
Neuroscienza
Gli inibitori in neuroscienze sono composti progettati per modulare l'attività di proteine, enzimi o recettori specifici all'interno del sistema nervoso. Questi inibitori sono cruciali per studiare i meccanismi molecolari alla base della funzione neuronale, della trasmissione sinaptica e delle malattie neurodegenerative. Mirando ai recettori dei neurotrasmettitori, ai canali ionici e alle vie di segnalazione, gli inibitori in neuroscienze aiutano a esplorare la funzione cerebrale e a sviluppare strategie terapeutiche per disturbi neurologici come l'Alzheimer, il Parkinson e l'epilessia. Presso CymitQuimica, offriamo una vasta gamma di inibitori in neuroscienze di alta qualità per supportare la tua ricerca in neurobiologia, neurofarmacologia e scienze cognitive.
Sottocategorie di "Neuroscienza"
- recettore 5-HT(1.025 prodotti)
- ACK(1 prodotti)
- AChR(645 prodotti)
- Citrato liasi ATP(17 prodotti)
- Recettore adrenergico(3.018 prodotti)
- BACE(37 prodotti)
- Beta amiloide(228 prodotti)
- CaMK(73 prodotti)
- COX(600 prodotti)
- Recettore della dopamina(445 prodotti)
- Ricettore GABA(372 prodotti)
- Gamma-secretasi(61 prodotti)
- GluR(265 prodotti)
- GlyT(26 prodotti)
- Recettore dell'istamina(385 prodotti)
- LRRK2(43 prodotti)
- Recettore della melatonina(26 prodotti)
- NMDAR(10 prodotti)
- Recettore OX(41 prodotti)
- Recettore degli oppioidi(327 prodotti)
Mostrare 12 più sottocategorie
Trovati 5530 prodotti di "Neuroscienza"
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SDZ 205-557 hydrochloride
CAS:5-HT3/5-HT4 receptor antagonistFormula:C14H22Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:337.248011-6561
CAS:1,1-Diphenyl-4-(pyrrolidin-1-yl)but-2-yn-1-ol is an anticholinergic agent that has the potential for the research of bronchial asthma [1].Formula:C20H21NOColore e forma:SolidPeso molecolare:291.39LY 206130
CAS:LY 206130 is an antagonist of serotonin 5-HT1A.Formula:C17H24N2O2Colore e forma:SolidPeso molecolare:288.38(RS)-Minesapride
CAS:Minesapride is a serotonin receptor agonist.Formula:C21H31ClN4O5Purezza:98%Colore e forma:SolidPeso molecolare:454.95(R)-VU 6008667
CAS:(R)-VU 6008667 is devoid of M5 NAM activity (IC50>10 μM).Formula:C24H17ClF2N2O2Colore e forma:SolidPeso molecolare:438.85YM 114
CAS:YM 114 is an anatagonist of 5-HT(3) receptor.Formula:C16H18ClN3OPurezza:98%Colore e forma:SolidPeso molecolare:303.79ML 10375
CAS:ML 10375 is an antagonist of 5-HT4 receptor.Formula:C17H25ClN2O3Colore e forma:SolidPeso molecolare:340.85COR627
CAS:COR627 is the GABA receptor positive allosteric modulator.Formula:C20H27NO3SPurezza:98%Colore e forma:SolidPeso molecolare:361.5RGH 1756
CAS:RGH 1756 is an atypical antipsychotic with high affinity to dopamine D(3) receptors that leads to c-Fos induction in a unique pattern.Formula:C26H30N4O2SPurezza:98%Colore e forma:SolidPeso molecolare:462.61Hexocyclium metilsulfate
CAS:Hexocyclium metilsulfate has anti-gastric secretory effects in humans.Formula:C21H36N2O5SPurezza:98%Colore e forma:SolidPeso molecolare:428.59HUHS2002
CAS:HUHS2002 is a free fatty acid derivative that works as a potentiator of GluA1 AMPA receptor responses and α7 ACh receptor responses.Formula:C17H24O3Purezza:98%Colore e forma:SolidPeso molecolare:276.37AZ4800
CAS:AZD4800 is a gamma secretase modulators.Formula:C24H29N5O3Colore e forma:SolidPeso molecolare:435.52NGX-267
CAS:NGX-267, a muscarinic M1 agonist, is used potentially for the treatment of Xerostomia, Alzheimer's disease and cognitive.Formula:C10H18N2OSColore e forma:SolidPeso molecolare:214.33LY2607540
CAS:LY2607540 is a metabotropic glutamate 2 potentiator with potential anxiolytic/antidepressant properties (EC(50) = 23 and 13 nM, respectively).Formula:C24H24F3N3O4Purezza:98%Colore e forma:SolidPeso molecolare:475.46γ-secretase modulator 1
CAS:gamma-secretase modulator 1 is a modulator of γ secretase and can be used in studies about the treatment of Alzheimer's disease.Formula:C24H24N4OSPurezza:99.75% - 99.96%Colore e forma:SolidPeso molecolare:416.54Prifuroline
CAS:Prifuroline is an agent of antiarrhythmic.Formula:C14H16N2OPurezza:98%Colore e forma:SolidPeso molecolare:228.29N,N-Dipropyldopamine (hydrobromide)
CAS:N,N-Dipropyldopamine is a dopamine agonist reducing DOPA and locomotion in rats and mice, reversible by spiroperidol.Formula:C14H24BrNO2Colore e forma:SolidPeso molecolare:318.255AF-DX 384 free base
CAS:AF-DX 384 free base is an M2 mAChR and M4 mAChR antagonist, useful in research on neurodivisions and diseases such as Parkinson's.Formula:C27H38N6O2Purezza:98%Colore e forma:SolidPeso molecolare:478.63GTS-21
