Proteasi/Proteasoma
Gli inibitori delle proteasi e del proteasoma sono composti che bloccano l'attività delle proteasi e del proteasoma, che sono coinvolti nella degradazione e nel turnover delle proteine. Questi inibitori sono fondamentali per studiare la regolazione dell'omeostasi proteica, il controllo del ciclo cellulare e l'apoptosi. Gli inibitori delle proteasi e del proteasoma vengono anche utilizzati nel trattamento di malattie come il cancro, dove la degradazione anomala delle proteine svolge un ruolo nella progressione della malattia. Inibendo le proteasi o il proteasoma, questi composti possono indurre la morte cellulare nelle cellule tumorali e sono strumenti critici sia per la ricerca di base che per lo sviluppo terapeutico. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle proteasi e del proteasoma di alta qualità per supportare la tua ricerca in biochimica, biologia cellulare e sviluppo di farmaci.
Sottocategorie di "Proteasi/Proteasoma"
- Acetil-CoA carbossilasi(38 prodotti)
- Cisteina proteasi(111 prodotti)
- DPP-4(27 prodotti)
- Glutaminasi(46 prodotti)
- Proteasi HIV(506 prodotti)
- PAI-1(26 prodotti)
- Inibitori della proteasi(50 prodotti)
- Ricettore attivato dalla proteasi(55 prodotti)
- Proteasoma(85 prodotti)
- Proteasi serina(54 prodotti)
- p97(15 prodotti)
Mostrare 3 più sottocategorie
Trovati 984 prodotti di "Proteasi/Proteasoma"
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AZD-9684
CAS:AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis.Formula:C10H14N2O2SColore e forma:SolidPeso molecolare:226.3TNK2-IN-1
CAS:TNK2-IN-1 is a TNK2 inhibitor (IC50: 224 nM) that can be used in cancer research.Formula:C23H24N6O2Colore e forma:SolidPeso molecolare:416.48ITX-4520
CAS:ITX-4520 novel highly potent, orally bioavailable inhibitor of hepatitis C virus (HCV) entry.Formula:C24H23F2N3OSColore e forma:SolidPeso molecolare:439.52K 579
CAS:K 579 is a dipeptidyl peptidase IV inhibitor.Formula:C17H24N6OPurezza:98%Colore e forma:SolidPeso molecolare:328.41L 722151
CAS:L 722151 is an FXIIIa inhibitor.Formula:C8H9ClN2O5S3Purezza:98%Colore e forma:SolidPeso molecolare:344.82PTIQ
CAS:MMP-3 expression inhibitorFormula:C13H17NO3Purezza:98%Colore e forma:SolidPeso molecolare:235.28Chymase-IN-1
CAS:Chymase-IN-1 is a selective, orally active inhibitor of human mast cell chymase (IC50: 29 nM).Formula:C20H15ClNO4PSPurezza:99.17%Colore e forma:SolidPeso molecolare:431.83Ref: TM-T10811
1mg155,00€5mg369,00€10mg525,00€25mg787,00€50mg1.054,00€100mg1.415,00€500mg2.802,00€1mL*10mM (DMSO)404,00€BAY-678 racemate
CAS:BAY-678 racemate: orally active, selective cell-permeable HNE inhibitor with IC50 of 20 nM.Formula:C20H15F3N4O2Purezza:98%Colore e forma:SolidPeso molecolare:400.35ADAMTS-5-IN-2
CAS:ADAMTS-5-IN-2 is a potent inhibitor of ADAMTS-5, exhibiting an IC50 of 0.71 µM, and holds potential for osteoarthritis research.Formula:C17H15N3OSColore e forma:SolidPeso molecolare:309.39Cofrogliptin
CAS:Cofrogliptin (HSK7653) is a DPP-4 inhibitor with hypoglycemic effects, which can be used to study type 2 diabetes (T2D).Formula:C18H19F5N4O3SColore e forma:SolidPeso molecolare:466.43Ref: TM-T62985
1mg73,00€5mg160,00€10mg250,00€25mgPrezzo su richiesta50mgPrezzo su richiesta1mL*10mM (DMSO)Prezzo su richiestaSafironil
CAS:Safironil, a novel antifibrotic, competitively inhibits collagen synthesis and modulates fibrosis, impacting type I/III collagen levels.Formula:C15H23N3O4Purezza:99.83%Colore e forma:SolidPeso molecolare:309.36Ref: TM-T67961
1mg64,00€5mg136,00€10mg192,00€25mg334,00€50mg477,00€100mg662,00€200mg892,00€1mL*10mM (DMSO)137,00€WNK-IN-7
CAS:WNK-IN-7 is a potent and selective WNK1 kinase inhibitor.Formula:C26H29N3OPurezza:98%Colore e forma:SolidPeso molecolare:399.53Adafosbuvir PM
CAS:Adafosbuvir PM (AL-335 PM) is a small molecule NS5B inhibitor that can be used to study chronic hepatitis C.Formula:C10H13FN2O6Purezza:98.39%Colore e forma:SolidPeso molecolare:276.22Cysteine protease inhibitor-2
CAS:Cysteine protease inhibitor from US20070032499A1; halts DCT116 at 6.5μM, PC3 at 4.4μM.Formula:C13H5N5OPurezza:98%Colore e forma:SolidPeso molecolare:247.21BR351 precursor
CAS:BR351 precursor is a precursor of BR351. BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).Formula:C27H32N2O8S2Purezza:98%Colore e forma:SolidPeso molecolare:576.68RS-104966
CAS:RS-104966 is an inhibitor of collagenase that acts by inducing the conformational change in the side-chains of the S1 pocket of MMP-1.Formula:C19H21NO6SPurezza:98%Colore e forma:SolidPeso molecolare:391.44THDP-17
CAS:THDP-17 is a inhibitor of glutaminase. THDP-17 shows a partial uncompetitive inhibition in vitro.Formula:C12H16N2SPurezza:98%Colore e forma:SolidPeso molecolare:220.33Ono-3307 mesylate
CAS:no-3307 mesylate is a protease inhibitor that inhibits a variety of proteases and may be used to study pancreatitis.Formula:C15H18N4O7S2Purezza:97.60% - 98.16%Colore e forma:SolidPeso molecolare:430.46Thrombin inhibitor 6
CAS:Thrombin Inhibitor 6, with an IC 50 of 1 nM, acts as a potent anticoagulant by inhibiting thrombin.Formula:C18H19ClN4O2SColore e forma:SolidPeso molecolare:390.89LY 135305
CAS:LY 135305 is a inhibition of spontaneous metastasis.Formula:C19H20ClNPurezza:98%Colore e forma:SolidPeso molecolare:297.82Batimastat sodium salt
