-101
CAS :MG-101 (Calpain inhibitor I) is a cell-permeable and potent inhibitor of cysteine proteases including calpains and lysosomal cathepsins.Formule :C20H37N3O4Degré de pureté :98% - ≥98%Couleur et forme :SolidMasse moléculaire :383.53CGGRGD acetate(1260223-44-6 free base)
RGD-based CGGRGD acetate with N-terminal cysteine; synthesized via solid-phase, modified PCL fiber with CBT for ammoniation.Formule :C21H37N9O11SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :623.65Acetosyringone
CAS :Acetosyringone (AS), a phenol from wounded plants, has analgesic, antipyretic, and anti-inflammatory properties.Formule :C10H12O4Degré de pureté :99.39% - 99.92%Couleur et forme :Light Brown PowderMasse moléculaire :196.2DMOG
CAS :DMOG (Dimethyloxalylglycine), an antagonist of the α-ketoglutarate cofactor, is an inhibitor for HIF prolyl hydroxylase.
Formule :C6H9NO5Degré de pureté :80.23% - 99.98%Couleur et forme :SolidMasse moléculaire :175.143-Methyltoxoflavin
CAS :3-Methyltoxoflavin (3-methyl toxoflavin) is an effective inhibitor of protein disulfide isomerase (PDI) and its IC50 value is 170 nM.Formule :C8H9N5O2Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :207.19Dehydrocostuslactone
CAS :Dehydrocostuslactone, from Aucklandia, offers anti-inflammatory, anticancer, and more health benefits.Formule :C15H18O2Degré de pureté :99.46% - 99.8%Couleur et forme :White PowderMasse moléculaire :230.3Ref: TM-TN6718
1mg56,00€5mg104,00€10mg147,00€25mg260,00€50mg391,00€100mg587,00€200mg823,00€1mL*10mM (DMSO)90,00€AZD0156
CAS :AZD0156 , an effective and specific inhibitors of ATM kinase, is potential antineoplastic activities and chemo-/radio-sensitizing.
Formule :C26H31N5O3Degré de pureté :99.13% - 99.87%Couleur et forme :SolidMasse moléculaire :461.56Tetrahydrocurcumin
CAS :Tetrahydrocurcumin (HZIV 81-2), a major metabolite of curcumin, has strong antioxidant and cardioprotective properties.Formule :C21H24O6Degré de pureté :97.81% - 98.82%Couleur et forme :Solid PowderMasse moléculaire :372.41Stearic acid
CAS :Stearic acid reduces tumor load, cuts visceral fat, gels foods/pharma, boosts insulin signaling, and ups milk yield without weight impact.Formule :C18H36O2Degré de pureté :99.40% - 99.81%Couleur et forme :White Solid LeafletsMasse moléculaire :284.482-Hydroxy-2-methylbutanoic acid
CAS :2-Hydroxy-2-methylbutyric acid is an unusual metabolite found in the urine of patients with 2-hydroxyglutaric aciduria and maple syrup urine disease.Formule :C5H10O3Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :118.132'-FUCOSYLLACTOSE
CAS :2'-FUCOSYLLACTOSE (2'-Fucosyl-D-lactose) is a fucose-containing oligosaccharide.Formule :C18H32O15Degré de pureté :98.31% - 99.96%Couleur et forme :SolidMasse moléculaire :488.44Aticaprant
CAS :Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.Formule :C26H27FN2O2Degré de pureté :99.9% - 99.97%Couleur et forme :SolidMasse moléculaire :418.5Ref: TM-TQ0082
1mg40,00€2mg52,00€5mg88,00€10mg126,00€25mg259,00€50mg406,00€100mg607,00€1mL*10mM (DMSO)87,00€kauran-16,17-diol
CAS :Kauran-16,17-diol, a natural diterpenoid product, exhibits anti-tumoral and apoptosis-inducing activities by inhibiting NO production in LPS-induced RAW 264.7
Formule :C20H34O2Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :306.48Limonin
CAS :Limonin (Citrolimonin) is a triterpenoid enriched in citrus fruits, which has antivirus and antitumor ability.Formule :C26H30O8Degré de pureté :99.65% - 99.66%Couleur et forme :White To Slightly Off White PowderMasse moléculaire :470.51(Z)-LFM-A13
CAS :(Z)-LFM-A13(IC50=2.5 μM), a specific Bruton's tyrosine kinase (BTK), is more than 100-fold specificity than other protein kinases, such as JAK1, JAK2, HCK, EGFR, and IRK.Formule :C11H8Br2N2O2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :360Guanosine 5'-triphosphate trisodium salt
CAS :5'-GTP trisodium salt activates G proteins, regulates cell proliferation/apoptosis, and aids DNA/RNA biosynthesis.Formule :C10H13N5Na3O14P3Degré de pureté :98.74% - 99.45%Couleur et forme :White PowderMasse moléculaire :589.13Adenosine monophosphate