CAS:GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.Formula:C19H20N2O2Purezza:98%Colore e forma:SolidPeso molecolare:308.37Lintopride
CAS:Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.Formula:C14H19ClN4O2Purezza:98%Colore e forma:SolidPeso molecolare:310.78Astrophloxine
CAS:Astrophloxine is a fluorescent imaging probe that targets antiparallel dimers.Astrophloxine can be used to detect aggregated Aβ in brain tissue andFormula:C27H33IN2Purezza:99.89%Colore e forma:SolidPeso molecolare:512.47PD-102807
CAS:PD-102807 is a selective and competitive M4 muscarinic receptor antagonist for Parkinson's disease research, inhibit airway smooth muscle (ASM) contraction.Formula:C23H24N2O4Purezza:98.90%Colore e forma:SolidPeso molecolare:392.45Camylofine
CAS:Camylofine (Avacan) is an antimuscarinic, used for relaxing smooth muscle.Formula:C19H32N2O2·2HClPurezza:98%Colore e forma:SolidPeso molecolare:393.4(S)-SNAP5114
CAS:(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.Formula:C30H35NO6Purezza:98.20%Colore e forma:SolidPeso molecolare:505.6Ref: TM-T16831
5mg49,00€10mg73,00€25mg152,00€50mg213,00€100mg309,00€200mg423,00€1mL*10mM (DMSO)49,00€5-HT3 antagonist 2
CAS:5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.Formula:C18H21N3OPurezza:98%Colore e forma:SolidPeso molecolare:295.383α,21-Dihydroxy-5α-pregnan-20-one
CAS:3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.Formula:C21H34O3Purezza:98.00%Colore e forma:SolidPeso molecolare:334.495-Carboxamidotryptamine maleate
CAS:5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.Formula:C15H17N3O5Purezza:99.88%Colore e forma:SolidPeso molecolare:319.31(Rac)-VU 6008667
CAS:(Rac)-VU 6008667 is a selective M5 NAM with IC50 of 1.8 μM, high CNS penetration.Formula:C24H17ClF2N2O2Purezza:99.82%Colore e forma:SolidPeso molecolare:438.85Zatosetron maleate
CAS:Zatosetron maleate(LY 277359 maleate) is a potent and selective serotonin 5HT3 receptor antagonist for the study of acute migraine.Formula:C23H29ClN2O6Purezza:98.07%Colore e forma:SolidPeso molecolare:464.94mHTT-IN-2
CAS:mHTT-IN-2 (compound 27) is a potent inhibitor of mutant huntingtin protein (mHTT), with an EC50 value of 0.066 μM.Formula:C20H22FN7OPurezza:98%Colore e forma:SolidPeso molecolare:395.43ETAP
CAS:ETAP, a dual inhibitor of both monoamine oxidase A (MAO-A) and monoamine oxidase B (MAO-B), exhibits antidepressant-like effects and is utilized in the researchFormula:C18H17N3OPurezza:98%Colore e forma:SolidPeso molecolare:291.35LRRK2-IN-10
CAS:LRRK2-IN-10 (compound 34) is a potent, mutation-selective, brain-penetrant inhibitor targeting G2019S-LRRK2 kinase with IC50 values of 11 nM for G2019S-LRRK2Formula:C20H15N5OPurezza:98%Colore e forma:SolidPeso molecolare:341.37MAO-B-IN-22
CAS:MAO-B-IN-22 (compound 6h) represents a powerful MAO-B inhibitor, boasting an IC50 value of 0.014 μM, and exhibits high antioxidant activity alongside effectiveFormula:C20H18FNO2Purezza:98%Colore e forma:SolidPeso molecolare:323.36MAO-B-IN-21
CAS:MAO-B-IN-21: MAO-B inhibitor with antioxidant, anti-amyloid aggregation, neuroprotective properties, BBB permeable, improves memory in Alzheimer's mice.Formula:C24H25ClN2O4Purezza:98%Colore e forma:SolidPeso molecolare:440.92S 14506 hydrochloride
CAS:S 14506 hydrochloride is a 5-HT1A receptor full agonist.Formula:C24H27ClFN3O2Purezza:99.92%Colore e forma:SolidPeso molecolare:443.94ELN318463 racemate
CAS:ELN318463 racemate (ELN 318463 racemate) is the racemate of ELN318463 which is an amyloid precursor protein (APP) selective γ-secretase inhibitor.Formula:C19H20BrClN2O3SPurezza:99.69%Colore e forma:SolidPeso molecolare:471.8Ref: TM-T11178L
1mg154,00€5mg370,00€10mg583,00€25mg858,00€50mg1.170,00€100mg1.575,00€1mL*10mM (DMSO)424,00€Bitopertin (R enantiomer)
CAS:Bitopertin R enantiomer (RG1678 R enantiomer) is the R-enantiomer of Bitopertin.Formula:C21H20F7N3O4SPurezza:98%Colore e forma:SolidPeso molecolare:543.46Anxiolytic/nonsedative agent-1
CAS:TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.Formula:C18H15N3O4Purezza:98.61%Colore e forma:SolidPeso molecolare:337.33Ref: TM-T23445
1mg64,00€2mg96,00€5mg115,00€10mg150,00€25mg330,00€50mg472,00€100mg655,00€500mg1.293,00€(R,R)-Glycopyrrolate
CAS:(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.Formula:C19H28BrNO3Purezza:98%Colore e forma:SolidPeso molecolare:398.34SB-269970
CAS:SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).Formula:C18H28N2O3SPurezza:98%Colore e forma:SolidPeso molecolare:352.49SCH-23390 maleate