CAS:Batimastat (BB-94) sodium salt is a broad-spectrum MMP inhibitor (IC50s: 3, 4, 4, 6, and 20 nM for MMP-1, MMP-2, MMP-9, MMP-7, and MMP-3).Formula:C23H31N3NaO4S2Purezza:98%Colore e forma:SolidPeso molecolare:500.63RWJ-58643 HCl
CAS:RWJ 58643 inhibits beta-tryptase & trypsin; at 100µg with budesonide 200µg, reduces symptoms & IL-5; high doses cause late eosinophilia.Formula:C20H27ClN6O4SColore e forma:SolidPeso molecolare:482.984CA 074
CAS:CA 074 is a potent inhibitor of cathepsin B with a Ki value of 2 to 5 nM.CA 074 inhibits ischemic hippocampal neuronal death in primates and attenuates
Formula:C18H29N3O6Purezza:97.80%Colore e forma:SolidPeso molecolare:383.44XMU-MP-2
CAS:XMU-MP-2 is a potent and selective protease inhibitor with anticancer activity that inhibits the growth of oncogenic BRK-driven tumors in a mouse xenograft
Formula:C32H33F3N8O2Purezza:99.29%Colore e forma:SolidPeso molecolare:618.65HCV-IN-37
CAS:HCV-IN-37: potent HCV inhibitor, stable in rat plasma post-oral dose (15 mg/kg), blocks virus entry phase.Formula:C31H35F2N5Colore e forma:SolidPeso molecolare:515.64KIN1400
CAS:KIN1400 activates IRF3, boosts antiviral immunity, stimulates IFNbeta, and inhibits WNV, DV, and HCV.Formula:C24H17F2N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:449.47AZD-1236
CAS:AZD1236 is a selective inhibitor for human MMP-9/MMP-12, less effective in rodents, and reduces lung injury and inflammation.Formula:C15H19ClN4O5SColore e forma:SolidPeso molecolare:402.852',5-Difluoro-2'-deoxycytidine
CAS:2',5-Difluoro-2'-deoxycytidine has potent anti-HCV activity and toxicity to rRNA.Formula:C9H11F2N3O4Purezza:98%Colore e forma:SolidPeso molecolare:263.2Butabindide
CAS:Butabindide (UCL-1397) selectively inhibits TPP II, protecting CCK-8, with Ki of 10 μM (TPP I) and 7 nM (TPP II).Formula:C17H25N3O2Colore e forma:SolidPeso molecolare:303.4Garvagliptin
CAS:Garvagliptin has antidiabetic activity.Formula:C18H23F2N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:399.46FK-448 Free base
CAS:FK-448 Free base is an effective and specific inhibitor of chymotrypsin, with an IC50 of 720 nM.Formula:C25H30N2O3Purezza:98%Colore e forma:SolidPeso molecolare:406.52BMS-986094
CAS:INX 08189 is an RNA-directed RNA polymerase (NS5B) inhibitor.Formula:C30H39N6O9PColore e forma:SolidPeso molecolare:658.64BR351
CAS:BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).Formula:C20H25FN2O5SPurezza:98%Colore e forma:SolidPeso molecolare:424.49LB-30057
CAS:LB-30057 is used as an oral thrombin inhibitor.Formula:C26H31N5O3SPurezza:98%Colore e forma:SolidPeso molecolare:493.62EI-1
CAS:EI-1 is an inhibitor of Hepatitis C virus entry.Formula:C16H19F3N6O3Colore e forma:SolidPeso molecolare:400.36TNIK-IN-4
CAS:TNIK-IN-4: strong TNIK inhibitor, IC50 of 0.61 μM, suppresses HCT116 colorectal cancer cells.Formula:C20H16FN3O3Colore e forma:SolidPeso molecolare:365.36U 27391
CAS:U 27391 is a metalloproteinase inhibitor. It acts by inhibits the action of human recombinant interleukin-1beta and glycosaminoglycan synthesis.Formula:C23H36N4O5Purezza:98%Colore e forma:SolidPeso molecolare:448.56Lodelaben
CAS:Lodelaben (Declaben, SC-39026) is a reversible, non-competitive,specific inhibitor of human neutrophil elastase (HNE) with high potency (IC50=0.5 μM).Formula:C25H41ClO3Purezza:99.62% - >99.99%Colore e forma:SolidPeso molecolare:425.04MDL-101146, (S)-
CAS:MDL-101146, (S)- is an effective orally active inhibitor of human neutrophil elastase.Formula:C29H37F5N4O6Purezza:98%Colore e forma:SolidPeso molecolare:632.62IMB-26
CAS:IMB-26 is an HCV inhibitor (EC50: 2.1 μM) and has shown potent anti-HCV effects.Formula:C20H23BrN2O6Colore e forma:SolidPeso molecolare:467.31Desethyl KBT-3022
CAS:Desethyl KBT-3022 is an active metabolite of the antiplatelet compound KBT-3022.Formula:C23H20N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:420.48Gosogliptin
CAS:Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.Formula:C17H24F2N6OPurezza:99.74%Colore e forma:SolidPeso molecolare:366.41p-APMSF (hydrochloride)
CAS:p-APMSF irreversibly inhibits several serine proteases; Ki: 1.02-1.54 μM; selective over chymotrypsin and acetylcholinesterase.Formula:C8H10ClFN2O2SColore e forma:SolidPeso molecolare:252.69STOCK2S-26016
CAS:WNK-IN-B, a cell-permeable diaminoacridine, selectively inhibits WNK signaling in mpkDCT/MOVAS by targeting SPAK/OSR1 CCT domain.Formula:C20H19N3O2Colore e forma:SolidPeso molecolare:333.38PF-06279794
CAS:PF-06279794 is a potent, selective and ATP-competitive TNIK inhibitor.Formula:C22H20N4OColore e forma:SolidPeso molecolare:356.42AA9 TG2 inhibitor
CAS:AA9 is a novel transglutaminase (TG2) inhibitor.Formula:C32H36N4O5Colore e forma:SolidPeso molecolare:556.65Desirudin
CAS:Desirudin (CGP 39393) inhibits thrombin, prevents thrombosis, and is used in thrombocytopenia research.Colore e forma:SolidGemigliptin Tartrate(911637-19-9 free base)
CAS:Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).Formula:C22H25F8N5O8Purezza:>99.99%Colore e forma:SolidPeso molecolare:639.45GM 1489
CAS:GM 1489 is an MMP inhibitor, effective against MMP-1, -2, -3, -8, -9, reduces cancer cell invasion, and prevents ear thickening in mice.Formula:C27H33N3O4Colore e forma:SolidPeso molecolare:463.57Tanomastat
CAS:Tanomastat is an orally bioavailable and non-peptidic biphenyl matrix metalloproteinases inhibitor.Formula:C23H19ClO3SPurezza:98%Colore e forma:SolidPeso molecolare:410.91Cyclophilin inhibitor 3
