
Angiogenesi
Gli inibitori dell'angiogenesi sono composti che interferiscono con la formazione di nuovi vasi sanguigni, un processo cruciale nella crescita e metastasi del cancro. Inibendo l'angiogenesi, questi composti possono limitare l'apporto di sangue ai tumori, rallentandone o arrestando la crescita. Gli inibitori dell'angiogenesi sono fondamentali nella ricerca sul cancro e nello sviluppo terapeutico, offrendo approfondimenti sui meccanismi di progressione tumorale e potenziali trattamenti per il cancro e altre malattie legate all'angiogenesi. Presso CymitQuimica, offriamo un'ampia gamma di inibitori dell'angiogenesi di alta qualità per supportare le tue ricerche in oncologia e biologia vascolare.
Sottocategorie di "Angiogenesi"
- BTK(166 prodotti)
- Bcr-Abl(117 prodotti)
- EGFR(553 prodotti)
- FAK(72 prodotti)
- FLT(88 prodotti)
- Recettore del fattore di crescita dei fibroblasti (FGFR)(176 prodotti)
- JAK(243 prodotti)
- PDGFR(127 prodotti)
- RAAS(86 prodotti)
- Src(82 prodotti)
- Syk(37 prodotti)
- Trombina(51 prodotti)
- VDA(2 prodotti)
- VEGFR(236 prodotti)
Mostrare 6 più sottocategorie
Trovati 2277 prodotti di "Angiogenesi"
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Tofacitinib Citrate
CAS:Tofacitinib Citrate (CP-690550 citrate) is a a potent, cell-permeable inhibitor of JAK1/2/3 (IC50s: 1/20/112 nM).Formula:C22H28N6O8Purezza:99.19% - 99.75%Colore e forma:SolidPeso molecolare:504.49LDN193189
CAS:LDN193189 blocks BMP signaling by inhibiting ALK2/3; IC50: ALK1/2/3/6 = 0.8/0.8/5.3/16.7 nM.Formula:C25H22N6Purezza:98% - 99.86%Colore e forma:SolidPeso molecolare:406.48Vodobatinib
CAS:Vodobatinib (K-0706) is a novel 3rd generation (3G) TKI effective against wild-type and mutated BCR-ABL1 with limited off-target activity.Formula:C27H20ClN3O2Purezza:99.06% - 99.55%Colore e forma:SolidPeso molecolare:453.92Ref: TM-T8882
1mg34,00€5mg74,00€10mg110,00€25mg200,00€50mg323,00€100mg500,00€500mg1.209,00€1mL*10mM (DMSO)82,00€Upadacitinib
CAS:Upadacitinib (ABT-494), a selective JAK1 inhibitor, is researched for autoimmune diseases; IC50: 43 nM.Formula:C17H19F3N6OPurezza:98.96% - 99.94%Colore e forma:SolidPeso molecolare:380.37Ref: TM-T7503
2mg55,00€5mg89,00€10mg116,00€25mg198,00€50mg276,00€100mg389,00€200mg595,00€1mL*10mM (DMSO)44,00€Nilotinib monohydrochloride monohydrate
CAS:Nilotinib monohydrochloride monohydrate (Nilotinib (monohydrochloride monohydrate)) is significantly potent BCR-ABL against, is a second generation tyrosineFormula:C28H22F3N7O·HCl·H2OPurezza:99.93%Colore e forma:SolidPeso molecolare:583.99Belizatinib
CAS:Belizatinib (TSR-011) is an effective, oral and dual inhibitor of ALK (IC50: 0.7 nM, wild-type recombinant ALK) and TRKA, TRKB, and TRKC.Formula:C33H44FN5O3Purezza:99.33% - 99.44%Colore e forma:SolidPeso molecolare:577.73Ref: TM-T4257
1mg40,00€2mg54,00€5mg93,00€10mg133,00€25mg259,00€50mg358,00€100mg500,00€1mL*10mM (DMSO)105,00€KHS101 hydrochloride
CAS:KHS101 is a TACC3 inhibitor and can selectively induce a neuronal differentiation phenotype.Formula:C18H22ClN5SPurezza:99.6%Colore e forma:SolidPeso molecolare:375.92Ref: TM-T5170
2mg34,00€5mg52,00€10mg80,00€25mg147,00€50mg239,00€100mg350,00€200mg497,00€1mL*10mM (DMSO)58,00€Pyridone 6
CAS:Pyridone 6, a selective JAK1/2/3 and Tyk2 inhibitor with IC50s: JAK1=15 nM, JAK2=1 nM, JAK3 (Ki=5 nM), Tyk2=1 nM; weakly binds other kinases (130 nM-10 μM).Formula:C18H16FN3OPurezza:97.1% - 98.74%Colore e forma:SolidPeso molecolare:309.34Ref: TM-T3080
