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Prolil-idrossilasi HIF/HIF

Prolil-idrossilasi HIF/HIF

Il fattore inducibile dall'ipossia (HIF) è un fattore di trascrizione che svolge un ruolo cruciale nelle risposte cellulari ai bassi livelli di ossigeno (ipossia). L'attività di HIF è strettamente regolata dalle prolyl-idrossilasi HIF, che bersagliano HIF per la degradazione in condizioni normossiche. Gli inibitori della prolyl-idrossilasi HIF possono stabilizzare HIF, promuovendo l'espressione di geni coinvolti nell'angiogenesi, eritropoiesi e metabolismo. Questi inibitori sono di grande interesse per il trattamento di condizioni come anemia, malattie ischemiche e cancro. Presso CymitQuimica, offriamo inibitori di HIF/prolyl-idrossilasi HIF per supportare la tua ricerca in biologia dell'ipossia, terapia anticancro e regolazione metabolica.

Trovati 156 prodotti per "Prolil-idrossilasi HIF/HIF".

prodotti per pagina.
  • Chloramphenicol

    CAS:
    Chloramphenicol (Chloromycetin) is a broad-spectrum antibiotic that inhibits the biosynthesis of bacterial proteins. Cost-effective and quality-assured.
    Formula:C11H12Cl2N2O5
    Purezza:99.6% - 99.90%
    Colore e forma:White Solid
    Peso molecolare:323.129
  • Roxadustat

    CAS:
    Roxadustat (FG-4592) is an orally bioavailable, hypoxia-inducible factor prolyl hydroxylase inhibitor (HIF-PHI), with potential anti-anemic activity.
    Formula:C19H16N2O5
    Purezza:99% - 99.88%
    Colore e forma:Yellow Solid
    Peso molecolare:352.3407
  • EHP-101

    CAS:
    EHP-101 is a PPARγ/CB2 dual agonist with anti-inflammatory properties, inhibits fat formation, and combats diet-related obesity.
    Formula:C28H35NO3
    Purezza:98.36%
    Colore e forma:Solid
    Peso molecolare:433.5824
  • Citric acid trilithium salt tetrahydrate

    CAS:
    Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) , the active component of Lithium, is a medicine used in the therapy of
    Formula:C6H13Li3O11
    Purezza:99.88%
    Colore e forma:White Solid
    Peso molecolare:281.984
  • Tilorone dihydrochloride

    CAS:
    Tilorone dihydrochloride is an orally active interferon inducer, and has antineoplastic and anti-inflammatory actions.
    Formula:C25H36Cl2N2O3
    Purezza:98% - 99.86%
    Colore e forma:Orange Solid
    Peso molecolare:483.47
  • Glucosamine

    CAS:
    Glucosamine (Chitosamine) is used as a dietary supplement. Glucosamine has pharmacological effects on osteoarthritis cartilage. High-Quality, Low-Cost!
    Formula:C6H13NO5
    Purezza:99.68% - 99.8%
    Colore e forma:Solid
    Peso molecolare:179.1711
  • Amifostine

    CAS:
    Amifostine (Ethyol) anhydrous is a cytoprotective agent, acts as a free radical scavenging activity.
    Formula:C5H15N2O3PS
    Purezza:99.59% - 99.91%
    Colore e forma:White Solid
    Peso molecolare:214.22
  • Glucosamine hydrochloride

    CAS:
    Glucosamine hydrochloride (Chitosamine hydrochloride) is commonly used as a treatment for osteoarthritis, although its acceptance as a medical therapy varies.
    Formula:C6H13NO5·HCl
    Purezza:99.77% - 99.96%
    Colore e forma:White Solid
    Peso molecolare:215.63
  • Hydroxycitric acid tripotassium hydrate

    CAS:
    Hydroxycitric acid tripotassium hydrate (Potassium citrate monohydrate) effectively inhibits HIF, has antioxidation, anti-inflammation, and anti-tumor effects.
    Formula:C6H7K3O8
    Purezza:99.85%
    Colore e forma:White Solid Crystalline
    Peso molecolare:324.4099
  • Minocycline hydrochloride

    CAS:
    Minocycline HCl: tetracycline antibiotic, treats bacterial infections and acne, may cause acute or chronic hepatitis.
    Formula:C23H28ClN3O7
    Purezza:98.49% - >99.99%
    Colore e forma:Yellow Solid
    Peso molecolare:493.94
  • Deferoxamine Mesylate

    CAS:
    Deferoxamine Mesylate (DFOM) is an iron chelator and iron death inhibitor.
    Formula:C26H52N6O11S
    Purezza:94.68% - 99.94%
    Colore e forma:White Solid
    Peso molecolare:656.79
  • SYP-5

    CAS:
    SYP-5 is a novel inhibitor of HIF-1, suppresses tumor cells invasion and angiogenesis.
    Formula:C18H16O3S
    Purezza:98.31%
    Colore e forma:Solid
    Peso molecolare:312.383
  • Enarodustat

    CAS:
    Enarodustat (JTZ-951) is an orally active factor inhibitor of prolyl hydroxylase (EC50: 0.22 μM) and has the potential for renal anemia treatment.
    Formula:C17H16N4O4
    Purezza:99.73% - 99.75%
    Colore e forma:Solid
    Peso molecolare:340.3333
  • HIF-2α-IN-2

    CAS:
    HIF-2α-IN-2 is a hypoxia-inducible factor (HIF-2α) inhibitor (IC50: 16 nM in scintillation proximity assay).
    Formula:C17H13F2NO4S
    Purezza:99.24%
    Colore e forma:White Solid
    Peso molecolare:365.351
  • (-)-Hydroxycitric acid lactone

    CAS:
    (-)-Hydroxycitric acid lactone (Garcinia lactone) is an anti-obesity agent.(-)-Hydroxycitric acid lactone was a potent inhibitor of ATP citrate lyase, which
    Formula:C6H6O7
    Purezza:99.85% - 99.91%
    Colore e forma:White Solid
    Peso molecolare:190.1076
  • PT2399

    CAS:
    PT2399, an oral HIF-2 inhibitor, blocks HIF-2α/1β dimerization, showing strong in vivo antitumor effects.
    Formula:C17H10F5NO4S
    Purezza:98.8% - 99.45%
    Colore e forma:White Solid
    Peso molecolare:419.323
  • Hydralazine hydrochloride

    CAS:
    Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.
    Formula:C8H9ClN4
    Purezza:99.85% - 99.86%
    Colore e forma:White Solid
    Peso molecolare:196.64
  • Albendazole

    CAS:
    Albendazole (SKF-62979) is used as a drug indicated for the treatment of a variety of worm infestations.
    Formula:C12H15N3O2S
    Purezza:98.76% - 98.89%
    Colore e forma:Colorless Crystals Solid
    Peso molecolare:265.331
  • Oltipraz

    CAS:
    Oltipraz (RP 35972) is a synthetic dithiolethione with potential chemopreventive and anti-angiogenic properties.
    Formula:C8H6N2S3
    Purezza:98.79% - 99.77%
    Colore e forma:Solid
    Peso molecolare:226.34
  • Vadadustat

    CAS:
    Vadadustat is a novel, titratable, oral hypoxia-inducible factor prolyl hydroxylase (HIF-PH) inhibitor in development for the treatment of anemia.
    Formula:C14H11ClN2O4
    Purezza:99.02% - 99.80%
    Colore e forma:Solid
    Peso molecolare:306.701