CAS:Cyclophilin inhibitor 3 (compound 7c), a potent inhibitor of cyclophilin A (CypA), exhibited potent anti-HCV effects with an EC50 value of 4.2 μM.Formula:C34H38N4O6Colore e forma:SolidPeso molecolare:598.69Tyrosinase-IN-4
CAS:Tyrosinase-IN-4, a potent inhibitor, has uses in skin-whitening, food preservation, cosmetics, agriculture, and medicine.Formula:C15H9ClO3Colore e forma:SolidPeso molecolare:272.68DTS
CAS:DTS is a selective and isoform-specific RSK1 kinase inhibitor. It also has broad cancer therapeutic potential.Formula:C14H14S3Purezza:98%Colore e forma:SolidPeso molecolare:278.46CP4d inhibitor
CAS:CP4d is a novel reversible tg2 transamidase site-specific inhibitorFormula:C18H13N5O5Colore e forma:SolidPeso molecolare:379.33Prodipine hydrochloride
CAS:Prodipine hydrochloride for purified and plasma Dipeptidyl peptidase IV (DPP IV) from the rabbit (IC50 of 4.5 μM and 30 μM, respectively).Formula:C20H26ClNPurezza:98%Colore e forma:SolidPeso molecolare:315.88Grazoprevir sodium salt
CAS:Grazoprevir sodium salt is a selective Hepatitis C virus NS3/4a protease inhibitor with broad activity across genotypes and resistant variants.Formula:C38H50N6NaO9SPurezza:98%Colore e forma:SolidPeso molecolare:789.9JPM-OEt
CAS:JPM-OEt: broad-spectrum, covalent cysteine cathepsin inhibitor with antitumor effects.Formula:C20H28N2O6Purezza:98%Colore e forma:SolidPeso molecolare:392.45Ro 09-1679
CAS:Ro 09-1679 is a thrombin inhibitor.Formula:C22H39N9O6Purezza:98%Colore e forma:SolidPeso molecolare:525.6Cathepsin L/S-IN-1
Cathepsin L/S-IN-1 inhibits Cathepsin L & S (IC50: 4.10 & 1.79 μM) and reduces metastasis in pancreatic cancer cells.Formula:C29H33BrN4O4SColore e forma:SolidPeso molecolare:613.57HCV-IN-3
CAS:HCV-IN-3 is a hepatitis C virus (HCV) NS3/4a protein inhibitor (IC50: 20 μM; Kd: 29 μM).Formula:C13H11F2NOPurezza:98%Colore e forma:SolidPeso molecolare:235.23Calpain Inhibitor XII
CAS:Calpain Inhibitor XII (Z-L-Nva-CONH-CH2-2-Py) is a calpain I inhibitor that inhibits calpain II and cathepsin B.
Formula:C26H34N4O5Colore e forma:SolidPeso molecolare:482.57SA 152
CAS:SA 152 is an organophosphoric inhibitor.Formula:C19H12F12NO2PColore e forma:SolidPeso molecolare:545.26AZD5248
CAS:AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).Formula:C22H22N4O2Colore e forma:SolidPeso molecolare:374.44Plasma kallikrein-IN-3
CAS:Plasma kallikrein-IN-3 is a potent inhibitor (IC50: 0.15 μM) used in hereditary angioedema and diabetic eye disease research.Formula:C20H23N5O2Colore e forma:SolidPeso molecolare:365.43VA4 TG2 inhibitor
CAS:VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.Formula:C33H41N5O6SColore e forma:SolidPeso molecolare:635.77Kallikrein 5-IN-2
CAS:Kallikrein 5-IN-2 inhibits KLK5 (pIC50=7.1); may normalize skin shedding, lessen inflammation & itching.Formula:C23H22N6OColore e forma:SolidPeso molecolare:398.46Elastase-IN-1
CAS:Elastase-IN-1 (Compound Q11) is a non-toxic elastase inhibitor with an IC 50 of 0.897 μM [1].Formula:C17H12N4O3Colore e forma:SolidPeso molecolare:320.3Tyrosinase-IN-11
CAS:Tyrosinase-IN-11: potent inhibitor, IC50 - 50nM/64nM (L-tyrosinase/L-dopa), antioxidant, low toxicity, for hyperpigmentation study.Formula:C15H14O5Colore e forma:SolidPeso molecolare:274.27PMPA sodium
CAS:PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.Formula:C6H11Na4O7PPurezza:98%Colore e forma:SolidPeso molecolare:318.08Cysteine Protease inhibitor
CAS:Cysteine protease inhibitors are inhibitors of cysteine proteases. Target: Cysteine ProteaseFormula:C18H14N4OPurezza:98%Colore e forma:SolidPeso molecolare:302.33APC-366 HCl
CAS:APC-366 is a selective inhibitor of the mast cell tryptase that inhibits tryptase-induced histamine release from human tonsil and lung cells.Formula:C22H29ClN6O4Colore e forma:SolidPeso molecolare:476.96AL-9
CAS:AL-9 is a GT-1b and GT-2a replication inhibitor.Formula:C23H22N4O3Purezza:98%Colore e forma:SolidPeso molecolare:402.45RID-F
CAS:RID-F is an inhibitor of the nonpeptidic proteasome.Formula:C38H50N2O2Purezza:98%Colore e forma:SolidPeso molecolare:566.82BC-05
CAS:BC-05, an orally active inhibitor targeting CD13 and the proteasome, displays potent inhibition with IC50 values of 0.13 μM against human CD13 and 1.39 μM forFormula:C21H29BN2O9Purezza:98%Colore e forma:SolidPeso molecolare:464.27BMS-363131
CAS:BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of <1.7 nM.Formula:C28H40N6O5Purezza:97.99%Colore e forma:SolidPeso molecolare:540.65Tyrosinase-IN-7
CAS:Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.Formula:C15H10O5Purezza:99%Colore e forma:SolidPeso molecolare:270.24α-Glucosidase-IN-5
CAS:α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.Formula:C15H13NO3Colore e forma:SolidPeso molecolare:255.27GSK2793660 HCl
CAS:GSK2793660 is a irreversible covalent α,β-unsaturated amide based DPP1 inhibitor.Formula:C22H32ClN3O3Colore e forma:SolidPeso molecolare:421.96SAP2-IN-1
CAS:SAP2-IN-1 inhibits secreted aspartate protease 2 (IC50: 0.92 μM), doesn't work in vitro, and helps research infections.Formula:C34H29NO7Colore e forma:SolidPeso molecolare:563.6ND-322 HCl
CAS:ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.Formula:C15H16ClNO3S2Purezza:99.49%Colore e forma:SolidPeso molecolare:357.88Ref: TM-T28145
1mg152,00€5mg334,00€10mg492,00€25mg780,00€50mg1.044,00€100mg1.414,00€1mL*10mM (DMSO)349,00€HCV-IN-34
CAS:HCV-IN-35, an oral HCV blocker, has an EC50 of 0.010 μM and a CC50 of 7.5 μM, indicating strong antiviral effects.Formula:C31H36ClN5Colore e forma:SolidPeso molecolare:514.1Azo-Resveratrol