CAS:SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Formula:C21H22ClNO5Purezza:98%Colore e forma:SolidPeso molecolare:403.86Lesopitron dihydrochloride
CAS:Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.Formula:C15H23Cl3N6Purezza:98%Colore e forma:SolidPeso molecolare:393.74Tilapertin
CAS:Tilapertin is an oral glycine transporter type-1 inhibitor.Formula:C20H21F3N2O2Purezza:98%Colore e forma:SolidPeso molecolare:378.39PF-03463275 2HCl
CAS:PF-03463275 is an orally available, CNS-penetrant inhibitor of SLC6A9, a GlyT1 glycine transporter.Formula:C19H24Cl3FN4OPurezza:98%Colore e forma:SolidPeso molecolare:449.78(+)-Nipecotic acid
CAS:(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.Formula:C6H11NO2Purezza:99.38%Colore e forma:SolidPeso molecolare:129.16W-13 hydrochloride
CAS:W-13 hydrochloride (W-13 HCl) is a calmodulin antagonist.Formula:C14H18Cl2N2O2SPurezza:98.51%Colore e forma:White PowderPeso molecolare:349.28CP94253 hydrochloride
CAS:CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).Formula:C15H20ClN3OPurezza:99.78%Colore e forma:SolidPeso molecolare:293.79Ref: TM-T22689
5mg66,00€10mg90,00€25mg205,00€50mg334,00€100mg537,00€200mg745,00€1mL*10mM (DMSO)66,00€hMAO-B-IN-7
CAS:Compound 11n (hMAO-B-IN-7) is a potent inhibitor of human monoamine oxidase-B (hMAO-B) that can cross the blood-brain barrier (BBB). It demonstrates an IC 50 value of 0.79±0.05 μM and is useful in research related to Alzheimer's disease (AD) and Parkinson's disease (PD) [1].Formula:C23H19FN2O5Colore e forma:SolidPeso molecolare:422.41hMAO-B-IN-6
CAS:Compound 17d (hMAO-B-IN-6) is an effective and selective hMAO-B inhibitor, demonstrating an IC 50 of 67.02 nM. It significantly ameliorates cognitive deficits induced by Scopolamine in Alzheimer's disease (AD) mice [1].Formula:C19H20N2O5Colore e forma:SolidPeso molecolare:356.37AChE/BChE-IN-3
CAS:AChE/BChE-IN-3 (BMC-1) dual inhibitor: IC50 of 6.08 μM for elAChE, 0.383 μM for eqBChE.Formula:C15H24N2O3Colore e forma:SolidPeso molecolare:280.36(-)-Donepezil
CAS:(-)-Donepezil is an isomer of Donepezil -- a nootropic acting as an inhibitor of acetylcholinesterase.Formula:C24H29NO3Colore e forma:SolidPeso molecolare:379.49Bradanicline
CAS:Bradanicline: potent α7 nAChR agonist, EC50=17 nM, Ki=1.4 nM, used in cognitive disorder research.Formula:C22H23N3O2Colore e forma:SolidPeso molecolare:361.44Protriptyline
CAS:Protriptyline: Antidepressant, AChE inhibitor (IC50 0.06 mM), prevents Aβ aggregation; potential for depression and Alzheimer's.Formula:C19H21NColore e forma:SolidPeso molecolare:263.38SSAO inhibitor-3
CAS:SSAO inhibitor-3 targets human AOC1/SSAO in atherosclerosis, diabetes, obesity, CKD, and more, with IC50s of 0.1-10 μM/<10 nM.Formula:C15H23FN4O3Colore e forma:SolidPeso molecolare:326.37BuChE-IN-2
CAS:BuChE-IN-2 inhibits BuChE (IC50: 1.28 μM), NO (0.67 μM), Aβ, ROS, chelates Cu2+, penetrates BBB, used in Alzheimer's research.Formula:C28H20F4N6O3Colore e forma:SolidPeso molecolare:564.49Naronapride
CAS:Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.Formula:C27H41ClN4O5Colore e forma:SolidPeso molecolare:537.09Bopindolol (malonate)
CAS:Bopindolol is a non-selective β-adrenergic receptor antagonist.Formula:C26H32N2O7Colore e forma:SolidPeso molecolare:484.549SV5
CAS:SV5: potent anti-Alzheimer's, protects SHSY-5Y from Aβ1-42 death, stable with optimal pharmacology in plasma, antioxidant, neuroprotective.Formula:C21H30N2O4S2Colore e forma:SolidPeso molecolare:438.6MAO-B-IN-15
CAS:MAO-B-IN-15 selectively inhibits MAO-B, targeting Tyr 326 (IC50 = 13.5 μM), useful for Parkinson's research.Formula:C17H18FNO2Colore e forma:SolidPeso molecolare:287.33BChE-IN-9
CAS:BChE-IN-9 (Azepano-11-deoxo-glycyrrhetol) is a hybrid BChE inhibitor (Ki: 0.21 μM).Formula:C30H51NOColore e forma:SolidPeso molecolare:441.73AChE/BChE/MAO-B-IN-3
AChE/BChE/MAO-B-IN-3: potent MAO-B, AChE & BChE inhibitor; IC50: 0.0359μM (MAO-B), 0.0473/0.0782μM (AChE/BChE); possible Alzheimer's research use.Formula:C25H31N3O3Colore e forma:SolidPeso molecolare:421.53AChE-IN-20
CAS:AChE-IN-20: AChE inhibitor (IC50: 397.32 nM), hCA-I/II blocker (IC50: ~77 nM avg), α GLY suppressor (IC50: 52.08 nM).Formula:C22H20N8O6S2Colore e forma:SolidPeso molecolare:556.57Territrem B
CAS:Territrem B: A mycotoxin that irreversibly blocks AChE, causes tremors in mice at 0.21 mg/kg.Formula:C29H34O9Colore e forma:SolidPeso molecolare:526.57AP-521 (Free base)
CAS:AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.Formula:C20H18N2O3SColore e forma:SolidPeso molecolare:366.43Nelonicline citrate
