
Deidrogenasi
Le deidrogenasi sono enzimi coinvolti nelle reazioni di ossidoriduzione delle vie metaboliche, svolgendo un ruolo centrale nella produzione di energia e nella respirazione cellulare. Questi enzimi sono cruciali per processi come il ciclo dell'acido citrico, la glicolisi e l'ossidazione degli acidi grassi. Gli inibitori delle deidrogenasi sono strumenti importanti nello studio delle malattie metaboliche, del cancro e dello stress ossidativo. Presso CymitQuimica, offriamo una selezione completa di inibitori delle deidrogenasi per supportare la tua ricerca in metabolismo, biologia del cancro e biochimica.
Trovati 299 prodotti di "Deidrogenasi"
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Mycophenolic acid
CAS:Mycophenolic acid (Mycophenolate) is an inosine monophosphate dehydrogenase(IMPDH) inhibitor with anti-proliferative activity.Formula:C17H20O6Purezza:98.79% - 99.77%Colore e forma:SolidPeso molecolare:320.34SCD1 inhibitor-4
CAS:<p>SCD1 inhibitor-4 is stearoylCoA desaturase-1 (SCD1) inhibitor. SCD1 inhibitor-4 can be used for the research of diabetes.</p>Formula:C17H16F3N5OPurezza:99.71%Colore e forma:SolidPeso molecolare:363.34CAY10566
CAS:CAY10566 is a potent SCD1 inhibitor, orally bioavailable, with IC50s: HepG2 cells, 7.9nM; mouse, 4.5nM; human, 26nM.Formula:C18H17ClFN5O2Purezza:99.5% - 99.54%Colore e forma:SolidPeso molecolare:389.81CVT-10216
CAS:CVT-10216 inhibits ALDH2 (IC50: 29 nM) and ALDH-1 (IC50: 1.3 μM), reducing alcohol intake and anxiety in rats.Formula:C24H19NO7SPurezza:98.76%Colore e forma:SolidPeso molecolare:465.48KPLH1130
CAS:<p>KPLH1130, a PDK inhibitor, boosts glucose tolerance and reduces inflammation in high-fat diet mice.</p>Formula:C15H13N3O3Purezza:99.07%Colore e forma:SolidPeso molecolare:283.28MF-438
CAS:MF-438 is an effective and orally bioavailable stearoyl-CoA desaturase 1 (SCD1) inhibitor (EC50: 2.3 nM for rSCD1).Formula:C19H18F3N5OSPurezza:98.98% - 99.50%Colore e forma:SolidPeso molecolare:421.44LY 345899
CAS:<p>LY 345899 is a Folate analog and is a methylenetetrahydrofolate dehydrogenase and MTHFD2 inhibitor (IC50: 96 nM and 663 nM, respectively and a Ki: 18 nM for</p>Formula:C20H21N7O7Purezza:99.7%Colore e forma:SolidPeso molecolare:471.42BAY-2402234
CAS:BAY-2402234: a selective DHODH inhibitor targeting myeloid cancers with low-nanomolar potency.Formula:C21H18ClF5N4O4Purezza:98.9%Colore e forma:SolidPeso molecolare:520.84ML390
CAS:<p>ML390 exerts its potent differentiation effect on multiple leukemia models.</p>Formula:C21H21F3N2O3Purezza:99.76%Colore e forma:SolidPeso molecolare:406.4NCT-502
CAS:<p>NCT-502 (N-(4,6-dimethylpyridin-2-yl)-4-[5-(trifluoromethyl)pyridin-2-yl]piperazine-1-carbothioamide) is a human phosphoglycerate dehydrogenase inhibitor,</p>Formula:C18H20F3N5SPurezza:99.60%Colore e forma:SolidPeso molecolare:395.45PTC299
CAS:<p>PTC299 ((4-chlorophenyl) (1S)-6-chloro-1-(4-methoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carboxylate) is an orally active inhibitor of VEGFA mRNA</p>Formula:C25H20Cl2N2O3Purezza:99.72%Colore e forma:SolidPeso molecolare:467.34LDH-IN-1
CAS:LDH-IN-1 is a pyrazole-based human lactate dehydrogenase (LDH) inhibitor(IC50s of 32 and 27 nM for LDHA and LDHB, respectively).Formula:C30H26N4O4S2Purezza:99.6%Colore e forma:SolidPeso molecolare:570.68XEN723
CAS:XEN723 is a potent thiazolylimidazolidinone Stearoyl-CoA Desaturase (SCD1) inhibitor(IC50s of 45 and 524 nM in mouse and HepG2 cell, respectively).Formula:C21H20FN5O2SPurezza:99.5%Colore e forma:SolidPeso molecolare:425.48CBR-5884
CAS:CBR-5884: active PHGDH inhibitor, IC50=33μM, disrupts serine synthesis, selectively targets high-serine cancers.Formula:C14H12N2O4S2Purezza:99.97%Colore e forma:SolidPeso molecolare:336.39DHODH-IN-11
CAS:DHODH-IN-11 is a leflunomide derivative and weak dihydroorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.03.Formula:C15H11N3O2Purezza:98.14%Colore e forma:SolidPeso molecolare:265.27Adrenosterone
CAS:Adrenosterone (11-ketoandrostenedione) is a steroid hormone isolated from the adrenal cortex.Formula:C19H24O3Purezza:98.13% - 98.29%Colore e forma:SolidPeso molecolare:300.39Trilostane
CAS:Trilostane (Win 24540) is a synthetic derivative of androstane with adrenocortical suppressive properties.Formula:C20H27NO3Purezza:99.46% - >99.99%Colore e forma:Tan CrystalsPeso molecolare:329.43IDH-305
CAS:<p>IDH-305: Oral, mutation-specific IDH1 inhibitor, 200x selective for R132 mutants; IC50: 27/28/6.14 nM for R132H/C/WT.</p>Formula:C23H22F4N6O2Purezza:99.68%Colore e forma:SolidPeso molecolare:490.45RS 61443
CAS:<p>RS 61443 (Mycophenolate mofetil) is an immunosuppressant, a non-competitive, selective and reversible inhibitor of inosine monophosphate dehydrogenase (IMPDH)</p>Formula:C23H31NO7Purezza:99.37% - 99.91%Colore e forma:SolidPeso molecolare:433.5Mutant IDH1 inhibitor
CAS:<p>Mutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).</p>Formula:C25H34N6O3Purezza:98.3%Colore e forma:SolidPeso molecolare:466.58