CAS:Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor.Formula:C12H10N2O3Colore e forma:SolidPeso molecolare:230.22(Rac)-Tanomastat
CAS:Tanomastat (BAY 12-9566) is an oral biphenyl MMP inhibitor; blocks MMP-2, -3, -9, -13, with anti-invasive and anti-metastatic properties.Formula:C23H19ClO3SColore e forma:SolidPeso molecolare:410.91Glutaminase-IN-4
CAS:Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor (IC50: 2.3 μM).Formula:C23H22N6O2S2Colore e forma:SolidPeso molecolare:478.59L 658758
CAS:L 658758 is an inhibitor of serine proteinase.Formula:C16H20N2O9SColore e forma:SolidPeso molecolare:416.4(3S,4S)-A2-32-01
(3S,4S)-A2-32-01, a less active (S,S)-enantiomer of A2-32-01. A2-32-01 is a potent caseinolytic protein proteases (ClpP) inhibitor .Formula:C19H27NO2Colore e forma:SolidPeso molecolare:301.42MMP-1-IN-1
MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM .Formula:C14H17ClN2O3Colore e forma:SolidPeso molecolare:296.75NAAA-IN-2
CAS:NAAA-IN-2, a selective inhibitor with 50 nM IC50, targets NAAA, an enzyme hydrolyzing PEA/OEA, and may aid inflammation and pain studies.Formula:C11H13N3O2SColore e forma:SolidPeso molecolare:251.3TAPI-0
CAS:TAPI-0 is a matrix metalloprotease (MMP) and TACE inhibitor.Formula:C24H32N4O5Colore e forma:SolidPeso molecolare:456.53Tyrosinase-IN-10
CAS:Tyrosinase-IN-10 serves as a partially competitive inhibitor of tyrosinase, demonstrating an inhibition concentration (IC50) value of 1.6 μM against the enzyme'Formula:C16H12O4Colore e forma:SolidPeso molecolare:268.26Calpain-2-IN-1
CAS:Calpain-2-IN-1 is a selective calpain-2 inhibitor with Ki values of 181 nM for calpain-1 and 7.8 nM for calpain-2, applicable for neurodegenerative diseases a.Formula:C28H37N3O7Colore e forma:SolidPeso molecolare:527.61HCV-IN-35
CAS:HCV-IN-35 is a potent inhibitor of HCV and shows potential for infectious disease research.Formula:C30H36ClN5Colore e forma:SolidPeso molecolare:502.09Calpain Inhibitor XI
CAS:Calpain Inhibitor XI, a reversible covalent inhibitor of calpain-1, is utilized in the research of neurodegenerative disorders.Formula:C26H40N4O6Colore e forma:SolidPeso molecolare:504.62AM 4299 B
CAS:AM 4299 B is a novel inhibitor of a thiol protease.Formula:C16H27N3O7Purezza:98%Colore e forma:SolidPeso molecolare:373.4MDL 27399
CAS:MDL 27399 suppresses human neutrophil cathepsin G.Formula:C26H36N4O8Colore e forma:SolidPeso molecolare:532.59CAA0225
CAS:CAA0225 is a selective inhibitor of cathepsin L. CAA0225 is a probe for autophagic proteolysis.Formula:C28H29N3O5Colore e forma:SolidPeso molecolare:487.55Immunoproteasome inhibitor 1
CAS:Potent, reversible immunoproteasome inhibitor; Ki: β5c 1.18 μM, β1i 0.27 μM, β5i 1.91 μM; potential in treating cancer.Formula:C20H26N2O4Colore e forma:SolidPeso molecolare:358.43ADAMTS-5-IN-3
CAS:ADAMTS-5-IN-3 is a potent inhibitor of ADAMTS-5 and ADAMTS-4, used in research on ADAMTS-5 or ADAMTS-4 mediated diseases.Formula:C20H23Cl2N3O3Colore e forma:SolidPeso molecolare:424.32JO146
CAS:JO146为针对沙眼衣原体高温需要蛋白A(CtHtrA)的蛋白酶抑制剂，其对CtHtrA和人中性粒细胞弹性蛋白酶(HNE)的IC50值分别为21.86 μM和1.15 μM，可应用于细菌感染的抑制。Formula:C31H44N3O7PColore e forma:SolidPeso molecolare:601.67L-873724
CAS:L-873724: Selective, reversible cathepsin K inhibitor; IC50s—cat K: 0.2 nM, cat S: 178 nM, cat L: 264 nM, cat B: 5239 nM; inhibits bone resorption.Formula:C23H26F3N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:481.53(R)-ND-336
CAS:(R)-ND-336: potent, selective MMP-9 inhibitor (K i = 19 nM); inhibits MMP-2 (127 nM), MMP-14 (119 nM); studied for diabetic foot ulcers.Formula:C16H18ClNO3S2Colore e forma:SolidPeso molecolare:371.89MMP13-IN-4
CAS:MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].Formula:C21H17BrN4O5Purezza:98%Colore e forma:SolidPeso molecolare:485.29PF-00356231 hydrochloride
CAS:PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.Formula:C25H21ClN2O3SPurezza:98.39%Colore e forma:SolidPeso molecolare:464.96Ref: TM-T12414
1mg67,00€5mg177,00€10mg284,00€25mg464,00€50mg642,00€100mg853,00€500mgPrezzo su richiestaMMP-2/9-IN-1
CAS:MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.Formula:C14H16IN7SColore e forma:SolidPeso molecolare:441.29AZD6564
CAS:AZD6564 is a fibrinolysis inhibitor which acts via interference of a protein-protein interaction.Formula:C13H22N2O2Colore e forma:SolidPeso molecolare:238.33GLS1 Inhibitor-3
CAS:GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.Formula:C30H32N10O2SColore e forma:SolidPeso molecolare:596.71HCV-IN-36
CAS:HCV-IN-36: oral HCV inhibitor, EC50 0.016 μM, CC50 8.78 μM, potent antiviral.Formula:C30H36ClN5Colore e forma:SolidPeso molecolare:502.09BC-23
CAS:BC-23 (NSC 45382) is a proteasome inhibitor with antitumor and antimicrobial activity for the study of leukemia and small cell lung cancer.Formula:C21H14ClN3O4SPurezza:98%Colore e forma:SolidPeso molecolare:439.87BRD-8899
CAS:BRD-8899 is a STK33 inhibitor, with an IC 50 of 11 nM [1].Formula:C17H22N4O3SColore e forma:SolidPeso molecolare:362.45Tyrosinase-IN-5
CAS:Tyrosinase-IN-5 (16c) inhibits tyrosinase with 0.02 μM IC50, reduces melanogenesis, and is low-toxicity.Formula:C18H13N3O6Colore e forma:SolidPeso molecolare:367.31Efegatran sulfate
CAS:Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.Formula:C21H34N6O7SPurezza:≥98% - ≥98%Colore e forma:SolidPeso molecolare:514.6DPP-IV-IN-1