CAS:Nelonicline citrate (ABT-126) is a selective α7 nAChR agonist with a Ki of 12.3 nM, studied for schizophrenia and Alzheimer's.Formula:C23H27N3O8SColore e forma:SolidPeso molecolare:505.545-HT2A receptor agonist-2
CAS:Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.Formula:C20H21ClN2O3Colore e forma:SolidPeso molecolare:372.85RLH 033
CAS:RLH 033 is a selective ligand for the sigma 1 recognition site.Formula:C25H31ClN2O4Purezza:98%Colore e forma:SolidPeso molecolare:458.98BMS-902483
CAS:BMS-902483: potent α7 partial agonist; enhances rodent cognition; α7 EC50=9.3nM; 5-HT3A IC50=480nM.Formula:C18H20N4OPurezza:98%Colore e forma:SolidPeso molecolare:308.38PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Formula:C17H21N3Purezza:98%Colore e forma:SolidPeso molecolare:267.37AChE/BuChE-IN-1
CAS:AChE/BuChE-IN-1: BuChE inhibitor (IC50=0.48µM), weaker AChE blocker (IC50=7.16µM), ·OH scavenger (IC50=0.1674µM), may aid in AD research.Formula:C19H19NO4Colore e forma:SolidPeso molecolare:325.36J-104129 fumarate
CAS:J-104129 fumarate is a potent M3 muscarinic receptor antagonist.Formula:C28H40N2O6Colore e forma:SolidPeso molecolare:500.63mGluR2 modulator 4
CAS:Compound 47 is a potent mGluR2 enhancer with an EC50 of 0.8 μM, potentially useful for antipsychotic research.Formula:C18H18BrN3Colore e forma:SolidPeso molecolare:356.26Pralidoxime
CAS:Pralidoxime reactivates AChE blocked by nerve agents, aiding as an organophosphate poisoning antidote.Formula:C7H9N2OColore e forma:SolidPeso molecolare:137.16SGC-AAK1-1N
CAS:SGC-AAK1-1N is a potent and selective inhibitor of AAK1 (AP2 associated kinase 1) with an IC 50 of 1.8 μM [1].Formula:C20H22N4O3SColore e forma:SolidPeso molecolare:398.482-PAT
CAS:2-PAT: reversible MAO-A inhib., IC50=0.721 µM; MAO-B inactivator, IC50=14.6 µM; potential in Parkinson's/depression study.Formula:C13H15NColore e forma:SolidPeso molecolare:185.26(S)-VQW-765
(S)-VQW-765, oral α7 nAChR partial agonist, may improve cognition in Alzheimer's and schizophrenia.Formula:C19H22N2OColore e forma:SolidPeso molecolare:294.39Ph-HTBA
CAS:Ph-HTBA: high-affinity CaMKIIα modulator, brain-penetrant, Kd 757 nM, used in ischemia/neurodegeneration research.Formula:C19H18O3Colore e forma:SolidPeso molecolare:294.34VU 0360172 hydrochloride
CAS:positive allosteric modulator of mGlu5 receptorsFormula:C18H16ClFN2OPurezza:98%Colore e forma:SolidPeso molecolare:330.78VU0463841
CAS:VU0463841 is a mGlu5 negative allosteric modulators.
Formula:C13H8ClFN4OColore e forma:SolidPeso molecolare:290.68Flupyrimin
CAS:Flupyrimin is the insect nicotinic acetylcholine receptor (nAChR) antagonist [1].Formula:C13H9ClF3N3OColore e forma:SolidPeso molecolare:315.68BuChE-IN-7
BuChE-IN-7: selective hBuChe & eqBuChe inhibitor, IC50s 40/80 nM, boosts cognition & memory, and penetrates blood-brain barrier.Formula:C25H34N2O2Colore e forma:SolidPeso molecolare:394.55MAO-B-IN-14
CAS:MAO-B-IN-14 (Compound 9) is a potent and selective inhibitor of monoamine oxidase-B (MAO-B) with an IC 50 of 0.95 μM and a Ki of 0.55 μM for human MAO-B.Formula:C17H14O3SColore e forma:SolidPeso molecolare:298.36ZK93423
CAS:ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.Formula:C23H22N2O4Colore e forma:SolidPeso molecolare:390.43CP 135807
CAS:CP 135807 is a 5-HT1D receptor agonist.Formula:C19H21N5O2Purezza:98%Colore e forma:SolidPeso molecolare:351.4AFDX384
CAS:AFDX384 is potent M2/M4 selective antagonist.Formula:C28H42N6O5SColore e forma:SolidPeso molecolare:574.74VU6010572
CAS:VU6010572: potent, selective mGlu3 modulator, IC50 245 nM, high CNS penetration.Formula:C20H18FNO3Colore e forma:SolidPeso molecolare:339.36VU6001966
CAS:VU6001966: potent, selective mGlu2 inhibitor (IC50=78 nM), negative modulator, with good CNS penetration.Formula:C17H15FN4O2Purezza:98%Colore e forma:SolidPeso molecolare:326.33Aβ Fibrillization modulator 1
CAS:Aβ Fibrillization Modulator 1 stabilizes amyloid-beta (Aβ) monomers, preventing their aggregation into fibrils.Formula:C17H12N4O3SSeColore e forma:SolidPeso molecolare:431.33Bisindolylmaleimide VII
CAS:Bisindolylmaleimide VII is a selective inhibitor of protein kinase C.Formula:C27H27N5O2Colore e forma:SolidPeso molecolare:453.54DPNB-ABT594
DPNB-ABT594, a nitrobenzyl-caged ABT594, selectively activates α4β2 over α7 nAChRs; used to study Ca²⁺ signaling in MHb.Formula:C31H46ClN3O11Colore e forma:SolidPeso molecolare:672.16AChE-IN-12
CAS:AChE-IN-12 inhibited rat/eel AChE, crossed BBB, prevented Aβ1-42 aggregation, and has potential for Alzheimer's research.Formula:C33H41NO7Colore e forma:SolidPeso molecolare:563.68AC-42
CAS:AC-42 is an allosteric agonist of M1 muscarinic receptor.