CAS :AMP is a purine nucleotide, vital in cell signaling and energy regulation, and inhibits EC 3.1.3.11 and 3.1.3.1, also an A1 receptor agonist.Formule :C10H14N5O7PDegré de pureté :99.59% - 99.84%Couleur et forme :Crystals From Water + Acetone SolidMasse moléculaire :347.22Danofloxacin
CAS :Danofloxacin (Danofloxacin free base) is a fluoroquinolone antibiotic used in veterinary medicine.Formule :C19H20FN3O3Degré de pureté :99.77% - 99.8%Couleur et forme :SolidMasse moléculaire :357.38N-Hydroxypipecolic acid
CAS :N-Hydroxypipecolic acid (NHP) is a plant metabolite and a systemic acquired resistance (SAR) regulator.Formule :C6H11NO3Degré de pureté :98.23% - ≥95%Couleur et forme :SolidMasse moléculaire :145.16Ref: TM-T19458
2mg55,00€5mg88,00€10mg120,00€25mg178,00€50mg260,00€100mg334,00€200mg500,00€1mL*10mM (DMSO)87,00€DPCPX
CAS :DPCPX (PD 116948) is an A1 adenosine receptor antagonistFormule :C16H24N4O2Degré de pureté :99.23% - 99.93%Couleur et forme :White SolidMasse moléculaire :304.39Mezlocillin Sodium
CAS :Mezlocillin Sodium (Baycipen) is a penicillin beta-lactam antibiotic used in the treatment of bacterial infections caused by susceptible, usually gram-positiveFormule :C21H25N5O8S2·NaDegré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :561.56IOX2
CAS :IOX2 is a selective HIF PHD inhibitor, active in cells with 21 nM IC50 for PHD2/ELGN-1, not inhibiting FIH at 20uM.Formule :C19H16N2O5Degré de pureté :98% - 99.59%Couleur et forme :SolidMasse moléculaire :352.34DR2313
CAS :DR2313 is a competitive inhibitor of poly(ADP-ribose) polymerase (IC50: 0.20 and 0.24 μM for PARP-1 and PARP-2 respectively). It also has neuroprotective.Formule :C8H10N2OSDegré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :182.24Dolutegravir
CAS :Dolutegravir (GSK1349572), HIV integrase inhibitor with IC50 of 2.7 nM, partly effective against some raltegravir-resistant HIV strains.Formule :C20H19F2N3O5Degré de pureté :98.97% - 99.75%Couleur et forme :White To Pale Yellow SolidMasse moléculaire :419.38Ref: TM-T6198
1mg34,00€5mg71,00€10mg105,00€25mg168,00€50mg222,00€100mg295,00€200mg432,00€1mL*10mM (DMSO)65,00€Mirdametinib
CAS :Mirdametinib (PD325901) is an MEK inhibitor (IC50=0.33 nM) with selective, non-ATP-competitive, and oral activity.Formule :C16H14F3IN2O4Degré de pureté :99.11% - 99.63%Couleur et forme :White PowderMasse moléculaire :482.19Ref: TM-T6189
1g898,00€5mg51,00€10mg74,00€25mg127,00€50mg175,00€100mg273,00€200mg406,00€500mg662,00€1mL*10mM (DMSO)55,00€WZ-3146
CAS :WZ3146: EGFR(L858R/E746_A750) inhibitor, IC50=2 nM, selective, doesn't block ERBB2(T798I).Formule :C24H25ClN6O2Degré de pureté :97.15%Couleur et forme :SolidMasse moléculaire :464.95Ref: TM-T6733
1mg50,00€2mg71,00€5mg92,00€10mg170,00€25mg301,00€50mg484,00€100mg692,00€1mL*10mM (DMSO)101,00€Rhamnocitrin
CAS :Rhamnocitrin can enhance the immune function, improve the formation of spleen cells of mice serum hemolysin of chicken red blood cell immune.Formule :C16H12O6Degré de pureté :98.33% - 99.27%Couleur et forme :SolidMasse moléculaire :300.26Gap19
CAS :Gap19 is a peptide that corresponds to a sequence on the cytoplasmic loop (CL) of Cx43.Formule :C55H96N14O13Degré de pureté :97.67%Couleur et forme :SolidMasse moléculaire :1161.44Clitorin
CAS :Clitorin has free radical scavenging property. It shows significant interactions with CD38, it may have anti-hyperglycemic potential.Formule :C33H40O19Degré de pureté :99.55% - 99.83%Couleur et forme :SolidMasse moléculaire :740.66Histamine dihydrochloride
CAS :Ceplene (Histamine dihydrochloride) is a gastric stimulant, bronchial constrictor, vasodilator, and neurotransmitter.Formule :C5H9N3·2HClDegré de pureté :97.72% - >99.99%Couleur et forme :White PowderMasse moléculaire :184.07Pomolic acid
CAS :Pomolic acid has anti-cancer, anti-inflammatory and apoptotic activities, it can induce apoptosis in SK-OV-3 cells, which is mediated by the mitochondrial-Formule :C30H48O4Degré de pureté :96.84% - 99.79%Couleur et forme :SolidMasse moléculaire :472.7Amcasertib
CAS :Amcasertib (BBI503) is an orally administered investigational agent designed to inhibit cancer stem cell pathways via targeting stemness kinases.