CAS:DPP-IV-IN-1 is an effective inhibitor of dipeptidyl peptidase IV (DPP-IV), a serine protease (IC50: 4.6 nM).Formula:C11H18FN3O2Purezza:98%Colore e forma:SolidPeso molecolare:243.28SP-Chymostatin B
CAS:SP-Chymostatin B inhibits proteases like chymotrypsin and papain; less effective on human elastase; works at 100-200 μg/ml.Formula:C30H41N7O6Purezza:98%Colore e forma:SolidPeso molecolare:595.69Elasnin
CAS:Elasnin is a reversible inhibitor of elastase for human granulocyte and pancreatic enzymes with IC50 values of 1.3 and 30 µg/ml, respectively.Formula:C24H40O4Colore e forma:SolidPeso molecolare:392.57Ono 3307 Free Base
CAS:Ono 3307 Free Base is a new synthetic protease inhibitorFormula:C14H14N4O4SColore e forma:SolidPeso molecolare:334.35Proteasome-IN-1
CAS:Proteasome-IN-1 is an inhibitor of proteasome.Formula:C42H35N5O3Purezza:98%Colore e forma:SolidPeso molecolare:657.76A-933548
CAS:A-933548: potent calpain inhibitor, selective vs. cathepsins, stable, effective in cell assays.Formula:C25H21N5O3Purezza:98%Colore e forma:SolidPeso molecolare:439.47ASPER-29
CAS:ASPER-29, an Asperphenamate analog, inhibits cathepsins L/S with IC50s of 6.03/5.02 μM, useful in cancer migration/invasion research.Formula:C31H29BrN2O5SColore e forma:SolidPeso molecolare:621.54CAY10704
CAS:CAY10704: Potent HCV inhibitor, EC50=17 nM, low cytotoxicity, good in mice, liver-targeted, not hepatotoxic, weak against dengue.Formula:C18H20Cl2N2Colore e forma:SolidPeso molecolare:335.27DPP-4-IN-1
CAS:DPP-4-IN-1 inhibits DPP-4 with 49 nM IC50, ideal for diabetes study, akin to Alogliptin.Formula:C19H19ClN6Colore e forma:SolidPeso molecolare:366.85AA10 TG2 inhibitor
CAS:AA10 is an irreversible inhibitor of transglutaminase 2 (TG2).Formula:C32H36N4O5Colore e forma:SolidPeso molecolare:556.65PK44 phosphate
CAS:PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).Formula:C17H19F5N7O5PColore e forma:SolidPeso molecolare:527.349BAY8040
CAS:BAY8040 is a potent selective human neutrophilic elastase inhibitor with excellent potency and selectivity with promising pharmacokinetic characteristics.Formula:C21H16F3N5O2Colore e forma:SolidPeso molecolare:427.38Z-LLF-CHO
CAS:Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.Formula:C29H39N3O5Purezza:98%Colore e forma:SolidPeso molecolare:509.64VEL-0230
CAS:VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.Formula:C14H24NNaO5Colore e forma:SolidPeso molecolare:309.33NNGH
CAS:NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.Formula:C13H20N2O5SPurezza:98.41%Colore e forma:SolidPeso molecolare:316.37ZM223 hydrochloride (2031177-48-5 free base)
ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.Formula:C23H18ClF3N4O2S2Purezza:98%Colore e forma:SolidPeso molecolare:538.99Alicapistat
CAS:Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).Formula:C25H27N3O4Purezza:98%Colore e forma:SolidPeso molecolare:433.5Tyrosinase-IN-6
CAS:Tyrosinase-IN-6 (4B) is a potent tyrosinase inhibitor (IC50=3.80 μM) with good antioxidant activity.Formula:C24H31N3O2Colore e forma:SolidPeso molecolare:393.52Anticancer agent 82
CAS:Anticancer agent 82, a FiVe1 derivative, selectively targets VIM in cancer cells to disrupt mitosis, with improved oral bioavailability.Formula:C19H18Cl2N4OColore e forma:SolidPeso molecolare:389.28GS-9256
CAS:GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].Formula:C46H56ClF2N6O8PSPurezza:98%Colore e forma:SolidPeso molecolare:957.46Tyrosinase-IN-3
CAS:Tyrosinase-IN-3 inhibits melanin production; potential for skin whitening and food preservation.Formula:C21H23NO5Colore e forma:SolidPeso molecolare:369.41Gü2602
CAS:Gü2602 inhibits the cathepsin K zymogen autocatalytic activation that is a potent, reversible inhibitor of cathepsin K (CatK) with a Ki of 0.013 nM for matureFormula:C16H22N4O3Colore e forma:SolidPeso molecolare:318.37HCV-IN-33
CAS:HCV-IN-33 (Compound (S)-3i) is an inhibitor of HCV entry.Formula:C31H36ClN5Colore e forma:SolidPeso molecolare:514.1JNJ-10329670
CAS:JNJ 10329670 is a highly potent (Ki of approximately 30 nM), nonpeptidic, noncovalent inhibitor of human cathepsin S with immunosuppressive activity.Formula:C30H34ClF3N6O3SColore e forma:SolidPeso molecolare:651.14AGLME
CAS:AGLME is used in a direct enzymatic assay for activated Hageman factor measuring the ability of Hageman factor to hydrolyze the cpd.Formula:C11H21N3O4Colore e forma:SolidPeso molecolare:259.3Odalasvir
CAS:Odalasvir is a novel NS5A inhibitor for the treatment of hepatitis C.Formula:C60H72N8O6Colore e forma:SolidPeso molecolare:1001.26Cysteine Protease inhibitor hydrochloride
CAS:Cysteine Protease inhibitor hydrochloride is a cysteine protease inhibitor.Formula:C18H15ClN4OPurezza:98%Colore e forma:SolidPeso molecolare:338.79Tec-IN-21
CAS:Tec-IN-21 is an inhibitor of Tec kinase, it also blocks unconventional secretion of fibroblast growth factor 2 (FGF2).Formula:C16H15ClN4O2SPurezza:98%Colore e forma:SolidPeso molecolare:362.83Sheng Gelieting
CAS:CGT-8012 inhibits DP-IV enzyme, aiding type II diabetes research, with an IC50 of 87 nM.Formula:C17H16F6N4OColore e forma:SolidPeso molecolare:406.33ZD8321
CAS:ZD8321 is an effective inhibitor of human Neutrophil elastase (Ki: 13±1.7 nM).Formula:C18H28F3N3O5Purezza:98%Colore e forma:SolidPeso molecolare:423.43Atevirdine
CAS:Atevirdine is an HIV-1 reverse transcriptase inhibitor with antiviral activity for the study of the AIDS dementia complex (ADC).