Formula:C20H31NOColore e forma:SolidPeso molecolare:301.47BMS-911172
CAS:BMS-911172 is an adaptor associated kinase 1 (AAK1 kinase) inhibitor with an IC 50 of 35 nM.Formula:C16H19F2N3O3Colore e forma:SolidPeso molecolare:339.34CGS 12066B dimaleate
CAS:5-HT1B full agonistFormula:C25H25F3N4O8Purezza:98%Colore e forma:SolidPeso molecolare:566.48RX 801077
CAS:RX 801077 is a selective I2R agonist, Ki of 70.1 nM, with anti-inflammatory and neuroprotective properties for TBI research.Formula:C11H10N2OColore e forma:SolidPeso molecolare:186.21CP 93129 dihydrochloride
CAS:5-HT1B agonist, potent and highly selectiveFormula:C12H14ClN3OPurezza:98%Colore e forma:SolidPeso molecolare:251.71TC-N 22A
CAS:TC-N 22A is a strong, selective, oral active mGlu4 forward allosteric regulator (PAM) that can cross the blood-brain barrier.Formula:C14H13N5SPurezza:99.95%Colore e forma:SolidPeso molecolare:283.35Parapenzolate bromide
CAS:Parapenzolate bromide is an orally active mAChR antagonist. parapenzolate bromide is an anticholinergic and antitussive agent.Formula:C21H26BrNO3Colore e forma:SolidPeso molecolare:420.347ASP2535
CAS:ASP2535 is a potent, selective, orally bioavailable, brain permeable and centrally-active glycine transporter-1 (GlyT1) inhibitor.ASP2535 can improve cognitiveFormula:C22H18N6OPurezza:98%Colore e forma:SolidPeso molecolare:382.42SR 16584
CAS:α3β4 nAChR antagonistFormula:C17H22N2OPurezza:99.84%Colore e forma:SolidPeso molecolare:270.37GR 55562 dihydrochloride
CAS:5-HT1B (5-HT1Dβ) silent antagonistFormula:C23H27Cl2N3O2Purezza:99.45%Colore e forma:SolidPeso molecolare:448.39Prucalopride hydrochloride
CAS:Prucalopride hydrochloride is a selective agonist of the 5-HT4.Formula:C18H27Cl2N3O3Purezza:98%Colore e forma:SolidPeso molecolare:404.33Usmarapride free base
CAS:Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.Formula:C21H29N5O2Purezza:99.91% - 99.91%Colore e forma:SolidPeso molecolare:383.49Lu-AF11205
CAS:Lu-AF11205 is a potent positive allosteric modulator (PAM) of mGlu5 receptor.Formula:C17H16N2OSPurezza:98%Colore e forma:SolidPeso molecolare:296.39Fluoroclorgyline
CAS:Fluoroclorgyline is a specific inhibitor of monoamine oxidase A (MAO-A).Formula:C13H15ClFNOPurezza:98%Colore e forma:SolidPeso molecolare:255.72RS-0466
CAS:RS-0466 is an β-amyloid-induced cytotoxicity inhibitor.Formula:C17H17N5O2Purezza:98%Colore e forma:SolidPeso molecolare:323.35Suclofenide
CAS:Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.Formula:C16H13ClN2O4SPurezza:98%Colore e forma:SolidPeso molecolare:364.8SB 258585 hydrochloride
CAS:SB 258585 hydrochloride is a 5-HT6 receptor antagonist.Formula:C18H23ClIN3O3SPurezza:98%Colore e forma:SolidPeso molecolare:523.82(S)-HexylHIBO
CAS:Group I mGlu receptor antagonistFormula:C12H20N2O4Purezza:98%Colore e forma:SolidPeso molecolare:256.3CUMI-101
CAS:CUMI-101 is an agonist of 5-HT1A receptor.Formula:C19H27N5O3Colore e forma:SolidPeso molecolare:373.45HexylHIBO
CAS:HexylHIBO is a type I mGluR antagonist that inhibits mGlu1a and mGlu5a, with Kb values of 140 and 110 μM, respectively.HexylHIBO decreases sEPSC in rats.Formula:C12H20N2O4Purezza:99.55%Colore e forma:SolidPeso molecolare:256.3(S)-3-Carboxy-4-hydroxyphenylglycine
CAS:group I metabotropic glutamate receptor antagonist and group II mGlu agonistFormula:C9H9NO5Purezza:98%Colore e forma:SolidPeso molecolare:211.17JN403
CAS:JN403 is a selective agonist of nicotinic acetylcholine receptor alpha7.Formula:C16H21FN2O2Colore e forma:SolidPeso molecolare:292.35(4E)-SUN9221
CAS:(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity inFormula:C25H31FN4O3Purezza:97.79%Colore e forma:SolidPeso molecolare:454.54GS 39783
CAS:GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement andFormula:C15H23N5O2SPurezza:99.92%Colore e forma:SolidPeso molecolare:337.44mAChr-in-1
CAS:mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).Formula:C23H25IN2O2Purezza:98%Colore e forma:SolidPeso molecolare:488.36PD 118717
CAS:PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.Formula:C20H22N4O3Purezza:98%Colore e forma:SolidPeso molecolare:366.41KL8604166
CAS:KL8604166 (UCB-11056) is a potential puzzle compound.UCB-11056 amplifies the formation of inducible cyclic AMP in rat brain tissue.Formula:C12H21N5O2Purezza:99.21%Colore e forma:SolidPeso molecolare:267.33Ref: TM-T29038
1mg264,00€5mg650,00€10mg888,00€25mg1.369,00€50mg1.783,00€100mg2.250,00€1mL*10mM (DMSO)590,00€Metitepine
CAS:Metitepine is a serotonin receptor antagonist in the CNS used as an antipsychotic.Formula:C20H24N2S2Colore e forma:SolidPeso molecolare:356.554-Chloro Trazodone hydrochloride
CAS:4-Chloro Trazodone HCl is a Trazodone isomer, an antidepressant for anxiety disorders.Formula:C19H23Cl2N5OColore e forma:SolidPeso molecolare:408.32Hyoscyamine hydrobromide
