
Cromatina/Epigenetica
Gli inibitori della cromatina/epigenetica sono composti che modulano la struttura e la funzione della cromatina o interferiscono con le modificazioni epigenetiche, come la metilazione del DNA e la modifica degli istoni. Questi inibitori sono strumenti essenziali per studiare la regolazione dell'espressione genica e il ruolo dell'epigenetica in malattie come il cancro, i disturbi neurologici e le anomalie dello sviluppo. Mirando ai processi epigenetici, questi inibitori possono alterare i modelli di espressione genica e offrire nuove opportunità terapeutiche. Presso CymitQuimica, offriamo un'ampia selezione di inibitori della cromatina/epigenetica di alta qualità per supportare le tue ricerche in biologia molecolare, genetica ed epigenetica.
Sottocategorie di "Cromatina/Epigenetica"
Trovati 2592 prodotti di "Cromatina/Epigenetica"
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GSK360A
CAS:GSK360A is a novel prolyl hydroxylase (PHD) domain-containing enzyme inhibitor.Formula:C17H17FN2O5Purezza:98%Colore e forma:SolidPeso molecolare:348.33CPI-4203
CAS:CPI-4203 is a selective inhibitor of KDM5 demethylases.Formula:C16H14N4OColore e forma:SolidPeso molecolare:278.31Valemetostat tosylate
CAS:Valemetostat tosylate is a dual inhibitor of EZH1/2 and used in the research of relapsed/refractory peripheral T-cell lymphoma.Formula:C33H42ClN3O7SPurezza:98%Colore e forma:SolidPeso molecolare:660.22Givinostat hydrochloride monohydrate
CAS:Givinostat hydrochloride monohydrate (ITF2357) is an HDAC inhibitor.Formula:C24H27N3O4·HCl·H2OPurezza:97.97% - 99.51%Colore e forma:SolidPeso molecolare:475.97IDO1 and HDAC1 Inhibitor
CAS:IDO1 and HDAC1 Inhibitor is a dual IDO1 and HDAC1 inhibitor (IC50s: 69.0 nM and 66.5 nM).Formula:C25H22BrFN8O4Purezza:98%Colore e forma:SolidPeso molecolare:597.4BPTF-IN-1
CAS:BPTF-IN-1 (AU1), a BPTF bromodomain inhibitor with 2.8 μM affinity, shows higher selectivity over BRD4 and possesses antimalarial properties.Formula:C23H23FN6O3Colore e forma:SolidPeso molecolare:450.47KP-302
CAS:KP-302 is a selective PAD inhibitor, reversing physical disability in multiple sclerosis (MS) mice and clearing T-cell infiltration in the brain.
Formula:C20H23N5O2Purezza:99.77%Colore e forma:SolidPeso molecolare:365.43Ref: TM-T88080
1mg60,00€5mg127,00€10mg202,00€25mg416,00€50mg677,00€100mg1.074,00€200mg1.454,00€1mL*10mM (DMSO)140,00€HDAC-IN-49
HDAC-IN-49: potent, broad HDAC inhibitor; IC50s: 10-1880 nM for HDAC1-6; strong anti-leukemic, low toxicity to healthy cells.Formula:C26H27FN4O4Colore e forma:SolidPeso molecolare:478.52PIM-1 Inhibitor 2
CAS:PIM-1 Inhibitor 2 (PIM1-IN-2) is a potent Pim-1 inhibitor with potential anti-cancer activity, used in cancer research.Formula:C17H11ClN4OPurezza:98.81%Colore e forma:SolidPeso molecolare:322.75Sirt1/2-IN-1
CAS:Sirt1/2-IN-1 inhibits SIRT1 (IC50: 1.81 μg/mL) and SIRT2 (2.10 μg/mL), less on SIRT3 (20.5 μg/mL), with anticancer properties.Formula:C22H13ClN2OS2Colore e forma:SolidPeso molecolare:420.93JAK3-IN-1
CAS:JAK3-IN-1 is an orally active, selective and potent JAK3 inhibitor for the study of immune system disorders.Formula:C26H30ClN7O2Colore e forma:SolidPeso molecolare:508.02Arazine
CAS:Arazine, a cell-permeable G protein modulator, is an isoprenylcysteine methyltransferase substrate.Formula:C20H33NO3SPurezza:90%Colore e forma:SolidPeso molecolare:367.55NSC-311068
CAS:NSC-311068: A selective TET1 inhibitor, reducing 5hmC and AML cell viability with high TET1.Formula:C10H6N4O4SColore e forma:SolidPeso molecolare:278.24SHP2/HDAC-IN-1
CAS:SHP2/HDAC-IN-1: dual SHP2/HDAC inhibitor, IC50: 20.4 nM/25.3 nM, boosts antitumor immunity, aids cancer immunotherapy research.Formula:C34H35Cl2N7O3Colore e forma:SolidPeso molecolare:660.59SIRT5 inhibitor 5
CAS:SIRT5 inhibitor 5 is a selective and substrate-competitive SIRT5 inhibitor, which does not occupy the NAD+ binding pocket,cancer and metabolism-related disease.Formula:C21H14ClN3O3SPurezza:99.33%Colore e forma:SolidPeso molecolare:423.87AJH-836
CAS:AJH-836 is a compound that activates Munc13-1 and PKC ε/α, demonstrating a dissociation constant (Kd) of 4.5 nM for PKCα, and facilitates the translocation ofFormula:C22H38O5Purezza:98%Colore e forma:SolidPeso molecolare:382.53SIRT2-IN-9
CAS:SIRT2-IN-9: selective SIRT2 inhibitor; IC50=1.3μM; halts MCF-7 cell growth; for cancer study.Formula:C21H22N6OS2Purezza:97.6%Colore e forma:SolidPeso molecolare:438.57MS453
CAS:MS453 is a potent and selective SETD8 inhibitor with an IC50 value of 804 nM.Formula:C20H27N5O3Colore e forma:SolidPeso molecolare:385.46HDAC-IN-58
CAS:HDAC-IN-58, a selective HDAC6 inhibitor, exhibits potent inhibitory activity with an IC50 of 2.06 nM, rendering it suitable for research into chronicFormula:C16H13ClF2N4O3SPurezza:98%Colore e forma:SolidPeso molecolare:414.81SW155246
CAS:SW155246 is a potent and selective inhibitor of DNMT1 (DNA methyltransferase 1; IC50 of 1.2 μM).Formula:C16H11ClN2O5SPurezza:98.99%Colore e forma:SolidPeso molecolare:378.79