Formula:C21H25N5O2Purezza:98.20%Colore e forma:SolidPeso molecolare:379.46Tyrosinase-IN-2
CAS:Tyrosinase-IN-2, a potent tyrosinase inhibitor, may help in skin lightening and food preservation research.Formula:C8H8N4O2SPurezza:99.78%Colore e forma:SolidPeso molecolare:224.24Ref: TM-T60278
5mg48,00€10mg71,00€25mg135,00€50mg212,00€100mg340,00€200mg467,00€1mL*10mM (DMSO)49,00€PG-116800
CAS:PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.Formula:C24H27N3O7SPurezza:98.03% - 99.66%Colore e forma:SolidPeso molecolare:501.55TG-2-IN-1
CAS:TG-2-IN-1 (Compound D003) is a transglutaminase-2 ( TGM-2 ) inhibitor. TG-2-IN-1 can be used in myopia research[1].Formula:C8H13ClN2OSPurezza:98.43%Colore e forma:SolidPeso molecolare:220.72Cathepsin X-IN-1
CAS:Cathepsin X-IN-1 (compound 25) reduces the migration of PC-3 cell with low cytotoxic that is a potent inhibitor of Cathepsin X (IC 50 = 7.13 μM) [1].
Formula:C15H13N3O3SPurezza:99.34%Colore e forma:SolidPeso molecolare:315.35CPA inhibitor
CAS:CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM.Formula:C18H19NO4Purezza:99.94%Colore e forma:SolidPeso molecolare:313.35Ref: TM-T10876
1mg54,00€5mg118,00€10mg155,00€25mg263,00€50mg384,00€100mgPrezzo su richiesta1mL*10mM (DMSO)131,00€TG2-IN-3h
CAS:TG2-IN-3h is a highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (tg2) inhibitorFormula:C21H26N4O4SPurezza:99.34% - 99.76%Colore e forma:SolidPeso molecolare:430.522'-C-Methyladenosine
CAS:2'-C-Methyladenosine from C. renalis inhibits HCV, NS5B RNA synthesis (IC50: 0.3, 1.9µM), and LRV1 in L. guyanensis, L. braziliensis.Formula:C11H15N5O4Purezza:99.85%Colore e forma:SolidPeso molecolare:281.2720S Proteasome activator 1
CAS:20S Proteasome activator 1: IC50—0.3 μM (trypsin), 0.7 μM (chymotrypsin), 1.8 μM (caspase); reduces alpha-synuclein A53T, aids neurodegenerative studies.Formula:C27H19ClF2N2OSPurezza:99.82%Colore e forma:SolidPeso molecolare:492.97Gemigliptin
CAS:Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)Formula:C18H19F8N5O2Purezza:99.72%Colore e forma:SolidPeso molecolare:489.36Ref: TM-T7369
2mg38,00€5mg57,00€10mg93,00€25mg148,00€50mg245,00€100mg385,00€500mg873,00€1mL*10mM (DMSO)84,00€TY-51469
CAS:TY-51469 is an inhibitor of chymase (IC50s for simian and human chymases: 0.4 and 7.0 nM, respectively).Formula:C20H15FN2O6S4Purezza:99.65%Colore e forma:SolidPeso molecolare:526.6VRK-IN-1
CAS:VRK-IN-1 is a potent and selective inhibitor of cowpox-associated kinase 1 (VRK1), which can be used in the study of neurological disorders.Formula:C18H11F4NO2Purezza:99.18% - 99.25%Colore e forma:SolidPeso molecolare:349.28Ref: TM-T35863
1mg98,00€5mg225,00€10mg359,00€25mg710,00€50mg1.071,00€100mg1.431,00€200mg1.953,00€1mL*10mM (DMSO)245,00€UK-396082
CAS:UK-396082 is a TAFI inhibitor that inhibits Carboxypeptidase B and can be used in the study of thrombosis, atherosclerosis, cancer and fibrotic conditions.Formula:C12H21N3O2Purezza:99.89%Colore e forma:SolidPeso molecolare:239.31UPGL00004
CAS:UPGL00004: potent GAC inhibitor, IC50=29 nM, Kd=27 nM, suppresses triple-negative breast cancer cell growth.Formula:C25H26N8O2S2Purezza:97.93%Colore e forma:SolidPeso molecolare:534.66Lenacapavir
CAS:Lenacapavir (GS-6207) is the first HIV-1 capsid inhibitor approved by the U.S. Food and Drug Administration, the European Medicines Agency, and Health Canada for the treatment of MDR HIV-1 infection.Cost-effective and quality-assured.Formula:C39H32ClF10N7O5S2Purezza:99.61% - 99.87%Colore e forma:SolidPeso molecolare:968.28Ref: TM-T11465
1mg187,00€5mg376,00€10mg565,00€25mg998,00€50mg1.388,00€100mg1.882,00€200mg2.622,00€1mL*10mM (DMSO)615,00€BDCRB
BDCRB disrupts HCMV DNA maturation by altering terminase cleavage, extending packaging 30 kb until second site.Formula:C12H11BrCl2N2O4Purezza:99.41% - 99.85%Colore e forma:SoildPeso molecolare:398.04BILB-1941
CAS:BILB-1941 (BILB-1941ZW) is an inhibitor of HCV NS5B polymerase and can be used in studies about HCV infection.Formula:C34H34N4O4Purezza:99.51% - 99.65%Colore e forma:SolidPeso molecolare:562.66Ref: TM-T26815
1mg296,00€5mg718,00€10mg982,00€25mg1.485,00€50mg2.008,00€100mg2.637,00€1mL*10mM (DMSO)1.044,00€DB04760
CAS:DB04760: selective MMP-13 inhibitor, non-zinc-chelating, IC50=8nM, reduces paclitaxel neurotoxicity, anticancer.Formula:C22H20F2N4O2Purezza:99.93% - 99.99%Colore e forma:SolidPeso molecolare:410.42Ref: TM-T15055
1mg84,00€5mg205,00€10mg309,00€25mg522,00€50mg747,00€100mg1.035,00€500mg2.052,00€1mL*10mM (DMSO)178,00€JNJ-10311795
CAS:JNJ-10311795 (RWJ-355871) is an inhibitor of neutrophil elastase G and mast cell chymase, demonstrating significant anti-inflammatory effects.Formula:C40H35N2O6PPurezza:97.43%Colore e forma:SolidPeso molecolare:670.69Setrobuvir