1mg50,00€2mg71,00€5mg105,00€10mg173,00€25mg358,00€50mg587,00€100mg888,00€200mg1.198,00€1mL*10mM (DMSO)110,00€ML347
CAS:ML347 (LDN 193719)(DN193719) is a highly specific ALK1/2 inhibitor ( IC50: 46/32 nM), and the selectivity for ALK2 is >300-fold than ALK3.Formula:C22H16N4OPurezza:99.30% - ≥95%Colore e forma:SolidPeso molecolare:352.39PHA-680632
CAS:PHA-680632 is potent inhibitor of Aurora A, Aurora B and Aurora C with IC50 of 27 nM, 135 nM and 120 nM, respectively.Formula:C28H35N7O2Purezza:98.2%Colore e forma:SolidPeso molecolare:501.62Tolebrutinib
CAS:Tolebrutinib is an oral, selective BTK inhibitor, effective for MS research, with brain penetration and IC50s of 0.4/0.7 nM in cells.Formula:C26H25N5O3Purezza:98.4% - 98.82%Colore e forma:SolidPeso molecolare:455.51Ref: TM-T9125
2mg40,00€5mg71,00€10mg105,00€25mg177,00€50mg264,00€100mg434,00€200mg622,00€1mL*10mM (DMSO)80,00€Src Inhibitor 1
CAS:Src Inhibitor 1 (Src Kinase Inhibitor 1) is a potent and selective dual site Src tyrosine kinase inhibitor.Formula:C22H19N3O3Purezza:99.68% - >99.99%Colore e forma:SolidPeso molecolare:373.4Ref: TM-T3593
2mg38,00€5mg56,00€10mg94,00€25mg172,00€50mg268,00€100mg429,00€200mg615,00€1mL*10mM (DMSO)Prezzo su richiestaG5-7
CAS:G5-7 is an oral JAK2 inhibitor targeting EGFR/STAT3 phosphorylation with potential for glioma research.Formula:C22H19F2NO3Purezza:97.3%Colore e forma:SolidPeso molecolare:383.39Ref: TM-T8742
1mg35,00€5mg71,00€10mg96,00€25mg172,00€50mg248,00€100mg348,00€200mg470,00€1mL*10mM (DMSO)78,00€K02288
CAS:K 02288 is a novel small molecule inhibitor of ALK1/2/3/6.Formula:C20H20N2O4Purezza:98% - 99.83%Colore e forma:SolidPeso molecolare:352.38Alectinib hydrochloride
CAS:Alectinib hydrochloride (RO5424802 Hydrochloride) is a selective, and orally available inhibitor of ALK( IC50 : 1.9 nM)Formula:C30H35ClN4O2Purezza:99.74% - 99.96%Colore e forma:SolidPeso molecolare:519.08Gilteritinib
CAS:Gilteritinib (ASP2215) is a potent inhibitor at the FMS-related tyrosine kinase 3 (FLT3) and AXL tyrosine kinase receptors (IC50 = 0.29 nM and <1 nM,Formula:C29H44N8O3Purezza:97.75% - 99.90%Colore e forma:SolidPeso molecolare:552.71Ref: TM-T4409
1g1.288,00€1mg38,00€2mg52,00€5mg85,00€10mg114,00€25mg177,00€50mg261,00€100mg411,00€500mg954,00€GNF-2
CAS:GNF-2 is a highly selective non-ATP competitive inhibitor of Bcr-Abl.Formula:C18H13F3N4O2Purezza:98.17% - ≥95%Colore e forma:SolidPeso molecolare:374.32PF-04929113 Mesylate
CAS:PF-04929113 Mesylate (SNX-5422 Mesylate), a prodrug of SNX-2112, is an orally available Hsp90 inhibitor (Kd: 41 nM) and also induces Her-2 degradation (IC50: 37Formula:C26H34F3N5O7SPurezza:99% - 99.46%Colore e forma:SolidPeso molecolare:617.63Ref: TM-T4342
1mg73,00€2mg95,00€5mg150,00€10mg273,00€25mg396,00€50mg583,00€100mg832,00€500mg1.684,00€1mL*10mM (DMSO)220,00€Branebrutinib
CAS:Branebrutinib (BMS986195) is a potent, covalent inhibitor of Bruton's tyrosine kinase (BTK), >5,000-fold selective over all kinases outside of the Tec family.Formula:C20H23FN4O2Purezza:95.86% - 99.31%Colore e forma:SolidPeso molecolare:370.42PT-2385
CAS:PT-2385 is a selective HIF-2α inhibitor (Kd<50 nM).Formula:C17H12F3NO4SPurezza:98.91% - 99.55%Colore e forma:SolidPeso molecolare:383.34Ref: TM-T7848
1mg63,00€2mg93,00€5mg144,00€10mg222,00€25mg379,00€50mg532,00€100mg740,00€200mg982,00€1mL*10mM (DMSO)119,00€