CAS:Hyoscyamine hydrobromide is an agent of anticholinergic.Formula:C17H24BrNO3Purezza:98%Colore e forma:SolidPeso molecolare:370.28Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Formula:C19H26ClN3O2S2Colore e forma:SolidPeso molecolare:428.01Dexetimide HCl
CAS:Dexetimide HCl is a muscarinic antagonist that has been used to treat neuroleptic-induced parkinsonism. Benzetimide is the (-)-enantimorph of dexetimide.Formula:C23H27ClN2O2Colore e forma:SolidPeso molecolare:398.93(E/Z)-VU0029767
CAS:VU0029767 enhances M1 muscarinic receptor function, increasing acetylcholine potency and efficacy.Formula:C21H21N3O3Colore e forma:SolidPeso molecolare:363.41Atropine Oxide Hydrochloride
CAS:Atropine Oxide, a derivative of anticholinergic Atropine, treats poisonings, slow heart rate, and reduces saliva during surgery.Formula:C17H24ClNO4Colore e forma:SolidPeso molecolare:341.83Echothiophate chloride
CAS:Echothiophate: long-lasting cholinesterase inhibitor for chronic glaucoma treatment; binds irreversibly, inactivating the enzyme.Formula:C9H23ClNO3PSColore e forma:SolidPeso molecolare:291.7708N-Nitroso Fluoxetine
CAS:N-Nitroso fluoxetine is a derivative of fluoxetine.1It is genotoxic toS. typhimuriumwhen used at concentrations ranging from 0.06 to 0.12 mg/ml.Formula:C17H17F3N2O2Colore e forma:SolidPeso molecolare:338.32AZD-9164 bromide
CAS:AMG-221, a selective 11β-HSD1 inhibitor, suppresses enzyme activity, lowers glucose/insulin, and reduces weight in obese mice.Formula:C29H38BrFN2O2Colore e forma:SolidPeso molecolare:545.53TC-1698 dihydrochloride
CAS:TC-1698 dihydrochloride: selective α7 nicotinic agonist, with some β-receptor activity; neuroprotectant.Formula:C13H20Cl2N2Colore e forma:SolidPeso molecolare:275.22Octamylamine hydrochloride
CAS:Octamylamine hydrochloride is a P450 inhibitor.Formula:C13H30ClNColore e forma:SolidPeso molecolare:235.84AS19
CAS:AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).Formula:C18H25N3Purezza:98%Colore e forma:SolidPeso molecolare:283.41Epibatidine 2HCl
CAS:Epibatidine 2HCl is a potent nicotinic agonist.Formula:C11H15Cl3N2Purezza:98%Colore e forma:SolidPeso molecolare:281.61SCH-50910 free base
CAS:SCH-50910 is an antagonist of GABAB receptor.Formula:C8H15NO3Colore e forma:SolidPeso molecolare:173.21Profadol hydrochloride
CAS:Profadol hydrochloride acts as a mixed agonist-antagonist of the μ-opioid receptor with analgesic activity.Formula:C14H22ClNOPurezza:98%Colore e forma:SolidPeso molecolare:255.78Ro 15-1310
CAS:Ro 15-3505, a benzodiazepine receptor partial inverse agonist, has shown the ability to improve impaired recent memory of aged mice.Formula:C15H14ClN3O3Colore e forma:SolidPeso molecolare:319.74Benzoctamine
CAS:Benzoctamine: oral psychoactive with tranquillizing effects; boosts catecholamine turnover; enhances rat heart [3H]noradrenaline uptake.Formula:C18H19NColore e forma:SolidPeso molecolare:249.35YM 230888
CAS:Selective mGlu1 antagonistFormula:C19H28N4OSPurezza:98%Colore e forma:SolidPeso molecolare:360.52Altanserin hydrochloride
CAS:Altanserin hydrochloride is a 5-HT2A receptor antagonist.Formula:C22H23ClFN3O2SPurezza:98%Colore e forma:SolidPeso molecolare:447.955-Nonyloxytryptamine oxalate
CAS:5-HT1B agonistFormula:C21H32N2O5Purezza:98%Colore e forma:SolidPeso molecolare:392.49(R)-DOI hydrochloride
CAS:(R)-DOI hydrochloride is the salt form of 2,5-Dimethoxy-4-iodoamphetamine (DOI), a potent 5-HT2A and 5-HT2C receptor agonist, orally active and hallucinogenic.Formula:C11H17ClINO2Purezza:99.88% - >99.99%Colore e forma:SolidPeso molecolare:357.62Bemesetron
CAS:Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.Formula:C15H17Cl2NO2Purezza:99.77%Colore e forma:SolidPeso molecolare:314.21U 90042
CAS:GABAA receptor ligandFormula:C17H13ClN6OPurezza:98%Colore e forma:SolidPeso molecolare:352.78Nexopamil racemate
CAS:Nexopamil racemate((Rac)-Nexopamil) is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.Formula:C24H40N2O3Purezza:98.61%Colore e forma:SolidPeso molecolare:404.59Amitifadine hydrochloride
CAS:Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).Formula:C11H12Cl3NPurezza:98%Colore e forma:SolidPeso molecolare:264.58KW-6055
CAS:KW-6055 has anti-amnesic activity, is a benzylpyridine derivative.Formula:C16H17N3O3Purezza:98%Colore e forma:SolidPeso molecolare:299.32AS1069562
CAS:AS1069562 inhibits 5-HT/NE reuptake, boosts IGF-1, FGF2 mRNA in dorsal root ganglia, spinal cord.Formula:C20H23NO5SPurezza:98%Colore e forma:SolidPeso molecolare:389.46Dac 5945
CAS:DAC 5945 is a more effective muscarinic antagonist in the airways than in the heart.Formula:C19H30ClN3OPurezza:98%Colore e forma:SolidPeso molecolare:351.91Palonosetron
CAS:Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).Formula:C19H24N2OPurezza:98%Colore e forma:SolidPeso molecolare:296.41U-89843A
CAS:U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].Formula:C16H24ClN5Purezza:98%Colore e forma:SolidPeso molecolare:321.85SCH 50911