CAS:Setrobuvir (ANA-598) is an orally active non-nucleoside HCV NS5B polymerase inhibitor with inhibitory effects on de novo RNA synthesis and primer extension withFormula:C25H25FN4O6S2Purezza:99.95% - 99.97%Colore e forma:SolidPeso molecolare:560.62Ref: TM-T28762
1mg229,00€5mg570,00€10mg812,00€25mg1.216,00€50mg1.663,00€100mg2.242,00€500mg4.494,00€1mL*10mM (DMSO)737,00€Sovaprevir
CAS:Sovaprevir is a non-structural 3 (NS3) protease inhibitor with antiviral activity for the treatment of HCV infection.Formula:C43H53N5O8SPurezza:99.89%Colore e forma:SolidPeso molecolare:799.97Ref: TM-T28830
1mg253,00€5mg620,00€10mg884,00€25mg1.314,00€50mg1.773,00€100mg2.385,00€1mL*10mM (DMSO)982,00€Melagatran
CAS:Melagatran is an orally available, direct synthetic thrombin inhibitor that does not require endogenous cofactors other than thrombin.Cost-effective and quality-assured.Formula:C22H31N5O4Purezza:98.29% - >99.99%Colore e forma:SolidPeso molecolare:429.51Ref: TM-T11994
1mg487,00€5mg1.134,00€10mg1.468,00€25mg2.215,00€50mg2.962,00€100mg4.024,00€1mL*10mM (DMSO)1.071,00€MMP2-IN-3
CAS:MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 μM).Formula:C23H21N3OPurezza:99.38%Colore e forma:SolidPeso molecolare:355.43Ref: TM-T61271
1mg64,00€5mg132,00€10mg195,00€25mg315,00€50mg439,00€100mg590,00€200mg793,00€1mL*10mM (DMSO)140,00€Sirpiglenastat
CAS:Sirpiglenastat (DRP-104) is a glutamine antagonist, a prodrug of DON, with antitumor activity that acts by suppressing the adaptive immune system.Formula:C22H27N5O5Purezza:98.01% - 98.37%Colore e forma:SolidPeso molecolare:441.48Isatoribine
CAS:Isatoribine(ANA245) free base is a potent TLR7 receptor agonist with anti-hepatitis C virus infection activity for the study of HCV infection.Formula:C10H12N4O6SPurezza:98.99% - 99.75%Colore e forma:SolidPeso molecolare:316.29AGPS-IN-2i
CAS:AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.Formula:C18H17F2N3O2Purezza:98.92%Colore e forma:SolidPeso molecolare:345.34Ref: TM-T69685
1mg74,00€5mg188,00€10mg311,00€25mg525,00€50mg747,00€100mg1.017,00€1mL*10mM (DMSO)154,00€HIV-1 integrase inhibitor 8
CAS:HIV-1 integrase inhibitor 8 is an inhibitor of HIV-1 integrase. Integration is a required step in HIV replication [1].
Formula:C21H24O2Purezza:98.91%Colore e forma:SolidPeso molecolare:308.41MMP-2/MMP-9 Inhibitor I
CAS:MMP-2/MMP-9-IN-1: oral IV collagenase inhibitor; IC50: 0.24 μM (MMP-9), 0.31 μM (MMP-2); targets cancer.Formula:C21H19NO4SPurezza:99.98%Colore e forma:SolidPeso molecolare:381.44Ref: TM-T21512
1mg56,00€5mg119,00€10mg177,00€25mg356,00€50mg590,00€100mg888,00€200mg1.198,00€1mL*10mM (DMSO)133,00€MK-8325
CAS:MK-8325 is a potent and orally available HCV NS5A inhibitor with replicative activity against a wide range of genotypes.MK-8325 has demonstrated bioavailabilityFormula:C43H54Cl2F2N8O6SiPurezza:99.61%Colore e forma:SolidPeso molecolare:915.93BAY-43-9695
CAS:BAY-43-9695 is a non-nucleoside compound with anti-human cytomegalovirus (HCMV) activity. It is the major metabolite of BAY-38-4766.Formula:C22H25N3O4SPurezza:99.50% - 99.98%Colore e forma:SolidPeso molecolare:427.52BMS-929075
CAS:BMS-929075 is an orally active HCV NS5B replicase (HCV NS5B replicase) palm site variant inhibitor with potency, high oral bioavailability and pharmacokineticFormula:C31H24F2N4O3Purezza:99.81% - 99.94%Colore e forma:SolidPeso molecolare:538.54Ref: TM-T26863
1mg172,00€5mg432,00€10mg618,00€25mg973,00€50mg1.333,00€100mg1.791,00€500mg3.529,00€1mL*10mM (DMSO)538,00€(2RS)-FPMPA
CAS:(2RS)-FPMPA（FPMPA） has antiviral activity with an IC50 value of 1.85 μM measured in human MT12 cells infected with SHIV (DH4R).Formula:C9H13FN5O4PPurezza:99.9% - >99.99%Colore e forma:SolidPeso molecolare:305.2P32/98 hemifumarate
CAS:P32/98 hemifumarate is a DPP4 inhibitor with hypoglycemic properties and is used in the study of type 2 diabetes.Formula:C22H40N4O6S2Purezza:99.46%Colore e forma:SolidPeso molecolare:520.71CP-544439
CAS:CP-544439 is an inhibitor of matrix metalloproteinase-13, which has an effect on adipose tissue development.Formula:C18H19FN2O6SPurezza:95.02% - 98.66%Colore e forma:SolidPeso molecolare:410.42Uprifosbuvir
CAS:Uprifosbuvir is an inhibitor of uridine nucleotide analog HCV NS5B polymerase.Formula:C22H29ClN3O9PPurezza:99.73% - >99.99%Colore e forma:SolidPeso molecolare:545.91TS-021
CAS:TS-021 is a selective dipeptidyl peptidase 4 (DPP-4) inhibitor with antidiabetic activity for the study of type 2 diabetes.Formula:C17H24FN3O5SPurezza:>99.99% - >99.99%Colore e forma:SolidPeso molecolare:401.45Etarotene