Formule :C31H33N5O2SDegré de pureté :97.56% - >99.99%Couleur et forme :SolidMasse moléculaire :539.69Rhein 8-Glucoside
CAS :Rhein 8-Glucoside (Rhein-8-glucoside) has low laxative activity.Formule :C21H18O11Degré de pureté :96.11% - 99.71%Couleur et forme :SolidMasse moléculaire :446.36L-Asparaginase
CAS :L-Asparaginase, an enzyme for acute lymphoblastic leukemia treatment, is administered via injection.Formule :NADegré de pureté :97%Couleur et forme :SolidMasse moléculaire :N/AReactive Blue 4
CAS :Reactive Blue 4: An anthraquinone dye; phytotoxic, cytotoxic, genotoxic. Used as a colorimetric sensor for various analytes in water.Formule :C23H14Cl2N6O8S2Degré de pureté :99.701%Couleur et forme :SolidMasse moléculaire :637.43γ-Cyclodextrin
CAS :γ-Cyclodextrin (Ringdex C) is a cycloamylose composed of eight alpha-(1->4) linked D-glucopyranose units found in some foods.Formule :C48H80O40Degré de pureté :98.56%Couleur et forme :White Solid CrystallineMasse moléculaire :1297.12WSB1 Degrader 1
CAS :WSB1 Degrader 1 is a potent, orally active degrader of WD repeat and SOCS box-containing 1, exhibiting anti-cancer metastatic effects.Formule :C21H22N2O2Degré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :334.41IU1-248
CAS :IU1-248 is a derivative of IU1. IU1-248 is a potent and selective USP14 inhibitor with an IC50 of 0.83 μM[1].Formule :C20H23N3O2Degré de pureté :99.3%Couleur et forme :SolidMasse moléculaire :337.42Ref: TM-T9375
1mg50,00€5mg97,00€10mg160,00€25mg319,00€50mg449,00€100mg640,00€200mg893,00€1mL*10mM (DMSO)107,00€LL-37, Human acetate(154947-66-7 free base)
LL-37, Human acetate is a 37-residue, amphipathic, cathelicidin-derived antimicrobial peptide, which exhibits a broad spectrum of antimicrobial activity.Formule :C207H344N60O55Degré de pureté :96.60% - 99.72%Couleur et forme :SolidMasse moléculaire :4553.31Sphingomyelin
CAS :Sphingomyelin is a natural sphingolipid that existed in animal cell membranes. It implicates the regulation of transmembrane signaling.Formule :C41H83N2O6PDegré de pureté :98% - 98%Couleur et forme :SolidMasse moléculaire :731.097Phillyrin
CAS :Phillyrin (Forsythin) is a novel AMPK activator, has anti-obesity effects in nutritive obesity mice, it can prevent lipid accumulation in HepG2 cells.Formule :C27H34O11Degré de pureté :98.28% - 99.71%Couleur et forme :SolidMasse moléculaire :534.55BI-6015
CAS :BI 6015 is an antagonist of HNF4α. HNF4α is a nuclear receptor that regulates gene expression in the intestine cells, liver cells, and pancreas-β cells.
Formule :C15H13N3O4SDegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :331.35LPYFD-NH2 acetate
LPYFD-NH2 acetate shows some inhibitory effect on the aggregation of Abeta(1-42).Formule :C35H48N6O10Degré de pureté :96.51%Couleur et forme :SolidMasse moléculaire :712.79Ref: TM-T22932L
1mg66,00€5mg130,00€10mg187,00€25mg309,00€50mg439,00€100mg590,00€200mg793,00€1mL*10mM (DMSO)188,00€DDP-38003 trihydrochloride
DDP-38003 trihydrochloride is a novel, orally available histone lysine-specific demethylase 1A (KDM1A/LSD1) inhibitor with an IC50 of 84 nM.Formule :C21H29Cl3N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :459.84BCI hydrochloride
CAS :BCI hydrochloride ((E)-BCI hydrochloride) is a DUSP6 inhibitor that inhibits RANKL-mediated osteoclastogenesis and attenuates oophorectomy-induced bone loss.Formule :C22H24ClNODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :353.89(2S,3R,4S,5R)-2-Amino-3,4,5,6-tetrahydroxyhexanal hydrochloride
CAS :(2S,3R,4S,5R)-2-Amino-3,4,5,6-tetrahydroxyhexanal hydrochloride (D-Mannosamine hydrochloride) is a compound used in the development of mannosylated liposomes.Formule :C6H14ClNO5Degré de pureté :99.13% - 99.67%Couleur et forme :Powder To Fine Crystals White/ColorlessMasse moléculaire :215.63