CAS:SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.Formula:C8H15NO3Purezza:98%Colore e forma:SolidPeso molecolare:173.21Mirisetron
CAS:Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.Formula:C24H31N3O2Purezza:99.88%Colore e forma:SolidPeso molecolare:393.52Tarafenacin D-tartrate
CAS:Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.Formula:C25H26F4N2O8Purezza:99.86%Colore e forma:SolidPeso molecolare:558.48BuChE-IN-6
CAS:BuChE-IN-6 inhibits BuChE (IC50: 0.46 μM eqBuChE, 0.51 μM hBuChE) and prevents Aβ 42 self-aggregation.Formula:C21H26N4O2Colore e forma:SolidPeso molecolare:366.46Sulfoxaflor
CAS:Sulfoxaflor (GF 2032) is an agonist of nAChR1 and nAChR2 subtypes and a systemic insecticide. Cost-effective and quality-assured.Formula:C10H10F3N3OSPurezza:99.56% - 99.98%Colore e forma:SolidPeso molecolare:277.27Ref: TM-T19940
1mg100,00€5mg275,00€10mg384,00€25mg572,00€50mg780,00€100mg1.018,00€250mg2.080,00€1mL*10mM (DMSO)245,00€LOX-IN-3
CAS:LOX-IN-3, an orally active inhibitor of lysyl oxidase (LOX), holds potential application in the fields of fibrosis, cancer, and angiogenesis research[1].Formula:C13H13FN2O2SColore e forma:SolidPeso molecolare:280.32ML289
CAS:ML289 is a potent CNS-penetrant mGlu3 modulator with IC50 of 0.66 μM, >15-fold selectivity over mGlu2, and inactive against mGlu5.Formula:C22H23NO3Purezza:99.54%Colore e forma:SolidPeso molecolare:349.42Ref: TM-T23000
5mg48,00€10mg75,00€25mg138,00€50mg212,00€100mg320,00€200mg445,00€1mL*10mM (DMSO)49,00€Alaproclate
CAS:Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.Formula:C13H18ClNO2Purezza:98.29% - 98.64%Colore e forma:SolidPeso molecolare:255.74ML352
CAS:ML352 inhibits choline transporter noncompetitively; Ki of 92 nM in human CHT, 166 nM in mouse synaptosomes.Formula:C21H29N3O4Purezza:99.15%Colore e forma:SolidPeso molecolare:387.47Methiothepin maleate
CAS:Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.Formula:C24H28N2O4S2Purezza:98%Colore e forma:SolidPeso molecolare:472.62RS 56812 hydrochloride
CAS:5-HT3 partial agonistFormula:C18H22ClN3O2Purezza:98.62%Colore e forma:SolidPeso molecolare:347.84A-794282
CAS:A-794282 is a selective antagonist of mGluR1.Formula:C19H18N4OSPurezza:99.87%Colore e forma:SolidPeso molecolare:350.44MAO-IN-M30 dihydrochloride
CAS:MAO-IN-M30 dihydrochloride: potent, brain-specific MAO-A/B inhibitor, iron chelator with antioxidant effects, counters Parkinson's in mice.Formula:C14H16Cl2N2OPurezza:99.83%Colore e forma:SolidPeso molecolare:299.2Ref: TM-T38034
1mg34,00€2mg43,00€5mg65,00€10mg90,00€25mg161,00€50mg230,00€100mg319,00€500mgPrezzo su richiesta2-Iodomelatonin
CAS:2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map melatonin sites in brain/tissues.Formula:C13H15IN2O2Purezza:99.7%Colore e forma:SolidPeso molecolare:358.17Ref: TM-T10073
10mg43,00€25mg79,00€50mg118,00€100mg178,00€200mg268,00€500mgPrezzo su richiesta1mL*10mM (DMSO)34,00€Tracazolate hydrochloride
CAS:Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.Formula:C16H25ClN4O2Purezza:99.52%Colore e forma:SolidPeso molecolare:340.85TIK-301
CAS:TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM
Formula:C14H17ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:280.75L-694,247
CAS:L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.Formula:C20H21N5O3SPurezza:98.36%Colore e forma:White SolidPeso molecolare:411.48VU0155041 sodium
CAS:VU0155041 sodium is a positive allosteric modulator of mGluR4 that promotes extinction in male rats.Formula:C14H14Cl2NNaO3Purezza:98%Colore e forma:SolidPeso molecolare:338.16HOCPCA
CAS:HOCPCA: potent, selective GHB site ligand; 27x higher affinity than GHB; crosses blood-brain barrier.Formula:C6H8O3Purezza:98%Colore e forma:SolidPeso molecolare:128.13CC4
CAS:Selective α6β2/α4β2 partial agonist; Ki: 12/26nM (rat); poor α3β4/α7 affinity; stimulates dopamine release; reduces nicotine self-admin in rats.Formula:C24H30N4O2Colore e forma:SolidPeso molecolare:406.52SCH 57790
CAS:SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.Formula:C25H31N3O2SPurezza:99.12% - 99.69%Colore e forma:SolidPeso molecolare:437.6WAY208466 dihydrochloride
CAS:WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.Formula:C17H20Cl2FN3O2SPurezza:98.43% - 99.56%Colore e forma:SolidPeso molecolare:420.33LP44 hydrochloride
CAS:LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Formula:C27H38ClN3OSPurezza:98.06%Colore e forma:SolidPeso molecolare:488.13Tropatepine
CAS:Tropatepine: oral anticholinergic, treats extrapyramidal symptoms, anti-Parkinson's.Formula:C22H23NSColore e forma:SolidPeso molecolare:333.49q-FTAA
CAS:q-FTAA targets Aβ1-42 fibrils (330-630 nM) and ADPBC (300-500 nM), useful in Alzheimer's disease research.Formula:C21H14O6S4Colore e forma:SolidPeso molecolare:490.59Neopterin, L-erythro-