CAS:Etarotene (Arotinoid ethyl sulphone) is an ethylsulfonyl derivative of aloe acid with differentiation-inducing and potentially antitumor activity.Etarotene is aFormula:C25H32O2SPurezza:99.58% - 99.98%Colore e forma:SolidPeso molecolare:396.59BMS-538305 HCl
CAS:BMS-538305 is a potent, selective inhibitor of dipeptidyl peptidase IV (DPP-IV).Formula:C17H27ClN2O2Colore e forma:SolidPeso molecolare:326.86AZD-9819
CAS:AZD-9819 is a neutrophil elastase (HNE) inhibitor applicable for research into chronic obstructive pulmonary disease (COPD).Formula:C25H19F3N6O2Purezza:100% - 99.18%Colore e forma:SolidPeso molecolare:492.45(Rac)-Neurodegenerative Disorder-Targeting Compound 1
CAS:(Rac)-Neurodegenerative Disorder-Targeting Compound 1 is a calpain inhibitor.Formula:C28H28N4O4Colore e forma:SolidPeso molecolare:484.55Ro 31-9790
CAS:Ro 31-9790 is a synthetic inhibitor of metalloproteinase (MMP).Formula:C15H29N3O4Purezza:98%Colore e forma:SolidPeso molecolare:315.41Thrombin inhibitor 1
CAS:Thrombin inhibitor 1 is a potent inhibitor of thrombin (Ki: 0.66 nM, 2xaPTT=0.43 μM).Formula:C22H20Cl2F2N4O3Purezza:98%Colore e forma:SolidPeso molecolare:497.32AA74-1
CAS:AA74-1 is a potent, selective APEH inhibitor that significantly enhances T-cell proliferation by inhibiting APEH activity [1].Formula:C16H28N4O2Purezza:98%Colore e forma:SolidPeso molecolare:308.42JW 480
CAS:JW480 is a potent and selective inhibitor of KIAA1363, a serine hydrolase enzyme.Formula:C22H23NO2Purezza:99.72%Colore e forma:SolidPeso molecolare:333.42Ref: TM-T22883
2mg35,00€5mg49,00€10mg79,00€25mg160,00€50mg259,00€100mg416,00€200mg587,00€1mL*10mM (DMSO)57,00€Flovagatran sodium
CAS:Flovagatran sodium, a thrombin inhibitor, is used potentially for the treatment of thrombosis.Formula:C27H36BN3NaO7Purezza:98%Colore e forma:SolidPeso molecolare:548.4BAY-320
CAS:BAY-320 is a Bub1 inhibitor. With an IC50 of 680 nM for human Bub1 in the presence of 2 mM ATP.Formula:C26H26F2N6O2Purezza:98%Colore e forma:SolidPeso molecolare:492.52SQ 32056
CAS:SQ 32056 is a cathepsin E inhibitor.Formula:C37H56N4O5Purezza:98%Colore e forma:SolidPeso molecolare:636.86BMS-189664 HCl
CAS:BMS-189664 HCl is a selective and orally active thrombin active site inhibitor.Formula:C22H35ClN6O4SPurezza:98%Colore e forma:SolidPeso molecolare:515.07Tyropeptin A-4
CAS:Tyropeptin A-4 is used as a proteasome inhibitor.Formula:C31H41N3O6Purezza:98%Colore e forma:SolidPeso molecolare:551.67NS5A-IN-3
CAS:NS5A-IN-3 is a potent NS5A inhibitor with high efficacy against HCV 1b, good activity on 3a, and strong metabolic stability; superior to daclatasvir.Formula:C44H44N6O8Purezza:98%Colore e forma:SolidPeso molecolare:784.86NS5A-IN-2
CAS:NS5A-IN-2, a potent inhibitor, is highly effective against HCV 1b and shows increased activity for GT 3a with good metabolic stability.Formula:C46H45N7O7Purezza:98%Colore e forma:SolidPeso molecolare:807.89TP0556351
CAS:TP0556351: potent MMP2 inhibitor with 0.2 nM IC50, reduces collagen in pulmonary fibrosis mice.Formula:C50H70N10O16Purezza:98%Colore e forma:SolidPeso molecolare:1067.15LM-030
CAS:LM-030, also known as BPR277, is a novel inhibitor of kallikrein-related peptidase 7 (KLK7) and epidermal elastase 2 (ELA2).Formula:C46H72N8O12Colore e forma:SolidPeso molecolare:929.11HCV-IN-44
CAS:HCV-IN-44 (compound 28) is an inhibitor of the HCV NS5B protein, efficacious in suppressing HCV virus replication and useful for researching HCV infection [1].Formula:C24H26FN3O5SColore e forma:SolidPeso molecolare:487.54MMP3 inhibitor 1
CAS:MMP3 inhibitor 1 is a potent and highly selective inhibitor of MMP-3 (IC50 of 1 nM).Formula:C23H31N3O6SPurezza:98%Colore e forma:SolidPeso molecolare:477.57(1R,4S)-Yimitasvir diphosphate
CAS:Yimitasvir diphosphate, also known as Emitasvir, is an orally-administered inhibitor of the hepatitis C virus (HCV) nonstructural protein 5A (NS5A).Formula:C49H64N8O14P2Colore e forma:SolidPeso molecolare:1051.03MMP13-IN-3
CAS:MMP13-IN-3 is an oral, selective MMP-13 inhibitor with IC50 of 1 nM, >1000x selective, for osteoarthritis treatment.Formula:C24H22N4O5Purezza:99.76%Colore e forma:SolidPeso molecolare:446.46Ref: TM-T16124
1mg93,00€5mg205,00€10mg334,00€25mg587,00€50mg802,00€100mg1.108,00€1mL*10mM (DMSO)227,00€MeOSuc-AAPV-CMK
CAS:MeOSuc-AAPV-CMK (Elastase Inhibitor III) serves as an inhibitor of elastase, as well as cathepsin G and proteinase 3, and impedes leukocyte elastase-mediatedFormula:C22H35ClN4O7Colore e forma:SolidPeso molecolare:502.99Ecallantide
CAS:Ecallantide (DX-88) is a recombinant inhibitor specifically targeting plasma kallikrein, which serves to impede the synthesis of bradykinin.Formula:C305H448N88O91S8Colore e forma:SolidPeso molecolare:7059.88