CAS:Neopterin, L-erythro- can be used as a cholinergic receptor.Formula:C9H11N5O4Colore e forma:SolidPeso molecolare:253.21A-850002
CAS:A-850002 is a bioactive chemical.Formula:C18H16N4OSColore e forma:SolidPeso molecolare:336.41S16961
CAS:S16961 (S169611) is an agonist of nicotinic receptor.Formula:C41H71NO6Purezza:99.69%Colore e forma:SolidPeso molecolare:674.01RJR-2429
CAS:RJR-2429 is a potent AChR agonist.Formula:C12H16N2Colore e forma:SolidPeso molecolare:188.27W-5 hydrochloride
CAS:W-5 hydrochloride (N-(6-Aminohexyl)-1-naphthalenesulfonamide HCl) is a potent calmodulin antagonist.Formula:C16H23ClN2O2SPurezza:99.35%Colore e forma:Off-White Crystalline SolidPeso molecolare:342.88DBO-83
CAS:DBO-83, an agonist of nicotinic acetylcholine receptors (nAChRs), has anti-amnesic and antinociceptive activities.Formula:C10H15Cl3N4Purezza:98%Colore e forma:SolidPeso molecolare:297.61OPC-14523 hydrochloride
CAS:OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.Formula:C23H29Cl2N3O2Purezza:99.60%Colore e forma:SolidPeso molecolare:450.4ST1936
CAS:ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.Formula:C13H17ClN2Purezza:98%Colore e forma:SolidPeso molecolare:236.74Ref: TM-T23396
1mg44,00€5mg111,00€10mg178,00€25mg316,00€50mg470,00€100mg682,00€200mg954,00€1mL*10mM (DMSO)123,00€GAT107
CAS:GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.Formula:C18H17BrN2O2SPurezza:99.33%Colore e forma:SolidPeso molecolare:405.31MAO-B-IN-23
CAS:MAO-B-IN-23, also known as Compound 11f, is a reversible and competitive monoamine oxidase B (MAO-B) inhibitor with an IC50 value of 1.44 μM and a Ki of 0.51 μMFormula:C19H18BrNOPurezza:98%Colore e forma:SolidPeso molecolare:356.26E2730
CAS:E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.Formula:C9H8F4N2O2SPurezza:98.22% - 98.54%Colore e forma:SolidPeso molecolare:284.23L 858051
CAS:L 858051 activates adenylate cyclase. It also inhibits glucose transport in rat adipocytes.Formula:C29H48N2O7Colore e forma:SolidPeso molecolare:536.7MFZ 10-7 hydrochloride
CAS:MFZ 10-7 hydrochloride is a highly potent and selective negative allosteric modulator of mGluR5 NAMFormula:C15H10ClFN2Purezza:98%Colore e forma:SolidPeso molecolare:272.71Phenoxypropazine
CAS:Phenoxypropazine, a potent monoamine oxidase (MAO) inhibitor, is utilized in depression research.Formula:C9H14N2OColore e forma:SolidPeso molecolare:166.22DMeOB
CAS:DMeOB (3,3'-Dimethoxybenzaldazine) is a negative regulator with mGluR5 agonist activity and is used in the study of neurological disorders.Formula:C16H16N2O2Purezza:98.34%Colore e forma:SolidPeso molecolare:268.31Phaclofen
CAS:GABAB antagonistFormula:C9H13ClNO3PPurezza:99.32%Colore e forma:White SolidPeso molecolare:249.63Ifoxetine sulfate
CAS:Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.Formula:C13H19NO2H2O4SPurezza:98%Colore e forma:SolidPeso molecolare:270.34PNU-96391
CAS:PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.Formula:C15H23NO2SPurezza:99.53%Colore e forma:SolidPeso molecolare:281.41Ref: TM-T28435
1mg73,00€5mg146,00€10mg210,00€25mg319,00€50mg447,00€100mg600,00€200mg800,00€1mL*10mM (DMSO)138,00€Aβ42-IN-2
CAS:Aβ42-IN-2 is a γ-secretase modulator. Aβ42-IN-2 has an IC 50 of 6.5 nM for Αβ 42. Aβ42-IN-2 can be used for the Alzheimer's disease research[1].Formula:C24H26N6O2Purezza:98.09% - 99.87%Colore e forma:SolidPeso molecolare:430.5Ref: TM-T9641
1mg42,00€5mg94,00€10mg134,00€25mg215,00€50mg304,00€100mg420,00€200mg582,00€1mL*10mM (DMSO)93,00€Glemanserin
CAS:Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.Formula:C20H25NOPurezza:99.93%Colore e forma:SolidPeso molecolare:295.42Ref: TM-T22964
1mg38,00€5mg84,00€10mg119,00€25mg259,00€50mg409,00€100mg605,00€500mg1.288,00€1mL*10mM (DMSO)84,00€(RS)-4-Carboxyphenylglycine
CAS:(RS)-4-Carboxyphenylglycine is a racemic mixture. (S)-4-Carboxyphenylglycine is a selective mGlu1α receptor antagonist.Formula:C9H9NO4Purezza:97.22% - >99.99%Colore e forma:SolidPeso molecolare:195.17MHP 133
CAS:MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).Formula:C17H20ClN5O3Purezza:98%Colore e forma:SolidPeso molecolare:377.83S 24795
CAS:S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.Formula:C14H13BrINOPurezza:99.934%Colore e forma:SolidPeso molecolare:418.07Ref: TM-T23286
5mg44,00€10mg66,00€25mg138,00€50mg215,00€100mg338,00€200mg480,00€1mL*10mM (DMSO)48,00€Chlorisondamine chloride
CAS:Chlorisondamine chloride: a nicotinic antagonist, mainly for animal research, former antihypertensive.Formula:C14H20Cl6N2Colore e forma:SolidPeso molecolare:429.03AZD 3043
CAS:AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.Formula:C19H29NO5Purezza:98.19% - 99.55%Colore e forma:SolidPeso molecolare:351.44SB 272183
CAS:SB 272183 is a highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drug.Formula:C29H28ClN5OPurezza:98%Colore e forma:SolidPeso molecolare:498.02

